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Drug interaction list


Query:
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN)

Interactions: 1383 hits    [ ATC classification | Therapeutic category ]

C00304  Kanamycin (P) unclassified
C01946  Oleandomycin; Amimycin; Landomycin; Matromycin; Romicil (P) unclassified
C06456  Phosphonoformate; Foscarmet; Foscarnet (P) unclassified
C07005  Flunisolide; Flunisolide anhydrous (P) unclassified
C07051  Indinavir (P) unclassified
C07370  Prednisone; 1,2-Dehydrocortisone; 17,21-Dihydroxypregna-1,4-diene-3,11,20-trione (P) unclassified
D00058  gamma-Aminobutyric acid (JAN); Gammalon (TN) (P) unclassified
D00063  Tobramycin (JP18/USP); Tobi (TN); Tobracin (TN); Tobrex (TN); Bethkis (TN) (P) unclassified
D00088  Hydrocortisone (JP18/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) (P) unclassified
D00104  Chloramphenicol (JP18/USP/INN); Amphicol (TN); Chloromycetin (TN); Econochlor (TN) (P) unclassified
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) (CI,P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4
D00109  Aspirin (JP18/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) (P) unclassified
D00118  Naproxen (JP18/USP/INN); Naprosyn (TN) (P) unclassified
D00120  Sulindac (JP18/USP/INN); Clinoril (TN) (P) unclassified
D00126  Ibuprofen (JP18/USP/INN); Advil (TN); Motrin (TN) (P) unclassified
D00127  Piroxicam (JP18/USP/INN); Feldene (TN) (P) unclassified
D00129  Calcitriol (JAN/USP/INN); Rocaltrol (TN) (P) unclassified
D00130  Diflunisal (JAN/USP/INN); Dolobid (TN) (P) unclassified
D00132  Ketoprofen (JP18/USP/INN); Orudis (TN) (P) unclassified
D00136  Haloperidol (JP18/USP/INN); Haldol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00140  Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) (P) unclassified
D00141  Indomethacin (USP); Indometacin (JP18/INN); Aconip (TN); Indocin (TN) (P) unclassified
D00142  Methotrexate (JP18/USP/INN); Otrexup (TN); Xatmep (TN) (P) unclassified
D00151  Mefenamic acid (JP18/USP/INN); Ponstel (TN) (P) unclassified
D00158  Tolmetin sodium (JAN/USP); Tolmetin sodium dihydrate; Tolectin (TN) (P) unclassified
D00163  Chenodiol (USAN); Chenodeoxycholic acid (JP18/INN); Chenix (TN) (P) unclassified
D00165  Hydrocortisone acetate (JP18/USP); Cortifoam (TN); U-cort (TN) (P) unclassified
D00169  Meclofenamate sodium (USP); Meclofenamate sodium monohydrate; Meclomen (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4
D00186  Ciprofloxacin (JP18/USP/INN); Cipro (TN); Otiprio (TN) (P) unclassified
D00203  Amphotericin B (JP18/USP/INN); Ambisome (TN); Amphotec (TN); Fungizone (TN) (P) unclassified
D00210  Norfloxacin (JP18/USP/INN); Noroxin (TN) (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00212  Vancomycin (USP); Vancocin (TN) (P) unclassified
D00218  Acetazolamide (JP18/USP/INN); Diamox (TN) (P) unclassified
D00224  Allopurinol (JP18/USP/INN); Zyloprim (TN) (P) unclassified
D00235  Atenolol (JP18/USP/INN); Tenormin (TN) (P) unclassified
D00238  Azathioprine (JP18/USP/INN); Azasan (TN); Imuran (TN); Jayempi (TN) (P) unclassified
D00244  Betamethasone (JP18/USP/INN); Celestone (TN); Rinderon (TN) (P) unclassified
D00246  Budesonide (JP18/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00251  Captopril (JP18/USP/INN); Apopril (TN); Capoten (TN) (P) unclassified
D00252  Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00255  Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00276  Clarithromycin (JP18/USP/INN); Biaxin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00279  Clofibrate (JP18/USP/INN); Atromid-S (TN) (P) unclassified
D00280  Clonazepam (JP18/USP/INN); Klonopin (TN) (P) unclassified
D00282  Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) (P) CYP inhibition: CYP3A4
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00285  Co-Trimoxazole (BAN); Sulfamethoxazole and trimethoprim; Bactrim (TN); Septra (TN) (P) unclassified
D00289  Danazol (JP18/USP/INN); Danocrine (TN) (P) unclassified
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00298  Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) (P) Transporter inhibition: ABCB1
D00304  Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) (P) unclassified
D00315  Etodolac (JP18/USP/INN); Lodine (TN) (P) unclassified
D00319  Felodipine (JP18/USP/INN); Plendil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP3A4
D00324  Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00325  Fluocinonide (JP18/USP/INN); Lidex (TN); Vanos (TN) (P) unclassified
D00328  Flurandrenolide (USP); Fludroxycortide (JAN/INN); Cordran (TN) (P) unclassified
D00330  Flurbiprofen (JP18/USP/INN); Ansaid (TN) (P) unclassified
D00331  Furosemide (JP18/USP/INN); Frusemide; Lasix (TN) (P) unclassified
D00333  Ganciclovir (JAN/USP/INN); Cytovene (TN); Vitrasert (TN); Zirgan (TN) (P) unclassified
D00334  Gemfibrozil (JAN/USP/INN); Lopid (TN) (P) unclassified
D00340  Hydrochlorothiazide (JP18/USP/INN); Esidrix (TN); Microzide (TN) (P) unclassified
D00346  Isoniazid (JP18/USP/INN); Laniazid (TN) (P) unclassified
D00349  Isradipine (USP/INN); Dynacirc (TN) (P) unclassified
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00354  Lamotrigine (JAN/USP/INN); Lamictal (TN) (P) unclassified
D00357  Losartan potassium (JP18/USP); Cozaar (TN) (P) unclassified
D00359  Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00362  Lisinopril (USP); Lisinopril hydrate (JP18); Lisinopril dihydrate; Prinivil (TN); Zestril (TN) (P) unclassified
D00369  Melphalan (JP18/USP/INN); Alkeran (TN) (P) unclassified
D00371  Theophylline (JP18); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) (P) unclassified
D00372  Thiabendazole (USP); Tiabendazole (JAN/INN); Mintezol (TN) (P) unclassified
D00375  Mephenytoin (USP/INN); Mesantoin (TN) (P) unclassified
D00377  Mesalamine (USP); Mesalazine (JP18/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) (P) unclassified
D00378  Timolol (USAN); Timolol hemihydrate; Betimol (TN) (P) unclassified
D00383  Trandolapril (JAN/USP/INN); Mavik (TN) (P) unclassified
D00385  Triamcinolone (JP18/USP/INN); Aristocort (TN); Kenacort (TN) (P) unclassified
D00386  Triamterene (JP18/USP/INN); Dyrenium (TN) (P) unclassified
D00392  Trimethadione (JP18/INN); Tridione (TN) (P) unclassified
D00399  Valproic acid (USP); Depakene (TN) (P) unclassified
D00400  Valsartan (JP18/USP/INN); Diovan (TN) (P) unclassified
D00404  Methsuximide (USP); Mesuximide (INN); Celontin (TN) (P) unclassified
D00407  Methylprednisolone (JP18/USP/INN); Medrol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00409  Metronidazole (JP18/USP/INN); Flagyl (TN); Noritate (TN); Nuvessa (TN); Vandazole (TN) (P) unclassified
D00416  Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00421  Ramipril (USP/INN); Altace (TN) (P) unclassified
D00425  Nabumetone (JP18/USP/INN); Relafen (TN) (P) unclassified
D00426  Risperidone (JP18/USP/INN); Risperdal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) unclassified
D00428  Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) (P) unclassified
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D00432  Nadolol (JP18/USP/INN); Corgard (TN) (P) unclassified
D00434  Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00437  Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00438  Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00442  Octreotide (USAN/INN) (P) unclassified
D00443  Spironolactone (JP18/USP/INN); Aldactone (TN) (P) unclassified
D00448  Sulfasalazine (USP/INN); Salazosulfapyridine (JP18); Azulfidine (TN) (P) unclassified
D00452  Suprofen (JAN/USP/INN); Profenal (TN) (P) unclassified
D00458  Quetiapine fumarate (JP18/USP); Seroquel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00459  Quinapril hydrochloride (JP18/USP); Accupril (TN) (P) unclassified
D00463  Oxaprozin (JP18/USP/INN); Daypro (TN) (P) unclassified
D00472  Prednisolone (JP18/USP/INN); Delta-cortef (TN) (P) unclassified
D00473  Prednisone (USP); Prednisone monohydrate; Deltasone (TN); Meticorten (TN); Rayos (TN) (P) unclassified
D00474  Primidone (JP18/USP/INN); Mysoline (TN) (P) unclassified
D00476  Probucol (JP18/USP/INN); Lorelco (TN) (P) unclassified
D00483  Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) (P) unclassified
D00491  Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00495  Paramethadione (INN); Paradione (TN) (P) unclassified
D00496  Penicillamine (JAN/USP/INN); Cuprimine (TN); Depen (TN) (P) unclassified
D00504  Phenacemide (JAN/INN); Phenurone (TN) (P) unclassified
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) unclassified
D00508  Phensuximide (USP/INN); Milontin (TN) (P) unclassified
D00510  Phenylbutazone (JP18/USP/INN); Azolid (TN) (P) unclassified
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) unclassified
D00513  Pindolol (JP18/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) (P) unclassified
D00519  Chlorothiazide (JAN/USP/INN); Diuril (TN) (P) unclassified
D00522  Candesartan (USAN/INN) (P) unclassified
D00523  Irbesartan (JP18/USP/INN); Avapro (TN) (P) unclassified
D00533  Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) (P) unclassified
D00535  Vigabatrin (JAN/USP/INN); Sabril (TN) (P) unclassified
D00536  Felbamate (USPINN); Felbatol (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00538  Zonisamide (JP18/USP/INN); Excegran (TN) (P) unclassified
D00539  Ethosuximide (JP18/USP/INN); Zarontin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00553  Prilocaine (USP/INN); Propitocaine (JAN) (P) unclassified
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00556  Aminopyrine (JAN); Aminophenazone (INN) (P) unclassified
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00565  Fenofibrate (JP18/USP/INN); Antara (TN); Lipantil (TN); Lipofen (TN); Tricor (TN); Triglide (TN) (P) unclassified
D00566  Sodium salicylate (JP18/USP); Salsonin (TN) (P) unclassified
D00567  Celecoxib (JP18/USP/INN); Celebrex (TN); Onsenal (TN) (P) unclassified
D00568  Rofecoxib (JAN/USAN/INN); Vioxx (TN) (P) unclassified
D00570  Colchicine (JP18/USP); Colchicine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D00578  Voriconazole (JP18/USP/INN); Vfend (TN) (P) unclassified
D00579  Foscarnet sodium (USP/INN); Foscavir (TN) (P) unclassified
D00594  Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) (P) unclassified
D00597  Acebutolol hydrochloride (JP18/USP); Sectral (TN) (P) unclassified
D00598  Betaxolol hydrochloride (JP18/USP); Betoptic (TN); Kerlone (TN) (P) unclassified
D00599  Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) (P) unclassified
D00601  Metoprolol tartrate (JP18/USP); Lopressor (TN) (P) unclassified
D00602  Penbutolol sulfate (JP18/USP); Levatol (TN) (P) unclassified
D00603  Timolol maleate (JP18/USP); Blocadren (TN); Istalol (TN); Timoptic (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00616  Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00617  Nicardipine hydrochloride (JP18/USAN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00618  Nisoldipine (JAN/USAN/INN); Sular (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D00620  Benazepril hydrochloride (JAN/USP); Lotensin (TN) (P) unclassified
D00621  Enalapril maleate (JP18/USP); Renivace (TN); Vasotec (TN) (P) unclassified
D00622  Fosinopril sodium (USP); Monopril (TN) (P) unclassified
D00623  Moexipril hydrochloride (USP); Univasc (TN) (P) unclassified
D00624  Perindopril erbumine (JAN/USP); Aceon (TN) (P) unclassified
D00626  Candesartan cilexetil (JP18/USP); Atacand (TN) (P) unclassified
D00627  Telmisartan (JP18/USP/INN); Micardis (TN) (P) unclassified
