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Drug interaction list


Query:
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN)

Interactions: 379 hits    [ ATC classification | Therapeutic category ]

C07051  Indinavir (P) unclassified
C07521  Thiopental (P) unclassified
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) (P) Enzyme: CYP3A4
D00125  Etoposide (JP18/USP/INN); Vepesid (TN) (P) unclassified
D00140  Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) (P) unclassified
D00168  Cytarabine (JP18/USP/INN); ARA-C; Depocyt (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00208  Mitomycin (USP/INN); Mitomycin C (JP18); MMC; Jelmyto (TN); Mitomycin (TN); Muamycin (TN) (P) unclassified
D00210  Norfloxacin (JP18/USP/INN); Noroxin (TN) (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (CI,P) CYP induction: CYP3A4
D00214  Dactinomycin (USP); Actinomycin D (JP18); Cosmegen (TN) (P) unclassified
D00251  Captopril (JP18/USP/INN); Apopril (TN); Capoten (TN) (P) unclassified
D00252  Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00275  Cisplatin (JP18/USP/INN); Platinol (TN) (P) unclassified
D00276  Clarithromycin (JP18/USP/INN); Biaxin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00282  Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) (P) CYP inhibition: CYP3A4
D00287  Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) (P) Enzyme: CYP3A4
D00288  Dacarbazine (JAN/USP/INN); DTIC-Dome (TN) (P) unclassified
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4
D00295  Cimetidine (JP18/USP/INN); Tagamet (TN) (P) CYP inhibition: CYP3A4
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP3A4
D00323  Flucytosine (JP18/USP/INN); Ancobon (TN) (P) unclassified
D00326  Fluoxetine (USAN/INN); Fluoxetine (TN) (P) unclassified
D00341  Hydroxyurea (USP); Hydroxycarbamide (JAN/INN); Droxia (TN); Hydrea (TN); Siklos (TN) (P) unclassified
D00343  Ifosfamide (JAN/USP/INN); Ifex (TN) (P) Enzyme: CYP3A4
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00362  Lisinopril (USP); Lisinopril hydrate (JP18); Lisinopril dihydrate; Prinivil (TN); Zestril (TN) (P) unclassified
D00383  Trandolapril (JAN/USP/INN); Mavik (TN) (P) unclassified
D00395  Troglitazone (JAN/USAN/INN); Rezulin (TN) (P) unclassified
D00416  Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00421  Ramipril (USP/INN); Altace (TN) (P) unclassified
D00422  Ranitidine (USAN/INN); Ranitidine (TN) (P) unclassified
D00424  Rifabutin (JAN/USP/INN); Mycobutin (TN) (P) Enzyme: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) unclassified
D00430  Secobarbital (USP/INN); Seconal (TN) (P) unclassified
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4
D00459  Quinapril hydrochloride (JP18/USP); Accupril (TN) (P) unclassified
D00474  Primidone (JP18/USP/INN); Mysoline (TN) (P) unclassified
D00491  Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) (P) Enzyme: CYP3A4
D00499  Pentobarbital (USP/INN); Nembutal (TN) (P) unclassified
D00500  Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) (P) unclassified
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) unclassified
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) unclassified
D00533  Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) (P) unclassified
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00555  Amobarbital (JP18/INN); Isomytal (TN) (P) unclassified
D00578  Voriconazole (JP18/USP/INN); Vfend (TN) (P) unclassified
D00584  Fluorouracil (JP18/USP/INN); 5-FU (TN); Adrucil (TN); Carac (TN); Fluoroplex (TN) (P) unclassified
D00585  Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) (P) Enzyme: CYP3A4
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00620  Benazepril hydrochloride (JAN/USP); Lotensin (TN) (P) unclassified
D00621  Enalapril maleate (JP18/USP); Renivace (TN); Vasotec (TN) (P) unclassified
D00622  Fosinopril sodium (USP); Monopril (TN) (P) unclassified
D00623  Moexipril hydrochloride (USP); Univasc (TN) (P) unclassified
D00624  Perindopril erbumine (JAN/USP); Aceon (TN) (P) unclassified
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4
D00673  Ranitidine hydrochloride (JP18/USP); Zantac (TN) (P) unclassified
D00698  Aprobarbital (INN); Alurate (TN) (P) unclassified
D00699  Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) (P) unclassified
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) unclassified
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00707  Fomepizole (JAN/USAN/INN); Antizol (TN) (P) CYP inhibition: CYP3A4
D00712  Methohexital sodium (USP); Brevital sodium (TN) (P) unclassified
