G Protein-coupled receptors
Rhodopsin family
Acetylcholine (muscarinic)
Adrenaline
alpha1a-adrenergic receptor [HSA:148] [KO:K04135]
alpha1-adrenergic receptor [HSA:146 147 148] [KO:K04137 K04136 K04135]
Epinephrine [ATC:A01AD01 B02BC09 C01CA24 R01AA14 R03AA01 S01EA01]
D00095 Epinephrine (USP/INN) D00996 Epinephrine hydrochloride (JAN) D02149 Epinephrine bitartrate (JAN/USP)
Agonist Agonist Agonist
Etilefrine [ATC:C01CA01]
Norepinephrine [ATC:C01CA03]
Norfenefrine [ATC:C01CA05]
Phenylephrine [ATC:C01CA06 R01AA04 R01AB01 R01BA03 S01FB01 S01GA05]
Oxedrine [ATC:C01CA08 S01GA06]
Metaraminol [ATC:C01CA09]
Methoxamine [ATC:C01CA10]
Midodrine [ATC:C01CA17]
Arbutamine [ATC:C01CA22]
Ephedrine [ATC:C01CA26 R01AA03 R01AB05 R03CA02 S01FB02]
Prazosin [ATC:C02CA01]
Indoramin [ATC:C02CA02]
Trimazosin [ATC:C02CA03]
Doxazosin [ATC:C02CA04]
Urapidil [ATC:C02CA06]
Ketanserin [ATC:C02KD01]
Phentolamine [ATC:C04AB01 V03AB36]
Tolazoline [ATC:C04AB02 M02AX02]
Nicergoline [ATC:C04AE02]
Phenoxybenzamine [ATC:C04AX02]
Moxisylyte [ATC:C04AX10 G04BE06]
Ifenprodil [ATC:C04AX28]
Labetalol [ATC:C07AG01]
Carvedilol [ATC:C07AG02]
Methylergometrine [ATC:G02AB01]
Ergot alkaloids [ATC:G02AB02]
Ergometrine [ATC:G02AB03]
Alfuzosin [ATC:G04CA01]
Tamsulosin [ATC:G04CA02]
Terazosin [ATC:G04CA03]
Silodosin [ATC:G04CA04]
Dihydroergotamine [ATC:N02CA01]
Ergotamine [ATC:N02CA02]
Levomepromazine [ATC:N05AA02]
Sertindole [ATC:N05AE03]
Pimozide [ATC:N05AG02]
Clozapine [ATC:N05AH02]
Asenapine [ATC:N05AH05]
Olanzapine [ATC:N05AH03]
Quetiapine [ATC:N05AH04]
Risperidone [ATC:N05AX08]
Mianserin [ATC:N06AX03]
Oxymetazoline [ATC:R01AA05 R01AB07 S01GA04]
Tetryzoline [ATC:R01AA06 R01AB03 S01GA02]
Xylometazoline [ATC:R01AA07 R01AB06 S01GA03]
Naphazoline [ATC:R01AA08 R01AB02 S01GA01]
Tramazoline [ATC:R01AA09]
Pseudoephedrine [ATC:R01BA02]
Dipivefrine [ATC:S01EA02]
Dapiprazole [ATC:S01EX02]
Amidephrine
Amosulalol
Arotinolol
Bunazosin
Bunitrolol
Dipivefrin
Guanadrel
Medroxalol
Methylephedrine
Naftopidil
Pelanserin
Setiptiline
alpha2b-adrenergic receptor [HSA:151] [KO:K04139]
alpha2-adrenergic receptor [HSA:150 151 152] [KO:K04138 K04139 K04140]
Methyldopa [ATC:C02AB01 C02AB02]
Clonidine [ATC:C02AC01 N02CX02 S01EA04]
Guanfacine [ATC:C02AC02]
Rilmenidine [ATC:C02AC06]
Yohimbin [ATC:G04BE04]
Tizanidine [ATC:M03BX02]
Piribedil [ATC:N04BC08]
Chlorpromazine [ATC:N05AA01]
Dexmedetomidine [ATC:N05CM18]
Mirtazapine [ATC:N06AX11]
Apraclonidine [ATC:S01EA03]
Brimonidine [ATC:S01EA05]
Aptazapine
Atipamezole
Delequamine
Detomidine
Fluparoxan
Guanabenz
Levonordefrin
Medetomidine
Romifidine
Xylazine; Veterinary
beta1-adrenergic receptor [HSA:153] [KO:K04141]
Isoprenaline [ATC:C01CA02 R03AB02 R03CB01]
Dobutamine [ATC:C01CA07]
Prenalterol [ATC:C01CA13]
Xamoterol [ATC:C01CX07]
Buphenine [ATC:C04AA02 G02CA02]