D00629  Nitrendipine (JP18/USAN/INN); Baypress (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00631  Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00634  Bisoprolol fumarate (JP18/USP); Zebeta (TN) (P) unclassified
D00635  Metoprolol succinate (USP); Toprol XL (TN) (P) unclassified
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00644  Esmolol hydrochloride (JAN/USP); Brevibloc (TN) (P) unclassified
D00649  Amiloride hydrochloride (USP); Midamor (TN) (P) unclassified
D00650  Bendroflumethiazide (JAN/USP/INN); Naturetin (TN) (P) unclassified
D00651  Benzthiazide (JAN/INN); Exna (TN) (P) unclassified
D00654  Hydroflumethiazide (JAN/USP/INN); Saluron (TN) (P) unclassified
D00656  Methyclothiazide (JAN/USP/INN); Enduron (TN) (P) unclassified
D00657  Polythiazide (JAN/USAN/INN); Renese (TN) (P) unclassified
D00658  Trichlormethiazide (JP18/USP/INN); Naqua (TN) (P) unclassified
D00661  Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00670  Donepezil hydrochloride (JP18/USP); Aricept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00687  Salmeterol xinafoate (JAN/USP); Serevent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00689  Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18); Beclovent (TN); Qnasl (TN); Vanceril (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00690  Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) unclassified
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00708  Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) (P) unclassified
D00709  Levetiracetam (JAN/USP/INN); Keppra (TN); E keppra (TN) (P) unclassified
D00710  Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) (P) unclassified
D00722  Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18); Ditropan (TN); Gelnique (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00726  Metoclopramide (JP18/INN); Elieten (TN); Terperan (TN) (P) unclassified
D00727  Olsalazine sodium (USAN); Dipentum (TN) (P) unclassified
D00734  Ursodiol (USP); Ursodeoxycholic acid (JP18/INN); Actigall (TN); Urso (TN) (P) unclassified
D00742  Etanercept (USAN/INN); Etanercept (genetical recombination) (JAN); Etanercept (genetical recombination) [Etanercept biosimilar 1] (JAN); Etanercept (genetical recombination) [Etanercept biosimilar 2] (JAN); Enbrel (TN) (P) unclassified
D00749  Leflunomide (JAN/USP/INN); Arava (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00751  Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00752  Mycophenolate mofetil (JAN/USP); Cellcept (TN) (P) unclassified
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D00754  Thalidomide (JAN/USP/INN); Thalomid (TN); Thaled (TN) (P) unclassified
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00809  Amitriptyline hydrochloride (JP18/USP); Elavil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00810  Choline salicylate (JAN/USAN/INN); Arthropan (TN) (P) unclassified
D00813  Ketorolac tromethamine (USP); Acular (TN); Toradol (TN) (P) unclassified
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) unclassified
D00824  Fluvoxamine maleate (JP18/USP); Luvox (TN) (P) CYP inhibition: CYP3A4
D00827  Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) (P) unclassified
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00851  Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) (P) unclassified
D00854  Quinupristin and dalfopristin; Synercid (TN) (P) CYP inhibition: CYP3A4
D00865  Amikacin sulfate (JP18/USP); Amikin (TN) (P) unclassified
D00866  Kanamycin sulfate (USP); Kanamycin monosulfate (JP18); Kantrex (TN) (P) unclassified
D00867  Netilmicin sulfate (JAN/USP); Netromycin (TN) (P) unclassified
D00868  Paromomycin sulfate (JAN/USP); Humatin (TN) (P) unclassified
D00869  Spectinomycin hydrochloride (USP); Spectinomycin hydrochloride hydrate (JP18); Trobicin (TN) (P) unclassified
D00880  Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) (P) unclassified
D00881  Econazole nitrate (JAN/USP); Ecoza (TN); Spectazole (TN) (P) unclassified
D00882  Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) (P) unclassified
D00885  Oxiconazole nitrate (JAN/USAN); Oxistat (TN) (P) unclassified
D00886  Sulconazole nitrate (JAN/USP); Exelderm (TN) (P) unclassified
D00887  Atorvastatin calcium anhydorous; Lipitor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D00888  Terconazole (USP/INN); Terazol 3 (TN) (P) unclassified
D00889  Cerivastatin sodium (JAN/USAN); Baycol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00890  Tioconazole (JAN/USP/INN); Vagistat-1 (TN) (P) unclassified
D00892  Fluvastatin sodium (JAN/USP); Lescol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00893  Pravastatin sodium (JP18/USP); CS-514; Pravachol (TN) (P) unclassified
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00903  Diclofenac potassium (USP); Cambia (TN); Cataflam (TN); Zipsor (TN) (P) unclassified
D00904  Diclofenac sodium (JP18/USP); Solaraze (TN); Voltaren (TN) (P) unclassified
D00926  Vancomycin hydrochloride (JP18/USP); Vancoled (TN); Vancocin (TN) (P) unclassified
D00961  Bicalutamide (JP18/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00968  Fenoprofen calcium (JAN/USP); Nalfon (TN) (P) unclassified
D00969  Meloxicam (JAN/USP/INN); Mobic (TN) (P) unclassified
D00970  Naproxen sodium (USP); Anaprox (TN) (P) unclassified
D00971  Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) (P) unclassified
D00972  Betamethasone sodium phosphate (JP18/USP); Celestone (TN) (P) unclassified
D00973  Cortisone acetate (JP18/USP); Cortone acetate (TN) (P) unclassified
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00976  Hydrocortisone cypionate (P) unclassified
D00977  Hydrocortisone sodium phosphate (JP18/USP); Hydrocortone phosphate (TN) (P) unclassified
D00978  Hydrocortisone sodium succinate (JP18/USP); A-hydrocort (TN); Solu-cortef (TN) (P) unclassified
D00979  Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00980  Prednisolone acetate (JP18/USP/INN); Econopred (TN); Pred forte (TN) (P) unclassified
D00981  Prednisolone sodium phosphate (JP18/USP); Pediapred (TN) (P) unclassified
D00982  Prednisolone tebutate (JAN/USP); Hydeltra-TBA (TN) (P) unclassified
D00983  Triamcinolone acetonide (JP18/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) (P) unclassified
D00984  Triamcinolone diacetate (JAN/USP); Aristocort (TN) (P) unclassified
D00985  Triamcinolone hexacetonide (USP/INN); Aristospan (TN) (P) unclassified
D00986  Fludrocortisone acetate (JP18/USP); Florinef acetate (TN) (P) unclassified
D00992  Gold sodium thiomalate (USP); Sodium aurothiomalate (JP18); Myochrysine (TN) (P) unclassified
D01025  Levobunolol hydrochloride (JAN/USP); Betagan (TN) (P) unclassified
D01026  Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) (P) unclassified
D01028  Ticlopidine hydrochloride (JP18/USP); Ticlid (TN) (P) unclassified
D01037  1,4-Dimethyl-7-isopropylazulene (JAN); Guaiazulene; Azunol (TN) (P) unclassified
D01049  Nimesulide (JAN/INN) (P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01063  Gentamicin sulfate (JP18/USP); Garamycin (TN); Gentacin (TN) (P) unclassified
D01069  Cilazapril (USAN); Cilazapril hydrate (JP18); Inhibace (TN) (P) unclassified
D01072  Chloramphenicol palmitate (JP18/USP); Chloromycetin palmitate (TN) (P) unclassified
D01078  Telithromycin (JAN/USAN/INN); Ketek (TN) (P) unclassified
D01087  Methyl salicylate (JP18/NF); Methyl salicylate (TN) (P) unclassified
D01092  Lanoconazole (JP18/INN); Latoconazole; Astat (TN) (P) unclassified
D01098  Maxacalcitol (JAN/USAN/INN); Oxarol (TN); Prezios (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01104  Barnidipine hydrochloride (JAN); Hypoca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01115  Eplerenone (JP18/USAN/INN); Inspra (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01119  Temocapril hydrochloride (JP18/USAN); Acecol (TN) (P) unclassified
D01122  Ibuprofen piconol (JP18/USAN); Staderm (TN) (P) unclassified
D01125  Calcipotriene (USP); Calcipotriol (JAN); Dovonex (TN) (P) unclassified
D01145  Azelnidipine (JP18/INN); Calblock (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01148  Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01154  Potassium acetate (JAN/USP); Potassium acetate (TN) (P) unclassified
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D01164  Aripiprazole (JAN/USP/INN); Abilify (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01173  Cilnidipine (JP18/INN); Atelec (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01176  Blonanserin (JAN/INN); AD 5423 (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01182  Alprenolol hydrochloride (JP18/USAN); Regletin (TN) (P) unclassified
D01183  Tolfenamic acid (JAN/INN); Clotam (TN) (P) unclassified
D01185  Protizinic acid (JAN/INN) (P) unclassified
D01189  Metiazinic acid (JAN/INN) (P) unclassified
D01190  Ethylphenacemide (JAN); Pheneturide (INN) (P) unclassified
D01196  Acetazolamide sodium (JAN); Diamox (TN) (P) unclassified
D01204  Olmesartan medoxomil (JP18/USP); Benicar (TN); Olmetec (TN) (P) Transporter inhibition: ABCB1
D01208  Aluminum clofibrate (JAN/INN); Alfibrate (TN) (P) unclassified
D01212  Simfibrate (JAN/INN); Cholesolvin (TN) (P) unclassified
D01213  Tolvaptan (JAN/USAN/INN); Samsca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) (CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01229  Paramethasone acetate (JAN/USAN); Haldrone (TN) (P) unclassified
D01235  Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) (P) CYP inhibition: CYP3A4
D01239  Prednisolone sodium succinate (JP18/USP); Kohakusanin (TN) (P) unclassified
D01240  Deslanoside (JP18/USP/INN); Cedilanid-d (TN) (P) unclassified
D01241  Penflutizide (JAN/INN) (P) unclassified
D01243  Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) (P) unclassified
D01246  Benzylhydrochlorothiazide (JAN); Behyd (TN) (P) unclassified
D01247  Ethiazide (JAN/INN) (P) unclassified
D01252  Alclofenac (JAN/USP/INN); Mervan (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01256  Cyclothiazide (JAN/USAN/INN); Anhydron (TN) (P) unclassified
D01266  Difluprednate (JAN/USAN/INN); Durezol (TN) (P) unclassified
D01267  Floctafenine (JAN/USAN/INN); Idarac (TN) (P) unclassified
D01271  Bufexamac (JAN/INN); Anderm (TN) (P) unclassified
D01272  Clobetasol propionate (JP18/USP); Clobex (TN); Cormax (TN); Olux (TN) (P) unclassified
D01273  Clobetasone butyrate (JAN/USAN); Kindavate (TN) (P) unclassified
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01289  Suxibuzone (JAN/INN) (P) unclassified
D01298  Potassium gluconate (JAN/USP); Gluconsan-K (TN) (P) unclassified
D01300  Clinofibrate (JP18/INN); Lipoclin (TN) (P) unclassified
D01303  Flunarizine hydrochloride (JAN/USAN) (P) unclassified
D01305  Feprazone (JAN/INN) (P) unclassified
D01308  Halcinonide (JAN/USP/INN); Halog (TN) (P) unclassified
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01325  Tiaprofenic acid (JAN/INN); Surgam (TN) (P) unclassified
D01327  Diflorasone diacetate (JP18/USP); Florone (TN); Psorcon (TN) (P) unclassified
D01330  Clidanac (JAN/INN) (P) unclassified
D01339  Midecamycin (JP18/INN); Medemycin (TN) (P) CYP inhibition: CYP3A4
D01341  Tiaramide hydrochloride (JP18/USAN); Solantal (TN) (P) unclassified
D01344  Fenbufen (JP18/USAN/INN) (P) unclassified
D01350  Streptomycin sulfate (JP18/USP); Streptomycin sulfate (TN) (P) unclassified
D01353  Emorfazone (JP18/INN); Pentoil (TN) (P) unclassified
D01357  Betamethasone valerate (JP18/USP); Beta-Val (TN); Luxiq (TN); Rinderon-V (TN) (P) unclassified