D00713  Thiamylal sodium (JP18); Surital (TN) (P) unclassified
D00714  Thiopental sodium (JP18/USP/INN); Pentothal (TN) (P) unclassified
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (P) Enzyme: CYP3A4 / Target: MTOR / CYP inhibition: CYP3A4
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00823  Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) (P) unclassified
D00824  Fluvoxamine maleate (JP18/USP); Luvox (TN) (P) CYP inhibition: CYP3A4
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00851  Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) (P) unclassified
D00854  Quinupristin and dalfopristin; Synercid (TN) (P) CYP inhibition: CYP3A4
D00879  Rifapentine (USAN/INN); Priftin (TN) (P) CYP induction: CYP3A4
D00882  Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) (P) unclassified
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) Enzyme: CYP3A4
D00895  Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) (P) unclassified
D00896  Efavirenz (JAN/USP/INN); Sustiva (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00960  Anastrozole (JP18/USP/INN); Arimidex (TN) (P) CYP inhibition: CYP3A4
D00961  Bicalutamide (JP18/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01059  Nimustine hydrochloride (JAN); Nidran (TN) (P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01068  Vinblastine sulfate (JP18/USP); Exal (TN); Velban (TN) (P) Enzyme: CYP3A4
D01069  Cilazapril (USAN); Cilazapril hydrate (JP18); Inhibace (TN) (P) unclassified
D01071  Hexobarbital (JAN/INN) (P) unclassified
D01078  Telithromycin (JAN/USAN/INN); Ketek (TN) (P) unclassified
D01119  Temocapril hydrochloride (JP18/USAN); Acecol (TN) (P) unclassified
D01155  Gemcitabine hydrochloride (JAN/USP); Gemzar (TN) (P) unclassified
D01211  Leucovorin calcium (USP); Calcium folinate (JP18); Uzel (TN); Wellcovorin (TN) (P) unclassified
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01235  Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) (P) CYP inhibition: CYP3A4
D01236  Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4
D01264  Daunorubicin hydrochloride (JP18/USP); Cerubidine (TN) (P) unclassified
D01275  Doxorubicin hydrochloride (JP18/USP); Adriacin (TN); Adriamycin (TN); Doxil (TN); Rubex (TN) (P) unclassified
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01280  Warfarin potassium (JP18); Athrombin-K (TN) (P) unclassified
D01309  Doxifluridine (JP18/INN); Furtulon (TN) (P) unclassified
D01310  Secobarbital sodium (JAN/USP); Seconal sodium (TN) (P) unclassified
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01339  Midecamycin (JP18/INN); Medemycin (TN) (P) CYP inhibition: CYP3A4
D01361  Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) (P) unclassified
D01363  Carboplatin (JP18/USP/INN); Paraplatin (TN) (P) unclassified
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) unclassified
D01404  Sobuzoxane (JAN); Perazolin (TN) (P) unclassified
D01416  Nedaplatin (JAN/INN); Aqupla (TN) (P) unclassified
D01425  Lopinavir (JAN/USP/INN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP3A4
D01510  Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01549  Imidapril hydrochloride (JP18); Tanatril (TN) (P) unclassified
D01615  Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01632  Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01633  Enocitabine (JAN/INN); Sunrabin (TN) (P) unclassified
D01636  Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) (P) CYP inhibition: CYP3A4
D01667  Delapril hydrochloride (JAN/USAN); Adecut (TN) (P) unclassified
D01740  Barbital (JP18/INN); Barbital (TN) (P) unclassified
D01747  Idarubicin hydrochloride (JP18/USP); Idamycin (TN) (P) unclassified
D01760  Ranimustine (JAN/INN); Cymerin (TN) (P) unclassified
D01769  Vindesine sulfate (JAN/USAN); Fildesin (TN) (P) unclassified
D01790  Oxaliplatin (JAN/USP/INN); Eloxatin (TN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01900  Alacepril (JP18/INN); Cetapril (TN) (P) unclassified
D01907  Fludarabine phosphate (JAN/USP); Fludara (TN) (P) unclassified
D01911  Aclarubicin hydrochloride (JP18); Aclacinon (TN) (P) unclassified
D01935  Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) (P) Enzyme: CYP3A4
D01948  Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) CYP inhibition: CYP3A4
D02009  Erythromycin lactobionate (JP18/USP); Erythrocin (TN) (P) unclassified
D02063  Peplomycin sulfate (JP18/USAN); Pepleo (TN) (P) unclassified
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) CYP induction: CYP3A4
