Target-based Classification of Drugs

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 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
       CHRM [HSA:1128 1129 1131 1132 1133] [KO:K04129 K04130 K04131 K04132 K04133]
         D08389  Pirenzepine (INN)
         D01297  Pirenzepine hydrochloride (USAN)
         D05276  Pirenzepine hydrochloride hydrate (JP18) <JP>
         D08160  Mebeverine (INN)
         D04868  Mebeverine hydrochloride (USAN)
         D07821  Dihexyverine (INN)
         D03824  Dihexyverine hydrochloride (USAN)
         D07079  Difemerine (INN)
         D08382  Piperidolate (INN)
         D01165  Piperidolate hydrochloride (JAN) <JP>
         D03088  Benzilonium bromide (USAN/INN)
         D07081  Penthienate bromide (NF XIII)
         D00481  Propantheline bromide (JP18/USP/INN) <JP>
         D07083  Otilonium bromide (INN)
         D00721  Methanthelinium bromide (INN)
         D05535  Poldine methylsulfate (USAN)
         D00720  Mepenzolate bromide (JP18/INN) <JP>
         D01532  Bevonium methylsulfate (JAN)
         D07084  Pipenzolate bromide (INN)
         D01201  Tiemonium iodide (JAN/INN)
         D01377  Prifinium bromide (JAN/INN)
         D02535  Timepidium bromide hydrate (JP18) <JP>
         D07070  Fenpiverinium bromide (INN)
         D01538  Valethamate bromide (JAN)
         D00113  Atropine (USP)
         D02069  Atropine sulfate (JP18/USP) <JP/US>
         D00147  Hyoscyamine (USP)
         D00719  Hyoscyamine sulfate (USP)
         D01648  Hyoscyamine methylbromide (JAN)
         D04479  Hyoscyamine hydrobromide (USP)
         D01451  Scopolamine butylbromide (JP18) <JP>
         D01077  Methylatropine nitrate (USAN)
         D03814  Atropine methylbromide (JAN)
         D01976  N-Methylscopolamine methylsulfate (JAN) <JP>
         D07951  Fentonium bromide (INN)
         D07099  Cimetropium bromide (JAN/INN)
         D02070  Homatropine methylbromide (USP)
         D00138  Scopolamine (INN) <US>
         D02071  Scopolamine hydrobromide (USP) <JP>
         D10939  Glycopyrronium tosylate (USAN) <JP/US>
         D00465  Oxybutynin (USAN/INN) <US>
         D00722  Oxybutynin chloride (USP) <JP/US>
         D08441  Propiverine (INN)
         D01007  Propiverine hydrochloride (JP18) <JP>
         D00765  Rocuronium bromide (JAN/USP/INN) <JP/US>
         D08418  Pridinol (INN)
         D02064  Pridinol mesilate (JAN) <JP>
         D08419  Pridinol hydrochloride
         D08638  Trihexyphenidyl (INN)
         D00787  Trihexyphenidyl hydrochloride (JP18/USP) <JP/US>
         D00779  Biperiden (JAN/USP/INN)
         D02246  Biperiden hydrochloride (JP18/USP) <JP>
         D02247  Biperiden lactate (JAN/USP) <JP>
         D08209  Metixene (INN)
         D01871  Methixene hydrochloride (USAN)
         D08425  Procyclidine (INN)
         D00782  Procyclidine hydrochloride (USP)
         D08426  Profenamine (INN)
         D01118  Profenamine hydrochloride (JAN)
         D03276  Profenamine hibenzate (JAN)
         D03711  Dexetimide (USAN/INN)
         D07804  Dexetimide hydrochloride
         D07301  Phenglutarimide (INN)
         D08157  Mazaticol (INN)
         D03264  Mazaticol hydrochloride hydrate (JAN)
         D07302  Bornaprine (INN)
         D07303  Tropatepine (INN)
         D08653  Tropatepine hydrochloride
         D07511  Benzatropine (INN)
         D00778  Benztropine mesylate (USP) <US>
         D04087  Ethybenztropine (USAN)
         D00270  Chlorpromazine (USP/INN)
         D00789  Chlorpromazine hydrochloride (JP18/USP) <JP/US>
         D03274  Chlorpromazine hibenzate (JAN)
         D04034  Chlorpromazine phenolphthalinate (JAN) <JP>
         D09819  Chlorpromazine tannate (JAN)
         D00524  Carbachol (JAN/USP/INN) <US>
         D01000  Bethanechol chloride (JP18/USP) <JP/US>
         D07349  Choline alfoscerate (INN)
         D02212  Ipratropium bromide (USP) <JP/US>