D01361  Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) (P) unclassified
D01366  Bezafibrate (JP18/USAN/INN); Bezatol SR (TN) (P) unclassified
D01367  Fluorometholone (JP18/USP/INN); NSC 33001; Fluor-op (TN); Fml (TN); Oxylone (TN) (P) unclassified
D01370  Cladribine (JAN/USP/INN); Leustatin (TN); Mavenclad (TN) (P) unclassified
D01372  Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01380  Isopropylantipyrine (JP18); Propyphenazone (INN); Yoshipyrin (TN) (P) unclassified
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) unclassified
D01387  Amcinonide (JAN/USP/INN); Cyclocort (TN) (P) unclassified
D01394  Epirizole (JP18/USAN); Mebron (TN) (P) unclassified
D01397  Ampiroxicam (JP18/INN); Flucam (TN) (P) unclassified
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01402  Betamethasone acetate (JAN/USP) (P) unclassified
D01410  Benzydamine hydrochloride (JAN/USAN); Tantum (TN) (P) unclassified
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01425  Lopinavir (JAN/USP/INN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP3A4
D01434  Deprodone propionate (JAN); Allomidon (TN) (P) unclassified
D01437  Nifenazone (JAN/INN) (P) unclassified
D01441  Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01442  Hydrocortisone succinate (JP18) (P) unclassified
D01454  Bupranolol hydrochloride (JP18) (P) unclassified
D01464  Flumethasone pivalate (USP); Flumetasone pivalate (JAN/BAN); Locorten (TN) (P) unclassified
D01466  Ethenzamide (JP18/INN); Ethenzamide (TN) (P) unclassified
D01471  Esatenolol (JAN/INN); (S)-Atenolol (P) unclassified
D01472  Tacalcitol hydrate (JP18); Bonalfa high (TN); Curatoderm (TN) (P) unclassified
D01475  Flurbiprofen axetil (JAN); FP 83; Ropion (TN) (P) unclassified
D01480  Isoconazole nitrate (JAN); Adestan-G (TN) (P) unclassified
D01492  Bucumolol hydrochloride (JP18) (P) unclassified
D01504  Bufetolol hydrochloride (JP18); Adobiol (TN) (P) unclassified
D01510  Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01512  Befunolol hydrochloride (JAN); Bentos (TN) (P) unclassified
D01513  Alminoprofen (JP18/INN); Minalfen (TN) (P) unclassified
D01518  Alfacalcidol (JAN/INN); Alsiodol (TN) (P) unclassified
D01523  Arbekacin sulfate (JP18); Habekacin (TN) (P) unclassified
D01545  Aceclofenac (JAN/INN); Aceclofenac (TN) (P) unclassified
D01547  Zaltoprofen (JP18/INN); CN 100; Peon (TN) (P) unclassified
D01549  Imidapril hydrochloride (JP18); Tanatril (TN) (P) unclassified
D01553  Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01557  Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) (P) unclassified
D01562  Aranidipine (JAN/INN); Sapresta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01565  Indometacin farnesil (JAN); Infree (TN) (P) unclassified
D01566  Gusperimus trihydrochloride (USAN); Gusperimus hydrochloride (JAN); Spanidin (TN) (P) unclassified
D01567  Ketophenylbutazone (JAN); Kebuzone (INN) (P) unclassified
D01578  Pranoprofen (JP18/INN); Elicapric (TN) (P) unclassified
D01581  Flufenamic acid (JAN/USAN/INN); Arlef (TN) (P) unclassified
D01582  Acemetacin (JP18/INN); Rantudil (TN) (P) unclassified
D01583  Pirfenidone (JAN/USAN/INN); Esbriet (TN) (P) unclassified
D01594  Bendazac (JAN/USAN/INN); Iwazac (TN) (P) unclassified
D01604  Efonidipine hydrochloride ethanolate (JAN); Efonidipine hydrochloride ethanol; Efonidipine hydrochloride; NZ 105 ethanolate; Landel (TN) (P) unclassified
D01614  Acetylkitasamycin (JP18); Neo-leucomycin H (TN) (P) unclassified
D01615  Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01618  Neomycin sulfate (USP); Fradiomycin sulfate (JP18); Mycifradin (TN); Neo-fradin (TN); Sofratulle (TN) (P) unclassified
D01619  Hydrocortisone butyrate (JP18/USP); Locoid (TN) (P) unclassified
D01620  Neticonazole hydrochloride (JAN); Atolant (TN) (P) unclassified
D01632  Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01636  Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) (P) CYP inhibition: CYP3A4
D01637  Betamethasone dipropionate (JP18/USP); Diprolene (TN); Rinderon-DP (TN); Sernivo (TN) (P) unclassified
D01656  Brovincamine fumarate (JAN); Sabromin (TN) (P) unclassified
D01661  Bucolome (JAN/INN); Paramidin (TN) (P) unclassified
D01662  Falecalcitriol (JAN/INN); Hornel (TN) (P) unclassified
D01664  Omoconazole nitrate (JAN/USAN) (P) unclassified
D01667  Delapril hydrochloride (JAN/USAN); Adecut (TN) (P) unclassified
D01675  Felbinac (JP18/USAN/INN); Dolinac (TN); Felbinac (TN) (P) unclassified
D01689  Loteprednol etabonate (JAN/USAN); Lotemax (TN) (P) unclassified
D01693  Dehydrocholic acid (JP18/USP/INN); Purified dehydrocholic acid (JP18); Decholin (TN) (P) unclassified
D01703  Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01706  Migrenin (JP18); Migrenin (TN) (P) unclassified
D01708  Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01709  Loxoprofen sodium hydrate (JP18); Lorfenamin (TN); Loxonin (TN) (P) unclassified
D01710  Roxithromycin (JP18/USAN/INN); Rulide (TN) (P) unclassified
D01712  Theophylline sodium acetate (JAN) (P) unclassified
D01718  Mofezolac (JAN/INN); Mofezolac (TN) (P) unclassified
D01741  Celiprolol hydrochloride (JAN/USAN); Selectol (TN) (P) unclassified
D01744  Brotizolam (JP18/USAN/INN); Lendormin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01745  Domperidone (JP18/USAN/INN); Motilium (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01753  Dibekacin sulfate (JP18); Panimycin (TN) (P) unclassified
D01762  Dipyrone (USAN); Sulpyrine hydrate (JP18); Metamizole sodium salt monohydrate; Sulpyrine (TN) (P) unclassified
D01764  Diflucortolone valerate (JP18); Afusona (TN) (P) unclassified
D01765  Proglumetacin maleate (JAN); Miridacin (TN) (P) unclassified
D01767  Tenoxicam (JAN/USAN/INN); Tilcotil (TN) (P) unclassified
D01775  Bifonazole (JP18/USAN/INN); Mycospor (TN) (P) unclassified
D01776  Antipyrine (JP18/USP); Phenazone (INN) (P) unclassified
D01787  Sulthiame (USAN); Sultiame (JP18); Ospolot (TN) (P) unclassified
D01788  Amfenac sodium (USAN); Amfenac sodium hydrate (JAN); Fenazox (TN) (P) unclassified
D01794  Bopindolol malonate (JAN); Sandonorm (TN) (P) unclassified
D01795  Tilisolol hydrochloride (JAN); Selecal (TN) (P) unclassified
D01806  Oxprenolol hydrochloride (JP18/USP); Okuspurecol (TN) (P) unclassified
D01811  Salicylamide (JAN/USP/INN); Salicylamide (TN) (P) unclassified
D01820  Alclometasone dipropionate (JAN/USP); Aclovate (TN) (P) unclassified
D01821  Micronomicin sulfate (JP18); Sagamicin (TN); Santemycin (TN) (P) unclassified
D01823  Ufenamate (JAN/INN); Flufenamic acid butyl ester; Combec (TN) (P) unclassified
D01825  Fluocinolone acetonide (JP18/USP/INN); Fluocet (TN); Retisert (TN); Synalar (TN) (P) unclassified
D01826  Isepamicin sulfate (JP18); Isepacin (TN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01841  Felbinac ethyl (JAN); LM 001 (P) unclassified
D01847  Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN) (P) unclassified
D01849  Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) (P) unclassified
D01851  Mepranoprofen arbamel (JAN); Y-23023 (P) unclassified
D01862  Pitavastatin calcium (JAN); NK 104; Livalo (TN) (CI,P) unclassified
D01865  Pelubiprofen (JAN/INN) (P) unclassified
D01866  Lornoxicam (JAN/USAN/INN); Lorcam (TN) (P) unclassified
D01868  Bekanamycin sulfate (JP18); AKM; Kanendomycin (TN) (P) unclassified
D01874  Vedaprofen (JAN/USAN/INN) (P) unclassified
D01881  Astromicin sulfate (JAN/USAN); Fortimicin (TN) (P) unclassified
D01886  Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) (P) unclassified
D01896  Cilostazol (JP18/USP/INN); Pletal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01897  Rokitamycin (JAN/INN); Ricamycin (TN) (P) unclassified
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01900  Alacepril (JP18/INN); Cetapril (TN) (P) unclassified
D01908  Nilvadipine (JP18/USAN/INN); Nivadil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01915  Rosuvastatin calcium (JP18/USP); ZD 4522; Crestor (TN) (CI,P) unclassified
D01922  Pratosartan (JAN/INN); KD 3-671 (P) unclassified
D01933  Vatanidipine hydrochloride (JAN); AE 0047; Calbren (TN) (P) unclassified
D01943  Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) (P) unclassified
D01948  Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01958  Indenolol hydrochloride (JP18) (P) unclassified
D01963  Ibufenac (JAN/USAN/INN); Dytransin (TN) (P) unclassified
D01966  Ezetimibe (JAN/USP/INN); Zetia (TN) (P) unclassified
D01969  Gallopamil hydrochloride (JAN) (P) unclassified
D01974  Tilmacoxib (JAN/USAN/INN) (P) unclassified
D01975  Fentiazac (JAN/USAN/INN) (P) unclassified
D01977  Gefitinib (JP18/USAN/INN); Iressa (TN) (P) unclassified
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) CYP inhibition: CYP3A4
D01998  Prednisolone farnesylate (JAN); PNF 21; Farnerate (TN) (P) unclassified
D02000  Kitasamycin tartrate (JP18); Leucomycin tartrate (TN) (P) unclassified
D02002  Isoniazid sodium methanesulfonate hydrate (JAN); Isoniazid sodium methanesulfonate monohydrate; Isoniazid sodium methanesulfonate; IHMS; Neoiscotin (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02009  Erythromycin lactobionate (JP18/USP); Erythrocin (TN) (P) unclassified
D02032  Betamethasone butyrate propionate (JAN); Antebate (TN) (P) unclassified
D02045  Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02060  Potassium chloride (JP18/USP); K-dur (TN); KCL (TN); Kaon-Cl (TN); Klor-con (TN); Klotrix (TN) (P) unclassified
D02061  Cyclopenthiazide (JAN/USAN/INN); Navidrex (TN) (P) unclassified
D02075  Sodium gualenate (INN); Sodium guaiazulenesulfonate; Azunol ST (TN) (P) unclassified
D02077  Potassium bicarbonate (USP); Potassium hydrogencarbonate; Potassium hydrogen carbonate; K-vescent (TN) (P) unclassified
D02081  Metipranolol hydrochloride; Optipranolol (TN) (P) unclassified
D02082  Eprosartan mesylate (USAN); Teveten (TN) (P) unclassified
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) CYP induction: CYP3A4
D02097  Tiagabine hydrochloride (USP); Gabitril (TN) (P) unclassified
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02110  Indomethacin sodium (USP); Indometacin sodium hydrate (JAN); Indomethacin sodium trihydrate; Indometacin sodium; Indocin I.V. (TN) (P) unclassified
D02112  Heparin sodium (JP18/USP/INN); Parnaparin sodium (INN); Liquemin sodium (TN) (P) unclassified
D02114  Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02115  Methotrexate sodium; Trexall (TN); Rasuvo (TN) (P) unclassified
D02134  Azithromycin hydrate (JP18); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) (P) Transporter inhibition: ABCB1
D02142  Teicoplanin (JP18/USAN/INN); Tagocid (TN) (P) unclassified
D02156  Prednisolone hemisuccinate (USP); Prednisolone succinate (JP18) (P) unclassified
D02165  Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02169  Croconazole hydrochloride (JP18); Pilzcin (TN) (P) unclassified
D02174  Dexamethasone acetate (JAN/USP); Decadronal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02181  Sisomicin sulfate (JAN/USP); Siseptin (TN) (P) unclassified
D02184  Erythromycin stearate (JP18/USP); Bristamycin (TN) (P) unclassified
D02185  Chloramphenicol sodium succinate (JP18/USP); Chloromycetin succinate (TN) (P) unclassified
D02186  Oleandomycin phosphate (JAN); Matromycin (TN) (P) unclassified
D02209  Ribostamycin sulfate (JP18); Vistamycin (TN) (P) unclassified
D02213  Metoclopramide hydrochloride (JAN); Metoclopramide dihydrochloride monohydrate; Primperan (TN); Reglan (TN) (P) unclassified
D02216  Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP18); Ciloxan (TN); Cipro (TN); Proquin XR (TN) (P) unclassified
