KEGG   DRUG: D00332Help
Entry
D00332                      Drug                                   

Name
Gabapentin (JAN/USAN/INN);
Neurontin (TN);
Gralise (TN)
Product
  Generic
GABAPENTIN (AMERISOURCEBERGEN DRUG CORPORATION), GABAPENTIN (Acella Pharmaceuticals), GABAPENTIN (Actavis Elizabeth LLC), GABAPENTIN (Actavis Elizabeth LLC), GABAPENTIN (Actavis Pharma Manufacturing Pvt Ltd. (SOD)), GABAPENTIN (Aidarex Pharmaceuticals LLC), GABAPENTIN (Aidarex Pharmaceuticals LLC), GABAPENTIN (Allied Pharma), GABAPENTIN (American Health Packaging), GABAPENTIN (American Health Packaging), GABAPENTIN (American Health Packaging), GABAPENTIN (Amneal Pharmaceuticals), GABAPENTIN (Amneal Pharmaceuticals of NY LLC), GABAPENTIN (Aphena Pharma Solutions - Tennessee), GABAPENTIN (Aphena Pharma Solutions - Tennessee), GABAPENTIN (Apotex Corp.), GABAPENTIN (Apotex Corp.), GABAPENTIN (Ascend Laboratories), GABAPENTIN (Aurobindo Pharma Limited), GABAPENTIN (Aurobindo Pharma Limited), GABAPENTIN (AvKARE), GABAPENTIN (Blenheim Pharmacal), GABAPENTIN (Blenheim Pharmacal), GABAPENTIN (Blenheim Pharmacal), GABAPENTIN (BluePoint Laboratories), GABAPENTIN (Breckenridge Pharmaceutical), GABAPENTIN (Bryant Ranch Prepack), GABAPENTIN (Bryant Ranch Prepack), GABAPENTIN (Bryant Ranch Prepack), GABAPENTIN (Bryant Ranch Prepack), GABAPENTIN (Bryant Ranch Prepack), GABAPENTIN (Cadila Healthcare Limited), GABAPENTIN (Camber Pharmaceuticals), GABAPENTIN (Camber Pharmaceuticals), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Cardinal Health), GABAPENTIN (Clinical Solutions Wholesale), GABAPENTIN (Clinical Solutions Wholesale), GABAPENTIN (Clinical Solutions Wholesale), GABAPENTIN (Contract Pharmacy Services-PA), GABAPENTIN (Contract Pharmacy Services-PA), GABAPENTIN (Direct Rx), GABAPENTIN (Dispensing Solutions), GABAPENTIN (Exelan Pharmaceuticals), GABAPENTIN (Exelan Pharmaceuticals), GABAPENTIN (Gen-Source Rx), GABAPENTIN (Glenmark Generics), GABAPENTIN (Golden State Medical Supply), GABAPENTIN (Golden State Medical Supply), GABAPENTIN (Golden State Medical Supply), GABAPENTIN (Greenstone LLC), GABAPENTIN (H.J. Harkins Company), GABAPENTIN (H.J. Harkins Company), GABAPENTIN (Hi-Tech Pharmacal), GABAPENTIN (Hikma Pharmaceutical), GABAPENTIN (Hikma Pharmaceutical), GABAPENTIN (Keltman Pharmaceuticals), GABAPENTIN (Kiel Laboratories), GABAPENTIN (Lake Erie Medica & Surgical Supply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical & Surgical S6758upply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical & Surgical Supply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical & Surgical Supply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical & Surgical Supply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical & Surgical Supply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical & Surgical Supply DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical DBA Quality Care Products LLC), GABAPENTIN (Lake Erie Medical DBA Quality Care Products LLC), GABAPENTIN (Liberty Pharmaceuticals), GABAPENTIN (MARKSANS PHARMA LIMITED), GABAPENTIN (Major Pharmaceuticals), GABAPENTIN (Major Pharmaceuticals), GABAPENTIN (McKesson Contract Packaging), GABAPENTIN (McKesson Contract Packaging), GABAPENTIN (McKesson Contract Packaging), GABAPENTIN (McKesson Packaging Services a business unit of McKesson Corporation), GABAPENTIN (McKesson Packaging Services a business unit of McKesson Corporation), GABAPENTIN (McKesson Packaging Services a business unit of McKesson Corporation), GABAPENTIN (MedVantx), GABAPENTIN (MedVantx), GABAPENTIN (MedVantx), GABAPENTIN (Medsource Pharmaceuticals), GABAPENTIN (Mylan Pharmaceuticals), GABAPENTIN (Mylan Pharmaceuticals), GABAPENTIN (NCS HealthCare of KY), GABAPENTIN (NCS HealthCare of KY), GABAPENTIN (NCS HealthCare of KY), GABAPENTIN (New Horizon Rx Group), GABAPENTIN (NorthStar Rx LLC), GABAPENTIN (NorthStar Rx LLC), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (PD-Rx Pharmaceuticals), GABAPENTIN (Pharmaceutica North America), GABAPENTIN (Pharmaceutica North America), GABAPENTIN (Pharmaceutica North America), GABAPENTIN (Physicians Total Care), GABAPENTIN (Physicians Total Care), GABAPENTIN (Preferred Pharmaceuticals), GABAPENTIN (Preferred Pharmaceuticals), GABAPENTIN (Preferred Pharmaceuticals), GABAPENTIN (Preferred Pharmaceuticals), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (REMEDYREPACK), GABAPENTIN (Ranbaxy Pharmaceuticals), GABAPENTIN (Rebel Distributors Corp), GABAPENTIN (Rebel Distributors Corp), GABAPENTIN (Rebel Distributors Corp), GABAPENTIN (Rebel Distributors Corp.), GABAPENTIN (Rebel Distributors Corp.), GABAPENTIN (STAT RX USA LLC), GABAPENTIN (STAT RX USA LLC), GABAPENTIN (STAT RX USA LLC), GABAPENTIN (STAT Rx USA LLC), GABAPENTIN (STAT Rx USA LLC), GABAPENTIN (Solco healthcare U.S.), GABAPENTIN (St Marys Medical Park Pharmacy), GABAPENTIN (St Marys Medical Park Pharmacy), GABAPENTIN (Sun Pharmaceutical Industries Limited), GABAPENTIN (Sun Pharmaceutical Industries Limited), GABAPENTIN (Taro Pharmaceuticals U.S.A.), GABAPENTIN (Teva Pharmaceuticals USA), GABAPENTIN (Teva Pharmaceuticals USA), GABAPENTIN (Unit Dose Services), GABAPENTIN (Unit Dose Services), GABAPENTIN (Unit Dose Services), GABAPENTIN (Unit Dose Services), GABAPENTIN (Unit Dose Services), GABAPENTIN (West-ward Pharmaceutical Corp), GABAPENTIN (West-ward Pharmaceutical Corp), GABAPENTIN (Zydus Pharmaceuticals (USA))
Formula
C9H17NO2
Exact mass
171.1259
Mol weight
171.2368
Structure
Mol fileKCF fileDB searchJmolKegDraw
Activity
Anticonvulsant
Remark
Therapeutic category: 
ATC code: 
Comment
GABA [CPD:C00334] analogue
Target
calcium channel, CACN alpha-2 delta blocker  [HSA:781 9254 55799 93589] [KO:K04858 K04859 K04860 K04861]
  Pathway
hsa04010  MAPK signaling pathway  
 
