Target-based Classification of Drugs

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 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
     Adrenaline
     Dopamine
     Histamine
       HRH1 [HSA:3269] [KO:K04149]
         D08587  Thonzylamine (INN)
         D01801  Thonzylamine hydrochloride (JAN/USAN)
         D08183  Mepyramine (INN)
         D05660  Pyrilamine maleate (USP)
         D07194  Thenalidine (INN)
         D08645  Tripelennamine (INN)
         D02091  Tripelennamine hydrochloride (USP)
         D06246  Tripelennamine citrate
         D07195  Chloropyramine (INN)
         D07679  Chloropyramine hydrochloride
         D00494  Promethazine (JAN/INN)
         D00480  Promethazine hydrochloride (JP18/USP) <JP/US>
         D01242  Promethazine teoclate (JAN/INN)
         D03290  Promethazine methylenedisalicylate (JAN) <JP>
         D08432  Promethazine maleate
         D08768  Promethazine hibenzate <JP>
         D07196  Tolpropamine (INN)
         D07853  Dimetindene (INN)
         D01343  Dimethindene maleate (USAN)
         D03535  Clemastine (USAN)
         D00666  Clemastine fumarate (JP18/USP) <JP/US>
         D07197  Bamipine (INN)
         D07492  Bamipine dihydrochloride
         D07493  Bamipine lactate
         D08355  Pheniramine (INN)
         D01174  Pheniramine maleate (JAN/USP)
         D08091  Isothipendyl (INN)
         D01143  Isothipendyl hydrochloride (JAN)
         D00300  Diphenhydramine (JP18/INN) <JP>
         D00669  Diphenhydramine hydrochloride (JP18/USP) <JP/US>
         D02419  Diphenhydramine salicylate (JAN)
         D03285  Diphenhydramine tannate (JP18)
         D03360  Diphenhydramine laurylsulfate (JAN) <JP>
         D03854  Diphenhydramine citrate (USP)
         D07198  Chlorphenoxamine (INN)
         D07684  Chlorphenoxamine hydrochloride
         D07875  Doxepin (INN)
         D00814  Doxepin hydrochloride (USP) <US>
         D00774  Orphenadrine citrate (USP) <US>
         D07854  Dimetotiazine (INN)
         D01902  Fonazine mesylate (USAN) <JP>
         D02599  Orphenadrine hydrochloride
         D00270  Chlorpromazine (USP/INN)
         D00789  Chlorpromazine hydrochloride (JP18/USP) <JP/US>
         D03274  Chlorpromazine hibenzate (JAN)
         D04034  Chlorpromazine phenolphthalinate (JAN) <JP>
         D09819  Chlorpromazine tannate (JAN)
         D00454  Olanzapine (JAN/USP/INN) <JP/US>
         D06623  Olanzapine pamoate (USAN) <US>
         D08054  Hydroxyzine (INN)
         D00672  Hydroxyzine hydrochloride (JP18/USP) <JP/US>
         D01096  Hydroxyzine pamoate (JP18/USP) <JP/US>
         D08297  Opipramol (INN)
         D01477  Opipramol hydrochloride (JAN/USAN)
         D08216  Mianserin (INN)
         D01358  Mianserin hydrochloride (JAN/USAN) <JP>
         D07522  Betahistine (INN)
         D01592  Betahistine mesilate (JP18) <JP>
         D03102  Betahistine hydrochloride (USP)
         D01295  Cinnarizine (JAN/USAN/INN)
         D07734  Cinnarizine dihydrochloride
         D08117  Levocabastine (INN)
         D01717  Levocabastine hydrochloride (JAN/USP) <JP>
         D07483  Azelastine (INN)
         D00659  Azelastine hydrochloride (JP18/USP) <JP/US>
         D07458  Antazoline (INN)
         D02950  Antazoline phosphate (USP)
         D07459  Antazoline hydrochloride
         D08293  Olopatadine (INN)
         D01192  Olopatadine hydrochloride (JP18/USP) <JP/US>
         D03166  Bromodiphenhydramine hydrochloride (USP)
         D07862  Diphenylpyraline (INN)
         D01172  Diphenylpyraline hydrochloride (JAN)
         D01627  Diphenylpyraline teoclate (JAN)
         D07617  Carbinoxamine (INN)
         D01336  Carbinoxamine maleate (JAN/USP) <US>
         D09808  Carbinoxamine diphenyldisulfonate (JAN)
         D07878  Doxylamine (INN)
         D02327  Doxylamine succinate (USP)
         D00520  Dimenhydrinate (JP18/USP/INN) <JP/US>
         D07543  Brompheniramine (INN)
         D00663  Brompheniramine maleate (USP)
         D07803  Dexchlorpheniramine (INN)
         D00668  Dexchlorpheniramine maleate (USP) <JP/US>
         D07398  Chlorphenamine (INN)
         D00665  Chlorpheniramine maleate (JP18/USP) <JP>
         D03475  Chlorpheniramine polistirex (USAN)
         D03704  Dexbrompheniramine maleate (USP)
         D07400  Histapyrrodine (INN)
         D07125  Alimemazine (INN)
         D02245  Trimeprazine tartrate (USP) <JP>
         D04979  Methdilazine (INN)
         D04980  Methdilazine hydrochloride (USP)
         D01324  Mequitazine (JP18/INN) <JP>
         D07401  Oxomemazine (INN)
         D07547  Buclizine (INN)
         D02089  Buclizine hydrochloride (USAN)
         D03621  Cyclizine (INN)
         D02090  Cyclizine lactate (BAN)
         D03622  Cyclizine hydrochloride (USP)
         D08163  Meclozine (BAN)
         D01317  Meclizine hydrochloride (JAN/USP) <US>
         D07662  Cetirizine (INN)
         D00664  Cetirizine hydrochloride (JP18/USP) <JP/US>
         D07402  Levocetirizine (USAN/INN)
         D08118  Levocetirizine dihydrochloride (USP) <JP/US>
         D07765  Cyproheptadine (INN)
         D02234  Cyproheptadine hydrochloride (JP18/USP) <JP/US>
         D08353  Phenindamine (INN)
         D02148  Phenindamine tartrate (USAN)
         D08648  Triprolidine (INN)
         D01782  Triprolidine hydrochloride (USP)
         D07403  Pyrrobutamine (BAN)
         D07482  Azatadine (INN)
         D00662  Azatadine maleate (USP)
         D00234  Astemizole (JAN/USP/INN)
         D00521  Terfenadine (JAN/USAN/INN)
         D00364  Loratadine (JAN/USP/INN) <JP>
         D08161  Mebhydrolin (INN)
         D01786  Mebhydrolin napadisilate (JAN)
         D07404  Deptropine (INN)
         D07790  Deptropine citrate
         D08105  Ketotifen (INN)
         D01332  Ketotifen fumarate (JP18/USAN) <JP>
         D02760  Acrivastine (USAN/INN)
         D01478  Ebastine (JP18/USAN/INN) <JP>
         D07406  Pimethixene (INN)
         D07900  Epinastine (INN)
         D01713  Epinastine hydrochloride (JAN) <JP/US>
         D01117  Mizolastine (JAN/INN)
         D07958  Fexofenadine (INN)
         D00671  Fexofenadine hydrochloride (JP18/USP) <JP/US>
         D03693  Desloratadine (JAN/USP/INN) <JP/US>
         D07407  Rupatadine (INN)
         D08497  Rupatadine fumarate (JAN) <JP>
         D09570  Bilastine (JAN/INN) <JP>
         D10230  Quifenadine (INN)
         D10510  Sequifenadine
         D07890  Emedastine (INN)
         D02249  Emedastine difumarate (JP18/USP) <JP>
         D06552  Alcaftadine (JAN/USAN/INN) <US>
         D04445  Histamine phosphate (USP) <US>
         D01460  Homochlorcyclizine hydrochloride (JP18) <JP>
         D01654  Bepotastine besylate (USAN) <JP/US>
         D01701  Difeterol hydrochloride (JAN)
         D02067  Diphenylimidazole (JAN)
         D03056  Barmastine (USAN/INN)
         D03491  Cidoxepin hydrochloride (USAN)
         D03568  Closiramine aceturate (USAN)
         D03620  Cycliramine maleate (USAN)
         D03893  Dorastine hydrochloride (USAN)
         D03963  Efletirizine dihydrochloride (USAN)
         D04055  Esmirtazapine maleate (USAN)
         D04494  Icotidine (USAN)
         D05196  Noberastine (USAN/INN)
         D05664  Pyroxamine maleate (USAN)
         D05742  Rocastine hydrochloride (USAN)
         D05769  Rotoxamine (USAN/INN)
         D06012  Tazifylline hydrochloride (USAN)
         D06021  Tecastemizole (USAN/INN)
         D06063  Temelastine (USAN/INN)
         D06084  Tesmilifene hydrochloride (USAN)
         D06376  Zolamine hydrochloride (USAN)
         D07532  Bisulepin
         D07533  Bisulepin hydrochloride
         D07860  Dioxopromethazine hydrochloride
         D07889  Embramine (INN)
         D08040  Histamine (DCF) <US>
         D08041  Homochlorcyclizine (INN)
         D08305  Orphenadrine (INN)
         D08967  Phenyltoloxamine citrate (USP)
         D09705  Bepotastine (USAN/INN)
         D09747  Difeterol phosphate (JAN)
         D09748  Difeterol (JAN/INN)
         D09838  Broizine (JAN)
       HRH2 [HSA:3274] [KO:K04150]
       HRH3 [HSA:11255] [KO:K04151]
       HRH4 [HSA:59340] [KO:K04152]
     Serotonin
     Trace amine
     Angiotensin
     Bradykinin
     Cholecystokinin
     Endothelin
     Follicle stimulating hormone
     Ghrelin
     Gonadotropin-releasing hormone
     Lutropin-choriogonadotropic hormone
     Melanocortin
     Motilin
     Neuropeptide Y
     Opioid
     Orexin
     Oxytocin
     Relaxin
     Somatostatin
     Tachykinin
     Thrombin
     Thyrotropin-releasing hormone
     Vasopressin
     Purine / pyrimidine
     Adenosine
     Cysteinyl leukotriene
     Free fatty acid
     Leukotriene
     Lysophosphatidic acid
     Prostaglandin
     Prostacyclin
     Sphingolipid
     Thromboxane
     Cannabinoid
     Melatonin
     Platelet activating factor
     R-spondin
   Secretin receptor family
   Metabotropic glutamate receptor family
   Frizzled / Smoothened family
   Others
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 17, 2024

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