D02219  Terbinafine hydrochloride (JP18/USP); Lamisil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02250  Octreotide acetate (JAN); Octreotide diacetate; Sandostatin (TN) (P) unclassified
D02258  Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D02264  Dipotassium glycyrrhizinate (JAN); Glycyrrhizinate dipotassium; Neubormitin (TN) (P) unclassified
D02267  Foscarnet sodium hydrate (JAN); Foscarnet sodium hexahydrate; Trisodium phosphonoformate hexahydrate; Foscavir (TN) (P) unclassified
D02269  Kitasamycin (JP18/USAN); Leucomycin (TN) (P) unclassified
D02286  Betamethasone benzoate (USP); Uticort (TN) (P) unclassified
D02287  Clocortolone pivalate (USP); Cloderm (TN) (P) unclassified
D02288  Hydrocortisone valerate (USP); Westcort (TN) (P) unclassified
D02289  Medrysone (USAN); HMS (TN) (P) unclassified
D02290  Flurbiprofen sodium (USP); Ocufen (TN) (P) unclassified
D02322  Apramycin (USAN/INN) (P) unclassified
D02338  Acebutolol (USAN/INN) (P) unclassified
D02341  Meclofenamic acid (USAN/INN) (P) unclassified
D02342  Bisoprolol (JAN/USAN/INN) (P) unclassified
D02350  Fenoprofen (USAN/INN) (P) unclassified
D02355  Tolmetin (USAN/INN) (P) unclassified
D02356  Verapamil (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D02358  Metoprolol (USAN/INN) (P) unclassified
D02372  Perospirone hydrochloride hydrate (JAN); Lullan (TN) (P) unclassified
D02374  Metipranolol (USAN/INN) (P) unclassified
D02375  Terbinafine (USAN/INN); Lamasil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02389  Primidolol (USAN/INN) (P) unclassified
D02420  Acetylspiramycin (JP18); Spiramycin II; Acetylspiramycin (TN) (P) unclassified
D02453  Flumethiazide (INN); Ademol (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02490  Tylosin (USP/INN); TS; Tylan (TN) (P) unclassified
D02492  Tilmicosin (USP/INN); TMS; Micotil (TN) (P) unclassified
D02493  Tilmicosin phosphate (USAN); TP (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) unclassified
D02501  Caspofungin acetate (JAN/USAN); Cancidas (TN) (P) unclassified
D02512  Dihydrostreptomycin sulfate (USP) (P) unclassified
D02523  Erythromycin acistrate (USAN); Erasis (TN) (P) unclassified
D02524  Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) (P) unclassified
D02525  Erythromycin propionate (USAN) (P) unclassified
D02537  Dronedarone (INN) (P) unclassified
D02542  Tobramycin sulfate (USP); Nebcin (TN) (P) unclassified
D02543  Amikacin (USP/INN) (P) unclassified
D02544  Sisomicin (USAN/INN) (P) unclassified
D02545  Isepamicin (USAN/INN) (P) unclassified
D02554  Rifaximin (JAN/USAN/INN); Xifaxan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 / Transporter inhibition: ABCB1
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D02556  Ravuconazole (prop.INN) (P) unclassified
D02557  Chlormidazole (INN) (P) unclassified
D02582  Fenticonazole (INN) (P) unclassified
D02583  Fenticonazole nitrate (USAN); Lomexin (TN) (P) unclassified
D02584  Aliconazole (INN) (P) unclassified
D02585  Vibunazole; Bay N-7133 (P) unclassified
D02586  Alteconazole (INN) (P) unclassified
D02587  Metildigoxin (JP18); Lanirapid (TN) (P) Transporter inhibition: ABCB1
D02591  Dexamethasone acefurate (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02592  Dexamethasone beloxil (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02596  Tocilizumab (USAN/INN); Tocilizumab (genetical recombination) (JAN); Actemra (TN) (P) unclassified
D02597  Adalimumab (USAN/INN); Adalimumab (genetical recombination) (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 1] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 2] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 3] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 4] (JAN); Adalimumab-adaz; Adalimumab-adbm; Adalimumab-afzb; Adalimumab-atto; Adalimumab-bwwd; Adalimumab-fkjp; Adalimumab-aaty; Adalimumab-aacf; Adalimumab-aqvh; Humira (TN); Abrilada (TN); Amjevita (TN); Cyltezo (TN); Hadlima (TN); Hyrimoz (TN) (P) unclassified
D02598  Infliximab (USAN/INN); Infliximab (genetical recombination) (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 1] (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 2] (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 3] (JAN); Infliximab-dyyb; Infliximab-abda; Infliximab-axxq; Remicade (TN); Inflectra (TN); Renflexis (TN); Avsola (TN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02629  Fluspirilene (USAN/INN); Imap (TN) (P) unclassified
D02630  Penfluridol (USAN/INN); Semap (TN) (P) unclassified
D02633  Lomerizine hydrochloride (JAN); Terranas (TN) (P) unclassified
D02689  Ramelteon (JAN/USAN/INN); Rozerem (TN) (P) unclassified
D02690  Cholestyramine resin (USP); Colestyramine (JAN/INN); Questran (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02706  Sodium gualenate hydrate (JAN); Azulene sulfonate sodium hydrate; Sodium guaiazulene sulfonate; Azunol (TN) (P) unclassified
D02709  Valdecoxib (USAN/INN); Bextra (TN) (P) unclassified
D02714  Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D02715  Balsalazide disodium (USP); Colazide (TN) (P) unclassified
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02765  Adaprolol maleate (USAN) (P) unclassified
D02766  Valpromide (INN); Depamide (TN) (P) unclassified
D02800  Alefacept (USAN/INN); Amevive (TN) (P) unclassified
D02802  Alemtuzumab (USAN/INN); Alemtuzumab (genetical recombination) (JAN); Campath (TN); Lemtrada (TN) (P) unclassified
D02834  Alprenoxime hydrochloride (USAN) (P) unclassified
D02838  Althiazide (USAN); Altizide (INN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02910  Amiodarone (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02914  Amlodipine maleate (USAN); Amvaz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02934  Anakinra (USAN/INN); Kineret (TN) (P) unclassified
D02944  Anirolac (USAN/INN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02980  Adomiparin sodium (USAN); Ardeparin sodium (USAN/INN); Semuloparin sodium (USAN/INN); Normiflo (TN) (P) unclassified
D02994  Rituximab (USAN/INN); Rituximab (genetical recombination) (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 1] (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 2] (JAN); Rituximab-abbs; Rituximab-pvvr; Rituximab-arrx; Rituxan (TN); Riabni (TN); Truximab (TN) (P) unclassified
D03023  Azaconazole (USAN/INN) (P) unclassified
D03033  Azathioprine sodium (USP); Imuran (TN) (P) unclassified
D03058  Basiliximab (USAN/INN); Basiliximab (genetical recombination) (JAN); Simulect (TN) (P) unclassified
D03063  BCG vaccine (USP); Freeze-dried BCG vaccine (for percutaneous use) (JP18); BCG vaccine (TN) (CI) unclassified
D03067  Belfosdil (USAN/INN) (P) unclassified
D03068  Belimumab (USAN); Belimumab (genetical recombination) (JAN); Benlysta (TN); LymphoStat-B (TN) (P) unclassified
D03077  Benazeprilat (USAN/INN) (P) unclassified
D03080  Benoxaprofen (USAN/INN); Oraflex (TN) (P) unclassified
D03098  Berythromycin (USAN/INN); Erythromycin B (P) unclassified
D03104  Betamicin sulfate (USAN) (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03150  Bortezomib (JAN/USAN/INN); Velcade (TN) (P) unclassified
D03163  Bromfenac sodium (USAN); Bromfenac sodium hydrate (JP18); Bromfenac sodium sesquihydrate; Bromday (TN); Prolensa (TN); Xibrom (TN); Yellox (TN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03170  Bucindolol hydrochloride (USAN) (P) unclassified
D03177  Bunolol hydrochloride (USAN) (P) unclassified
D03189  Buthiazide (USAN); Butizide (INN) (P) unclassified
D03190  Butikacin (USAN/INN) (P) unclassified
D03198  Butoxamine hydrochloride (USAN) (P) unclassified
D03203  Abatacept (USAN/INN); Abatacept (genetical recombination) (JAN); Orencia (TN) (P) unclassified
D03204  Abetimus sodium (USAN) (P) unclassified
D03208  Aliskiren (USAN/INN); Rasilez (TN) (CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D03218  Axitinib (JAN/USAN); Inlyta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03222  Belatacept (USAN/INN); Nulojix (TN) (P) unclassified
D03253  Brecanavir (USAN) (P) unclassified
D03254  Flufenamate aluminum (JAN); Flufenamic acid aluminum; Opyrin (TN) (P) unclassified
D03256  Valganciclovir hydrochloride (JAN/USP); Valcyte (TN) (P) unclassified
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03262  Kanamycin sulfate (JP18); Kanamycin sulfate (TN) (P) unclassified
D03301  Prednisolone valerate acetate (JAN); PDL; Spirazon (TN) (P) unclassified
D03325  Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03337  Reviparin sodium (JAN); Clivarine (TN) (P) unclassified
D03353  Dalteparin sodium (JAN/USP/INN); Ardeparin sodium; Fragmin (TN) (P) unclassified
D03363  Canrenone (USAN) (P) unclassified
D03385  Carbaspirin calcium (USAN); Carbasalate calcium (INN) (P) unclassified
D03410  Carprofen (USP/INN); Rimadyl (TN) (P) unclassified
D03415  Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03440  Ceronapril (USAN/INN) (P) unclassified
D03441  Certolizumab pegol (USAN/INN); Certolizumab pegol (genetical recombination) (JAN); Cimzia (TN) (P) unclassified
D03449  Cetamolol hydrochloride (USAN) (P) unclassified
D03461  Chloramphenicol pantothenate complex (USAN/INN); Pantofenicol (TN) (P) unclassified
D03471  Chlorothiazide sodium (USP); Diuril (TN) (P) unclassified
D03489  Cicloprofen (USAN/INN) (P) unclassified
D03490  Cicloprolol hydrochloride (USAN) (P) unclassified
D03521  Ciprofibrate (USAN/INN) (P) unclassified
D03526  Cisconazole (USAN/INN) (P) unclassified
D03536  Clentiazem maleate (JAN/USAN) (P) unclassified
D03540  Cliprofen (USAN/INN) (P) unclassified
D03541  Clocortolone acetate (USAN) (P) unclassified
D03560  Clopirac (USAN/INN) (P) unclassified
D03561  Cloprednol (USAN/INN); Cloradryn (TN) (P) unclassified
D03594  Cortivazol (USAN) (P) unclassified
D03601  Crilvastatin (USAN/INN) (P) unclassified
D03639  Daclizumab (USAN/INN); Zenapax (TN); Zinbryta (TN) (P) unclassified
D03643  Dalvastatin (USAN/INN) (P) unclassified
D03652  Darbufelone mesylate (USAN) (P) unclassified
D03655  Darodipine (USAN/INN) (P) unclassified
D03656  Darunavir (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP induction: CYP3A4
D03671  Deflazacort (USAN/INN); Emflaza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D03673  Deligoparin sodium (USAN/INN) (P) unclassified
D03674  Enoxaparin sodium (JAN/USP/INN); Lovenox (TN) (P) unclassified
D03689  Deracoxib (USAN) (P) unclassified
D03696  Desonide (USP/INN); Desowen (TN); Verdeso (TN) (P) unclassified
D03697  Desoximetasone (USP/INN); Topicort (TN) (P) unclassified
D03710  Etoricoxib (USAN/INN) (P) unclassified
D03712  Firocoxib (USAN/INN); Equioxx (TN) [veterinary] (P) unclassified
D03714  Lumiracoxib (USAN/INN) (P) unclassified
D03715  Dexibuprofen (USAN/INN) (P) unclassified
D03716  Parecoxib (USAN/INN) (P) unclassified
D03717  Parecoxib sodium (USAN); Dynastat (TN) (P) unclassified
D03718  Dexibuprofen lysine (USAN); Dexibuprofen lysine monohydrate; Doctrin (TN) (P) unclassified
D03727  Dexpemedolac (USAN/INN) (P) unclassified
D03729  Dexpropranolol hydrochloride (USAN) (P) unclassified
D03752  Quinapril (INN) (P) unclassified
D03753  Perindopril (USAN/INN) (P) unclassified
D03756  Indolapril hydrochloride (USAN) (P) unclassified
D03758  Libenzapril (USAN/INN) (P) unclassified
D03759  Diacetolol hydrochloride (USAN) (P) unclassified
D03760  Pentopril (USAN/INN) (P) unclassified
D03763  Pivopril (USAN/INN) (P) unclassified
D03765  Spirapril hydrochloride (USAN); Renormax (TN) (P) unclassified
D03767  Zofenopril calcium (USAN); Zoprace (TN) (P) unclassified