D02102  Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02126  Primaquine phosphate (JAN/USP); Primaquine (TN) (P) unclassified
D02131  Tegafur and uracil; Uftoral (TN) (P) unclassified
D02165  Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) (P) Enzyme: CYP3A4
D02166  Mitoxantrone hydrochloride (JAN/USP); Novantron (TN) (P) unclassified
D02168  Topotecan hydrochloride (USAN); Nogitecan hydrochloride (JAN); Hycamtin (TN); Potactasol (TN) (P) unclassified
D02174  Dexamethasone acetate (JAN/USP); Decadronal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02177  Bleomycin sulfate (JP18/USP); Blenoxane (TN) (P) unclassified
D02184  Erythromycin stearate (JP18/USP); Bristamycin (TN) (P) unclassified
D02197  Vincristine sulfate (JP18/USP); VCR; Marqibo (TN); Oncovin (TN); Vincasar (TN); Vincrex (TN) (P) unclassified
D02214  Epirubicin hydrochloride (JP18/USP); EPI; Ellence (TN) (P) unclassified
D02252  Amobarbital sodium (JAN/USP); Amytal sodium (TN) (P) unclassified
D02253  Pentobarbital calcium (JP18); Ravona (TN) (P) unclassified
D02356  Verapamil (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02372  Perospirone hydrochloride hydrate (JAN); Lullan (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) unclassified
D02523  Erythromycin acistrate (USAN); Erasis (TN) (P) unclassified
D02524  Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) (P) unclassified
D02525  Erythromycin propionate (USAN) (P) unclassified
D02537  Dronedarone (INN) (P) unclassified
D02554  Rifaximin (JAN/USAN/INN); Xifaxan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) CYP inhibition: CYP3A4
D02556  Ravuconazole (prop.INN) (P) unclassified
D02591  Dexamethasone acefurate (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02592  Dexamethasone beloxil (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02618  Butobarbital (BAN); Butethal; Neonal (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) Enzyme: CYP3A4
D02817  Allobarbital (USAN/INN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03046  Cytarabine ocfosfate hydrate (JAN); Cytarabine ocfosphate hydrate; Fosteabine sodium monohydrate; Starasid (TN) (P) unclassified
D03077  Benazeprilat (USAN/INN) (P) unclassified
D03098  Berythromycin (USAN/INN); Erythromycin B (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03180  Butabarbital (USP); Secbutabarbital (BAN) (P) unclassified
D03182  Butalbital (USP/INN); Sandoptal (TN) (P) unclassified
D03229  Bleomycin hydrochloride (JP18); BLM; Bleo (TN) (P) unclassified
D03230  Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) (P) unclassified
D03250  Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) (P) unclassified
D03440  Ceronapril (USAN/INN) (P) unclassified
D03503  Cimetidine hydrochloride (USP); Cimetidine hydrochloride (TN) (P) CYP inhibition: CYP3A4
D03656  Darunavir (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP induction: CYP3A4
D03752  Quinapril (INN) (P) unclassified
D03753  Perindopril (USAN/INN) (P) unclassified
D03756  Indolapril hydrochloride (USAN) (P) unclassified
D03758  Libenzapril (USAN/INN) (P) unclassified
D03760  Pentopril (USAN/INN) (P) unclassified
D03763  Pivopril (USAN/INN) (P) unclassified
D03765  Spirapril hydrochloride (USAN); Renormax (TN) (P) unclassified
D03767  Zofenopril calcium (USAN); Zoprace (TN) (P) unclassified
D03769  Enalaprilat (USP); Enalaprilat dihydrate; Vasotec (TN) (P) unclassified
D03772  Fosinoprilat (USAN/INN) (P) unclassified
D03773  Quinaprilat (USAN/INN) (P) unclassified
D03775  Spiraprilat (USAN/INN) (P) unclassified
D03776  Zofenoprilat arginine (USAN) (P) unclassified
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03846  Dimethyl fumarate (JAN/USAN); Tecfidera (TN) (P) unclassified
D03914  Dronedarone hydrochloride (USP); Multaq (TN) (P) unclassified
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4
D04054  Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate (P) unclassified
D04059  Mepenzolate bromide and phenobarbital; Trancolon P (TN) (P) unclassified
D04077  Eterobarb (USAN/INN); Antilon (TN) (P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04187  Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) (P) unclassified
D04307  Proxyphylline, ephedrine hydrochloride and phenobarbital; Asthmolysin D (TN) (P) unclassified
D04475  Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) (P) unclassified
D04477  Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) (P) unclassified
D04536  Influenza virus vaccine (USP); FluShield (TN); Fluarix quadrivalent (TN) (P) unclassified
