| C00989 |
4-Hydroxybutanoic acid; 4-Hydroxybutanoate; 4-Hydroxybutyric acid |
(P) unclassified |
| C01089 |
(R)-3-Hydroxybutanoate; (R)-3-Hydroxybutanoic acid; (R)-3-Hydroxybutyric acid; D-beta-Hydroxybutyric acid |
(P) unclassified |
| C03197 |
(S)-3-Hydroxybutanoate |
(P) unclassified |
| C05984 |
2-Hydroxybutanoic acid; 2-Hydroxybutyrate; 2-Hydroxybutyric acid |
(P) unclassified |
| C06790 |
Trichloroethene; Trichloroethylene; TCE |
(P) unclassified |
| C07521 |
Thiopental |
(P) unclassified |
| C13827 |
Chloroform |
(P) unclassified |
| C17721 |
Vinyl ether |
(P) unclassified |
| C17722 |
Narcobarbital |
(P) unclassified |
| C17723 |
Metabutethamine |
(P) unclassified |
| C17725 |
Heptabarbital |
(P) unclassified |
| D00033 |
Phenol (JP16/USP); Liquefied phenol (JP16); Phenol for disinfection (JP16); Phenol, liquefied; Paoscle (TN); Phenol (TN); Liquefied phenol (TN); Phenol for disinfection (TN) |
(P) unclassified |
| D00049 |
Nicotinic acid (JP16/INN); Niacin (USP); Niacor (TN); Niaspan (TN) |
(P) unclassified |
| D00059 |
Levodopa (JP16/USP/INN); Dopar (TN) |
(P) Target: DRD2 DRD3 |
| D00068 |
Anhydrous ethanol (JP16); Alcohol (USP); Dehydrated ethanol; Ethyl alcohol; Dehydrated ethanol (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D00095 |
Adrenaline (JP16); Epinephrine (USP/INN); Adrenalin (TN); Auvi-q (TN); Epipen (TN) |
(CI) Target: ADRA1D ADRA1B ADRA1A |
| D00102 |
Nitrous oxide (JP16/USP); Nitrous oxide (TN) |
(P) unclassified |
| D00110 |
Cocaine (USP); Cocaine (TN) |
(P) unclassified |
| D00136 |
Haloperidol (JP16/USP/INN); Haldol (TN) |
(P) Enzyme: CYP2D6 CYP3A4 CYP1A2 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00138 |
Scopolamine (INN); Transderm scop (TN) |
(P) unclassified |
| D00140 |
Erythromycin (JP16/USP/INN); EM; Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00197 |
Reserpine (JP16/USP/INN); Apoplon (TN); Serpalan (TN) |
(P) unclassified |
| D00211 |
Rifampicin (JP16/INN); Rifampin (USP); Rifadin (TN); Rimactane (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP2D6 |
| D00225 |
Alprazolam (JP16/USP/INN); Xanax (TN) |
(P) Enzyme: CYP3A4 |
| D00228 |
Amoxapine (JP16/USP/INN); Asendin (TN) |
(P) Enzyme: CYP2D6 CYP1A2 CYP3A4 / CYP inhibition: CYP2D6 |
| D00241 |
Baclofen (JP16/USP/INN); Kemstro (TN); Lioresal (TN) |
(P) unclassified |
| D00250 |
Capsaicin (JAN/USP); Zostrix (TN) |
(P) unclassified |
| D00252 |
Carbamazepine (JP16/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00253 |
Carbidopa hydrate - levodopa mixt; Parcopa (TN); Sinemet (TN) |
(P) unclassified |
| D00265 |
Chloral hydrate (JP16/USP); Noctec (TN) |
(P) unclassified |
| D00267 |
Chlordiazepoxide (JP16/USP/INN); Libritabs (TN) |
(P) unclassified |
| D00270 |
Chlorpromazine (USP/INN); Thorazine (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00276 |
Clarithromycin (JP16/USP/INN); CAM; Biaxin (TN) |
(CI) Enzyme: CYP3A4 |
| D00280 |
Clonazepam (JP16/USP/INN); Klonopin (TN) |
(P) unclassified |
| D00282 |
Clotrimazole (JP16/USP/INN); Lotrimin (TN); Mycelex (TN) |
(CI) unclassified |
| D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) Enzyme: CYP1A2 CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D00293 |
Diazepam (JP16/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 |
| D00294 |
Diazoxide (JAN/USP/INN); Hyperstat (TN) |
(P) unclassified |
| D00308 |
Droperidol (JP16/USP/INN); Droleptan (TN); Inapsine (TN) |
(P) Target: DRD2 |
| D00311 |
Estazolam (JP16/USAN/INN); ProSom (TN) |
(P) Enzyme: CYP3A4 |
| D00320 |
Fentanyl (JAN/USAN/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 |
| D00322 |
Fluconazole (JP16/USAN/INN); Diflucan (TN) |
(CI,P) Enzyme: CYP3A4 |
| D00329 |
Flurazepam (JAN/INN); Insumin (TN) |
(P) unclassified |
| D00338 |
Halazepam (USAN/INN); Paxipam (TN) |
(P) unclassified |
| D00350 |
Itraconazole (JP16/USAN); Itrizole (TN); Sporanox (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00351 |
Ketoconazole (JP16/USP); Nizoral (TN); Xolegel (TN) |
(CI) Enzyme: CYP3A4 |
| D00358 |
Lidocaine (JP16/USP/INN); Dentipatch (TN); Xylocaine (TN) |
(P) Enzyme: CYP1A2 CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D00365 |
Lorazepam (JP16/USP/INN); Ativan (TN) |
(P) unclassified |
| D00370 |
Temazepam (USP/INN); Restoril (TN) |
(P) Enzyme: CYP3A4 |
| D00373 |
Thioridazine (USP/INN); Mellaril-S (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00374 |
Tiotixene (JAN); Thiothixene (USP); Navane (TN) |
(P) Target: DRD2 |
| D00376 |
Meprobamate (JAN/USP/INN); Equanil (TN); Miltown (TN) |
(P) unclassified |
| D00387 |
Triazolam (JAN/USP/INN); Halcion (TN) |
(P) Enzyme: CYP3A4 |
| D00388 |
Triclofos sodium (JP16/USAN); Tricloryl (TN) |
(P) unclassified |
| D00390 |
Triflupromazine (USP/INN); Vesprin (TN) |
(P) Target: DRD2 |
| D00402 |
Methocarbamol (JAN/USP/INN); Delaxin (TN); Robaxin (TN) |
(P) unclassified |
| D00403 |
Levomepromazine (USAN/INN); Methotrimeprazine (USP); Levoprome (TN) |
(P) Enzyme: CYP2D6 / Target: ADRA1D ADRA1B ADRA1A DRD2 / CYP inhibition: CYP2D6 |
| D00416 |
Miconazole (JP16/USP/INN); Monistat (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00426 |
Risperidone (JP16/USAN/INN); Risperdal (TN) |
(P) Enzyme: CYP2D6 CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 / CYP inhibition: CYP2D6 |
| D00427 |
Ritonavir (JAN/USAN/INN); Norvir (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP2D6 |
| D00429 |
Saquinavir (JAN/USP/INN); Fortovase (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00430 |
Secobarbital (USP/INN); Seconal (TN) |
(P) unclassified |
| D00454 |
Olanzapine (JAN/USAN/INN); Zyprexa (TN) |
(P) Enzyme: CYP1A2 CYP2D6 / Target: ADRA1D ADRA1B ADRA1A DRD2 DRD3 / CYP inhibition: CYP2D6 |
| D00457 |
Quazepam (JAN/USP/INN); Doral (TN) |
(P) Enzyme: CYP3A4 |
| D00458 |
Quetiapine fumarate (JP16/USAN); Seroquel (TN) |
(P) Enzyme: CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 DRD3 |
| D00464 |
Oxazepam (JAN/USP/INN); Serax (TN) |
(P) unclassified |
| D00470 |
Prazepam (JP16/USAN/INN); Centrax (TN) |
(P) unclassified |
| D00474 |
Primidone (JP16/USP/INN); Mysoline (TN) |
(P) unclassified |
| D00479 |
Prochlorperazine maleate (JP16/USP); Compazine (TN) |
(P) Target: DRD2 |
| D00480 |
Promethazine hydrochloride (JP16/USP); Phenergan (TN); Promethegan (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D00493 |
Prochlorperazine (JAN/USP/INN); Compro (TN) |
(P) Target: DRD2 |
| D00498 |
Pentazocine (JP16/USP/INN); Fortral (TN) |
(P) unclassified |
| D00499 |
Pentobarbital (USP/INN); Nembutal (TN) |
(P) unclassified |
| D00500 |
Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) |
