| D00049 |
Nicotinic acid (JP16/INN); Niacin (USP); Niacor (TN); Niaspan (TN) |
(P) unclassified |
| D00163 |
Chenodeoxycholic acid (JP16/INN); Chenodiol (USAN); Chenix (TN) |
(P) unclassified |
| D00184 |
Ciclosporin (JP16); Cyclosporine (USP); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: SLCO1B1 ABCB11 |
| D00279 |
Clofibrate (JP16/USP/INN); Atromid-S (TN) |
(CI1) unclassified |
| D00298 |
Digoxin (JP16/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) unclassified |
| D00322 |
Fluconazole (JP16/USAN/INN); Diflucan (TN) |
(P) Enzyme: CYP3A4 |
| D00565 |
Fenofibrate (JAN/INN); Antara (TN); Lipantil (TN); Lipofen (TN); Tricor (TN); Triglide (TN) |
(CI1,P) unclassified |
| D00578 |
Voriconazole (JAN/USAN/INN); Vfend (TN) |
(P) Enzyme: CYP3A4 |
| D00734 |
Ursodeoxycholic acid (JP16/INN); Ursodiol (USP); Actigall (TN); Urso (TN) |
(P) unclassified |
| D00896 |
Efavirenz (JAN/INN); Sustiva (TN) |
(P) Enzyme: CYP3A4 |
| D01080 |
Daptomycin (JAN/USAN/INN); Cubicin (TN) |
(P) unclassified |
| D01160 |
Saquinavir mesilate (JAN); Saquinavir mesylate (USP); Invirase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: SLCO1B1 |
| D01227 |
Bosentan hydrate (JAN); Bosentan (USAN); Tracleer (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 / Transporter inhibition: ABCB11 |
| D01240 |
Deslanoside (JP16/USP/INN); Cedilanid-d (TN) |
(P) unclassified |
| D01291 |
Nicomol (JP16/INN); Cholexamin (TN) |
(P) unclassified |
| D01300 |
Clinofibrate (JP16/INN); Lipoclin (TN) |
(CI1,P) unclassified |
| D01366 |
Bezafibrate (JP16/USAN/INN); Bezatol SR (TN) |
(CI1,P) unclassified |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) Enzyme: CYP3A4 |
| D01754 |
Niceritrol (JP16/INN); Perycit (TN) |
(P) unclassified |
| D02587 |
Metildigoxin (JP16); Lanirapid (TN) |
(P) unclassified |
| D04121 |
Exenatide (JAN/USAN/INN); Byetta (TN) |
(P) unclassified |
| D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |