KEGG icon

Drug interaction list


Query:
D00706  Zolpidem tartrate (JP18/USP); Ambien (TN); Intermezzo (TN)

Interactions: 268 hits    [ ATC classification | Therapeutic category ]

C00989  4-Hydroxybutanoic acid; 4-Hydroxybutanoate; 4-Hydroxybutyric acid (P) unclassified
C06807  Acetophenazine (P) unclassified
C07521  Thiopental (P) unclassified
C17723  Metabutethamine (P) unclassified
D00033  Phenol (JP18/USP); Liquefied phenol (JP18); Phenol for disinfection (JP18); Phenol, liquefied; Paoscle (TN); Phenol (TN); Liquefied phenol (TN); Phenol for disinfection (TN) (P) unclassified
D00102  Nitrous oxide (JP18/USP); Nitrous oxide (TN) (P) unclassified
D00110  Cocaine (USP); Cocaine (TN) (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00241  Baclofen (JP18/USP/INN); Kemstro (TN); Lioresal (TN) (P) unclassified
D00250  Capsaicin (JAN/USP); Zostrix (TN) (P) unclassified
D00270  Chlorpromazine (USP/INN); Thorazine (TN) (P) unclassified
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4 / Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4
D00358  Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) (P) Enzyme: CYP1A2 CYP3A4
D00373  Thioridazine (USP/INN); Mellaril-S (TN) (P) unclassified
D00390  Triflupromazine (USP/INN); Vesprin (TN) (P) unclassified
D00403  Methotrimeprazine (USP); Levomepromazine (USAN/INN); Levoprome (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00430  Secobarbital (USP/INN); Seconal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4
D00474  Primidone (JP18/USP/INN); Mysoline (TN) (P) unclassified
D00479  Prochlorperazine maleate (JP18/USP); Compazine (TN) (P) unclassified
D00493  Prochlorperazine (JAN/USP/INN); Compro (TN) (P) unclassified
D00498  Pentazocine (JP18/USP/INN); Fortral (TN) (P) unclassified
D00499  Pentobarbital (USP/INN); Nembutal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00500  Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00503  Perphenazine (JP18/USP/INN); Trilafon (TN) (P) unclassified
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) unclassified
D00542  Halothane (JP18/USP/INN); Fluothane (TN) (P) Enzyme: CYP3A4
D00543  Enflurane (JP18/USP/INN); Ethrane (TN) (P) unclassified
D00544  Methoxyflurane (USP/INN); Penthrane (TN) (P) Enzyme: CYP3A4
D00545  Isoflurane (JP18/USP/INN); Forane (TN) (P) unclassified
D00546  Desflurane (JAN/USP/INN); Suprane (TN) (P) unclassified
D00547  Sevoflurane (JP18/USAN/INN); Ultane (TN) (P) unclassified
D00548  Etomidate (USP/INN); Amidate (TN) (P) Target: GABRA1
D00549  Propofol (JAN/USP/INN); Diprivan (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4 / Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00551  Tetracaine (USP/INN); Amethocaine; Amethocaine (TN) (P) unclassified
D00552  Benzocaine (USP/INN); Ethyl aminobenzoate (JP18); Parathesin (TN) (P) unclassified
D00553  Prilocaine (USP/INN); Propitocaine (JAN) (P) unclassified
D00555  Amobarbital (JP18/INN); Isomytal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00578  Voriconazole (JP18/USP/INN); Vfend (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) Enzyme: CYP3A4
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4
D00698  Aprobarbital (INN); Alurate (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00699  Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00711  Ketamine hydrochloride (JP18/USP); Ketalar (TN) (P) unclassified
D00712  Methohexital sodium (USP); Brevital sodium (TN) (P) Target: GABRA1
D00713  Thiamylal sodium (JP18); Surital (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00714  Thiopental sodium (JP18/USP/INN); Pentothal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D00732  Chloroprocaine hydrochloride (USP); Clorotekal (TN); Iheezo (TN); Nesacaine (TN) (P) unclassified
D00733  Dibucaine (USP); Cinchocaine (INN); Nupercaine (TN) (P) unclassified
D00735  Dyclonine hydrochloride (USP); Dyclone (TN); Dyclopro (TN) (P) unclassified
D00737  Etidocaine hydrochloride; Duranest (TN) (P) unclassified