(P) unclassified |
| D00502 |
Pergolide mesilate (JAN); Pergolide mesylate (USP); Permax (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00503 |
Perphenazine (JP16/USP/INN); Trilafon (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00506 |
Phenobarbital (JP16/USP/INN); Luminal (TN) |
(P) CYP induction: CYP1A2 CYP3A4 |
| D00514 |
Dexmedetomidine (USAN/INN); Dexdor (TN); Precedex (TN) |
(P) unclassified |
| D00515 |
Nitroglycerin (JP16/USP); Glyceryl trinitrate; Minitran (TN); Nitro-bid (TN); Nitro-dur (TN); Nitromist (TN); Transderm-nitro (TN) |
(P) unclassified |
| D00516 |
Isosorbide dinitrate (JP16/USP/INN); Dilatrate-sr (TN); Isordil (TN) |
(P) unclassified |
| D00520 |
Dimenhydrinate (JP16/USP/INN); Dramamine (TN) |
(P) unclassified |
| D00530 |
Zaleplon (JAN/USAN/INN); Sonata (TN) |
(P) Enzyme: CYP3A4 |
| D00531 |
Nitrazepam (JP16/USAN/INN); Benzalin (TN); Nitrazepam (TN) |
(P) unclassified |
| D00532 |
Glutethimide (JAN/INN); Doriden (TN) |
(P) unclassified |
| D00537 |
Topiramate (JAN/USAN/INN); Topamax (TN); Trokendi xr (TN) |
(P) Enzyme: CYP3A4 |
| D00542 |
Halothane (JP16/USP/INN); Fluothane (TN) |
(P) Enzyme: CYP3A4 |
| D00543 |
Enflurane (JP16/USP/INN); Ethrane (TN) |
(P) unclassified |
| D00545 |
Isoflurane (JP16/USP/INN); Forane (TN) |
(P) unclassified |
| D00546 |
Desflurane (JAN/USP/INN); Suprane (TN) |
(P) unclassified |
| D00547 |
Sevoflurane (JP16/USAN/INN); Ultane (TN) |
(P) Enzyme: CYP3A4 |
| D00548 |
Etomidate (USAN/INN); Amidate (TN) |
(P) unclassified |
| D00549 |
Propofol (JAN/USAN/INN); Diprivan (TN) |
(P) unclassified |
| D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN) |
(P) Enzyme: CYP3A4 |
| D00551 |
Tetracaine (USP/INN); Amethocaine; Amethocaine (TN) |
(P) unclassified |
| D00552 |
Ethyl aminobenzoate (JP16); Benzocaine (USP/INN); Parathesin (TN) |
(P) unclassified |
| D00553 |
Propitocaine (JAN); Prilocaine (USP/INN) |
(P) unclassified |
| D00555 |
Amobarbital (JP16/INN); Isomytal (TN) |
(P) unclassified |
| D00557 |
Methaqualone (JAN/USAN/INN) |
(P) unclassified |
| D00559 |
Pramipexole hydrochloride hydrate (JAN); Pramipexole hydrochloride (USAN); Mirapex (TN) |
(P) Target: DRD2 DRD3 |
| D00560 |
Pimozide (JP16/USP/INN); Orap (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / Target: ADRA1D ADRA1B ADRA1A DRD2 DRD3 / CYP inhibition: CYP2D6 |
| D00561 |
Sertindole (USAN/INN); SerLect (TN) |
(P) Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D00578 |
Voriconazole (JAN/USAN/INN); Vfend (TN) |
(CI) Enzyme: CYP3A4 |
| D00604 |
Clonidine hydrochloride (JP16/USP); Catapres (TN) |
(P) unclassified |
| D00605 |
Guanabenz acetate (JP16/USP); Wytensin (TN) |
(P) unclassified |
| D00613 |
Fenoldopam mesylate (USP); Corlopam (TN) |
(P) unclassified |
| D00630 |
Isosorbide mononitrate (JP16/USP/INN); Imdur (TN); Ismo (TN) |
(P) unclassified |
| D00631 |
Bepridil hydrochloride hydrate (JAN); Bepridil hydrochloride (USAN); Vascor (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D00633 |
Dopamine hydrochloride (JP16/USP); Actopamin (TN); Intropin (TN) |
(P) Target: DRD2 DRD3 |
| D00664 |
Cetirizine hydrochloride (JP16/USAN); Zyrtec (TN) |
(P) unclassified |
| D00665 |
Chlorpheniramine maleate (JP16/USP); Chlor-trimeton (TN); Teldrin (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D00666 |
Clemastine fumarate (JP16/USP); Tavist (TN) |
(P) unclassified |
| D00668 |
d-Chlorpheniramine maleate (JP16); Dexchlorpheniramine maleate (USP); Mylaramine (TN); Polaramine (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D00669 |
Diphenhydramine hydrochloride (JP16/USP); Benadryl (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D00672 |
Hydroxyzine hydrochloride (JP16/USP); Atarax (TN); Vistaril (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP2D6 |
| D00679 |
Ergotamine tartrate (JP16/USP); Ergomar (TN) |
(P) Enzyme: CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D00693 |
Chlordiazepoxide hydrochloride (JAN/USP); Librium (TN) |
(P) unclassified |
| D00694 |
Clorazepate dipotassium (JP16/USP); Tranxene (TN) |
(P) unclassified |
| D00695 |
Flurazepam hydrochloride (USP); Flurazepam dihydrochloride; Dalmane (TN) |
(P) unclassified |
| D00696 |
Midazolam hydrochloride (USAN); Versed (TN) |
(P) Enzyme: CYP3A4 |
| D00698 |
Aprobarbital (INN); Alurate (TN) |
(P) unclassified |
| D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) unclassified |
| D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) CYP induction: CYP1A2 CYP3A4 |
| D00702 |
Buspirone hydrochloride (USP); Buspar (TN) |
(P) unclassified |
| D00704 |
Ethchlorvynol (JAN/USP/INN); Placidyl (TN) |
(P) unclassified |
| D00705 |
Paraldehyde (USP); Paral (TN) |
(P) unclassified |
| D00706 |
Zolpidem tartrate (JP16/USAN); Ambien (TN); Intermezzo (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
| D00711 |
Ketamine hydrochloride (JP16/USP); Ketalar (TN) |
(P) unclassified |
| D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) unclassified |
| D00713 |
Thiamylal sodium (JP16); Surital (TN) |
(P) unclassified |
| D00714 |
Thiopental sodium (JP16/USP/INN); Pentothal (TN) |
(P) unclassified |
| D00726 |
Metoclopramide (JP16/INN); Elieten (TN); Terperan (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00732 |
Chloroprocaine hydrochloride (USP); Nesacaine (TN) |
(P) unclassified |
| D00733 |
Dibucaine (USP); Cinchocaine (INN); Nupercaine (TN) |
(P) unclassified |
| D00735 |
Dyclonine hydrochloride (USP); Dyclone (TN) |
(P) unclassified |
| D00737 |
Etidocaine hydrochloride; Duranest (TN) |
(P) unclassified |
| D00738 |
Mepivacaine hydrochloride (JP16/USP); Carbocaine (TN); Polocaine (TN); Scandonest plain (TN) |
(P) unclassified |
| D00740 |
Procaine hydrochloride (JP16/USP); Novocain (TN) |
(P) unclassified |
| D00741 |
Tetracaine hydrochloride (JP16/USP); Protocaine hydrochloride (TN) |
(P) unclassified |
| D00754 |
Thalidomide (JAN/USP/INN); Thalomid (TN); Thaled (TN) |
(P) unclassified |
| D00770 |
Chlorphenesin carbamate (JP16/USAN); Maolate (TN) |
(P) unclassified |
| D00776 |
Tizanidine hydrochloride (JP16/USAN); Zanaflex (TN) |
(P) Enzyme: CYP1A2 |
| D00780 |
Bromocriptine mesilate (JP16); Bromocriptine mesylate (USP); Parlodel (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D00784 |
Ropinirole hydrochloride (JAN/USAN); Requip (TN) |
(P) Enzyme: CYP1A2 / Target: DRD2 |
| D00787 |
Trihexyphenidyl hydrochloride (JP16/USP); Artane (TN) |
(P) unclassified |
| D00788 |
Acetophenazine maleate (USAN); Tindal (TN) |
(P) unclassified |
| D00789 |
