D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) |
(P) unclassified |
D00184 |
Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) unclassified |
D00235 |
Atenolol (JP18/USP/INN); Tenormin (TN) |
(P) Enzyme: CYP2D6 |
D00255 |
Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) |
(P) Enzyme: CYP2D6 |
D00276 |
Clarithromycin (JP18/USP/INN); Biaxin (TN) |
(P) unclassified |
D00295 |
Cimetidine (JP18/USP/INN); Tagamet (TN) |
(P) CYP inhibition: CYP2D6 |
D00298 |
Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) unclassified |
D00322 |
Fluconazole (JP18/USP/INN); Diflucan (TN) |
(P) unclassified |
D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) Enzyme: CYP2D6 |
D00432 |
Nadolol (JP18/USP/INN); Corgard (TN) |
(P) unclassified |
D00443 |
Spironolactone (JP18/USP/INN); Aldactone (TN) |
(P) unclassified |
D00480 |
Promethazine hydrochloride (JP18/USP); Phenergan (TN); Promethegan (TN) |
(P) Enzyme: CYP2D6 |
D00483 |
Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) |
(P) Enzyme: CYP2D6 |
D00513 |
Pindolol (JP18/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) |
(P) Enzyme: CYP2D6 |
D00515 |
Nitroglycerin (JP18/USP); Glyceryl trinitrate; Minitran (TN); Nitro-bid (TN); Nitro-dur (TN); Nitromist (TN); Transderm-nitro (TN) |
(P) unclassified |
D00545 |
Isoflurane (JP18/USP/INN); Forane (TN) |
(P) unclassified |
D00547 |
Sevoflurane (JP18/USAN/INN); Ultane (TN) |
(P) unclassified |
D00598 |
Betaxolol hydrochloride (JP18/USP); Betoptic (TN); Kerlone (TN) |
(P) unclassified |
D00599 |
Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) |
(P) Enzyme: CYP2D6 |
D00600 |
Labetalol hydrochloride (JP18/USP); Normodyne (TN); Trandate (TN) |
(P) unclassified |
D00601 |
Metoprolol tartrate (JP18/USP); Lopressor (TN) |
(P) Enzyme: CYP2D6 |
D00603 |
Timolol maleate (JP18/USP); Blocadren (TN); Istalol (TN); Timoptic (TN) |
(P) Enzyme: CYP2D6 |
D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) unclassified |
D00631 |
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) |
(P) Enzyme: CYP2D6 / Target: CACNA1C CACNA1D CACNA1F CACNA1S / CYP inhibition: CYP2D6 |
D00634 |
Bisoprolol fumarate (JP18/USP); Zebeta (TN) |
(P) unclassified |
D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) unclassified |
D00638 |
Flecainide acetate (JP18/USP); Tambocor (TN) |
(P) Enzyme: CYP2D6 |
D00639 |
Mexiletine hydrochloride (JP18/USP); Mexitil (TN) |
(P) Enzyme: CYP2D6 |
D00644 |
Esmolol hydrochloride (JAN/USP); Brevibloc (TN) |
(P) unclassified |
D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) unclassified |
D00765 |
Rocuronium bromide (JAN/USP/INN); Zemuron (TN) |
(P) unclassified |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
D01025 |
Levobunolol hydrochloride (JAN/USP); Betagan (TN) |
(P) unclassified |
D01026 |
Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) |
(P) unclassified |
D01162 |
Verteporfin (JAN/USP/INN); Visudyne (TN) |
(P) unclassified |
D01177 |
Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) |
(P) unclassified |
D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) unclassified |
D01240 |
Deslanoside (JP18/USP/INN); Cedilanid-d (TN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) unclassified |
D01337 |
Epoprostenol sodium (JAN/USAN); Flolan (TN); Veletri (TN) |
(P) unclassified |
D01369 |
Bevantolol hydrochloride (JAN/USAN); Calvan (TN); Vantol (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) unclassified |
D01469 |
Amosulalol hydrochloride (JP18); Lowgan (TN) |
(P) unclassified |
D01504 |
Bufetolol hydrochloride (JP18); Adobiol (TN) |
(P) unclassified |
D01554 |
Pilsicainide hydrochloride hydrate (JP18); Pilsicainide hydrochloride; SUN 1165 (TN); Sunrythm (TN) |