         D01946  Oxitropium bromide (JAN/INN)
         D08837  Aclidinium bromide (JAN/USAN/INN) <JP/US>
         D10181  Umeclidinium bromide (JAN/USAN) <JP/US>
         D00999  Acetylcholine chloride (JP18/USP/INN) <JP/US>
         D07759  Cyclopentolate (INN)
         D01002  Cyclopentolate hydrochloride (JP18/USP) <JP/US>
         D01004  Homatropine hydrobromide (JP18/USP)
         D00397  Tropicamide (JP18/USP/INN) <JP/US>
         D04970  Methacholine chloride (JAN/USP/INN) <JP/US>
         D00232  Anisotropine methylbromide (USAN)
         D00715  Methscopolamine bromide (USP) <US>
         D00716  Clidinium bromide (USP/INN)
         D01175  Carpronium chloride (JAN/INN) <JP>
         D01231  Piroheptine hydrochloride (JAN) <JP>
         D01315  Methylbenactyzium bromide (JP18/INN)
         D01318  Diphenidol hydrochloride (USAN) <JP>
         D01359  Etomidoline (JAN/INN)
         D01463  Diponium bromide (JAN/INN)
         D01491  Butropium bromide (JP18/INN) <JP>
         D01521  Pipethanate hydrochloride (JAN)
         D01600  Diphenylpiperidinomethyldioxolan iodide (JAN)
         D01815  Oxapium iodide (JP18/INN)
         D01955  Aclatonium napadisilate (JAN)
         D01987  Pipethanate ethobromide (JAN)
         D02417  Flutropium bromide (JAN)
         D02603  Diethazine hydrochloride
         D03011  Atropine oxide hydrochloride (USAN)
         D03076  Benapryzine hydrochloride (USAN)
         D03087  Benzetimide hydrochloride (USAN)
         D03858  Diphenidol (USAN/INN)
         D03859  Diphenidol pamoate (USAN)
         D03970  Elantrine (USAN)
         D03979  Elucaine (USAN)
         D04116  Eucatropine hydrochloride (USP XXXII)
         D04434  Heteronium bromide (USAN/INN)
         D05012  Metoquizine (USAN/INN)
         D05035  Milameline hydrochloride (USAN)
         D05360  Parapenzolate bromide (USAN/INN)
         D05418  Pentapiperium methylsulfate (USAN)
         D05452  Phencarbamide (USAN)
         D05628  Propenzolate hydrochloride (USAN)
         D05703  Rapacuronium bromide (USAN/INN)
         D06015  Tazomeline citrate (USAN)
         D06061  Tematropium methylsulfate (USAN)
         D06175  Tofenacin hydrochloride (USAN)
         D06192  Toquizine (USAN)
         D06217  Triampyzine sulfate (USAN)
         D07477  Atropine oxide (INN)
         D07513  Benzetimide (INN)
         D07823  Diethazine (INN)
         D08384  Pipethanate (INN)
         D08395  Piroheptine (INN)
         D08595  Tiemonium methylsulfate
         D09402  Darotropium bromide (USAN/INN)
         D09752  Carpronium chloride hydrate (JAN) <JP>
         D10180  Umeclidinium (USAN)
         D10545  Batefenterol (USAN)
         D10546  Batefenterol succinate (USAN)
         D11383  Blarcamesine (USAN)
         D11549  Blarcamesine hydrochloride (USAN)
       CHRM1 [HSA:1128] [KO:K04129]
       CHRM2 [HSA:1129] [KO:K04130]
       CHRM3 [HSA:1131] [KO:K04131]
       CHRM4 [HSA:1132] [KO:K04132]
     Adrenaline
     Dopamine
     Histamine
     Serotonin
     Trace amine
     Angiotensin
     Bradykinin
     Cholecystokinin
     Endothelin
     Follicle stimulating hormone
     Ghrelin
     Gonadotropin-releasing hormone
     Lutropin-choriogonadotropic hormone
     Melanocortin
     Motilin
     Neuropeptide Y
     Opioid
     Orexin
     Oxytocin
     Relaxin
     Somatostatin
     Tachykinin
     Thrombin
     Thyrotropin-releasing hormone
     Vasopressin
     Purine / pyrimidine
     Adenosine
     Cysteinyl leukotriene
     Free fatty acid
     Leukotriene
     Lysophosphatidic acid
     Prostaglandin
     Prostacyclin
     Sphingolipid
     Thromboxane
     Cannabinoid
     Melatonin
     Platelet activating factor
     R-spondin
   Secretin receptor family
   Metabotropic glutamate receptor family
   Frizzled / Smoothened family
   Others
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: March 14, 2024

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