KEGG   DRUG: セレコキシブHelp
エントリ  
D00567                      Drug                                   

一般名   
セレコキシブ (JAN);
Celecoxib (JAN/USAN/INN)
商品名   
米国の商品 
  後発品
CELECOXIB (Actavis Pharma), CELECOXIB 200 MG (Aidarex Pharmaceuticals LLC), CELECOXIB (Aidarex Pharmaceuticals LLC), CELECOXIB (Alembic Pharmaceuticals), CELECOXIB (Alembic Pharmaceuticals Limited), CELECOXIB (American Health Packaging), CELECOXIB (Amneal Pharmaceuticals LLC), CELECOXIB (Aphena Pharma Solutions - Tennessee), CELECOXIB (Aphena Pharma Solutions - Tennessee), CELECOXIB (Apotex Corp.), CELECOXIB (Aurobindo Pharma Limited), CELECOXIB (Blenheim Pharmacal), CELECOXIB (Blenheim Pharmacal), CELECOXIB (Blenheim Pharmacal), CELECOXIB (Blenheim Pharmacal), CELECOXIB (Blenheim Pharmcal), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Bryant Ranch Prepack), CELECOXIB (Cambridge Therapeutics Technologies), CELECOXIB (Cardinal Health), CELECOXIB (Cipla USA), CELECOXIB (DIRECT RX), CELECOXIB (Denton Pharma), CELECOXIB (DirectRX), CELECOXIB (Golden State Medical Supply), CELECOXIB (Greenstone LLC), CELECOXIB (Jubilant Cadista Pharmaceuticals), CELECOXIB (Lake Erie Medical DBA Quality Care Products LLC), CELECOXIB (Lake Erie Medical DBA Quality Care Products LLC), CELECOXIB (Lake Erie Medical DBA Quality Care Products LLC), CELECOXIB (Lake Erie Medical DBA Quality Care Products LLC), CELECOXIB (Lake Erie Medical DBA Quality Care Products LLC), CELECOXIB (Lake Erie Medical DBA Quality Care Products LLC), CELECOXIB (Lupin Pharmaceuticals), CELECOXIB (Macleods Pharmaceuticals Limited), CELECOXIB (Major Pharmaceuticals), CELECOXIB (Mas Management Group), CELECOXIB (Medsource Pharmaceuticals), CELECOXIB (Micro Labs Limited), CELECOXIB (Mylan Institutional), CELECOXIB (Mylan Pharmaceuticals), CELECOXIB (NorthStar RxLLC), CELECOXIB (NuCare Pharmaceuticals), CELECOXIB (NuCare Pharmaceuticals), CELECOXIB (NuCare Pharmaceuticals), CELECOXIB (NuCare Pharmaceuticals), CELECOXIB (NuCare Pharmaceuticals), CELECOXIB (NuCare Pharmaceuticals), CELECOXIB (PD-Rx Pharmaceuticals), CELECOXIB (PD-Rx Pharmaceuticals), CELECOXIB (PD-Rx Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB 200 MG (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Preferred Pharmaceuticals), CELECOXIB (Proficient Rx LP), CELECOXIB (Proficient Rx LP), CELECOXIB (Proficient Rx LP), CELECOXIB (Proficient Rx LP), CELECOXIB (Proficient Rx LP), CELECOXIB (Proficient Rx LP), CELECOXIB (Proficient Rx LP), CELECOXIB 200 MG (Proficient Rx LP), CELEXIB 100-EZS (PureTek Corporation), CELECOXIB (QPharma), CELECOXIB (REMEDYREPACK), CELECOXIB (REMEDYREPACK), CELECOXIB (RPK Pharmaceuticals), CELECOXIB (RedPharm Drug), CELECOXIB (RedPharm Drug), CELECOXIB (RedPharm Drug), CELECOXIB (RedPharm Drug), CELECOXIB (RxChange), CELECOXIB 200 MG (SYDON LABS LLC), CELECOXIB 200 MG (SYDON LABS LLC), CELECOXIB 100 MG (SYDON LABS LLC), CELECOXIB 50 MG (SYDON LABS LLC), CELECOXIB 400 MG (SYDON LABS LLC), CELECOXIB (St. Mary's Medical Park Pharmacy), CELECOXIB (St. Mary's Medical Park Pharmacy), CELECOXIB (St. Mary's Medical Park Pharmacy), CELECOXIB (St. Mary's Medical Park Pharmacy), CELECOXIB (Teva Pharmaceuticals USA), CELECOXIB (Torrent Pharmaceuticals Limited), CELECOXIB (Trigen Laboratories), CELECOXIB (Unit Dose Services), CELECOXIB (Unit Dose Services), CELECOXIB (Unit Dose Services)
組成式   
C17H14F3N3O2S
質量    
381.0759
分子量   
381.3722
構造式   
Mol fileKCF fileDB search
Simcomp    SIMCOMP
クラス   
抗炎症薬
 DG01504  非ステロイド性抗炎症薬 (NSAID)
  DG01907  コキシブ系抗炎症薬
 DG01922  選択的COX2阻害薬
  DG01907  コキシブ系抗炎症薬
酵素基質
 DG01642  CYP2C9により代謝される薬剤
酵素阻害
 DG01645  CYP2D6阻害薬
コード   
同一コード: C07589
薬効分類: 1149
ATCコード: L01XX33 M01AH01
商品: D00567<JP/US>
効能    
鎮痛薬, 抗炎症薬, シクロオキシゲナーゼ2阻害薬
ターゲット 
PTGS2 (COX2) [HSA:5743] [KO:K11987]
  パスウェイ
hsa00590  アラキドン酸の代謝
代謝    
Enzyme: CYP2C9 [HSA:1559]
相互作用  
CYP inhibition: CYP2D6 [HSA:1565]
Drug interaction
構造マップ 
map07112  1,2-ジフェニル置換ファミリー
map07219  シクロオキシナーゼ (COX) 阻害薬
階層分類  
医療用医薬品の薬効分類 [BR:jp08301]
 1  神経系及び感覚器官用医薬品
  11  中枢神経系用薬
   114  解熱鎮痛消炎剤
    1149  その他の解熱鎮痛消炎剤
     D00567  セレコキシブ (JAN)
医療用医薬品のATC分類 [BR:jp08303]
 L 抗悪性腫瘍薬と免疫調節薬
  L01 抗悪性腫瘍薬
   L01X その他の抗悪性腫瘍薬
    L01XX その他の抗悪性腫瘍薬
     L01XX33 セレコキシブ
      D00567  セレコキシブ (JAN) <JP/US>
 M 筋骨格系
  M01 抗炎症及び抗リウマチ製剤
   M01A 抗炎症及び抗リウマチ製剤、非ステロイド系
    M01AH コキシブ
     M01AH01 セレコキシブ
      D00567  セレコキシブ (JAN) <JP/US>
医療用医薬品のUSP分類 [BR:jp08302]
 鎮痛薬
  非ステロイド系抗炎症薬
   セレコキシブ
    D00567  セレコキシブ (JAN)
 抗炎症薬
  非ステロイド系抗炎症薬
   セレコキシブ
    D00567  セレコキシブ (JAN)
Target-based classification of drugs  [BR:br08310]
 Enzymes
  Oxidoreductases (EC1)
   Prostaglandin synthase
    PTGS2 (COX2)
     D00567  Celecoxib (JAN/USAN/INN) <JP/US>
治療薬の医薬品クラス [jp08360.html]
 リウマチ・痛風治療薬
  D00567
 麻酔薬・鎮痛薬と抗炎症薬
  D00567
日本の新薬 [jp08318.html]
 新有効成分含有医薬品
  D00567
BRITE hierarchy
リンク   
CAS: 169590-42-5
PubChem: 7847633
ChEBI: 41423
ChEMBL: CHEMBL118
DrugBank: DB00482
PDB-CCD: CEL[PDBj]
LigandBox: D00567

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