D03769  Enalaprilat (USP); Enalaprilat dihydrate; Vasotec (TN) (P) unclassified
D03772  Fosinoprilat (USAN/INN) (P) unclassified
D03773  Quinaprilat (USAN/INN) (P) unclassified
D03775  Spiraprilat (USAN/INN) (P) unclassified
D03776  Zofenoprilat arginine (USAN) (P) unclassified
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03812  Diflucortolone (USAN) (P) unclassified
D03813  Diflucortolone pivalate (USAN) (P) unclassified
D03816  Tenivastatin calcium (USAN) (P) unclassified
D03820  Dutasteride (JAN/USP/INN); Avodart (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03830  Diltiazem malate (USAN); Tiamate (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03839  Droxinavir hydrochloride (USAN) (P) unclassified
D03840  Palinavir (USAN/INN) (P) unclassified
D03842  Telinavir (USAN/INN) (P) unclassified
D03843  Tipranavir disodium (USAN) (P) unclassified
D03844  Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) (P) unclassified
D03846  Dimethyl fumarate (JAN/USAN); Tecfidera (TN) (P) unclassified
D03865  Dirithromycin (USP/INN); Dynabac (TN) (P) unclassified
D03883  Doconazole (USAN/INN) (P) unclassified
D03914  Dronedarone hydrochloride (USP); Multaq (TN) (P) unclassified
D03936  Econazole (USAN/INN) (P) unclassified
D03940  Eculizumab (USAN/INN); Eculizumab (genetical recombination) (JAN); Soliris (TN) (P) unclassified
D03959  Efalizumab (USAN/INN); Raptiva (TN) (P) unclassified
D03960  Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) (P) unclassified
D03978  Eltrombopag olamine (JAN/USAN); Promacta (TN) (P) unclassified
D03997  Enilconazole (USAN/INN) (P) unclassified
D04003  Enolicam sodium (USAN); Enolicam sodium monohydrate (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D04033  Epithiazide (USAN); Epitizide (INN) (P) unclassified
D04040  Eprosartan (USAN/INN) (P) unclassified
D04054  Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate (P) unclassified
D04059  Mepenzolate bromide and phenobarbital; Trancolon P (TN) (P) unclassified
D04102  Etofenamate (USAN/INN) (P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D04126  Saralasin acetate (USAN); Sarenin (TN) (P) unclassified
D04142  Fenclofenac (USAN/INN) (P) unclassified
D04144  Fenclorac (USAN/INN) (P) unclassified
D04145  Fendosal (USAN/INN); Alnovin (TN) (P) unclassified
D04148  Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04187  Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) (P) unclassified
D04190  Flestolol sulfate (USAN) (P) unclassified
D04193  Flordipine (USAN/INN) (P) unclassified
D04201  Flucloronide (USAN); Fluclorolone acetonide (INN) (P) unclassified
D04206  Flufenisal (USAN/INN) (P) unclassified
D04208  Flumethasone (USAN); Flumetasone (INN) (P) unclassified
D04214  Flunisolide acetate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04217  Fluocortin butyl (USAN) (P) unclassified
D04218  Fluocortolone (USAN/INN) (P) unclassified
D04219  Fluocortolone caproate (USAN) (P) unclassified
D04221  Fluorometholone acetate (USP); Fluorometholone 17-acetate; Flarex (TN) (P) unclassified
D04225  Fluperolone acetate (USAN); Methral (TN) (P) unclassified
D04243  Forasartan (USAN/INN) (P) unclassified
D04244  Formocortal (USAN/INN); Deflamene (TN) (P) unclassified
D04260  Fostedil (USAN/INN) (P) unclassified
D04273  Furaprofen (USAN/INN) (P) unclassified
D04277  Furobufen (USAN/INN) (P) unclassified
D04300  Ganaxolone (USAN/INN); Ztalmy (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04301  Ganciclovir sodium (USAN); Cytovene IV (TN) (P) unclassified
D04358  Golimumab (USAN/INN); Golimumab (genetical recombination) (JAN); Simponi (TN) (P) unclassified
D04409  Halobetasol propionate (USP); Ulobetasol propionate; Ultravate (TN) (P) unclassified
D04411  Halofenate (USAN/INN) (P) unclassified
D04427  Heparin calcium (JP18); Nadroparin calcium (INN); Calciparin; Calciparine (TN) (P) unclassified
D04446  Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04447  Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04463  Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04467  Hydrocortisone hemisuccinate (USP) (P) unclassified
D04482  Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) (P) unclassified
D04483  Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) (P) unclassified
D04484  Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) (P) unclassified
D04489  Ibritumomab tiuxetan (USAN/INN); Ibritumomab tiuxetan (genetical recombination) (JAN); Zevalin (TN) (P) unclassified
D04490  Ibuprofen aluminum (USAN) (P) unclassified
D04530  Indoprofen (USAN/INN) (P) unclassified
D04536  Influenza virus vaccine (USP); FluShield (TN); Fluarix quadrivalent (TN) (P) unclassified
D04624  Isoconazole (USAN/INN) (P) unclassified
D04638  Isoxepac (USAN/INN); Artil (TN) (P) unclassified
D04639  Isoxicam (USAN/INN); Maxicam (TN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04657  Lacidipine (USAN/INN); Motens (TN) (P) unclassified
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04687  Lenalidomide (JAN/USAN/INN); Revlimid (TN) (P) unclassified
D04710  Levobetaxolol hydrochloride (USAN); Betaxon (TN) (P) unclassified
D04725  Lexithromycin (USAN/INN) (P) unclassified
D04733  Lidoflazine (USAN/INN); Angex (TN) (P) unclassified
D04736  Lifibrate (USAN/INN) (P) unclassified
D04737  Lifibrol (USAN/INN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (CI,P) unclassified
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04863  Mavacoxib (USAN) (P) unclassified
D04866  Freeze-dried live attenuated measles vaccine (JP18) (CI) unclassified
D04888  Medroxalol (USAN/INN) (P) unclassified
D04889  Medroxalol hydrochloride (USAN) (P) unclassified
D04896  Megalomicin potassium phosphate (USAN) (P) unclassified
D04948  Potassium L-aspartate (JAN); Potassium aspartate; L-Aspartate potassium; Aspara K (TN) (P) unclassified
D04952  Potassium aspartate and magnesium aspartate (JAN/USAN); Aspara (TN) (P) unclassified
D04976  Methalthiazide (USAN) (P) unclassified
D04977  Parnaparin sodium (JP18); Lowhepa (TN) (P) unclassified
D05000  Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05001  Methylprednisolone sodium phosphate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05002  Methylprednisolone suleptanate (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05008  Metoclopramide hydrochloride (USP); Metoclopramide monohydrochloride monohydrate; Clopra (TN); Reglan (TN) (P) unclassified
D05011  Metoprolol fumarate (USP); Lopressor (TN) (P) unclassified
D05016  Metronidazole hydrochloride (USAN); Flagyl I.V. (TN) (P) unclassified
D05017  Metronidazole phosphate (USAN) (P) unclassified
D05024  Mibefradil dihydrochloride (USAN); Posicor (TN) (P) unclassified
D05089  Freeze-dried live attenuated mumps vaccine (JP18); Freeze-dried live attenuated mumps vaccine (TN) (CI) unclassified
D05092  Muromonab-CD3 (JAN/USAN/INN); Orthoclone okt3 (TN) (P) unclassified
D05094  Mycophenolate mofetil hydrochloride (USAN); Cellcept (TN) (P) unclassified
D05095  Mycophenolate sodium (USP); Myfortic (TN) (P) unclassified
D05096  Mycophenolic acid (USAN/INN); Mycophenolic acid (TN) (P) unclassified
D05102  Nafenopin (USAN/INN) (P) unclassified
D05121  Naproxol (USAN/INN) (P) unclassified
D05127  Nebivolol (USAN/INN) (P) unclassified
D05128  Nebramycin (USAN) (P) unclassified
D05140  Framycetin (INN); Fradiomycin B; Neomycin B; FRM (P) unclassified
D05141  Neomycin palmitate (USAN) (P) unclassified
D05142  Neomycin undecylenate (USAN) (P) unclassified
D05143  Nepafenac (JAN/USAN/INN); Nevanac (TN) (P) unclassified
D05153  Neutramycin (USAN) (P) unclassified
D05181  Aspirin aluminum (JP18) (P) unclassified
D05182  Influenza HA vaccine (JP18) (P) unclassified
D05218  Ocrelizumab (USAN); Ocrelizumab (genetical recombination) (JAN); Ocrevus (TN) (P) unclassified
D05230  Octreotide pamoate (USAN) (P) unclassified
D05246  Olmesartan (USAN/INN) (P) Transporter inhibition: ABCB1
D05248  Freeze-dried inactivated tissue culture ravies vaccine (JP18) (P) unclassified
D05268  Orconazole nitrate (USAN) (P) unclassified
D05319  Oxyphenbutazone hydrate; Tandearil (TN) (P) unclassified
D05345  Pamatolol sulfate (USAN) (P) unclassified
D05351  Josamycin propionate (JP18); Josamy (TN) (P) CYP inhibition: CYP3A4
D05367  Parconazole hydrochloride (USAN) (P) unclassified
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (P) unclassified
D05404  Pemedolac (USAN/INN) (P) unclassified
D05425  Pentisomicin (USAN/INN) (P) unclassified
D05429  Aminophylline hydrate (JP18) (P) unclassified
D05442  Perhexiline maleate (USAN) (P) unclassified
D05451  Phenbutazone sodium glycerate (USAN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP18) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05511  Piroxicam betadex (USAN) (P) unclassified
D05512  Piroxicam cinnamate (USAN) (P) unclassified
D05513  Piroxicam olamine (USAN) (P) unclassified
D05515  Pirprofen (USAN/INN) (P) unclassified
D05538  Mozenavir (INN) (P) unclassified
D05544  Live oral polimyelitis vaccine (JAN); Poliovirus vaccine live oral; Orimune (TN) (CI) unclassified
D05587  Practolol (USAN) (P) unclassified
D05598  Pravadoline maleate (USAN) (P) unclassified
D05601  Prednicarbate (USP/INN); Dermatop (TN) (P) unclassified
D05619  Prodolic acid (USAN/INN) (P) unclassified
D05621  Progabide (USAN/INN); Gabren (TN) (P) unclassified
D05629  Propikacin (USAN) (P) unclassified
D05640  Prorenoate potassium (USAN/INN) (P) unclassified
D05713  Relomycin (USAN/INN) (P) unclassified
D05717  Repromicin (USAN/INN) (P) unclassified
D05719  Resocortol butyrate (USAN) (P) unclassified
D05729  Rimexolone (USP/INN); Vexol (TN) (P) unclassified
D05757  Rosaramicin (USAN/INN) (P) unclassified
D05758  Rosaramicin butyrate (USAN) (P) unclassified
D05759  Rosaramicin propionate (USAN) (P) unclassified
D05760  Rosaramicin sodium phosphate (USAN) (P) unclassified
D05761  Rosaramicin stearate (USAN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05788  Salcolex (USAN); Salcolex tetrahydrate (P) unclassified
D05789  Salethamide maleate (USAN) (P) unclassified
D05791  Salicylate meglumine (USAN) (P) unclassified
D05793  Salnacedin (USAN/INN) (P) unclassified
D05800  Saperconazole (USAN/INN) (P) unclassified
D05801  Saprisartan potassium (USAN) (P) unclassified
D05811  Sedecamycin (USAN/INN) (P) unclassified
D05830  Sermetacin (USAN/INN) (P) unclassified
D05908  Spiramycin (JAN/USAN/INN); Rovamycin (TN) (P) unclassified
D05912  Spiroxasone (USAN/INN) (P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05937  Sudoxicam (USAN/INN) (P) unclassified
D05995  Talmetacin (USAN/INN) (P) unclassified
D05998  Talosalate (USAN/INN) (P) unclassified
D06010  Tasosartan (USAN/INN) (P) unclassified
D06060  Teludipine hydrochloride (USAN) (P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06076  Teprotide (USAN/INN) (P) unclassified
D06082  Tesicam (USAN) (P) unclassified
D06102  Theofibrate (USAN); Etofylline clofibrate (INN); Duolip (TN) (P) unclassified
D06103  Theophylline (USP); Theophylline monohydrate; Accurbron (TN) (P) unclassified
D06104  Theophylline sodium glycinate (USP); Asbron (TN) (P) unclassified
D06133  Tibric acid (USAN/INN) (P) unclassified
D06143  Tifurac sodium (USAN) (P) unclassified
D06156  Tiopinac (USAN/INN) (P) unclassified
D06171  Tixocortol pivalate (USAN) (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06209  Treloxinate (USAN/INN) (P) unclassified
D06216  Triamcinolone acetonide sodium phosphate (USAN) (P) unclassified
D06254  Trospectomycin sulfate (USAN) (P) unclassified
D06258  Tulathromycin (JAN/USAN/INN) (P) unclassified
