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Remark |
G Protein-coupled receptors
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Cytokine receptors
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Nuclear receptors
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Ion channels
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Transporters
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ABC transporters
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Solute carrier family
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SLC5
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SLC6
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SLC6A1 (GABA transporter 1) [HSA:6529] [KO:K05034]
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SLC6A2 (noradrenalin transporter) [HSA:6530] [KO:K05035]
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Mazindol [ATC:A08AA05]
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Sibutramine [ATC: A08AA10]
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D08513 Sibutramine (INN)
D02571 Sibutramine hydrochloride hydrate (JAN); Sibutramine hydrochloride (USAN)
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Inhibitor
Inhibitor
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Cocaine [ATC:N01BC01 R02AD03 S01HA01 S02DA02]
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Desipramine [ATC:N06AA01]
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Imipramine [ATC:N06AA02]
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Clomipramine [ATC:N06AA04]
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Trimipramine [ATC:N06AA06]
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Lofepramine [ATC:N06AA07]
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Amitriptyline [ATC:N06AA09]
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Nortriptyline [ATC:N06AA10]
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Amoxapine [ATC:N06AA17]
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Maprotiline [ATC:N06AA21]
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Nomifensine [ATC:N06AX04]
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Viloxazine [ATC:N06AX09]
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Venlafaxine [ATC:N06AX16]
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Milnacipran [ATC:N06AX17]
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Reboxetine [ATC:N06AX18]
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Duloxetine [ATC:N06AX21]
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Desvenlafaxine [ATC:N06AX23]
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Amfetamine [ATC:N06BA01]
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Dexamfetamine [ATC:N06BA02]
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Metamfetamine [ATC:N06BA03]
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Atomoxetine [ATC:N06BA09]
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Lisdexamfetamine [ATC:N06BA12]
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Amitifadine
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Amitriptylinoxide
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Edivoxetine
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Esreboxetine
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Imipraminoxid
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Levomilnacipran
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Nisoxetine
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Pyrovalerone
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SLC6A3 (dopamine transporter) [HSA:6531] [KO:K05036]
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Dexfenfluramine [ATC:A08AA04]
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Mazindol [ATC:A08AA05]
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Sibutramine [ATC:A08AA10]
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D08513 Sibutramine (INN)
D02571 Sibutramine hydrochloride hydrate (JAN); Sibutramine hydrochloride (USAN)
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Inhibitor
Inhibitor
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Cocaine [ATC:R02AD03]
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Amfetamine [ATC:N06BA01]
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Dexamfetamine [ATC:N06BA02]
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Metamfetamine [ATC:N06BA03]
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Lisdexamfetamine [ATC:N06BA12]
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Amfonelic acid
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Amitifadine
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Bicifadine
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Ioflupane I 123
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Pyrovalerone
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SLC6A4 (serotonin transporter) [HSA:6532] [KO:K05037]
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Mazindol [ATC:A08AA05]
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Sibutramine [ATC:A08AA10]
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D08513 Sibutramine (INN)
D02571 Sibutramine hydrochloride hydrate (JAN); Sibutramine hydrochloride (USAN)
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Inhibitor
Inhibitor
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Dapoxetine [ATC:G04BX14]
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Trazodone [ATC:N06AX05]
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Cocaine [ATC:N01BC01 R02AD03 S01HA01 S02DA02]
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Desipramine [ATC:N06AA01]
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Imipramine [ATC:N06AA02]
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Clomipramine [ATC:N06AA04]
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Lofepramine [ATC:N06AA07]
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Amitriptyline [ATC:N06AA09]
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Nortriptyline [ATC:N06AA10]
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Dosulepin [ATC:N06AA16]
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Fluoxetine [ATC:N06AB03]
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Citalopram [ATC:N06AB04]
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Paroxetine [ATC:N06AB05]
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Sertraline [ATC:N06AB06]
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Fluvoxamine [ATC:N06AB08]
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Escitalopram [ATC:N06AB10]
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Trazodone [ATC:N06AX05]
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Viloxazine [ATC:N06AX09]
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Venlafaxine [ATC:N06AX16]
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Milnacipran [ATC:N06AX17]
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Duloxetine [ATC:N06AX21]
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Desvenlafaxine [ATC:N06AX23]
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Vilazodone [ATC:N06AX24]
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Amitifadine
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Amitriptylinoxide
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Bicifadine
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Levomilnacipran
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SLC6A9 (glycine transporter type 1) (GlyT1) [HSA:6536] [KO:K05038]
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SLC9
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SLC12
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SLC22
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SLC29
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Major facilitator superfamily
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Others
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Enzymes
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Protein kinases
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Cytokines
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Others
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