D00203 |
Amphotericin B (JP18/USP/INN); Ambisome (TN); Amphotec (TN); Fungizone (TN) |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) unclassified |
D00235 |
Atenolol (JP18/USP/INN); Tenormin (TN) |
(P) Enzyme: CYP2D6 |
D00255 |
Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) |
(P) Enzyme: CYP2D6 |
D00295 |
Cimetidine (JP18/USP/INN); Tagamet (TN) |
(P) CYP inhibition: CYP2D6 |
D00298 |
Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) unclassified |
D00432 |
Nadolol (JP18/USP/INN); Corgard (TN) |
(P) unclassified |
D00483 |
Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) |
(P) Enzyme: CYP2D6 |
D00513 |
Pindolol (JP18/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) |
(P) Enzyme: CYP2D6 |
D00598 |
Betaxolol hydrochloride (JP18/USP); Betoptic (TN); Kerlone (TN) |
(P) unclassified |
D00599 |
Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) |
(P) Enzyme: CYP2D6 |
D00600 |
Labetalol hydrochloride (JP18/USP); Normodyne (TN); Trandate (TN) |
(P) unclassified |
D00601 |
Metoprolol tartrate (JP18/USP); Lopressor (TN) |
(P) Enzyme: CYP2D6 |
D00616 |
Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) |
(P) unclassified |
D00619 |
Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) unclassified |
D00634 |
Bisoprolol fumarate (JP18/USP); Zebeta (TN) |
(P) unclassified |
D00644 |
Esmolol hydrochloride (JAN/USP); Brevibloc (TN) |
(P) unclassified |
D00738 |
Mepivacaine hydrochloride (JP18/USP); Carbocaine (TN); Polocaine (TN); Scandonest plain (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00765 |
Rocuronium bromide (JAN/USP/INN); Zemuron (TN) |
(P) unclassified |
D00776 |
Tizanidine hydrochloride (JP18/USP); Zanaflex (TN) |
(P) unclassified |
D00809 |
Amitriptyline hydrochloride (JP18/USP); Elavil (TN) |
(P) Enzyme: CYP2D6 |
D00811 |
Clomipramine hydrochloride (JP18/USP); Anafranil (TN) |
(P) Enzyme: CYP2D6 |
D00815 |
Imipramine hydrochloride (JP18/USP); Tofranil (TN) |
(P) Enzyme: CYP2D6 |
D00818 |
Maprotiline hydrochloride (JP18/USP); Ludiomil (TN) |
(P) Enzyme: CYP2D6 |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
D01026 |
Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) |
(P) unclassified |
D01179 |
Duloxetine hydrochloride (JAN/USP); Cymbalta (TN); Yentreve (TN) |
(P) CYP inhibition: CYP2D6 |
D01240 |
Deslanoside (JP18/USP/INN); Cedilanid-d (TN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) unclassified |
D01280 |
Warfarin potassium (JP18); Athrombin-K (TN) |
(P) unclassified |
D01369 |
Bevantolol hydrochloride (JAN/USAN); Calvan (TN); Vantol (TN) |
(P) unclassified |
D01469 |
Amosulalol hydrochloride (JP18); Lowgan (TN) |
(P) unclassified |
D01504 |
Bufetolol hydrochloride (JP18); Adobiol (TN) |
(P) unclassified |
D01691 |
Nipradilol (JAN/INN); Hypadil (TN) |
(P) unclassified |
D01741 |
Celiprolol hydrochloride (JAN/USAN); Selectol (TN) |
(P) unclassified |
D01830 |
Arotinolol hydrochloride (JP18); Almarl (TN) |
(P) unclassified |
D01847 |
Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN) |
(P) unclassified |
D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP2D6 |
D02106 |
Arsenic trioxide (JP18/USAN); Trisenox (TN) |
(P) unclassified |
D02260 |
Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18); Paxil (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
D02342 |
Bisoprolol (JAN/USAN/INN) |
(P) unclassified |
D02567 |
Escitalopram oxalate (JAN/USP); Lexapro (TN) |
(P) Enzyme: CYP2D6 / CYP inhibition: CYP2D6 |
D02587 |
Metildigoxin (JP18); Lanirapid (TN) |
(P) unclassified |
D02740 |
Lidocaine and prilocaine; Lidocaine and propitocaine; Emla (TN); Oraqix (TN); Lidocaine and prilocaine (TN) |
(P) unclassified |
D03658 |
Dasatinib (JAN/INN) |
(P) unclassified |
D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) unclassified |
D05277 |
Formoterol fumarate hydrate (JP18); Formoterol fumarate dihydrate; Atock (TN); Foradil (TN) |
(P) unclassified |
D05380 |
Pazopanib hydrochloride (JAN/USAN); Votrient (TN) |
(P) unclassified |
D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) unclassified |
D06407 |
Vandetanib (JAN/USAN/INN); Caprelsa (TN) |
(P) unclassified |
D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) unclassified |
D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) unclassified |
D06637 |
Romidepsin (JAN/USAN/INN); Istodax (TN) |
(P) unclassified |
D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) unclassified |
D09535 |
Mirabegron (JAN/USAN/INN); Myrbetriq (TN) |
(P) CYP inhibition: CYP2D6 |
D09595 |
Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) |
(P) unclassified |
D09701 |
Abiraterone acetate (JAN/USP); Zytiga (TN) |
(P) unclassified |
D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(P) Enzyme: CYP2D6 |
D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) unclassified |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP2D6 |
D10019 |
Panobinostat lactate (JAN); Farydak (TN) |
(P) CYP inhibition: CYP2D6 |
D10255 |
Anagrelide hydrochloride hydrate (JAN); Anagrelide hydrochloride monohydrate; Agrylin (TN) |
(P) unclassified |
D10501 |
Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) |
(P) unclassified |
D10506 |
Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) |
(P) unclassified |
D10514 |
Dacomitinib (USAN); Dacomitinib hydrate (JAN); Vizimpro (TN) |
(P) CYP inhibition: CYP2D6 |
D10533 |
Umeclidinium bromide and vilanterol; Anoro (TN) |
(P) Enzyme: CYP2D6 |
D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
D10993 |
Tucidinostat (JAN/USAN/INN); Hiyasta (TN) |
(P) unclassified |
D11027 |
Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) |
(P) unclassified |
D11035 |
Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) |
(P) unclassified |
D11036 |
Glycopyrrolate and formoterol; Bevespi (TN) |
(P) unclassified |
D11062 |
Osilodrostat phosphate (JAN/USAN); Isturisa (TN) |
(P) Enzyme: CYP2D6 |
D11584 |
Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) |
(P) unclassified |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP2D6 |
D11708 |
Givosiran sodium (JAN); Givlaari (TN) |
(P) unclassified |