Alprenolol [ATC:C07AA01]
Oxprenolol [ATC:C07AA02]
Pindolol [ATC:C07AA03]
Propranolol [ATC:C07AA05]
Sotalol [ATC:C07AA07]
Timolol [ATC:C07AA06 S01ED01]
Nadolol [ATC:C07AA12]
Mepindolol [ATC:C07AA14]
Carteolol [ATC:C07AA15 S01ED05]
Tertatolol [ATC:C07AA16]
Bopindolol [ATC:C07AA17]
Bupranolol [ATC:C07AA19]
Penbutolol [ATC:C07AA23]
Cloranolol [ATC:C07AA27]
Practolol [ATC:C07AB01]
Metoprolol [ATC:C07AB02]
Atenolol [ATC:C07AB03]
Acebutolol [ATC:C07AB04]
Betaxolol [ATC:C07AB05 S01ED02]
Bevantolol [ATC:C07AB06]
Bisoprolol [ATC:C07AB07]
Celiprolol [ATC:C07AB08]
Esmolol [ATC:C07AB09]
Epanolol [ATC:C07AB10]
S-atenolol [ATC:C07AB11]
Nebivolol [ATC:C07AB12]
Talinolol [ATC:C07AB13]
Levobunolol [ATC:S01ED03]
Metipranolol [ATC:S01ED04]
Befunolol [ATC:S01ED06]
Adaprolol
Alprenoxime
Bucindolol
Bufetolol
Bunolol
Butopamine
Cetamolol
Cicloprolol
Cimaterol
Denopamine
Dexpropranolol
Diacetolol
Flestolol
Indenolol
Landiolol
Levdobutamine
Levobetaxolol
Nipradilol
Pamatolol
Primidolol
Talibegron
Tilisolol
beta2-adrenergic receptor [HSA:154] [KO:K04142]
Dopexamine [ATC:C01CA14]
Isoxsuprine [ATC:C04AA01]
Ritodrine [ATC:G02CA01]
Fenoterol [ATC:G02CA03]
Orciprenaline [ATC:R03AB03 R03CB03]
Salbutamol [ATC:R03AC02 R03CC02]
Terbutaline [ATC:R03AC03 R03CC03]
Rimiterol [ATC:R03AC05]
Hexoprenaline [ATC:R03AC06 R03CC05]
Isoetarine [ATC:R03AC07 R03CC06]
Pirbuterol [ATC:R03AC08 R03CC07]
Tretoquinol [ATC:R03AC09 R03CC09]
Carbuterol [ATC:R03AC10 R03CC10]
Tulobuterol [ATC:R03AC11 R03CC11]
Salmeterol [ATC:R03AC12]
Formoterol [ATC:R03AC13]
Clenbuterol [ATC:R03AC14 R03CC13]
Reproterol [ATC:R03AC15 R03CC14]
Procaterol [ATC:R03AC16 R03CC08]
Bitolterol [ATC:R03AC17]
Indacaterol [ATC:R03AC18]
Methoxyphenamine [ATC:R03CB02]
Bambuterol [ATC:R03CC12]
Abediterol
Albuterol
Arformoterol
Butoxamine
Carazolol
Clorprenaline
Colterol
Milveterol
Isoetharine
Levalbuterol
Levosalbutamol
Mabuterol
Metaproterenol
Olodaterol
Picumeterol
Ractopamine
Sibenadet
Soterenol
Vilanterol
Zinterol
beta3-adrenergic receptor [HSA:155] [KO:K04143]
Amibegron
Fasobegron
Mirabegron
Ritobegron
Solabegron
Dopamine
Histamine
Serotonin
Tachykinin / neurokinin
Ghrelin
Orexin
Neuropeptide Y
Opioid
Angiotensin
Bradykinin
Endothelin
Lutropin-choriogonadotropic hormone
Follicle stimulating hormone
Oxytocin
Vasopressin
Melanocortin
Gonadotropin-releasing hormone
Somatostatin
Thyrotropin-releasing hormone
Cholecystokinin
Motilin
Thrombin
Purine / pyrimidine
Adenosine
Prostaglandin
Prostacyclin
Leukotriene
Thromboxane
Cysteinyl leukotriene
Sphingolipid
Cannabinoid
Platelet activating factor
Melatonin
Secretin receptor family
Metabotropic glutamate receptor family
Others
Cytokine receptors
Nuclear receptors
Ion channels
Transporters
Enzymes
Protein kinases
Cytokines
Target-based Classification of Drugs Target-based Classification of Drugs