Target-based Classification of Drugs

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     Remark
 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
     Adrenaline
       alpha1a-adrenergic receptor [HSA:148] [KO:K04135]
       alpha1-adrenergic receptor [HSA:146 147 148] [KO:K04137 K04136 K04135]
         Epinephrine [ATC:A01AD01 B02BC09 C01CA24 R01AA14 R03AA01 S01EA01]
         Adrenalone  [ATC:A01AD06 B02BC05]
         Etilefrine [ATC:C01CA01]
         Norepinephrine [ATC:C01CA03]
         Norfenefrine [ATC:C01CA05]
         Phenylephrine [ATC:C01CA06 R01AA04 R01AB01 R01BA03 S01FB01 S01GA05]
         Oxedrine [ATC:C01CA08 S01GA06]
         Metaraminol [ATC:C01CA09]
         Methoxamine [ATC:C01CA10]
         Midodrine [ATC:C01CA17]
         Arbutamine [ATC:C01CA22]
         Ephedrine [ATC:C01CA26 R01AA03 R01AB05 R03CA02 S01FB02]
         Prazosin [ATC:C02CA01]
         Indoramin [ATC:C02CA02]
         Trimazosin [ATC:C02CA03]
         Doxazosin [ATC:C02CA04]
         Urapidil [ATC:C02CA06]
         Ketanserin [ATC:C02KD01]
         Phentolamine [ATC:C04AB01 V03AB36]
         Tolazoline [ATC:C04AB02 M02AX02]
         Nicergoline [ATC:C04AE02]
         Phenoxybenzamine [ATC:C04AX02]
         Moxisylyte [ATC:C04AX10 G04BE06]
         Ifenprodil [ATC:C04AX28]
         Labetalol [ATC:C07AG01]
         Carvedilol [ATC:C07AG02]
         Methylergometrine [ATC:G02AB01]
         Ergot alkaloids [ATC:G02AB02]
         Ergometrine [ATC:G02AB03]
         Alfuzosin [ATC:G04CA01]
         Tamsulosin [ATC:G04CA02]
         Terazosin [ATC:G04CA03]
         Silodosin [ATC:G04CA04]
         Dihydroergotamine [ATC:N02CA01]
         Ergotamine [ATC:N02CA02]
         Levomepromazine [ATC:N05AA02]
         Sertindole [ATC:N05AE03]
         Pimozide [ATC:N05AG02]
         Clozapine [ATC:N05AH02]
         Asenapine [ATC:N05AH05]
         Olanzapine [ATC:N05AH03]
         Quetiapine [ATC:N05AH04]
         Risperidone [ATC:N05AX08]
         Mianserin [ATC:N06AX03]
         Oxymetazoline [ATC:R01AA05 R01AB07 S01GA04]
         Tetryzoline [ATC:R01AA06 R01AB03 S01GA02]
         Xylometazoline [ATC:R01AA07 R01AB06 S01GA03]
         Naphazoline [ATC:R01AA08 R01AB02 S01GA01]
         Tramazoline [ATC:R01AA09]
         Pseudoephedrine [ATC:R01BA02]
           D08449  Pseudoephedrine (INN)
           D00485  Pseudoephedrine hydrochloride (USP)
           D05648  Pseudoephedrine polistirex (USAN)
           D05649  Pseudoephedrine sulfate (USP)
Agonist
Agonist
Agonist
Agonist
         Dipivefrine [ATC:S01EA02]
         Dapiprazole [ATC:S01EX02]
         Amidephrine
         Amosulalol
         Arotinolol
         Bunazosin
         Bunitrolol
         Dipivefrin
         Guanadrel
         Medroxalol
         Methylephedrine
         Naftopidil
         Pelanserin
         Setiptiline
       alpha2b-adrenergic receptor [HSA:151] [KO:K04139]
       alpha2-adrenergic receptor [HSA:150 151 152] [KO:K04138 K04139 K04140]
         Epinephrine [ATC:A01AD01 B02BC09 C01CA24 R01AA14 R03AA01 S01EA01]
         Norepinephrine [ATC:C01CA03]
         Oxedrine [ATC:C01CA08 S01GA06]
         Metaraminol [ATC:C01CA09]
         Ephedrine [ATC:C01CA26 R01AA03 R01AB05 R03CA02 S01FB02]
         Methyldopa [ATC:C02AB01 C02AB02]