(P) unclassified |
D01565 |
Indometacin farnesil (JAN); Infree (TN) |
(P) unclassified |
D01691 |
Nipradilol (JAN/INN); Hypadil (TN) |
(P) unclassified |
D01741 |
Celiprolol hydrochloride (JAN/USAN); Selectol (TN) |
(P) unclassified |
D01830 |
Arotinolol hydrochloride (JP18); Almarl (TN) |
(P) unclassified |
D01847 |
Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN) |
(P) unclassified |
D01902 |
Fonazine mesylate (USAN); Dimetotiazine mesilate (JAN); Banistyl (TN) |
(P) unclassified |
D01935 |
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) |
(P) unclassified |
D01943 |
Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) |
(P) unclassified |
D01973 |
Eletriptan hydrobromide (JAN/USAN); Relpax (TN) |
(P) unclassified |
D01992 |
Tandospirone citrate (JAN/USAN); SM 3997; Sediel (TN) |
(P) unclassified |
D02019 |
Magnesium sulfate hydrate and glucose; Magnesol (TN) |
(P) unclassified |
D02274 |
Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18); Dantrium (TN); Ryanodex (TN) |
(P) unclassified |
D02342 |
Bisoprolol (JAN/USAN/INN) |
(P) unclassified |
D02587 |
Metildigoxin (JP18); Lanirapid (TN) |
(P) unclassified |
D02714 |
Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) |
(P) unclassified |
D03290 |
Promethazine methylenedisalicylate (JAN); Pyrethia (TN) |
(P) Enzyme: CYP2D6 |
D04046 |
Salicylamide, acetaminophen, anhydrous caffeine and promethazine methylenedisalicylate; PL (TN) |
(P) unclassified |
D04187 |
Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) |
(P) unclassified |
D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(P) unclassified |
D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) CYP inhibition: CYP2D6 |
D06213 |
Treprostinil (JAN/USAN/INN); Remodulin (TN) |
(P) unclassified |
D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) unclassified |
D07505 |
Latanoprost and timolol maleate; Xalacom (TN) |
(P) unclassified |
D08493 |
Dorzolamide hydrochloride and timolol maleate (JP18); Cosopt (TN) |
(P) Enzyme: CYP2D6 |
D08768 |
Promethazine hibenzate; Hiberna (TN) |
(P) Enzyme: CYP2D6 |
D09535 |
Mirabegron (JAN/USAN/INN); Myrbetriq (TN) |
(P) CYP inhibition: CYP2D6 |
D09701 |
Abiraterone acetate (JAN/USP); Zytiga (TN) |
(P) unclassified |
D09815 |
Travoprost and timolol maleate; Duotrav (TN) |
(P) unclassified |
D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(P) Enzyme: CYP2D6 |
D09994 |
Selexipag (JAN/USAN/INN); Uptravi (TN) |
(P) unclassified |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP2D6 |
D10298 |
Brimonidine tartrate and timolol maleate; Combigan (TN); Aibeta (TN) |
(P) unclassified |
D10512 |
Brinzolamide and timolol maleate; Azorga (TN) |
(P) Enzyme: CYP2D6 |
D10514 |
Dacomitinib (USAN); Dacomitinib hydrate (JAN); Vizimpro (TN) |
(P) CYP inhibition: CYP2D6 |
D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) unclassified |
D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
D10569 |
Tafluprost and timolol maleate; Tapcom (TN) |
(P) unclassified |
D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP2D6 |
D10804 |
Carteolol and latanoprost; Mikeluna (TN) |
(P) unclassified |
D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
D11027 |
Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) |
(P) unclassified |
D11190 |
Vosoritide (USAN/INN); Vosoritide (genetical recombination) (JAN); Voxzogo (TN) |
(P) unclassified |
D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP2D6 |
D11708 |
Givosiran sodium (JAN); Givlaari (TN) |
(P) unclassified |
D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) unclassified |
D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(P) unclassified |