D06273  Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06315  Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06347  Yellow fever vaccine (USP); YF-Vax (TN) (CI) unclassified
D06363  Ziconotide (USAN/INN); Prialt (TN) (P) unclassified
D06364  Zidometacin (USAN/INN) (P) unclassified
D06373  Zinoconazole hydrochloride (USAN) (P) unclassified
D06382  Zomepirac sodium (USAN); Zomepirac sodium dihydrate (P) unclassified
D06390  Azithromycin (USP); Zmax (TN) (P) Transporter inhibition: ABCB1
D06398  Tinzaparin sodium (USAN); Innohep (TN) (P) unclassified
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06405  Nalfurafine hydrochloride (JAN/USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06412  Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06466  Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) (CI) unclassified
D06475  Adsorbed hepatitis B vaccine (JP18); Bimmugen (TN) (P) unclassified
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06495  Octreotide acetate (USP); Sandostatin (TN) (P) unclassified
D06511  Freeze-dried smallpox vaccine prepared in cell culture (JP18) (CI) unclassified
D06512  Freeze-dried live attenuated rubella vaccine (JP18) (CI) unclassified
D06573  Carisbamate (USAN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06598  Gamithromycin (USAN/INN) (P) unclassified
D06606  Ibuprofen lysine (USAN); Ibuprofen L-lysine (JAN); Solufenum; Neoprofen (TN) (P) unclassified
D06622  Nebivolol hydrochloride (USAN); Bystolic (TN) (P) unclassified
D06630  Pramiconazole (USAN/INN) (P) unclassified
D06635  Rilonacept (USAN/INN); Arcalyst (TN) (P) unclassified
D06637  Romidepsin (JAN/USAN/INN); Istodax (TN) (P) unclassified
D06646  Epanolol (USAN/INN) (P) unclassified
D06673  Meprednisone (USP/INN) (P) unclassified
D06876  Hydrocortisone aceponate (INN); Efficort (TN) (P) unclassified
D06883  Sertaconazole (INN) (P) unclassified
D06886  Natalizumab (USAN/INN); Natalizumab (genetical recombination) (JAN); Tysabri (TN) (P) unclassified
D07073  Dexamethasone cipecilate (JAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07077  Ambrisentan (JAN/INN); Letairis (TN); Volibris (TN) (P) unclassified
D07082  Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) (CI,P) Transporter inhibition: ABCB1
D07116  Alclometasone (INN) (P) unclassified
D07141  Indobufen (INN) (P) unclassified
D07144  Dabigatran etexilate (USAN/INN); Pradaxa (TN) (P) Transporter inhibition: ABCB1
D07156  Alprenolol (INN) (P) unclassified
D07172  Mebutizide (INN) (P) unclassified
D07181  Mepindolol (INN) (P) unclassified
D07182  Tertatolol (INN) (P) unclassified
D07183  Cloranolol (INN) (P) unclassified
D07184  Talinolol (INN) (P) unclassified
D07185  Fendiline (INN) (P) unclassified
D07186  Ronifibrate (INN) (P) unclassified
D07187  Etofibrate (INN) (P) unclassified
D07188  Clofibride (INN) (P) unclassified
D07193  Flutrimazole (INN) (P) unclassified
D07201  Fluprednidene (INN) (P) unclassified
D07202  Halometasone (INN) (P) unclassified
D07203  Methylprednisolone aceponate (INN); Advantan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07219  Flunoxaprofen (INN) (P) unclassified
D07230  Prednylidene (INN) (P) unclassified
D07242  Flurithromycin (INN) (P) unclassified
D07262  Mofebutazone (INN); Monazone (TN) (P) unclassified
D07263  Clofezone (JAN/INN); Clofezone dihydrate (P) unclassified
D07264  Bumadizone (INN) (P) unclassified
D07265  Lonazolac (INN) (P) unclassified
D07266  Oxametacin (INN) (P) unclassified
D07267  Droxicam (INN) (P) unclassified
D07268  Ibuproxam (INN); Ibudros (TN) (P) unclassified
D07269  Dexketoprofen (INN) (P) unclassified
D07290  Dipyrocetyl (INN) (P) unclassified
D07291  Benorilate (INN); Benorylate (P) unclassified
D07292  Guacetisal (INN); Prontomucil (TN) (P) unclassified
D07293  Imidazole salicylate (INN); Selezen (TN) (P) unclassified
D07298  Barbexaclone (INN); Maliasin (TN) (P) unclassified
D07299  Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07300  Beclamide (INN) (P) unclassified
D07421  Aloxiprin (INN); Superpyrin (TN) (P) unclassified
D07432  Streptoduocin (BAN); Streptomycin sulfate and dihydrostreptomycin sulfate (P) unclassified
D07436  Afelimomab (INN) (P) unclassified
D07443  Amfenac (INN) (P) unclassified
D07447  Amiloride (INN); Amiclaran (TN) (P) unclassified
D07450  Amlodipine (USP/INN); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07453  Amtolmetin guacil (INN); Artromed (TN) (P) unclassified
D07462  Arbekacin (INN) (P) unclassified
D07464  Paramethasone (INN); Dillar (TN) (P) unclassified
D07467  Paromomycin (INN); Paromomycin (TN) (P) unclassified
D07470  Astromicin (INN) (P) unclassified
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07474  Atorvastatin (INN); Lipitor (TN); Sortis (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D07486  Azithromycin (INN); Azasite (TN); Azithromycin (TN) (P) Transporter inhibition: ABCB1
D07488  Balsalazide (INN) (P) unclassified
D07494  Barnidipine (INN); Vasexten (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07495  Beclometasone (INN); Beclometason (TN) (P) unclassified
D07496  Befunolol (INN) (P) unclassified
D07497  Bekanamycin (INN); Kanamycin B (P) unclassified
D07499  Benazepril (INN); Benazepril Sandoz (TN); Forteekor [veterinary] (TN) (P) unclassified
D07503  Bendazac lysine (BAN); Bendalina (TN) (P) unclassified
D07509  Benidipine (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07510  Adomiparin (USAN); Semuloparin (USAN); Heparin (BAN); Enoxaparin; Bemiparin; Parnaparin; Nadroparin; Heparin (TN) (P) unclassified
D07516  Benzydamine (INN); Apo-Benzydamine (TN) (P) unclassified
D07517  Benzydamine salicylate; Fulgium (TN) (P) unclassified
D07520  Bepridil (INN); Bepadin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07526  Betaxolol (INN); Betaxolol (TN) (P) unclassified
D07529  Binifibrate (INN); Biniwas (TN) (P) unclassified
D07537  Bopindolol (INN); Sandonorm (TN) (P) unclassified
D07538  Bosentan (INN) (CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07541  Bromfenac (INN) (P) unclassified
D07545  Brovincamine (INN); Sarbromin (TN) (P) unclassified
D07549  Bumadizone calcium salt hemihydrate; Desflam (TN); Eumotol (TN) (P) unclassified
D07564  Allopurinol sodium; Aloprim (TN) (P) unclassified
D07569  Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07578  Eldecalcitol (JAN/INN); Edirol (TN) (P) unclassified
D07579  Aspirin calcium salt; Notras (TN) (P) unclassified
D07580  Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) (P) unclassified
D07581  Aspirin magnesium salt; Mobidin (TN) (P) unclassified
D07582  Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) (P) unclassified
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07590  Bupranolol (INN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP induction: CYP3A4
D07598  Butoconazole (INN); Gynofort (TN) (P) unclassified
D07608  Carazolol (INN); Conducton (TN); Suacron [veterinary] (TN) (P) unclassified
D07612  Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) (P) unclassified
D07624  Carteolol (INN) (P) unclassified
D07626  Caspofungin (INN); Cancidas (TN) (P) unclassified
D07660  Celiprolol (INN); Celiprolol PCH (TN) (P) unclassified
D07661  Cerivastatin (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07674  Chloramphenicol stearate; Quemicetina (TN) (P) unclassified
D07675  Chloramphenicol succinate; Chloramphenicol ICN (TN) (P) unclassified
D07676  Chlormidazole hydrochloride; Unfungicid (TN) (P) unclassified
D07682  Clazosentan sodium (JAN/USAN); Pivlaz (TN) (P) unclassified
D07699  Cilazapril (INN); Inhibace (TN) (P) unclassified
D07702  Ciprofloxacin lactate; Ciproxin (TN) (P) unclassified
D07710  Clarithromycin lactobionate; Klacid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07715  Clobetasol (INN); Clobecort Amex (TN) (P) unclassified
D07717  Clobetasone (INN) (P) unclassified
D07719  Clocortolone (INN) (P) unclassified
D07723  Clofibric acid (INN) (P) unclassified
D07724  Magnesium clofibrate (INN); Clofibric acid magnesium salt; Clofibrate Magnesico Chobet (TN) (P) unclassified
D07749  Cortisone (INN); Cortisone (TN) (P) unclassified
D07752  Croconazole (INN) (P) unclassified
D07781  Delapril (INN); Delaket (TN) (P) unclassified
D07796  Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07797  Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07798  Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07799  Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07800  Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07801  Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07802  Dexamethasone phosphate; Decadron-phosphate (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07811  Dibekacin (INN) (P) unclassified
D07816  Diclofenac (USAN/INN); Solaraze (TN); Zorvolex (TN) (P) unclassified
D07817  Diclofenac diethylamine; Voltaren Emulgel (TN) (P) unclassified
D07818  Diclofenac epolamine; Diclofenac hydroxyethylpyrrolidine; Flector (TN) (P) unclassified
D07819  Diclofenac calcium; Voltaren Actingo Extra (TN) (P) unclassified
D07824  Diethylamine salicylate; Algesal (TN) (P) unclassified
D07827  Diflorasone (INN); Murode (TN) (P) unclassified
D07840  Dihydrostreptomycin (INN) (P) unclassified
D07845  Diltiazem (INN); Surazem (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07866  Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07869  Donepezil (JAN/INN); Donaz (TN); Allydone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07882  Eberconazole (INN) (P) unclassified
D07884  Eberconazole nitrate; Ebernet (TN) (P) unclassified
D07886  Efonidipine (INN) (P) unclassified
D07888  Eltenac (INN); Telzenac (TN) (P) unclassified
D07892  Enalapril (INN); Enalapril (TN) (P) unclassified
D07909  Erythromycin thiocyanate; Erythrocin (TN) (P) unclassified
D07910  Erythromycin stinoprate (INN); Erysec (TN) (P) unclassified
D07916  Esmolol (INN) (P) unclassified
D07943  Fendiline hydrochloride; Sensit (TN) (P) unclassified
D07945  Fenfluramine (INN); Ponderax (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07967  Fludrocortisone (INN); Astonin-H (TN) (P) unclassified
D07971  Flunarizine (INN); Sibelium (TN) (P) unclassified
D07972  Fluocortin (INN) (P) unclassified
D07973  Fluocortolone 21-pivalate; Fluocortolone pivalate; Ultradil (TN) (P) unclassified
D07980  Fluprednidene acetate; Fluprednidene 21-acetate; Decoderm (TN) (P) unclassified
D07981  Fluticasone (INN); Fluticaps (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07983  Fluvastatin (INN); Fluvas (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07984  Fluvoxamine (INN) (P) CYP inhibition: CYP3A4
D07991  Fosfosal (INN); Aydolid (TN) (P) unclassified
D07992  Fosinopril (INN); Monopril (TN) (P) unclassified
D07993  Fosphenytoin (INN) (P) CYP induction: CYP3A4
D07994  Framycetin sulfate; Neomycin B sulfate; Isofra (TN) (P) unclassified
D07999  Sodium furosemide; Frosemide sodium; Lasix (TN) (P) unclassified
D08001  Furosemide diolamine; Furosemide diethanolamine salt; Nuriban (TN) (P) unclassified
D08009  Gallopamil (INN) (P) unclassified
D08013  Gentamicin (BAN); Gentamicin (TN) (P) unclassified
D08021  Glucametacin (INN); Glucametan (TN) (P) unclassified
D08032  Gusperimus (INN); 15-Deoxyspergualin (P) unclassified
D08050  Hydroxychloroquine (INN); Polirreumin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08058  Ibuprofen arginine salt; Zafen (TN) (P) unclassified
D08059  Ibuprofen sodium; Ibuprofen sodium anhydrous; Esprenit (TN) (P) unclassified