         Clonidine [ATC:C02AC01 N02CX02 S01EA04]
         Guanfacine [ATC:C02AC02]
         Rilmenidine [ATC:C02AC06]
         Phentolamine [ATC:C04AB01 V03AB36]
         Tolazoline [ATC:C04AB02 M02AX02]
         Phenoxybenzamine [ATC:C04AX02]
         Methylergometrine [ATC:G02AB01]
         Ergot alkaloids [ATC:G02AB02]
         Ergometrine [ATC:G02AB03]
         Yohimbin [ATC:G04BE04]
         Tizanidine [ATC:M03BX02]
         Piribedil [ATC:N04BC08]
         Chlorpromazine [ATC:N05AA01]
         Levomepromazine [ATC:N05AA02]
         Asenapine [ATC:N05AH05]
         Dexmedetomidine [ATC:N05CM18]
         Mianserin [ATC:N06AX03]
         Mirtazapine [ATC:N06AX11]
         Pseudoephedrine [ATC:R01BA02]
           D08449  Pseudoephedrine (INN)
           D00485  Pseudoephedrine hydrochloride (USP)
           D05648  Pseudoephedrine polistirex (USAN)
           D05649  Pseudoephedrine sulfate (USP)
Agonist
Agonist
Agonist
Agonist
         Dipivefrine [ATC:S01EA02]
         Apraclonidine [ATC:S01EA03]
         Brimonidine [ATC:S01EA05]
         Dapiprazole [ATC:S01EX02]
         Aptazapine
         Atipamezole
         Delequamine
         Detomidine
         Dipivefrin
         Fluparoxan
         Guanabenz
         Guanadrel
         Levonordefrin
         Methylephedrine
         Medetomidine
         Romifidine
         Setiptiline
         Xylazine; Veterinary
       beta1-adrenergic receptor [HSA:153] [KO:K04141]
         Epinephrine [ATC:A01AD01 B02BC09 C01CA24 R01AA14 R03AA01 S01EA01]
         Isoprenaline [ATC:C01CA02 R03AB02 R03CB01]
         Norepinephrine [ATC:C01CA03]
         Dobutamine [ATC:C01CA07]
         Prenalterol [ATC:C01CA13]
         Arbutamine [ATC:C01CA22]
         Ephedrine [ATC:C01CA26 R01AA03 R01AB05 R03CA02 S01FB02]
         Xamoterol [ATC:C01CX07]
         Buphenine [ATC:C04AA02 G02CA02]
         Alprenolol [ATC:C07AA01]
         Oxprenolol [ATC:C07AA02]
         Pindolol [ATC:C07AA03]
         Propranolol [ATC:C07AA05]
         Sotalol [ATC:C07AA07]
         Timolol [ATC:C07AA06 S01ED01]
         Nadolol [ATC:C07AA12]
         Mepindolol [ATC:C07AA14]
         Carteolol [ATC:C07AA15 S01ED05]
         Tertatolol [ATC:C07AA16]
         Bopindolol [ATC:C07AA17]
         Bupranolol [ATC:C07AA19]
         Penbutolol [ATC:C07AA23]
         Cloranolol [ATC:C07AA27]
         Practolol [ATC:C07AB01]
         Metoprolol [ATC:C07AB02]
         Atenolol [ATC:C07AB03]
         Acebutolol [ATC:C07AB04]
         Betaxolol [ATC:C07AB05 S01ED02]
         Bevantolol [ATC:C07AB06]
         Bisoprolol [ATC:C07AB07]
         Celiprolol [ATC:C07AB08]
         Esmolol [ATC:C07AB09]
         Epanolol [ATC:C07AB10]
         S-atenolol [ATC:C07AB11]
         Nebivolol [ATC:C07AB12]
         Talinolol [ATC:C07AB13]
         Labetalol [ATC:C07AG01]
         Carvedilol [ATC:C07AG02]
         Pseudoephedrine [ATC:R01BA02]
           D08449  Pseudoephedrine (INN)
           D00485  Pseudoephedrine hydrochloride (USP)
           D05648  Pseudoephedrine polistirex (USAN)
           D05649  Pseudoephedrine sulfate (USP)
Agonist
Agonist
Agonist
Agonist
         Dipivefrine [ATC:S01EA02]
         Levobunolol [ATC:S01ED03]
         Metipranolol [ATC:S01ED04]
         Befunolol [ATC:S01ED06]
         Adaprolol