D00738  Mepivacaine hydrochloride (JP18/USP); Carbocaine (TN); Polocaine (TN); Scandonest plain (TN) (P) unclassified
D00740  Procaine hydrochloride (JP18/USP); Novocain (TN) (P) unclassified
D00741  Tetracaine hydrochloride (JP18/USP); Protocaine hydrochloride (TN) (P) unclassified
D00788  Acetophenazine maleate (USAN); Tindal (TN) (P) unclassified
D00789  Chlorpromazine hydrochloride (JP18/USP); Sonazine (TN) (P) unclassified
D00791  Fluphenazine hydrochloride (JAN/USP); Prolixin (TN) (P) unclassified
D00792  Fluphenazine enanthate (JP18/USP); Prolixin enanthate (TN) (P) unclassified
D00793  Fluphenazine decanoate (JAN/USP); Prolixin decanoate (TN) (P) unclassified
D00795  Mesoridazine besylate (USP); Serentil (TN) (P) unclassified
D00797  Promazine hydrochloride (USP); Sparine (TN) (P) unclassified
D00798  Thioridazine hydrochloride (JP18/USP); Mellaril (TN) (P) unclassified
D00799  Trifluoperazine hydrochloride (JAN/USP); Stelazine (TN) (P) unclassified
D00800  Triflupromazine hydrochloride (JAN/USP); Vesprin (TN) (P) unclassified
D00824  Fluvoxamine maleate (JP18/USP); Luvox (TN) (P) CYP inhibition: CYP1A2 CYP3A4
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00835  Alfentanil hydrochloride (USP); Alfenta (TN) (P) unclassified
D00845  Sufentanil citrate (USP); Dsuvia (TN); Sufenta (TN) (P) unclassified
D00961  Bicalutamide (JP18/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D01071  Hexobarbital (JAN/INN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D01130  Thiethylperazine maleate (JAN/USP); Norzine (TN) (P) unclassified
D01152  Oxethazaine (JP18/USAN); Oxetacaine (INN); Strocain (TN) (P) unclassified
D01177  Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) (P) unclassified
D01243  Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4 / Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D01280  Warfarin potassium (JP18); Athrombin-K (TN) (P) unclassified
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) Enzyme: CYP3A4 CYP1A2
D01310  Secobarbital sodium (JAN/USP); Seconal sodium (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D01355  Tramadol hydrochloride (JP18/USP); Ultram (TN) (P) Enzyme: CYP3A4
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4
D01412  Perazine maleate (JAN) (P) unclassified
D01447  Thioproperazine mesilate (JAN); Thioproperazine mesylate (P) unclassified
D01448  Trifluoperazine maleate (JAN); Trifluoperazine (TN) (P) unclassified
D01450  Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) (P) Enzyme: CYP3A4
D01485  Propericiazine (JAN); Periciazine; Neuleptil (TN) (P) unclassified
D01520  Levomepromazine hydrochloride (JAN/USAN); Nozinan (TN) (P) unclassified
D01740  Barbital (JP18/INN); Barbital (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D01768  Benoxinate hydrochloride (USP); Oxybuprocaine hydrochloride (JP18); Benoxil (TN) (P) unclassified
D01772  Ether (JP18/USP); Diethyl ether (P) unclassified
D01860  Perazine dimalonate (JAN) (P) unclassified
D01878  Tolycaine hydrochloride (JAN) (P) unclassified
D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN); Diethylaminoethyl p-butylaminobenzoate hydrochloride (JAN); Calvital liquid (TN); T cain (TN) (P) unclassified
D02022  Prochlorperazine mesilate (JAN); Prochlorperazine dimethanesulfonate; Novamin (TN) (P) unclassified
D02037  Perphenazine maleate (JP18); PZC (TN) (P) unclassified
D02086  Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) (P) Enzyme: CYP3A4 CYP1A2
D02098  Proparacaine hydrochloride (USP); Alcaine (TN); Ophthetic (TN) (P) unclassified
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02163  Fluphenazine maleate (JAN); Flumezin (TN) (P) unclassified
D02182  Cocaine hydrochloride (JP18/USP); Cocaine hydrochloride (TN) (P) unclassified
D02220  Dibucaine hydrochloride (JP18/USP); Nupercaine hydrochloride (TN); Percamin (TN) (P) unclassified
D02227  Pentazocine hydrochloride (JAN/USP); Sosegon (TN); Talacen (TN) (P) unclassified
D02248  Levomepromazine maleate (JP18/USAN); Hirnamin (TN) (P) unclassified