Chlorpromazine hydrochloride (JP16/USP); Sonazine (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00790 |
Chlorprothixene (JAN/USAN/INN); Taractan (TN) |
(P) unclassified |
| D00791 |
Fluphenazine hydrochloride (JAN/USP); Prolixin (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00792 |
Fluphenazine enanthate (JP16/USP); Prolixin enanthate (TN) |
(P) Target: DRD2 |
| D00793 |
Fluphenazine decanoate (JAN/USP); Prolixin decanoate (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00794 |
Loxapine succinate (USP); Loxitane (TN) |
(P) Target: DRD2 |
| D00795 |
Mesoridazine besylate (USP); Serentil (TN) |
(P) unclassified |
| D00796 |
Molindone hydrochloride (USP); Moban (TN) |
(P) Target: DRD2 |
| D00797 |
Promazine hydrochloride (USP); Sparine (TN) |
(P) Target: DRD2 |
| D00798 |
Thioridazine hydrochloride (JP16/USP); Mellaril (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D00799 |
Trifluoperazine hydrochloride (JAN/USP); Stelazine (TN) |
(P) Target: DRD2 |
| D00800 |
Triflupromazine hydrochloride (JAN/USP); Vesprin (TN) |
(P) Target: DRD2 |
| D00801 |
Lithium carbonate (JP16/USP); Eskalith (TN); Lithobid (TN) |
(P) unclassified |
| D00809 |
Amitriptyline hydrochloride (JP16/USP); Elavil (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D00811 |
Clomipramine hydrochloride (JP16/USP); Anafranil (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D00815 |
Imipramine hydrochloride (JP16/USP); Tofranil (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D00816 |
Nortriptyline hydrochloride (JP16/USP/INN); Pamelor (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D00818 |
Maprotiline hydrochloride (JP16/USP); Ludiomil (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D00820 |
Trazodone hydrochloride (JAN/USP); Desyrel (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D00824 |
Fluvoxamine maleate (JP16/USAN); Luvox (TN) |
(CI) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 CYP1A2 |
| D00825 |
Sertraline hydrochloride (JAN/USAN); Zoloft (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP2D6 |
| D00835 |
Alfentanil hydrochloride (USP); Alfenta (TN) |
(P) unclassified |
| D00836 |
Buprenorphine hydrochloride (JP16/USP); Buprenex (TN) |
(P) unclassified |
| D00842 |
Morphine sulfate hydrate (JP16); Morphine sulfate (USP); Morphine sulfate pentahydrate; Astramor PH (TN); Avinza (TN); Depodur (TN); Kadian (TN); MS contin (TN) |
(P) unclassified |
| D00845 |
Sufentanil citrate (USP); Sufenta (TN) |
(P) unclassified |
| D00851 |
Erythromycin estorate (JAN); Erythromycin estolate (USP); Ilosone (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00854 |
Quinupristin - dalfopristin mixt; Synercid (TN) |
(CI) Enzyme: CYP3A4 |
| D00874 |
Moxifloxacin hydrochloride (JAN/USAN); MFLX; Avelox (TN); Vigamox (TN) |
(P) unclassified |
| D00880 |
Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) |
(CI) unclassified |
| D00881 |
Econazole nitrate (JAN/USP); Spectazole (TN) |
(CI) unclassified |
| D00882 |
Miconazole nitrate (JP16/USP); MCZ; Micatin (TN); Monistat (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00885 |
Oxiconazole nitrate (JAN/USAN); Oxistat (TN) |
(CI) unclassified |
| D00886 |
Sulconazole nitrate (JAN/USP); Exelderm (TN) |
(CI) unclassified |
| D00888 |
Terconazole (USAN/INN); Terazol 3 (TN) |
(CI) unclassified |
| D00890 |
Tioconazole (JAN/USP/INN); Vagistat-1 (TN) |
(CI) unclassified |
| D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(CI) Enzyme: CYP3A4 |
| D00897 |
Indinavir sulfate (USAN); Crixivan (TN) |
(CI) Enzyme: CYP3A4 |
| D00899 |
Nelfinavir mesilate (JAN); Nelfinavir mesylate (USAN/INN); Viracept (TN) |
(CI) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D00969 |
Meloxicam (JAN/USAN/INN); Mobic (TN) |
(P) Enzyme: CYP3A4 |
| D00987 |
Cabergoline (JAN/USAN/INN); Cabaser (TN); Dostinex (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D01044 |
Flupentixol (INN); Flupenthixol; Depixol (TN) |
(P) Target: DRD2 |
| D01051 |
Spiperone (JAN/USAN); Spiropitan (TN) |
(P) Target: DRD2 |
| D01071 |
Hexobarbital (JAN/INN) |
(P) unclassified |
| D01096 |
Hydroxyzine pamoate (JP16/USP); Atarax-P (TN); Vistaril pamoate (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP2D6 |
| D01101 |
Bromperidol (JAN/USAN/INN); Impromen (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D01105 |
Moperone hydrochloride (JAN); Luvatren (TN) |
(P) Target: DRD2 |
| D01107 |
Milnacipran hydrochloride (JAN/USAN); Savella (TN); Toledomin (TN) |
(P) unclassified |
| D01118 |
Profenamine hydrochloride (JAN); Ethopropazine hydrochloride; Parkin (TN); Parsidol (TN) |
(P) unclassified |
| D01150 |
Methyprylon (JAN/INN); Noludar (TN) |
(P) unclassified |
| D01160 |
Saquinavir mesilate (JAN); Saquinavir mesylate (USP); Invirase (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01164 |
Aripiprazole (JAN/USAN/INN); Abilify (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D01172 |
Diphenylpyraline hydrochloride (JAN); Hispril (TN); Vena (TN) |
(P) unclassified |
| D01176 |
Blonanserin (JAN/INN); AD 5423 |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D01177 |
Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) |
(P) unclassified |
| D01179 |
Duloxetine hydrochloride (JAN/USAN); Cymbalta (TN) |
(P) Enzyme: CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D01205 |
Dexmedetomidine hydrochloride (JAN/USAN); Precedex (TN) |
(P) unclassified |
| D01219 |
Oxypertine (JAN/USAN/INN); Forit (TN) |
(P) unclassified |
| D01226 |
Sulpiride (JP16/USAN/INN); Dogmatyl (TN) |
(P) Target: DRD2 DRD3 |
| D01230 |
Flunitrazepam (JP16/USAN/INN); Rohypnol (TN) |
(P) unclassified |
| D01231 |
Piroheptine hydrochloride (JAN); Trimol (TN) |
(P) unclassified |
| D01243 |
Propitocaine hydrochloride (JAN); Prilocaine hydrochloride (USP); Citanest (TN) |
(P) unclassified |
| D01245 |
Bromazepam (JP16/USAN/INN); Lectopam (TN) |
(P) Enzyme: CYP3A4 |
| D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP2D6 |
| D01254 |
Tofisopam (JP16/INN); Emandaxin (TN) |
(P) Enzyme: CYP3A4 |
| D01268 |
Cloxazolam (JP16/INN); Sepazon (TN) |
(P) unclassified |
| D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(CI) Enzyme: CYP3A4 |
| D01277 |
Droxidopa (JP16/INN); Dops (TN) |
(P) unclassified |
| D01278 |
Oxazolam (JP16/INN); Serenal (TN) |
(P) unclassified |
| D01279 |
Flutoprazepam (JP16/INN); Restas (TN) |
(P) unclassified |
| D01285 |
Lofepramine hydrochloride (JAN/USAN); Amplit (TN) |
(P) unclassified |
| D01286 |
Flutazolam (JAN/INN); Coreminal (TN) |
(P) unclassified |
| D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
| D01292 |
Medazepam (JP16/INN); Pamnace (TN) |