D04539  Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) (P) unclassified
D04540  Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) (P) unclassified
D04547  Insulin, isophane (USP); Isophane insulin human (genetical recombination) injectable aqueous suspension (JP18); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (P) unclassified
D04866  Freeze-dried live attenuated measles vaccine (JP18) (CI) unclassified
D04985  Methohexital (USP/INN) (P) unclassified
D05024  Mibefradil dihydrochloride (USAN); Posicor (TN) (P) unclassified
D05152  Netupitant (USAN/INN) (P) unclassified
D05182  Influenza HA vaccine (JP18) (P) unclassified
D05351  Josamycin propionate (JP18); Josamy (TN) (P) CYP inhibition: CYP3A4
D05544  Live oral polimyelitis vaccine (JAN); Poliovirus vaccine live oral; Orimune (TN) (CI) unclassified
D05699  Ranitidine bismuth citrate (USAN); Tritec (TN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05932  Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) (P) unclassified
D06076  Teprotide (USAN/INN) (P) unclassified
D06106  Thiamylal (P) unclassified
D06399  Tegafur, gimeracil and oteracil potassium; Ts-1 (TN); Teysuno (TN) (P) unclassified
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4
D06466  Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) (CI) unclassified
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06503  Pemetrexed sodium hydrate (JAN); Pemetrexed disodium heptahydrate; Alimta (TN) (P) unclassified
D06512  Freeze-dried live attenuated rubella vaccine (JP18) (CI) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06887  Talbutal (INN); Lotusate (TN) (P) unclassified
D07073  Dexamethasone cipecilate (JAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07085  Bendamustine hydrochloride (JAN/USAN); Treanda (TN); Ribomustin (TN) (P) unclassified
D07100  Amrubicin hydrochloride (JAN/USAN); Calsed (TN) (P) unclassified
D07298  Barbexaclone (INN); Maliasin (TN) (P) unclassified
D07321  Vinylbital (INN); Vinylbitone (P) unclassified
D07322  Vinbarbital (INN) (P) unclassified
D07323  Cyclobarbital (INN); Ciclobarbital (TN) (P) unclassified
D07324  Proxibarbal (INN); Centralgol (TN) (P) unclassified
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07499  Benazepril (INN); Benazepril Sandoz (TN); Forteekor [veterinary] (TN) (P) unclassified
D07538  Bosentan (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP induction: CYP3A4
D07699  Cilazapril (INN); Inhibace (TN) (P) unclassified
D07710  Clarithromycin lactobionate; Klacid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07748  Conivaptan (INN) (P) unclassified
D07757  Cyclobarbital calcium (BAN); Phanodorn calcium (TN) (P) unclassified
D07781  Delapril (INN); Delaket (TN) (P) unclassified
D07782  Delavirdine (INN) (P) unclassified
D07796  Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07797  Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07798  Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07799  Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07800  Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07801  Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07802  Dexamethasone phosphate; Decadron-phosphate (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07866  Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) (P) Enzyme: CYP3A4
D07892  Enalapril (INN); Enalapril (TN) (P) unclassified
D07909  Erythromycin thiocyanate; Erythrocin (TN) (P) unclassified
D07910  Erythromycin stinoprate (INN); Erysec (TN) (P) unclassified
D07928  Ethinylestradiol propanesulfonate; Turisteron (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07984  Fluvoxamine (INN) (P) CYP inhibition: CYP3A4
D07992  Fosinopril (INN); Monopril (TN) (P) unclassified
D07993  Fosphenytoin (INN) (P) CYP induction: CYP3A4
D08068  Imidapril (INN); Hipertene (TN) (P) unclassified
D08080  Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP18); Insulin Humacart (TN) (P) unclassified
D08131  Lisinopril (INN); Zestril (TN) (P) unclassified
D08195  Methadone (BAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08217  Mibefradil (INN) (P) unclassified
D08225  Moexipril (INN) (P) unclassified
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08287  Norfloxacin nicotinate; Quinabic soluble powder (TN) [veterinary] (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08386  Pirarubicin hydrochloride; Pinorubin (TN); Therarubicin (TN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) CYP induction: CYP3A4
D08529  Spirapril (INN) (P) unclassified