D02252  Amobarbital sodium (JAN/USP); Amytal sodium (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D02253  Pentobarbital calcium (JP18); Ravona (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D02354  Thiethylperazine (USAN/INN) (P) unclassified
D02372  Perospirone hydrochloride hydrate (JAN); Lullan (TN) (P) unclassified
D02456  Aminobenzoic acid (USP); p-Aminobenzoic acid; RVPaba lipstick (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02604  Acepromazine maleate (USP) (P) unclassified
D02605  Methoxypromazine maleate (P) unclassified
D02607  Mepazine acetate (P) unclassified
D02608  Perazine fendizoate (JAN) (P) unclassified
D02609  Prochlorperazine edisylate (USP); Compazine syrup (TN) (P) unclassified
D02610  Thiethylperazine malate (JAN); Torecan (TN) (P) unclassified
D02611  Phenoperidine (INN) (P) unclassified
D02618  Butobarbital (BAN); Butethal; Neonal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D02642  Butaperazine (USAN) (P) unclassified
D02643  Butaperazine maleate (USAN) (P) unclassified
D02644  Carphenazine maleate (USAN); Proketazine (TN) (P) unclassified
D02653  Cyclophenazine hydrochloride (USAN) (P) unclassified
D02671  Mesoridazine (USAN/INN); Lidanar (TN) (P) unclassified
D02679  Piperacetazine (USAN/INN); Quide (TN) (P) unclassified
D02680  Pipotiazine palmitate (USAN); Piportil depot (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) Enzyme: CYP3A4
D02812  Aliflurane (USAN/INN) (P) unclassified
D02817  Allobarbital (USAN/INN) (P) unclassified
D02906  Aminobenzoate potassium (USP); Potaba (TN) (P) unclassified
D02907  Aminobenzoate sodium (USP); Sodium aminobenzoate (P) unclassified
D02941  Anileridine (USP/INN) (P) unclassified
D02942  Anileridine hydrochloride (USP); Leritine (TN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02991  Articaine hydrochloride (JAN/USP) (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03180  Butabarbital (USP); Secbutabarbital (BAN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D03182  Butalbital (USP/INN); Sandoptal (TN) (P) unclassified
D03274  Chlorpromazine hibenzate (JAN); Contomin (TN) (P) unclassified
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP inhibition: CYP1A2 / CYP induction: CYP3A4
D03719  Dexivacaine (USAN/INN) (P) unclassified
D03841  Nitrous oxide and oxygen; Anesoxyn (TN) (P) unclassified
D03852  Droperidol and fentanyl citrate; Innovar (TN) (P) Enzyme: CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4
D04034  Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) (P) unclassified
D04038  Perphenazine fendizoate (JAN); PZC (TN) (P) unclassified
D04048  Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) (P) Enzyme: CYP3A4 CYP1A2
D04077  Eterobarb (USAN/INN); Antilon (TN) (P) unclassified
D04088  Ethyl chloride (USP) (P) unclassified
D04095  Etidocaine (USAN/INN) (P) unclassified
D04237  Fluroxene (USAN); Fluoromar (TN) (P) unclassified
D04257  Fospropofol disodium (USAN); Aquavan (TN); Lusedra (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04965  Perphenazine hydrochloride; Perphenazine dihydrochloride; PZC intramuscular injection (TN) (P) unclassified
D04985  Methohexital (USP/INN) (P) Target: GABRA1
D05177  Nitisinone (JAN/USAN/INN); Orfadin (TN) (P) unclassified
D05208  Norflurane (USAN/INN) (P) unclassified
D05626  Propanidid (USAN/INN); Epontol (TN) (P) unclassified
D05665  Pyrrocaine (USAN/INN) (P) unclassified
D05743  Rodocaine (USAN) (P) unclassified
D05745  Roflurane (USAN/INN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05866  Sodium oxybate (USAN); Sodium gammahydroxybutyrate; Xyrem (TN) (P) unclassified
D05938  Sufentanil (USAN/INN) (P) unclassified
D06055  Teflurane (USAN/INN) (P) unclassified
D06106  Thiamylal (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D06405  Nalfurafine hydrochloride (JAN/USAN) (P) Enzyme: CYP3A4
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4
D06534  Phenolated water (JP18); Phenolated water for disinfection (JP18); Phenol hydrate; Phenol water (TN); Phenolated water for disinfection (TN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06887  Talbutal (INN); Lotusate (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D07065  Acepromazine (INN); Concentrat vo34 (TN) (P) unclassified