D08066  Imatinib (INN); Glamox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08067  Azilsartan medoxomil (USAN) (P) unclassified
D08068  Imidapril (INN); Hipertene (TN) (P) unclassified
D08074  Penbutolol (INN) (P) unclassified
D08078  Indenolol (INN) (P) unclassified
D08083  Vedolizumab (USAN); Vedolizumab (genetical recombination) (JAN); Entyvio (TN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08102  Ketoprofen lysine; Artrosilene (TN) (P) unclassified
D08103  Ketoprofen sodium; Orudis (TN) (P) unclassified
D08104  Ketorolac (INN); Toradol (TN) (P) unclassified
D08111  Lercanidipine (INN); Lercanil (TN) (P) unclassified
D08115  Levobunolol (INN) (P) unclassified
D08131  Lisinopril (INN); Zestril (TN) (P) unclassified
D08142  Lonazolac calcium salt; Argun (TN) (P) unclassified
D08146  Losartan (INN); Losartic (TN) (P) unclassified
D08147  Loteprednol (INN) (P) unclassified
D08149  Loxoprofen (INN) (P) unclassified
D08153  Mabuprofen (INN); Aldospray analgesico (TN) (P) unclassified
D08155  Manidipine (INN); Manidipine 6300; Artedil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08162  Meclofenamate sodium; Meclomen (TN) (P) unclassified
D08190  Dipyrone (BAN); Metamizole sodium; Vetalgin (TN) (P) unclassified
D08214  Metronidazole benzoate (USP); Elyzol (TN) (P) unclassified
D08217  Mibefradil (INN) (P) unclassified
D08219  Micronomicin (DCF) (P) unclassified
D08225  Moexipril (INN) (P) unclassified
D08227  Mometasone (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08260  Neomycin (INN); Fradiomycin; Neomycin; Kaomycine (TN) (P) unclassified
D08268  Netilmicin (INN); Netira (TN) (P) unclassified
D08270  Nicardipine (INN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08275  Niflumic acid (INN); Niflugel (TN) (P) unclassified
D08287  Norfloxacin nicotinate; Quinabic soluble powder (TN) [veterinary] (P) unclassified
D08295  Olsalazine (INN) (P) unclassified
D08296  Omoconazole (INN) (P) unclassified
D08313  Oxiconazole (INN) (P) unclassified
D08318  Oxprenolol (INN); Oxprenolol (TN) (P) unclassified
D08324  Oxyphenbutazone (INN); Reozon (TN); Oxyphenbutazone (TN) (P) unclassified
D08340  Perhexiline (INN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08363  Phenylbutazone calcium; Peralgin (TN) (P) unclassified
D08364  Phenylbutazone sodium; Ambene (TN) (P) unclassified
D08374  Piketoprofen (INN); Calmatel (TN) (P) unclassified
D08375  Piketoprofen hydrochloride; Triparsean (TN) (P) unclassified
D08410  Pravastatin (INN); Pravator (TN) (P) unclassified
D08412  Prednisolone pivalate; Prednisolone 21-pivalate; Ultracortenol (TN) (P) unclassified
D08413  Prednisolone sodium metazoate (USAN); Prednisolone metasulfobenzoate sodium; Prednisolone 21-(sodium 3-sulfobenzoate); Predenema (TN) (P) unclassified
D08414  Prednisolone 21-(sodium tetrahydrophthalate); Prednisolone sodium tetrahydrophthalate; Fenicort (TN) (P) unclassified
D08415  Prednisolone steaglate (BAN); Prednisolone 21-steaglate; Sintisone (TN) (P) unclassified
D08416  Prednisone acetate; Prednisone 21-acetate (P) unclassified
D08427  Proglumetacin (INN); Bruxel (TN) (P) unclassified
D08443  Propranolol (INN); Propranolol (TN) (P) unclassified
D08476  Resocortol (INN) (P) unclassified
D08478  Ribostamycin (INN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) CYP induction: CYP3A4
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08492  Rosuvastatin (INN); Creston (TN) (CI,P) unclassified
D08497  Rupatadine fumarate (JAN); Rinialer (TN); Rupafin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08501  Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) (P) unclassified
D08510  Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) (P) unclassified
D08525  Sotalol (INN); Darob mite (TN) (P) unclassified
D08526  Spectinomycin (INN); Adspec (TN); Prospec (TN) (P) unclassified
D08527  Spiramycin adipate; Rovamycina (TN); Spiramaicina (TN) (P) unclassified
D08528  Spiramycin embonate; Cofamix STS (TN) (P) unclassified
D08529  Spirapril (INN) (P) unclassified
D08531  Streptomycin (INN); Streptomycin (TN) (P) unclassified
D08535  Sulconazole (INN) (P) unclassified
D08554  Tacalcitol (INN); Bonalfa (TN) (P) unclassified
D08556  Tacrolimus (INN); Prograf (TN) (CI,P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4
D08566  Temocapril (INN) (P) unclassified
D08572  Tertatolol hydrochloride; Artex (TN) (P) unclassified
D08586  Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) (P) unclassified
D08588  Tiagabine (INN); Gabitril (TN) (P) unclassified
D08592  Tiaramide (INN) (P) unclassified
D08594  Ticlopidine (INN); Ticlopidin-Puren (TN) (P) unclassified
D08598  Tilisolol (INN) (P) unclassified
D08600  Timolol (INN); Timolol (TN); Betimol (TN) (P) unclassified
D08605  Tipranavir (INN); Aptivus (TN) (P) unclassified
D08610  Tixocortol (INN) (P) unclassified
D08630  Tribuzone (prop.INN); Benetazon (TN) (P) unclassified
D08657  Apricoxib (USAN/INN) (P) unclassified
D08660  Ulobetasol (INN); Halobetasol (P) unclassified
D08667  Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) (P) unclassified
D08686  Ziconotide acetate; Prialt (TN) (P) unclassified
D08688  Zofenopril (INN); Zofenil (TN) (P) unclassified
D08699  Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08776  Pneumococcal vaccine polyvalent; Pneumococcus vaccine; Pneumovax 23 (TN) (P) unclassified
D08777  Freeze-dried live attenuated varicella vaccine (CI) unclassified
D08804  Freeze-dried live attenuated measles-rubella combined vaccine; Mearubik (TN) (CI) unclassified
D08808  Anti-human thymocyte immunoglobulin, equine (JAN); Atgam (TN); Lymphoglobuline (TN) (P) unclassified
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08860  Apremilast (JAN/USAN); Otezla (TN) (P) unclassified
D08864  Azilsartan (JAN/USAN/INN); Azilva (TN) (P) unclassified
D08865  Azilsartan kamedoxomil (USAN); Edarbi (TN) (P) unclassified
D08879  Brivaracetam (JAN/USAN/INN); Briviact (TN) (P) unclassified
D08890  Choline fenofibrate (USAN/INN); Trilipix (TN) (P) unclassified
D08892  Clevidipine (USAN/INN); Clevidipine butyrate; Cleviprex (TN) (P) unclassified
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08964  Perampanel (USAN); Fycompa (TN) (P) unclassified
D08976  Pomalidomide (JAN/USAN/INN); Pomalyst (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09012  Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) Transporter inhibition: ABCB1
D09033  Voclosporin (JAN/USAN/INN); Lupkynis (TN) (P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4
D09190  Anti-human thymocyte immunoglobulin, rabbit (JAN); Thymoglobuline (TN) (P) unclassified
D09197  Valsartan and hydrochlorothiazide (JP18); Co-dio (TN) (P) unclassified
D09208  Cetilistat (JAN/USAN/INN); Oblean (TN) (P) unclassified
D09214  Ustekinumab (USAN/INN); Ustekinumab (genetical recombination) (JAN); Ustekinumab (genetical recombination) [Ustekinumab biosimilar 1] (JAN); Stelara (TN) (P) unclassified
D09215  Eslicarbazepine (USAN/INN) (P) CYP induction: CYP3A4
D09314  Ofatumumab (USAN/INN); Ofatumumab (genetical recombination) (JAN); Arzerra (TN); Kesimpta (TN) (P) unclassified
D09315  Canakinumab (USAN/INN); Canakinumab (genetical recombination) (JAN); Ilaris (TN) (P) unclassified
D09319  Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09360  Obeticholic acid (JAN/USAN/INN); Ocaliva (TN) (P) unclassified
D09394  Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) (P) CYP inhibition: CYP3A4
D09546  Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) (P) Transporter inhibition: ABCB1
D09568  Naproxcinod (USAN/INN) (P) unclassified
D09569  Ezogabine (USAN); Retigabine (INN); Potiga (TN) (P) unclassified
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) Transporter inhibition: ABCB1
D09587  Brentuximab vedotin (USAN/INN); Brentuximab vedotin (genetical recombination) (JAN); Adcetris (TN) (P) unclassified
D09588  Briakinumab (USAN/INN) (P) unclassified
D09594  Olmesartan medoxomil and azelnidipine; Rezaltas (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09595  Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) CYP induction: CYP3A4
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09642  Modithromycin (USAN/INN) (P) unclassified
D09669  Siltuximab (USAN/INN); Sylvant (TN) (P) unclassified
D09680  Teprotumumab (USAN/INN); Teprotumumab (genetical recombination) (JAN); Teprotumumab-trbw; Tepezza (TN) (P) unclassified
D09702  Albaconazole (USAN/INN) (P) unclassified
D09707  Dabigatran (USAN/INN) (P) Transporter inhibition: ABCB1
D09710  Edoxaban (USAN/INN) (P) Transporter inhibition: ABCB1
D09725  Emulsified influenza HA vaccine (A/H1N1); Arepanrix (H1N1) (TN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09733  Afatinib dimaleate (USAN); Afatinib maleate (JAN); Gilotrif (TN); Giotrif (TN) (P) Transporter inhibition: ABCB1
D09741  Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09743  Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09753  Saxagliptin hydrate (JAN); Onglyza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09760  Ibuprofen sodium (USAN); Ibuprofen sodium hydrate (P) unclassified
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09789  Kirenidipine hydrochloride (JAN) (P) unclassified
D09796  Hydrocortisone caproate (JAN) (P) unclassified
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09809  Tylosin acetate isovalerte (JAN) (P) unclassified
D09813  Lenalidomide hydrate (JAN); Revlimid (TN) (P) unclassified
D09843  Beradilol monoethyl maleate (JAN); TZC-5665 (P) unclassified
D09881  Cobicistat (JAN/USAN/INN); Tybost (TN) (P) Enzyme-Target: CYP3A4
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (CI,P) Transporter inhibition: ABCB1
D09919  Lenvatinib (USAN/INN) (P) Transporter inhibition: ABCB1
D09920  Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) (P) Transporter inhibition: ABCB1
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (P) unclassified
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (P) unclassified
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09967  Secukinumab (USAN/INN); Secukinumab (genetical recombination) (JAN); Cosentyx (TN) (P) unclassified
D09970  Tofacitinib (USAN); Tasocitinib (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09987  Vaniprevir (JAN/USAN/INN); Vanihep (TN) (CI) unclassified
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP induction: CYP3A4
D10001  Fingolimod (INN); Gilenya (TN) (P) unclassified
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10017  Naproxen etemesil (USAN) (P) unclassified
D10019  Panobinostat lactate (JAN); Farydak (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10021  Efinaconazole (JAN/USAN/INN); Clenafin (TN); Jublia (TN) (P) unclassified
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10032  Tylvalosin (USAN/INN) (P) unclassified
D10033  Tylosin tartrate (USP) (P) unclassified
D10034  Tylvalosin tartrate (USAN); Aiviosin [veterinary] (TN) (P) unclassified
D10061  Brodalumab (USAN); Brodalumab (genetical recombination) (JAN); Siliq (TN) (P) unclassified
D10071  Ixekizumab (USAN); Ixekizumab (genetical recombination) (JAN); Taltz (TN) (P) unclassified
D10080  Sirukumab (USAN); Sirukumab (genetical recombination) (JAN) (P) unclassified
D10081  Simeprevir (JAN/USAN) (P) Transporter inhibition: ABCB1
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10093  Asunaprevir (JAN/USAN); Sunvepra (TN) (CI) CYP induction: CYP3A4 / Transporter inhibition: ABCB1
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10135  Macitentan (JAN/USAN); Opsumit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D10147  Pasireotide (USAN) (P) unclassified
