Target-based Classification of Drugs

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 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
       CHRM [HSA:1128 1129 1131 1132 1133] [KO:K04129 K04130 K04131 K04132 K04133]
       CHRM1 [HSA:1128] [KO:K04129]
       CHRM2 [HSA:1129] [KO:K04130]
       CHRM3 [HSA:1131] [KO:K04131]
         D08325  Oxyphencyclimine (INN)
         D01006  Oxyphencyclimine hydrochloride (JAN)
         D07078  Rociverine (INN)
         D07820  Dicycloverine (INN)
         D00717  Dicyclomine hydrochloride (JAN/USP) <US>
         D00540  Glycopyrrolate (USP) <JP/US>
         D00723  Tridihexethyl chloride (BAN)
         D01005  Isopropamide iodide (JAN/USP/INN)
         D01003  Hexocyclium metilsulfate (INN)
         D06878  Diphemanil metilsulfate (INN)
         D00193  Dexpanthenol (USP/INN) <JP>
         D10938  Glycopyrronium (USAN)
         D00646  Tolterodine (USAN/INN)
         D01148  Tolterodine tartrate (JAN/USP) <JP/US>
         D08522  Solifenacin (INN)
         D01269  Solifenacin succinate (JAN/USAN/INN) <JP/US>
         D01103  Trospium chloride (JAN/USP/INN) <US>
         D03654  Darifenacin (USAN/INN)
         D01699  Darifenacin hydrobromide (JAN/USAN) <US>
         D07226  Fesoterodine (INN)
         D08923  Fesoterodine fumarate (JAN/USAN) <JP/US>
         D10853  Desfesoterodine (INN)
         D06273  Imidafenacin (JAN/INN) <JP>
         D00525  Pilocarpine (JAN/USP)
         D02200  Pilocarpine hydrochloride (JP18/USP) <JP/US>
         D05478  Pilocarpine nitrate (USP)
         D08376  Pilocarpine borate
         D07667  Cevimeline (INN)
         D00661  Cevimeline hydrochloride (USAN) <JP/US>
         D01929  Tiotropium bromide hydrate (JAN) <JP/US>
         D10978  Revefenacin (USAN/INN) <US>
         D01875  Tiquizium bromide (JAN/INN) <JP>
         D02876  Alvameline maleate (USAN)
         D04057  Esoxybutynin chloride (USAN)
         D10989  Sofpironium bromide (JAN/USAN/INN) <JP>
         D11900  Navafenterol (USAN)
         D11901  Navafenterol saccharinate (USAN)
       CHRM4 [HSA:1132] [KO:K04132]
     Adrenaline
     Dopamine
     Histamine
     Serotonin
     Trace amine
     Angiotensin
     Bradykinin
     Cholecystokinin
     Endothelin
     Follicle stimulating hormone
     Ghrelin
     Gonadotropin-releasing hormone
     Lutropin-choriogonadotropic hormone
     Melanocortin
     Motilin
     Neuropeptide Y
     Opioid
     Orexin
     Oxytocin
     Relaxin
     Somatostatin
     Tachykinin
     Thrombin
     Thyrotropin-releasing hormone
     Vasopressin
     Purine / pyrimidine
     Adenosine
     Cysteinyl leukotriene
     Free fatty acid
     Leukotriene
     Lysophosphatidic acid
     Prostaglandin
     Prostacyclin
     Sphingolipid
     Thromboxane
     Cannabinoid
     Melatonin
     Platelet activating factor
     R-spondin
   Secretin receptor family
   Metabotropic glutamate receptor family
   Frizzled / Smoothened family
   Others
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: March 26, 2024

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