D07122  Alfentanil (INN); Rapifen (TN) (P) unclassified
D07282  Alfaxalone (INN) (P) unclassified
D07284  Butanilicaine (INN) (P) unclassified
D07298  Barbexaclone (INN); Maliasin (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D07307  Cyamemazine (INN); Tercian (TN) (P) unclassified
D07308  Chlorproethazine (INN) (P) unclassified
D07321  Vinylbital (INN); Vinylbitone (P) unclassified
D07322  Vinbarbital (INN) (P) unclassified
D07323  Cyclobarbital (INN); Ciclobarbital (TN) (P) unclassified
D07324  Proxibarbal (INN); Centralgol (TN) (P) unclassified
D07468  Articaine (INN); Carticaine (P) unclassified
D07523  Betaine (JAN); Cystadane (TN) (P) unclassified
D07552  Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) (P) Enzyme: CYP3A4
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP induction: CYP3A4
D07678  Chloroprocaine (INN) (P) unclassified
D07685  Chlorproethazine hydrochloride; Neuriplege (TN) (P) unclassified
D07756  Cyamemazine tartrate; Tercian (TN) (P) unclassified
D07757  Cyclobarbital calcium (BAN); Phanodorn calcium (TN) (P) unclassified
D07865  Dixyrazine; Esucos (TN) (P) unclassified
D07881  Dyclonine (INN) (P) unclassified
D07977  Fluphenazine (INN); Moditen (TN) (P) unclassified
D08098  Ketamine (INN); Tekam (TN) (P) unclassified
D08116  Levobupivacaine (INN); Novabupi (TN) (P) Enzyme: CYP3A4 CYP1A2
D08127  Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) (P) Enzyme: CYP3A4 CYP1A2
D08181  Mepivacaine (INN); Carboplyin Dental (TN) (P) unclassified
D08311  Oxetacaine hydrochloride; Emoren (TN) (P) unclassified
D08319  Oxybuprocaine (INN); Monofree oxybuprocaine (TN) (P) unclassified
D08341  Perphenazine decanoate; Trilafon dekanoat (TN) (P) unclassified
D08342  Perphenazine enantate; Perphenazine enanthate; Trilafon (TN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) Target: GABRA1 GABRA2 GABRA3 GABRA4 GABRA5 GABRA6 GABRB1 GABRB2 GABRB3 GABRD GABRE GABRG1 GABRG2 GABRG3 GABRP GABRQ
D08385  Pipotiazine (INN); Piportil (TN) (P) unclassified
D08422  Procaine (INN); Solution of novocain (TN) (P) unclassified
D08430  Promazine (INN); Combelen [veterinary] (TN) (P) unclassified
D08448  Proxymetacaine (INN); Proparacaine (P) unclassified
D08473  Remifentanil (INN); Ultiva (TN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) CYP induction: CYP3A4
D08490  Ropivacaine (INN); Naropin (TN) (P) Enzyme: CYP3A4 CYP1A2
D08585  Thioproperazine (INN) (P) unclassified
D08636  Trifluoperazine (INN); Apo-trifluoperazine (TN) (P) unclassified
D08640  Trimecaine (INN); Mesidicain; Mesocain (P) unclassified
D08641  Trimecaine hydrochloride; Mesocain (TN) (P) unclassified
D09216  Thiopropazate (INN) (P) unclassified
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) Enzyme: CYP3A4
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09819  Chlorpromazine tannate (JAN) (P) unclassified
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP inhibition: CYP1A2 / CYP induction: CYP3A4
D09999  Tramadol hydrochloride and acetaminophen; Tramcet (TN) (P) Enzyme: CYP3A4
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) unclassified
D10811  Fentanyl hydrochloride (JAN); Ionsys (TN) (P) Enzyme: CYP3A4
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (P) unclassified
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) Enzyme: CYP3A4
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11027  Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11062  Osilodrostat phosphate (JAN/USAN); Isturisa (TN) (P) Enzyme: CYP3A4
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (P) unclassified
D11404  Asciminib hydrochloride (JAN/USAN); Scemblix (TN) (P) Enzyme: CYP3A4
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11708  Givosiran sodium (JAN); Givlaari (TN) (P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) CYP inhibition: CYP1A2
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (P) unclassified