         Alprenoxime
         Amosulalol
         Arotinolol
         Bucindolol
         Bucumolol
         Bufetolol
         Bunitrolol
         Bunolol
         Butopamine
         Cetamolol
         Cicloprolol
         Cimaterol
         Denopamine
         Dexpropranolol
         Diacetolol
         Dipivefrin
         Flestolol
         Indenolol
         Landiolol
         Levdobutamine
         Levobetaxolol
         Methylephedrine
         Medroxalol
         Nipradilol
         Pamatolol
         Primidolol
         Talibegron
         Tilisolol
       beta2-adrenergic receptor [HSA:154] [KO:K04142]
         Epinephrine [ATC:A01AD01 B02BC09 C01CA24 R01AA14 R03AA01 S01EA01]
         Isoprenaline [ATC:C01CA02 R03AB02 R03CB01]
         Norepinephrine [ATC:C01CA03]
         Dopexamine [ATC:C01CA14]
         Arbutamine [ATC:C01CA22]
         Ephedrine [ATC:C01CA26 R01AA03 R01AB05 R03CA02 S01FB02]
         Isoxsuprine [ATC:C04AA01]
         Buphenine [ATC:C04AA02 G02CA02]
         Alprenolol [ATC:C07AA01]
         Oxprenolol [ATC:C07AA02]
         Pindolol [ATC:C07AA03]
         Propranolol [ATC:C07AA05]
         Timolol [ATC:C07AA06 S01ED01]
         Sotalol [ATC:C07AA07]
         Nadolol [ATC:C07AA12]
         Mepindolol [ATC:C07AA14]
         Carteolol [ATC:C07AA15 S01ED05]
         Tertatolol [ATC:C07AA16]
         Bopindolol [ATC:C07AA17]
         Bupranolol [ATC:C07AA19]
         Penbutolol [ATC:C07AA23]
         Cloranolol [ATC:C07AA27]
         Labetalol [ATC:C07AG01]
         Carvedilol [ATC:C07AG02]
         Ritodrine [ATC:G02CA01]
         Fenoterol [ATC:G02CA03]
         Pseudoephedrine [ATC:R01BA02]
           D08449  Pseudoephedrine (INN)
           D00485  Pseudoephedrine hydrochloride (USP)
           D05648  Pseudoephedrine polistirex (USAN)
           D05649  Pseudoephedrine sulfate (USP)
Agonist
Agonist
Agonist
Agonist
         Orciprenaline [ATC:R03AB03 R03CB03]
         Salbutamol [ATC:R03AC02 R03CC02]
         Terbutaline [ATC:R03AC03 R03CC03]
         Rimiterol [ATC:R03AC05]
         Hexoprenaline [ATC:R03AC06 R03CC05]
         Isoetarine [ATC:R03AC07 R03CC06]
         Pirbuterol [ATC:R03AC08 R03CC07]
         Tretoquinol [ATC:R03AC09 R03CC09]
         Carbuterol [ATC:R03AC10 R03CC10]
         Tulobuterol [ATC:R03AC11 R03CC11]
         Salmeterol [ATC:R03AC12]
         Formoterol [ATC:R03AC13]
         Clenbuterol [ATC:R03AC14 R03CC13]
         Reproterol [ATC:R03AC15 R03CC14]
         Procaterol [ATC:R03AC16 R03CC08]
         Bitolterol [ATC:R03AC17]
         Indacaterol [ATC:R03AC18]
         Methoxyphenamine [ATC:R03CB02]
         Dipivefrine [ATC:S01EA02]
         Levobunolol [ATC:S01ED03]
         Metipranolol [ATC:S01ED04]
         Befunolol [ATC:S01ED06]
         Bambuterol [ATC:R03CC12]
         Abediterol
         Adaprolol
         Amosulalol
         Albuterol
         Alprenoxime
         Arformoterol
         Arotinolol
         Bucindolol
         Bucumolol
         Bufetolol
         Bunitrolol
         Bunolol
         Butoxamine
         Carazolol
         Cetamolol
         Cicloprolol
         Cimaterol
         Clorprenaline
         Colterol
         Dexpropranolol
         Diacetolol
         Dipivefrin
         Flestolol
         Indenolol