(P) unclassified |
| D01293 |
Ethyl loflazepate (JAN/INN); Meilax (TN) |
(P) Enzyme: CYP3A4 |
| D01310 |
Secobarbital sodium (JAN/USP); Seconal sodium (TN) |
(P) unclassified |
| D01316 |
Mexazolam (JAN/INN); Melex (TN) |
(P) Enzyme: CYP3A4 |
| D01321 |
Zotepine (JAN/INN); Setous (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D01324 |
Mequitazine (JP16/INN); Kitazemin (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D01328 |
Clotiazepam (JP16/INN); Rize (TN) |
(P) unclassified |
| D01332 |
Ketotifen fumarate (JP16/USAN); Zaditen (TN) |
(P) unclassified |
| D01348 |
Terguride (JAN/INN); Teluron (TN) |
(P) Target: DRD2 |
| D01354 |
Fludiazepam (JP16/INN); Erispan (TN) |
(P) unclassified |
| D01355 |
Tramadol hydrochloride (JAN/USAN); Ultram (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D01358 |
Mianserin hydrochloride (JAN/USAN); Tetramide (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / Target: ADRA1D ADRA1B ADRA1A / CYP inhibition: CYP2D6 |
| D01361 |
Erythromycin ethylsuccinate (JP16/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01372 |
Zopiclone (JAN/INN); Amoban (TN); Zopiclone (TN) |
(P) Enzyme: CYP3A4 |
| D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) unclassified |
| D01383 |
Pethidine hydrochloride (JP16); Meperidine hydrochloride (USP); Demerol (TN) |
(P) unclassified |
| D01389 |
Clofedanol hydrochloride (JP16); Chlophedianol hydrochloride (USAN); Coldrin (TN) |
(P) unclassified |
| D01391 |
Bromovalerylurea (JP16); Bromisoval (INN); Bromisovalum; Bromovalerylurea (TN); Bromural (TN); Brovarin (TN) |
(P) unclassified |
| D01399 |
Fentanyl citrate (JP16/USP); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 |
| D01408 |
Flurazepam hydrochloride (JP16); Flurazepam monohydrochloride; Dalmate (TN) |
(P) unclassified |
| D01412 |
Perazine maleate (JAN) |
(P) unclassified |
| D01425 |
Lopinavir (JAN/USAN/INN) |
(CI) CYP inhibition: CYP2D6 |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(CI) Enzyme: CYP3A4 |
| D01441 |
Imatinib mesilate (JAN); Imatinib mesylate (USAN); Gleevec (TN); Glivec (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D01447 |
Thioproperazine mesilate (JAN); Thioproperazine mesylate |
(P) Target: DRD2 |
| D01448 |
Trifluoperazine maleate (JAN); Trifluoperazine (TN) |
(P) Target: DRD2 |
| D01449 |
Carpipramine maleate (JAN); Defekton (TN) |
(P) unclassified |
| D01450 |
Bupivacaine hydrochloride hydrate (JP16); Bupivacaine hydrochloride (USP); Marcaine (TN) |
(P) Enzyme: CYP3A4 |
| D01451 |
Scopolamine butylbromide (JP16); Butylscopolamine bromide; Buscopan (TN) |
(P) unclassified |
| D01460 |
Homochlorcyclizine hydrochloride (JP16); Homochlorcyclizine dihydrochloride; SA 97 dihydrochloride; Homoclomin (TN) |
(P) unclassified |
| D01462 |
Lisuride maleate (JAN) |
(P) Target: DRD2 |
| D01465 |
Nizofenone fumarate (JAN); Ekonal (TN) |
(P) unclassified |
| D01468 |
Nemonapride (JAN/INN); Emilace (TN) |
(P) Target: DRD2 DRD3 |
| D01481 |
Dihydrocodeine phosphate (JP16); Dihydro (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D01482 |
Pipamperone hydrochloride (JAN) |
(P) Target: DRD2 |
| D01485 |
Propericiazine (JAN); Periciazine; Neuleptil (TN) |
(P) Target: DRD2 |
| D01496 |
Oxymetebanol (JAN); Drotebanol (INN); Metebanyl (TN) |
(P) unclassified |
| D01505 |
Talipexole hydrochloride (JAN); Domin (TN) |
(P) Target: DRD2 |
| D01514 |
Etizolam (JP16/INN); Sedekopan (TN) |
(P) Enzyme: CYP3A4 |
| D01520 |
Levomepromazine hydrochloride (JAN/USAN); Nozinan (TN) |
(P) Enzyme: CYP2D6 / Target: ADRA1D ADRA1B ADRA1A DRD2 / CYP inhibition: CYP2D6 |
| D01522 |
Tiapride hydrochloride (JP16); Gramalil (TN) |
(P) Target: DRD2 |
| D01546 |
Dosulepin hydrochloride (JAN); Dothiepin hydrochloride (USAN); Dosulepin (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D01548 |
Mosapramine hydrochloride (JAN); Cremin (TN) |
(P) Target: DRD2 |
| D01564 |
Rilmazafone hydrochloride hydrate (JAN); Rilmazafone hydrochloride dihydrate; Rilmazafone hydrochloride; Rhythmy (TN) |
(P) unclassified |
| D01593 |
Nimetazepam (JAN/INN); Erimin (TN) |
(P) unclassified |
| D01597 |
Clotiapine (JAN/INN); Clothiapine (USAN); Entumin (TN) |
(P) unclassified |
| D01657 |
Lormetazepam (JAN/USAN/INN); Loramet (TN) |
(P) unclassified |
| D01731 |
Potassium bromide (JP16); Potassium bromide (TN) |
(P) unclassified |
| D01740 |
Barbital (JP16/INN); Barbital (TN) |
(P) unclassified |
| D01744 |
Brotizolam (JP16/USAN/INN); Lendormin (TN) |
(P) Enzyme: CYP3A4 |
| D01745 |
Domperidone (JP16/USAN/INN); Motilium (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D01758 |
Haloxazolam (JP16/INN); Somelin (TN) |
(P) unclassified |
| D01773 |
Oxatomide (JAN/USAN/INN); Celtect (TN) |
(P) unclassified |
| D01782 |
Triprolidine hydrochloride hydrate (JAN); Triprolidine hydrochloride (USP); Venen (TN) |
(P) unclassified |
| D01785 |
Pirmenol hydrochloride hydrate (JAN); Pimenol (TN) |
(P) unclassified |
| D01807 |
Mebutamate (JAN/USAN); Capla (TN); Dormate (TN) |
(P) unclassified |
| D01860 |
Perazine dimalonate (JAN) |
(P) unclassified |
| D01871 |
Metixene hydrochloride (JAN); Methixene hydrochloride (USAN); Methixene hydrochloride hydrete; Trest (TN) |
(P) unclassified |
| D01879 |
Eptazocine hydrobromide (JAN); Sedapain (TN) |
(P) unclassified |
| D01898 |
Haloperidol decanoate (JAN/USAN); Halomonth (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D01901 |
Xenon (JAN); Xenopure (TN) |
(P) unclassified |
| D01902 |
Dimetotiazine mesilate (JAN); Fonazine mesylate (USAN); Banistyl (TN) |
(P) unclassified |
| D01939 |
Ziprasidone hydrochloride hydrate (JAN); Ziprasidone hydrochloride (USAN); Geodon (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D02004 |
Apomorphine hydrochloride hydrate (JAN); Apomorphine hydrochloride (USP); Apokyn (TN); Ixense (TN); Uprima (TN) |
(P) Target: DRD2 |
| D02008 |
Tadalafil (JAN/USAN/INN); Adcirca (TN); Cialis (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D02009 |
Erythromycin lactobionate (JP16/USP); EML; Erythrocin (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02022 |
Prochlorperazine mesilate (JAN); Prochlorperazine dimethanesulfonate; Novamin (TN) |
(P) Target: DRD2 |
| D02034 |
Setiptiline maleate (JAN); Tecipul (TN) |
(P) Target: ADRA1D ADRA1B ADRA1A |
| D02035 |
Timiperone (JAN); Tolopelon (TN) |
(P) Target: DRD2 |
| D02037 |
Perphenazine maleate (JP16); PZC (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D02055 |
Sodium bromide (JP16); Sodium bromide (TN) |
(P) unclassified |
| D02064 |
Pridinol mesilate (JAN); Pridinol methanesulfonate; Konlax (TN) |
(P) unclassified |