D08566  Temocapril (INN) (P) unclassified
D08616  Teneligliptin (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08688  Zofenopril (INN); Zofenil (TN) (P) unclassified
D08774  Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08837  Aclidinium bromide (JAN/USAN/INN); Tudorza pressair (TN); Eklira genuair (TN) (P) CYP inhibition: CYP3A4
D08876  Boceprevir (INN/USAN); Victrelis (TN) (P) unclassified
D08914  Eribulin mesylate (USAN); Eribulin mesilate (JAN); Halaven (TN) (P) Enzyme: CYP3A4
D09012  Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (P) unclassified
D09197  Valsartan and hydrochlorothiazide (JP18); Co-dio (TN) (P) unclassified
D09215  Eslicarbazepine (USAN/INN) (P) CYP induction: CYP3A4
D09347  Fostamatinib (USAN) (P) Enzyme: CYP3A4
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) Enzyme: CYP3A4
D09394  Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) (P) CYP inhibition: CYP3A4
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) CYP induction: CYP3A4
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) Enzyme: CYP3A4
D09725  Emulsified influenza HA vaccine (A/H1N1); Arepanrix (H1N1) (TN) (P) unclassified
D09727  Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) (P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4
D09756  Teneligliptin hydrobromide hydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09881  Cobicistat (JAN/USAN/INN); Tybost (TN) (P) Enzyme-Target: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP induction: CYP3A4
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10064  Dabrafenib (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10065  Daclatasvir (USAN) (P) Enzyme: CYP3A4
D10081  Simeprevir (JAN/USAN) (P) unclassified
D10093  Asunaprevir (JAN/USAN); Sunvepra (TN) (P) CYP induction: CYP3A4
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10105  Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) (P) Enzyme: CYP3A4
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10246  Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4
D10469  Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) (P) unclassified
D10519  Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10526  Trifluridine and tipiracil hydrochloride; Lonsurf (TN) (P) unclassified
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10570  Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) (P) unclassified
D10582  Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) (P) CYP inhibition: CYP3A4
D10596  Pemetrexed sodium hemipentahydrate (JAN); Pemetrexed disodium hemipentahydrate; Pemetrexed accord (TN) (P) unclassified
D10639  Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) (P) unclassified
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10644  Isavuconazonium (USAN) (P) unclassified
D10745  Ombitasvir, paritaprevir and ritonavir; Technivie (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10753  Atazanavir and cobicistat; Evotaz (TN) (P) Enzyme: CYP3A4
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (P) unclassified
D10756  Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) unclassified
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (P) unclassified
D10882  Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) (P) CYP induction: CYP3A4
D10895  Fosaprepitant (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11034  Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (P) unclassified
D11390  Daunorubicin and cytarabine; Vyxeos (TN) (P) unclassified
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11521  Lamivudine, nevirapine and zidovudine (P) unclassified
D11565  Grazoprevir (USAN/INN); Grazoprevir anhydrous (P) unclassified
D11567  Insulin degludec and liraglutide; Xultophy (TN) (P) unclassified
D11580  Perindopril arginine (P) unclassified
D11661  Bendamustine hydrochloride hydrate (JAN); Bendamustine hydrochloride monohydrate; Treakisym (TN) (P) unclassified
D11673  Berotralstat (USAN/INN) (P) CYP inhibition: CYP3A4
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11858  Omeprazole magnesium, amoxicillin and rifabutin; Talicia (TN) (P) unclassified
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11968  Teneligliptin hydrobromide (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) unclassified
D12015  St. John's wort; SJW (P) unclassified
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (P) Enzyme: CYP3A4
D12353  Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (P) unclassified
D12619  Ensitrelvir (USAN/INN) (P) unclassified
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4