         Methylephedrine
         Milveterol
         Isoetharine
         Levalbuterol
         Levosalbutamol
         Mabuterol
         Metaproterenol
         Medroxalol
         Nipradilol
         Olodaterol
         Pamatolol
         Primidolol
         Picumeterol
         Ractopamine
         Sibenadet
         Soterenol
         Talibegron
         Tilisolol
         Vilanterol
         Zinterol
       beta3-adrenergic receptor [HSA:155] [KO:K04143]
         Epinephrine [ATC:A01AD01 B02BC09 C01CA24 R01AA14 R03AA01 S01EA01]
         Isoprenaline [ATC:C01CA02 R03AB02 R03CB01]
         Norepinephrine [ATC:C01CA03]
         Arbutamine [ATC:C01CA22]
         Ephedrine [ATC:C01CA26 R01AA03 R01AB05 R03CA02 S01FB02]
         Buphenine [ATC:C04AA02 G02CA02]
         Alprenolol [ATC:C07AA01]
         Oxprenolol [ATC:C07AA02]
         Pindolol [ATC:C07AA03]
         Propranolol [ATC:C07AA05]
         Timolol [ATC:C07AA06 S01ED01]
         Nadolol [ATC:C07AA12]
         Mepindolol [ATC:C07AA14]
         Carteolol [ATC:C07AA15 S01ED05]
         Tertatolol [ATC:C07AA16]
         Bopindolol [ATC:C07AA17]
         Bupranolol [ATC:C07AA19]
         Penbutolol [ATC:C07AA23]
         Cloranolol [ATC:C07AA27]
         Labetalol [ATC:C07AG01]
         Carvedilol [ATC:C07AG02]
         Pseudoephedrine [ATC:R01BA02]
           D08449  Pseudoephedrine (INN)
           D00485  Pseudoephedrine hydrochloride (USP)
           D05648  Pseudoephedrine polistirex (USAN)
           D05649  Pseudoephedrine sulfate (USP)
Agonist
Agonist
Agonist
Agonist
         Dipivefrine [ATC:S01EA02]
         Levobunolol [ATC:S01ED03]
         Metipranolol [ATC:S01ED04]
         Befunolol [ATC:S01ED06]
         Adaprolol
         Alprenoxime
         Amibegron
         Amosulalol
         Arotinolol
         Bucindolol
         Bufetolol
         Bunitrolol
         Bunolol
         Cetamolol
         Cicloprolol
         Cimaterol
         Dexpropranolol
         Diacetolol
         Dipivefrin
         Fasobegron
         Flestolol
         Medroxalol
         Methylephedrine
         Mirabegron
         Nipradilol
         Primidolol
         Pamatolol
         Ritobegron
         Solabegron
         Talibegron
         Tilisolol
     Dopamine
     Histamine
     Serotonin
     Tachykinin / neurokinin
     Ghrelin
     Orexin
     Neuropeptide Y
     Opioid
     Angiotensin
     Bradykinin
     Endothelin
     Lutropin-choriogonadotropic hormone
     Follicle stimulating hormone
     Oxytocin
     Vasopressin
     Melanocortin
     Gonadotropin-releasing hormone
     Somatostatin
     Thyrotropin-releasing hormone
     Cholecystokinin
     Motilin
     Thrombin
     Purine / pyrimidine
     Adenosine
     Prostaglandin
     Prostacyclin
     Leukotriene
     Thromboxane
     Sphingolipid
     Free fatty acid
     Cannabinoid
     Platelet activating factor
     Melatonin
     Cysteinyl leukotriene
   Secretin receptor family
   Metabotropic glutamate receptor family
   Others
 
 Cytokine receptors
 
 Nuclear receptors
 
 Ion channels
 
 Transporters
 
 Enzymes
 
 Protein kinases
 
 Cytokines
 
 Others

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Last updated: July 9, 2014

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