| D02071 |
Scopolamine hydrobromide hydrate (JP16); Scopolamine hydrobromide (USP); Scopolamine hydrobromide trihydrate; Hysco (TN); Isopto hyoscine (TN) |
(P) unclassified |
| D02076 |
Brimonidine tartrate (JAN/USAN); Alphagan (TN) |
(P) unclassified |
| D02086 |
Lidocaine injection (JP16); Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D02100 |
Ziprasidone mesylate (USAN); Ziprasidone mesylate hydrate; Geodon (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D02101 |
Codeine phosphate hydrate (JP16); Codeine phosphate (USP); Codeine (TN) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP2D6 |
| D02106 |
Arsenic trioxide (JP16/USAN); Trisenox (TN) |
(P) unclassified |
| D02135 |
Levodopa - benserazide hydrochloride mixt; Madopar (TN) |
(P) unclassified |
| D02162 |
Chlorprothixene hydrochloride (JAN) |
(P) unclassified |
| D02163 |
Fluphenazine maleate (JAN); Flumezin (TN) |
(P) Target: DRD2 |
| D02175 |
Compound oxycodone (JP16); Pavinal (TN) |
(P) unclassified |
| D02182 |
Cocaine hydrochloride (JP16/USP); Cocaine hydrochloride (TN) |
(P) unclassified |
| D02184 |
Erythromycin stearate (JP16/USP); ES; Bristamycin (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02205 |
Ethylmorphine hydrochloride hydrate (JP16); Ethylmorphine hydrochloride dihydrate; Ethylmorphine hydrochloride (TN) |
(P) Enzyme: CYP3A4 |
| D02208 |
Sultopride hydrochloride (JAN); Sultopride monohydrochloride; Barnetil (TN) |
(CI,P) Target: DRD2 |
| D02211 |
Dihydroergotamine mesilate (JP16); Dihydroergotamine mesylate (USP); Migranal (TN) |
(P) Enzyme: CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D02213 |
Metoclopramide hydrochloride (JAN); Metoclopramide dihydrochloride monohydrate; Primperan (TN); Reglan (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D02227 |
Pentazocine hydrochloride (JAN/USP); Sosegon (TN); Talacen (TN) |
(P) unclassified |
| D02229 |
Sildenafil citrate (JAN/USAN); Revatio (TN); Viagra (TN) |
(P) Enzyme: CYP3A4 |
| D02234 |
Cyproheptadine hydrochloride (JP16/USP); Periactin (TN) |
(P) unclassified |
| D02236 |
Flupentixol dihydrochloride (JAN) |
(P) Target: DRD2 |
| D02245 |
Alimemazine tartrate (JP16); Trimeprazine tartrate (USP); Alimezine (TN) |
(P) unclassified |
| D02246 |
Biperiden hydrochloride (JP16/USP); Tasmolin (TN) |
(P) unclassified |
| D02247 |
Biperiden lactate (JAN/USP); Tasmolin (TN) |
(P) unclassified |
| D02248 |
Levomepromazine maleate (JP16/USAN); Hirnamin (TN) |
(P) Enzyme: CYP2D6 / Target: ADRA1D ADRA1B ADRA1A DRD2 / CYP inhibition: CYP2D6 |
| D02249 |
Emedastine difumarate (JP16/USP); Daren (TN); Emadine (TN) |
(P) unclassified |
| D02252 |
Amobarbital sodium (JAN/USP); Amytal sodium (TN) |
(P) unclassified |
| D02253 |
Pentobarbital calcium (JP16); Ravona (TN) |
(P) unclassified |
| D02260 |
Paroxetine hydrochloride hydrate (JAN); Paxil (TN) |
(CI) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D02271 |
Morphine hydrochloride hydrate (JP16); Morphine hydrochloride trihydrate; Anpec (TN) |
(P) unclassified |
| D02274 |
Dantrolene sodium hydrate (JP16); Dantrolene sodium (USAN); Dantrium (TN) |
(P) Enzyme: CYP1A2 |
| D02340 |
Loxapine (USAN/INN); Adasuve (TN) |
(P) Target: DRD2 |
| D02361 |
Propiomazine (USAN/INN) |
(P) unclassified |
| D02362 |
Paroxetine (USP/INN); Paroxetine (TN) |
(CI) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D02371 |
Clocapramine hydrochloride hydrate (JP16); Clofekton (TN) |
(P) Target: DRD2 |
| D02372 |
Perospirone hydrochloride hydrate (JAN); Lullan (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D02408 |
Trimipramine maleate (JAN/USAN); Surmontil (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D02497 |
Fosamprenavir (INN) |
(CI) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D02498 |
Lopinavir mixture with ritonavir; Lopinavir - ritonavir mixt; Kaletra (TN) |
(CI) unclassified |
| D02523 |
Erythromycin acistrate (USAN); EA; Erasis (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02524 |
Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02525 |
Erythromycin propionate (USAN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02555 |
Posaconazole (USAN/INN); Noxafil (TN) |
(CI) unclassified |
| D02567 |
Escitalopram oxalate (JAN/USAN); Lexapro (TN) |
(CI) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D02604 |
Acepromazine maleate (USP) |
(P) unclassified |
| D02608 |
Perazine fendizoate (JAN) |
(P) unclassified |
| D02609 |
Prochlorperazine edisylate (USP); Compazine syrup (TN) |
(P) Target: DRD2 |
| D02611 |
Phenoperidine (INN) |
(P) unclassified |
| D02612 |
Thiothixene hydrochloride (USP); Thiothixene dihydrochloride dihydrate; Tiotixene dihydrochloride; Thiothixene hydrochloride (TN) |
(P) Target: DRD2 |
| D02613 |
Clopenthixol (USAN) |
(P) Target: DRD2 |
| D02615 |
Chlorpromazine hydrochloride - promethazine hydrochloride - phenobarbital mixt; Vegetamin (TN) |
(P) unclassified |
| D02618 |
Butobarbital (BAN); Butethal; Neonal (TN) |
(P) unclassified |
| D02619 |
Carbromal (INN); Adalin (TN) |
(P) unclassified |
| D02621 |
Fluanisone (INN) |
(P) unclassified |
| D02622 |
Pipamperone (USAN/INN); Floropipamide |
(P) Target: DRD2 |
| D02623 |
Moperone (INN) |
(P) Target: DRD2 |
| D02624 |
Eszopiclone (JAN/USAN/INN); Estorra (TN); Lunesta (TN) |
(P) unclassified |
| D02625 |
Trifluperidol (USAN/INN); Triperidol (TN) |
(P) Target: DRD2 |
| D02626 |
Bromperidol decanoate (USAN) |
(P) Target: DRD2 |
| D02627 |
Benperidol (USAN/INN); Anquil (TN) |
(P) unclassified |
| D02629 |
Fluspirilene (USAN/INN); Imap (TN) |
(P) unclassified |
| D02630 |
Penfluridol (USAN/INN); Semap (TN) |
(P) unclassified |
| D02642 |
Butaperazine (USAN) |
(P) unclassified |
| D02643 |
Butaperazine maleate (USAN) |
(P) unclassified |
| D02666 |
Iloperidone (USAN/INN); Fanapt (TN) |
(P) Target: DRD2 |
| D02671 |
Mesoridazine (USAN/INN); Lidanar (TN) |
(P) unclassified |
| D02680 |
Pipotiazine palmitate (USAN); Piportil depot (TN) |
(P) unclassified |
| D02682 |
Remoxipride (USAN) |
(P) Target: DRD2 |
| D02683 |
Remoxipride hydrochloride (USAN) |
(P) Target: DRD2 |
| D02689 |
Ramelteon (JAN/USAN/INN); Rozerem (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
| D02713 |
Carpipramine hydrochloride hydrate (JAN); Carpipramine dihydrochloride; Defekton (TN) |
(P) unclassified |
| D02716 |
Pregabalin (JAN/USAN/INN); Lyrica (TN) |
(P) unclassified |
| D02717 |
Valnoctamide (USAN/INN); Axiquel (TN) |
(P) unclassified |
| D02740 |
Lidocaine - prilocaine mixt; Lidocaine - propitocaine mixt; Emla (TN); Oraqix (TN) |
(P) unclassified |
| D02770 |
Adinazolam (USAN/INN) |