Interaction
Drug interaction
Structure map
Anticonvulsants
Brite
Therapeutic category of drugs in Japan [BR:br08301]
 1  Agents affecting nervous system and sensory organs
  11  Agents affecting central nervous system
   113  Antiepileptics
    1139  Others
     D00332  Gabapentin (JAN/USAN/INN)
Anatomical Therapeutic Chemical (ATC) classification [BR:br08303]
 N NERVOUS SYSTEM
  N03 ANTIEPILEPTICS
   N03A ANTIEPILEPTICS
    N03AX Other antiepileptics
     N03AX12 Gabapentin
      D00332  Gabapentin (JAN/USAN/INN)
USP drug classification [BR:br08302]
 Anticonvulsants
  Gamma-aminobutyric Acid (GABA) Augmenting Agents
   Gabapentin
    D00332  Gabapentin (JAN/USAN/INN)
Target-based classification of drugs [BR:br08310]
 Ion channels
  Voltage-gated cation channels
   Ca2+ channel, CACN alpha-1, CaVx.x
    voltage-dependent calcium channel [HSA:781 9254 55799 93589] [KO:K04858 K04859 K04860 K04861]
     Gabapentin [ATC:N03AX12]
      D00332  Gabapentin (JAN/USAN/INN)
BRITE hierarchy
Other DBs
CAS: 
60142-96-3
PubChem: 
DrugBank: 
PDB-CCD: 
LigandBox: 
NIKKAJI: 
KCF data Show

ATOM        12
            1   C1z C    25.8300  -23.5200
            2   C1b C    25.8300  -22.1200
            3   C1x C    25.8300  -24.9200
            4   C1x C    24.6400  -22.8200
            5   C1b C    27.0200  -24.2200
            6   C6a C    27.0900  -21.4200
            7   C1x C    24.6400  -25.6200
            8   C1x C    23.3800  -23.5200
            9   N1a N    28.2800  -23.5900
            10  O6a O    27.0900  -20.0900
            11  O6a O    28.2800  -22.1900
            12  C1x C    23.3800  -24.9200
BOND        12
            1     1   2 1
            2     1   3 1
            3     1   4 1
            4     1   5 1
            5     2   6 1
            6     3   7 1
            7     4   8 1
            8     5   9 1
            9     6  10 2
            10    6  11 1
            11    7  12 1
            12    8  12 1

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