D10151  Plazomicin (USAN) (P) unclassified
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10172  Teriflunomide (USAN); Aubagio (TN) (P) unclassified
D10192  Recombinant adsorbed quadrivalent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil (TN); Silgard (TN) (P) unclassified
D10198  Calcipotriol hydrate (JAN); Calcipotriol monohydrate; Calcipotriene hydrate; Dovonex (TN) (P) unclassified
D10212  Recombinant adsorbed bivalent human papillomavirus-like particle vaccine (derived from Trichoplusia ni cells); Cervarix (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (P) unclassified
D10226  Sacubitril valsartan sodium hydrate (JAN); Sacubitril mixture with valsartan; Entresto (TN) (P) unclassified
D10243  Irbesartan and amlodipine besilate (JP18); Aimix (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10254  Esflurbiprofen (JAN) (P) unclassified
D10308  Baricitinib (JAN/USAN/INN); Olumiant (TN) (P) Transporter inhibition: ABCB1
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10385  Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10396  Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN); Ofev (TN) (P) Transporter inhibition: ABCB1
D10400  Tildrakizumab (USAN); Tildrakizumab (genetical recombination) (JAN); Tildrakizumab-asmn; Ilumya (TN) (P) unclassified
D10438  Guselkumab (USAN/INN); Guselkumab (genetical recombination) (JAN); Tremfya (TN) (P) unclassified
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10469  Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) (P) Transporter inhibition: ABCB1
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10492  Tildipirosin (USAN/INN); Zuprevo [veterinary] (TN) (P) unclassified
D10497  Pasireotide diaspartate; Signifor (TN) (P) unclassified
D10501  Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10505  Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D10506  Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10513  Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10519  Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10520  Rabeprazole, amoxicillin and metronidazole; Rabefine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10525  Valsartan and cilnidipine; Atedio (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10527  Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10528  Aldosterone (INN) (P) unclassified
D10533  Umeclidinium bromide and vilanterol; Anoro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10534  Calcipotriene and betamethasone dipropionate; Calcipotriol and betamethasone dipropionate; Dovobet (TN); Enstilar (TN); Taclonex (TN) (P) unclassified
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10556  Fimasartan (INN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10568  Pitavastatin calcium hydrate (JP18); Livalo (TN) (CI,P) unclassified
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10639  Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) (CI) Transporter inhibition: ABCB1
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10653  Peficitinib (USAN/INN) (P) unclassified
D10655  Plazomicin sulfate (USAN); Zemdri (TN) (P) unclassified
D10656  Polmacoxib (USAN/INN) (P) unclassified
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (CI,P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (P) unclassified
D10699  Cholic acid (JAN/USAN); Cholbam (TN) (P) unclassified
D10711  Pemafibrate (JAN); Parmodia (TN) (CI,P) unclassified
D10721  Peficitinib hydrobromide (JAN/USAN); Smyraf (TN) (P) unclassified
D10733  Talazoparib tosylate (USAN); Talazoparib tosilate (JAN); Talzenna (TN) (P) unclassified
D10745  Ombitasvir, paritaprevir and ritonavir; Technivie (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D10750  Isavuconazole (INN); Cresemba (TN) (P) unclassified
D10753  Atazanavir and cobicistat; Evotaz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (P) unclassified
D10756  Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) (P) unclassified
D10761  Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) unclassified
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10822  Ciprofloxacin hydrate (JAN); Ciprofloxacin hemiheptahydrate (P) unclassified
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (P) unclassified
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10871  Filgotinib (USAN/INN) (P) unclassified
D10872  Filgotinib hydrochloride (USAN) (P) unclassified
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10892  Esaxerenone (JAN/INN) (P) unclassified
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (P) unclassified
D10915  Cannabidiol (USAN/INN); CBD; Epidiolex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10930  Etrasimod (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10931  Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10944  Itacitinib (USAN/INN) (P) unclassified
D10945  Itacitinib adipate (JAN/USAN) (P) unclassified
D10967  Ozanimod hydrochloride (JAN/USAN); Zeposia (TN) (P) unclassified
D10968  Ozanimod (USAN/INN) (P) unclassified
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D10993  Tucidinostat (JAN/USAN/INN); Hiyasta (TN) (P) unclassified
D10994  Upadacitinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10995  Upadacitinib tartrate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11000  Vamorolone (USAN/INN); Agamree (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11014  Glecaprevir and pibrentasvir; Mavyret (TN) (P) Transporter inhibition: ABCB1
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11035  Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11052  Risankizumab (USAN/INN); Risankizumab (genetical recombination) (JAN); Risankizumab-rzaa; Skyrizi (TN) (P) unclassified
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11054  Ravulizumab (USAN/INN); Ravulizumab (genetical recombination) (JAN); Ultomiris (TN) (P) unclassified
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) unclassified
D11079  Satralizumab (USAN/INN); Satralizumab (genetical recombination) (JAN); satralizumab-mwge; Enspryng (TN) (P) unclassified
D11082  Anifrolumab (USAN); Anifrolumab (genetical recombination) (JAN); Anifrolumab-fnia; Saphnelo (TN) (P) unclassified
D11092  Pitavastatin magnesium; Zypitamag (TN) (CI,P) unclassified
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11095  Atorvastatin calcium propylene glycol solvate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D11106  Filgotinib maleate (JAN/USAN); Jyseleca (TN) (P) unclassified
D11120  Emapalumab (USAN/INN); Emapalumab (genetical recombination) (JAN); Emapalumab-lzsg; Gamifant (TN) (P) unclassified
D11123  Mirikizumab (USAN/INN); Mirikizumab (genetical recombination) (JAN); Mirikizumab-mrkz; Omvoh (TN) (P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11150  Cenobamate (USAN/INN); Xcopri (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11154  Diroximel fumarate (JAN/USAN/INN); Vumerity (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11204  Octreotide hydrochloride (USAN) (P) unclassified
D11215  Ponesimod (USAN/INN); Ponvory (TN) (P) unclassified
D11243  Ublituximab (USAN/INN); Briumvi (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (P) unclassified
D11397  Darvadstrocel (INN); Alofisel (TN) (P) unclassified
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11460  Siponimod (USAN/INN) (P) unclassified
D11470  Imlifidase (USAN/INN); Idefirix (TN) (P) unclassified
D11472  Remdesivir (JAN/USAN); Veklury (TN) (P) unclassified
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) Transporter inhibition: ABCB1
D11520  Ezetimibe and rosuvastatin; Roszet (TN); Rosuzet (TN) (CI) unclassified
D11525  Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) (P) unclassified
D11530  Sutimlimab (USAN/INN); Sutimlimab (genetical recombination) (JAN); Sutimlimab-jome; Enjaymo (TN) (P) unclassified
D11550  Bimekizumab (USAN/INN); Bimekizumab (genetical recombination) (JAN); Bimzelx (TN) (P) unclassified
D11565  Grazoprevir (USAN/INN); Grazoprevir anhydrous (CI) Transporter inhibition: ABCB1
D11568  Edoxaban tosylate (USAN) (P) Transporter inhibition: ABCB1
D11572  Beclomethasone dipropionate monohydrate; Beconase aq (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11580  Perindopril arginine (P) unclassified
D11584  Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) (P) unclassified
D11613  Pegcetacoplan (JAN/USAN/INN); Empaveli (TN) (P) unclassified
D11641  Danicopan (JAN/USAN/INN); Voydeya (TN) (P) unclassified
D11659  Tolvaptan sodium phosphate (JAN); Samtasu (TN) (P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1
D11696  Crovalimab (USAN/INN); Crovalimab (genetical recombination) (JAN); Piasky (TN) (P) unclassified
D11703  Opinercept (INN) (P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (P) unclassified
D11757  Inebilizumab (USAN/INN); Inebilizumab (genetical recombination) (JAN); Inebilizumab-cdon; Uplizna (TN) (P) unclassified
D11785  Oteseconazole (USAN/INN); Vivijoa (TN) (P) unclassified
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11815  Belumosudil (USAN) (P) unclassified
D11816  Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) (P) unclassified
D11817  Deucravacitinib (JAN/USAN); Sotyktu (TN) (P) unclassified
D11861  Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) (P) unclassified
D11862  Indacaterol and mometasone furoate; Atectura (TN) (P) unclassified
D11863  Human papillomavirus 9-valent vaccine, recombinant; Recombinant adsorbed 9-valent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil 9 (TN); Silgard 9 (TN) (P) unclassified
D11876  Efgartigimod alfa (USAN/INN); Efgartigimod alfa (genetical recombination) (JAN); Efgartigimod alfa-fcab; Vyvgart (TN) (P) unclassified
D11881  Amlodipine benzoate; Katerzia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) unclassified
D12015  St. John's wort; SJW (P) unclassified
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12066  Spesolimab (USAN/INN); Spesolimab (genetical recombination) (JAN); Spesolimab-sbzo; Spevigo (TN) (P) unclassified
D12182  Rozanolixizumab (USAN/INN); Rozanolixizumab (genetical recombination) (JAN); rozanolixizumab-noli; Rystiggo (TN) (P) unclassified
D12251  Iptacopan (USAN/INN) (P) unclassified
D12252  Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) (P) unclassified
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12311  Bortezomib hydrate (JAN) (P) unclassified
D12326  Opelconazole (USAN/INN) (P) unclassified
D12353  Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) (P) unclassified
D12356  Zilucoplan sodium (JAN); Zilbrysq (TN) (P) unclassified
D12357  Zilucoplan (USAN/INN) (P) unclassified
D12410  Landiolol (USAN/INN) (P) unclassified
D12438  Pitavastatin calcium and ezetimibe; Livazebe (TN) (CI) unclassified
D12487  Olokizumab (INN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (P) unclassified
D12595  Aspirin trelamine (USAN) (P) unclassified
D12596  Aspirin trelamine hydrochloride (USAN) (P) unclassified
D12597  Ibuprofen trelamine (USAN); Ibuprofen diethylaminoethyl ester (P) unclassified
D12598  Ibuprofen trelamine hydrochloride (USAN) (P) unclassified
D12609  Dasatinib laurylsulfate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12684  Efgartigimod alfa and hyaluronidase; Efgartigimod alfa (genetical recombination) and vorhyaluronidase alfa (genetical recombination); Efgartigimod alfa and hyaluronidase-qvfc; Vyvgard hytrulo (TN); Vyvdura (TN) (P) unclassified
D12747  Divozilimab (INN) (P) unclassified
D12748  Levilimab (INN) (P) unclassified
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4