(P) unclassified |
| D02771 |
Adinazolam mesylate (USAN) |
(P) unclassified |
| D02775 |
Adrogolide hydrochloride (USAN) |
(P) unclassified |
| D02798 |
Alcohol diluted (NF) |
(P) unclassified |
| D02817 |
Allobarbital (USAN/INN) |
(P) unclassified |
| D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(CI) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D02941 |
Anileridine (USP/INN) |
(P) unclassified |
| D02942 |
Anileridine hydrochloride (USP); Leritine (TN) |
(P) unclassified |
| D02968 |
Aprepitant (JAN/USAN/INN); Emend (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02991 |
Articaine hydrochloride (USAN) |
(P) unclassified |
| D02995 |
Asenapine maleate (USAN); Saphris (TN) |
(P) Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D03089 |
Benzoctamine hydrochloride (USAN) |
(P) unclassified |
| D03165 |
Bromocriptine (USAN/INN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D03214 |
Aplindore fumarate (USAN) |
(P) Target: DRD2 |
| D03253 |
Brecanavir (USAN) |
(CI) unclassified |
| D03260 |
Vardenafil hydrochloride hydrate (JAN); Levitra (TN) |
(P) unclassified |
| D03264 |
Mazaticol hydrochloride hydrate (JAN); Mazaticol hydrochloride; Pentona (TN) |
(P) unclassified |
| D03274 |
Chlorpromazine hibenzate (JAN); Contomin (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D03276 |
Profenamine hibenzate (JAN); Parkin (TN) |
(P) unclassified |
| D03290 |
Promethazine methylenedisalicylate (JAN); Pyrethia (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D03365 |
Nicotine (USP); Habitrol (TN) |
(P) Enzyme: CYP1A2 |
| D03444 |
Opium, powdered (JP16); Opium (USP) |
(P) unclassified |
| D03445 |
Opium alkaloids hydrochlorides (JP16); Pan opin (TN) |
(P) unclassified |
| D03494 |
Ciladopa hydrochloride (USAN); Tremerase (TN) |
(P) Target: DRD2 |
| D03556 |
Zuclopenthixol (INN); Clopixol (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D03562 |
Clorazepate monopotassium (USAN) |
(P) unclassified |
| D03656 |
Darunavir (USAN/INN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03785 |
Dichloralphenazone (USP) |
(P) unclassified |
| D03833 |
Indinavir (USAN); Indinavir hydrate |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN) |
(CI) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D03837 |
Fosamprenavir sodium (USAN) |
(CI) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D03839 |
Droxinavir hydrochloride (USAN) |
(CI) unclassified |
| D03840 |
Palinavir (USAN/INN) |
(CI) unclassified |
| D03841 |
Nitrous oxide - oxygen; Anesoxyn (TN) |
(P) unclassified |
| D03842 |
Telinavir (USAN/INN) |
(CI) unclassified |
| D03843 |
Tipranavir disodium (USAN) |
(CI) unclassified |
| D03852 |
Droperidol - fentanyl citrate mixt; Innovar (TN) |
(P) Enzyme: CYP3A4 |
| D03855 |
Pethidine hydrochloride - levallorphan tartrate mixt; Pethilorfan (TN) |
(P) unclassified |
| D03863 |
Opium alkaloids and atropine injection (JP16); Opium alkaloids hydrochloride - atropine sulfate hydrate mixt; Opiato (TN) |
(P) unclassified |
| D03866 |
Opium alkaloids and scopolamine injection (JP16); Weak opium alkaloids and scopolamine injection (JP16); Opium alkaloids hydrochloride - scopolamine hydrobromide hydrate mixt; Opisco (TN) |
(P) unclassified |
| D03869 |
Opium ipecac powder (JP16); Dover's powder (TN) |
(P) unclassified |
| D03872 |
Compound oxycodone and atropine injection (JP16); Pavinal atropine (TN) |
(P) unclassified |
| D03876 |
Morphine hydrochloride hydrate - atropine sulfate hydrate (JP16); Morphine and atropine (TN) |
(P) unclassified |
| D03891 |
Dopexamine (USAN/INN) |
(P) Target: DRD2 DRD3 |
| D03936 |
Econazole (USAN/INN) |
(CI) unclassified |
| D03975 |
Allylisopropylacetylurea; Apronal; Apronalide |
(P) unclassified |
| D04024 |
Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate (USAN); Tykerb (TN) |
(P) Enzyme: CYP3A4 |
| D04034 |
Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) |
(P) Target: DRD2 |
| D04038 |
Perphenazine fendizoate (JAN); PZC (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D04044 |
Chlorpheniramine maleate - acetaminophen - salicylamide - anhydrous caffeine mixt; LL (TN) |
(P) unclassified |
| D04046 |
Salicylamide - acetaminophen - anhydrous caffeine - promethazine methylenedisalicylate mixt; PL (TN) |
(P) unclassified |
| D04048 |
Ropivacaine hydrochloride hydrate (JAN); Ropivacaine hydrochloride (USP); Anapeine (TN) |
(P) Enzyme: CYP1A2 |
| D04052 |
Adrenaline - lidocaine hydrochloride mixt; Epinephrine - lidocaine hydrochloride mixt; Xylocaine (TN) |
(CI,P) Enzyme: CYP3A4 CYP1A2 |
| D04054 |
Erythromycin salnacedin (USAN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04059 |
Mepenzolate bromide - phenobarbital mixt; Trancolon P (TN) |
(P) unclassified |
| D04088 |
Ethyl chloride (USP) |
(P) unclassified |
| D04095 |
Etidocaine (USAN/INN) |
(P) unclassified |
| D04257 |
Fospropofol disodium (USAN); Aquavan (TN); Lusedra (TN) |
(P) unclassified |
| D04259 |
Diphenhydramine hydrochloride - diprophylline mixt; Travelmin (TN) |
(P) unclassified |
| D04261 |
Diphenhydramine salicylate - diprophylline mixt; Travelmin (TN) |
(P) unclassified |
| D04266 |
Benzylhydrochlorothiazide - Reserpine - Carbazochrome mixt; Behyd RA (TN) |
(P) unclassified |
| D04296 |
Diprophylline - methoxyphenamine hydrochloride - noscapine - chlorpheniramine maleate mixt; Asthma (TN) |
(P) unclassified |
| D04299 |
Diprophylline - ephedrine hydrochloride - papaverine hydrochloride - noscapine - diphenhydramine hydrochloride mixt; Asthpyllin (TN) |
(P) unclassified |
| D04307 |
Proxyphylline - ephedrine hydrochloride - phenobarbital mixt; Asthmolysin D (TN) |
(P) unclassified |
| D04313 |
Dihydrocodeine phosphate - dl-methylephedrine hydrochloride - Chlorpheniramine maleate mixt; Huscode (TN) |
(P) unclassified |
| D04324 |
Noscapine hydrochloride - dl-methylephedrine hydrochloride - diphenhydramine hydrochloride mixt; Sekiel (TN) |
(P) unclassified |
| D04336 |
Cherry bark extract - codeine phosphate hydrate mixt; Brocin codeine (TN) |
(P) unclassified |
| D04338 |
Dihydrocodeine phosphate - ephedrine hydrochloride - ammmonium chloride mixt; Sekicode (TN) |
(P) unclassified |
| D04447 |
Betamethasone - d-chlorpheniramine maleate mixt; Celestamine (TN) |
(P) unclassified |
| D04488 |
Ibopamine (USAN/INN) |
(P) Target: DRD2 |
| D04650 |
Ketazolam (USAN/INN) |
(P) unclassified |
| D04749 |
Lithium citrate (USP); Lithonate (TN) |
(P) unclassified |
| D04750 |
Lithium hydroxide (USP) |
(P) unclassified |
| D04813 |
Lidocaine hydrochloride - epinephrine bitartrate mixt; Ora (TN); Lidosite (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
| D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(P) Target: DRD2 |
| D04855 |
Ethanol for disinfection (JP16); Ethanol for disinfection (TN) |
(P) unclassified |
| D04882 |
Medazepam hydrochloride (USAN); Nobrium (TN) |
(P) unclassified |
| D04965 |
Perphenazine hydrochloride; Perphenazine dihydrochloride; PZC intramuscular injection (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D04985 |
Methohexital (USP/INN) |
(P) unclassified |
| D05008 |
Metoclopramide hydrochloride (USAN); Metoclopramide hydrochloride monohydrate; Clopra (TN); Reglan (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D05028 |
Midazolam maleate (USAN) |
(P) Enzyme: CYP3A4 |
| D05277 |
Formoterol fumarate hydrate (JP16); Formoterol fumarate dihydrate; Atock (TN); Foradil (TN) |
(P) unclassified |
| D05339 |
Paliperidone (JAN/USAN/INN); Invega (TN) |
(P) Target: DRD2 |
| D05340 |
Paliperidone palmitate (JAN/USAN) |
(P) Target: DRD2 |
| D05374 |
Paroxetine hydrochloride (USP); Paxil (TN) |
(CI) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D05375 |
Paroxetine mesylate (USAN); Pexeva (TN) |
(CI) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D05462 |
Oxycodone hydrochloride hydrate (JP16) |
(P) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D05538 |
Mozenavir (INN) |
(CI) unclassified |
| D05575 |
Pramipexole (USAN/INN) |
(P) Target: DRD2 DRD3 |
| D05626 |
Propanidid (USAN/INN); Epontol (TN) |
(P) unclassified |
| D05677 |
Quinelorane hydrochloride (USAN) |
(P) Target: DRD2 |
| D05682 |
Quinpirole hydrochloride (USAN) |
(P) Target: DRD2 DRD3 |
| D05768 |
Rotigotine (JAN/USAN/INN); Neupro (TN) |
(P) Target: DRD2 |
| D05832 |
Sibenadet hydrochloride (USAN); Viozan (TN) |
(P) Target: DRD2 |
| D05928 |
Stiripentol (JAN/USAN/INN) |
(P) Enzyme: CYP3A4 CYP1A2 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6 |
| D05938 |
Sufentanil (USAN/INN) |
(P) unclassified |
| D06338 |
Xenon Xe 127 (USP); Xenon, isotope of mass 127; Xenon Xe 127 (TN) |
(P) unclassified |
| D06339 |
Xenon Xe 133 (JAN/USP/INN); Xenon (133Xe); Xenon Xe 133 (TN) |
(P) unclassified |
| D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) Enzyme: CYP3A4 |
| D06405 |
Nalfurafine hydrochloride (JAN) |
(P) Enzyme: CYP3A4 |
| D06413 |
Nilotinib hydrochloride hydrate (JAN); Tasigna (TN) |
(P) Enzyme: CYP3A4 |
| D06414 |
Dasatinib hydrate (JAN); Dasatinib (USAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 |
| D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06499 |
Opium tincture (JP16); Opium tincture (TN) |
(P) unclassified |
| D06534 |
Phenolated water (JP16); Phenolated water for disinfection (JP16); Phenol hydrate; Phenol water (TN); Phenolated water for disinfection (TN) |
(P) unclassified |
| D06535 |
|
(P) unclassified |
| D06536 |
|
(P) unclassified |
| D06537 |
|
(P) unclassified |
| D06542 |
Ethanol (JP16); Ethanol (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D06597 |
Fosaprepitant meglumine (JAN); Fosaprepitant dimeglumine (USAN); Proemend (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06623 |
Olanzapine pamoate (USAN); Olanzapine pamoate monohydrate |
(P) Enzyme: CYP1A2 CYP2D6 / Target: ADRA1D ADRA1B ADRA1A DRD2 DRD3 / CYP inhibition: CYP2D6 |
| D06699 |
Japanese valerian (JP16); Powdered japanese valerian (JP16); Valerianae radix (TN) |
(P) unclassified |
| D06883 |
Sertaconazole (INN) |
(CI) unclassified |
| D06887 |
Talbutal (INN); Lotusate (TN) |
(P) unclassified |
| D07065 |
Acepromazine (INN); Concentrat vo34 (TN) |
(P) unclassified |
| D07122 |
Alfentanil (INN); Rapifen (TN) |
(P) unclassified |
| D07132 |
Buprenorphine (JAN/INN); Temgesic (TN) |
(P) unclassified |
| D07217 |
Quinagolide (INN/BAN) |
(P) Target: DRD2 |
| D07282 |
Alfaxalone (INN) |
(P) unclassified |
| D07283 |
Esketamine (INN) |
(P) unclassified |
| D07284 |
Butanilicaine (INN) |
(P) unclassified |
| D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) unclassified |
| D07307 |
Cyamemazine (INN); Tercian (TN) |
(P) unclassified |
| D07308 |
Chlorproethazine (INN) |
(P) unclassified |
| D07309 |
Melperone (INN); Bunil (TN) |
(P) unclassified |
| D07310 |
Amisulpride (INN); Deniban (TN); Solian (TN) |
(P) unclassified |
| D07311 |
Veralipride (INN); Agreal (TN) |
(P) unclassified |
| D07312 |
Levosulpiride (INN); Levopraid (TN) |
(P) Target: DRD2 DRD3 |
| D07313 |
Prothipendyl (INN) |
(P) unclassified |
| D07314 |
Pinazepam (INN); Domar (TN) |
(P) unclassified |
| D07315 |
Camazepam (INN) |
(P) unclassified |
| D07316 |
Captodiame (BAN) |
(P) unclassified |
| D07317 |
Emylcamate (INN) |
(P) unclassified |
| D07318 |
Mephenoxalone (INN); Dorsiflex (TN) |
(P) unclassified |
| D07319 |
Gedocarnil (INN) |
(P) unclassified |
| D07320 |
Etifoxine (INN/BAN) |
(P) unclassified |
| D07321 |
Vinylbital (INN); Vinylbitone |
(P) unclassified |
| D07322 |
Vinbarbital (INN) |
(P) unclassified |
| D07323 |
Cyclobarbital (INN); Ciclobarbital (TN) |
(P) unclassified |
| D07324 |
Proxibarbal (INN); Centralgol (TN) |
(P) unclassified |
| D07325 |
Chloralodol (INN); Chlorhexadol |
(P) unclassified |
| D07326 |
Loprazolam (INN); Dormonoct (TN) |
(P) unclassified |
| D07327 |
Doxefazepam (INN) |
(P) unclassified |
| D07328 |
Cinolazepam (INN); Gerodorm (TN) |
(P) unclassified |
| D07329 |
Pyrithyldione (INN) |
(P) unclassified |
| D07330 |
Clomethiazole (INN); Distraneurine (TN) |
(P) unclassified |
| D07331 |
Hexapropymate (INN); Merinax (TN) |
(P) unclassified |
| D07332 |
Methylpentynol (INN); Meparfynol; Methylparafynol; Atemorin (TN) |
(P) unclassified |
| D07333 |
Niaprazine (INN); Nopron (TN) |
(P) unclassified |
| D07460 |
Apomorphine (BAN); Uprima (TN) |
(P) Target: DRD2 |
| D07468 |
Articaine (INN); Carticaine |
(P) unclassified |
| D07471 |
Atazanavir (INN); Reyataz (TN) |
(CI) Enzyme: CYP3A4 |
| D07552 |
Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) |
(P) unclassified |
| D07583 |
Phenytoin - phenobarbital mixt; Aleviatin with phenobarbital (TN) |
(P) unclassified |
| D07593 |
Buspirone (INN); Gen-Buspirone (TN) |
(P) unclassified |
| D07598 |
Butoconazole (INN); Gynofort (TN) |
(CI) unclassified |
| D07678 |
Chloroprocaine (INN) |
(P) unclassified |
| D07685 |
Chlorproethazine hydrochloride; Neuriplege (TN) |
(P) unclassified |
| D07686 |
Chlorprothixene acetate; Truxal (TN) |
(P) unclassified |
| D07687 |
Chlorprothixene citrate; Truxal (TN) |
(P) unclassified |
| D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(CI) Enzyme: CYP3A4 |
| D07725 |
Clomethiazole edisilate; Heminevrin (TN) |
(P) unclassified |
| D07756 |
Cyamemazine tartrate; Tercian (TN) |
(P) unclassified |
| D07757 |
Cyclobarbital calcium (BAN); Phanodorn calcium (TN) |
(P) unclassified |
| D07837 |
Dihydroergotamine (INN); Neomigran (TN) |
(P) Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D07838 |
Dihydroergotamine tartrate; Divegal (TN) |
(P) Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D07865 |
Dixyrazine; Esucos (TN) |
(P) unclassified |
| D07868 |
Domperidone maleate; Domperidone (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D07870 |
Dopamine (INN); Medopa (TN) |
(P) Target: DRD2 DRD3 |
| D07881 |
Dyclonine (INN) |
(P) unclassified |
| D07906 |
Ergotamine (INN) |
(P) Enzyme: CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 |
| D07909 |
Erythromycin thiocyanate; Erythrocin (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07910 |
Erythromycin stinoprate (INN); Erysec (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07930 |
Etifoxine hydrochloride; Stresam (TN) |
(P) unclassified |
| D07976 |
Flupentixol decanoate; Fluanxol depot (TN) |
(P) Target: DRD2 |
| D07977 |
Fluphenazine (INN); Moditen (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D07984 |
Fluvoxamine (INN) |
(CI) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 CYP1A2 |
| D08035 |
Haloperidol lactate; Haldol (TN) |
(P) Target: DRD2 |
| D08054 |
Hydroxyzine (INN); Marex (TN) |
(P) CYP inhibition: CYP2D6 |
| D08057 |
Ibopamine hydrochloride; Scandine (TN) |
(P) Target: DRD2 |
| D08098 |
Ketamine (INN); Tekam (TN) |
(P) unclassified |
| D08116 |
Levobupivacaine (INN); Novabupi (TN) |
(P) unclassified |
| D08118 |
Levocetirizine hydrochloride (JAN/USAN); Levocetirizine dihydrochloride; Xyzal (TN) |
(P) unclassified |
| D08127 |
Lidocaine hydrochloride monohydrate; Lidocaine (TN) |
(P) Enzyme: CYP3A4 CYP1A2 CYP2D6 / CYP inhibition: CYP2D6 |
| D08132 |
Lisuride (INN) |
(P) Target: DRD2 |
| D08133 |
Lithium; Normothymin-E (TN) |
(P) unclassified |
| D08134 |
Lithium acetate; Quilonorm (TN) |
(P) unclassified |
| D08135 |
Lithium bromide; Lithium Microsol (TN) |
(P) unclassified |
| D08136 |
Lithium gluconate; Lithioderm (TN) |
(P) unclassified |
| D08137 |
Lithium sulfate; Lithionit (TN) |
(P) unclassified |
| D08145 |
Loprazolam mesilate; Loprazolam mesylate; Loprazolam methanesulfonate; Havlane (TN) |
(P) unclassified |
| D08148 |
Loxapine hydrochloride; Desconex (TN) |
(P) Target: DRD2 |
| D08170 |
Melatonin; Melatonina (TN) |
(P) Enzyme: CYP1A2 |
| D08172 |
Melperone hydrochloride; Buronil (TN) |
(P) unclassified |
| D08181 |
Mepivacaine (INN); Carboplyin Dental (TN) |
(P) unclassified |
| D08226 |
Molindone (INN) |
(P) Target: DRD2 |
| D08235 |
Mosapramine (INN) |
(P) Target: DRD2 |
| D08259 |
Nelfinavir (INN); Viracept (TN) |
(CI) Enzyme: CYP3A4 CYP2D6 / CYP inhibition: CYP2D6 |
| D08283 |
Nordazepam (INN); Calmday (TN) |
(P) Enzyme: CYP3A4 |
| D08313 |
Oxiconazole (INN) |
(CI) unclassified |
| D08339 |
Pergolide (INN); Permax (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D08341 |
Perphenazine decanoate; Trilafon dekanoat (TN) |
(P) Target: DRD2 |
| D08342 |
Perphenazine enantate; Perphenazine enanthate; Trilafon (TN) |
(P) Target: DRD2 |
| D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) CYP induction: CYP1A2 CYP3A4 |
| D08385 |
Pipotiazine (INN); Piportil (TN) |
(P) unclassified |
| D08422 |
Procaine (INN); Solution of novocain (TN) |
(P) unclassified |
| D08430 |
Promazine (INN); Combelen [veterinary] (TN) |
(P) unclassified |
| D08439 |
Propiomazine maleate; Propavan (TN) |
(P) unclassified |
| D08446 |
Prothipendyl hydrochloride; Dominal (TN) |
(P) unclassified |
| D08456 |
Quetiapine (INN); Norsic (TN) |
(P) Enzyme: CYP3A4 / Target: ADRA1D ADRA1B ADRA1A DRD2 DRD3 |
| D08457 |
Quinagolide hydrochloride (BAN); Norprolac (TN) |
(P) Target: DRD2 |
| D08473 |
Remifentanil (INN); Ultiva (TN) |
(P) unclassified |
| D08489 |
Ropinirole (USAN/INN); Ropitor (TN) |
(P) Enzyme: CYP1A2 / Target: DRD2 |
| D08490 |
Ropivacaine (INN); Naropin (TN) |
(P) Enzyme: CYP1A2 |
| D08510 |
Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) |
(CI) unclassified |
| D08535 |
Sulconazole (INN) |
(CI) unclassified |
| D08549 |
Sultopride (INN) |
(P) Target: DRD2 |
| D08558 |
Talipexole (INN) |
(P) Target: DRD2 |
| D08575 |
Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) |
(P) unclassified |
| D08585 |
Thioproperazine (INN) |
(P) Target: DRD2 |
| D08590 |
Tiapride (INN); Tiapridal (TN) |
(P) Target: DRD2 |
| D08605 |
Tipranavir (INN); Aptivus (TN) |
(CI) unclassified |
| D08634 |
Triclofos (INN); Neguvon [veterinary] (TN) |
(P) unclassified |
| D08636 |
Trifluoperazine (INN); Apo-trifluoperazine (TN) |
(P) Target: DRD2 |
| D08637 |
Trifluperidol hydrochloride; Triperidol (TN) |
(P) Target: DRD2 |
| D08687 |
Ziprasidone (INN); Zipradon (TN) |
(P) Enzyme: CYP3A4 / Target: DRD2 |
| D08690 |
Zolpidem (INN); Sanval (TN) |
(P) Enzyme: CYP3A4 CYP1A2 |
| D08691 |
Zuclopenthixol acetate; Cisordinol-acutard (TN) |
(P) Target: DRD2 |
| D08692 |
Zuclopenthixol decanoate; Clopixol depot (TN) |
(P) Target: DRD2 |
| D08693 |
Zuclopenthixol dihydrochloride; Clopixol (TN) |
(P) Enzyme: CYP2D6 / Target: DRD2 / CYP inhibition: CYP2D6 |
| D08695 |
dl-Methylephedrine hydrochloride - dihydrocodeine phosphate - diprophylline - diphenhydramine salicylate - acetaminophen - bromovalerylurea mixt; Coughcode N (TN) |
(P) unclassified |
| D08697 |
Platycodon fluidextract - glycyrrhiza extract - plantago herb extract - peony root extract - dihydrocodeine phosphate mixt; Opisezol codeine (TN) |
(P) unclassified |
| D08768 |
Promethazine hibenzate; Hiberna (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
| D08769 |
Diphenhydramine hydrochloride - calcium bromide mixt; Rescalmin (TN) |
(P) unclassified |
| D08774 |
Amoxicillin hydrate - clarithromycin - lansoprazole mixt; Lansap (TN) |
(CI) Enzyme: CYP3A4 |
| D09012 |
Telaprevir (JAN/USAN/INN); Incivek (TN) |
(CI) unclassified |
| D09216 |
Thiopropazate (INN) |
(P) unclassified |
| D09319 |
Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) |
(P) unclassified |
| D09535 |
Mirabegron (USAN/JAN); Myrbetriq (TN) |
(P) unclassified |
| D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) unclassified |
| D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) unclassified |
| D09819 |
Chlorpromazine tannate (JAN) |
(P) Target: DRD2 |
| D09958 |
Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) |
(P) unclassified |
| D09999 |
Tramadol hydrochloride - acetaminophen mixt; Tramcet (TN) |
(P) unclassified |
| E00839 |
Grapefruit juice |
(P) unclassified |
| E00840 |
Alcoholic beverage |
(P) unclassified |