C00304 |
Kanamycin |
(P) unclassified |
C01946 |
Oleandomycin; Amimycin; Landomycin; Matromycin; Romicil |
(P) unclassified |
C06456 |
Phosphonoformate; Foscarmet; Foscarnet |
(P) unclassified |
C07005 |
Flunisolide; Flunisolide anhydrous |
(P) unclassified |
C07051 |
Indinavir |
(P) unclassified |
C07370 |
Prednisone; 1,2-Dehydrocortisone; 17,21-Dihydroxypregna-1,4-diene-3,11,20-trione |
(P) unclassified |
D00058 |
gamma-Aminobutyric acid (JAN); Gammalon (TN) |
(P) unclassified |
D00063 |
Tobramycin (JP18/USP); Tobi (TN); Tobracin (TN); Tobrex (TN); Bethkis (TN) |
(P) unclassified |
D00088 |
Hydrocortisone (JP18/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) |
(P) unclassified |
D00104 |
Chloramphenicol (JP18/USP/INN); Amphicol (TN); Chloromycetin (TN); Econochlor (TN) |
(P) unclassified |
D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) |
(CI,P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4 |
D00109 |
Aspirin (JP18/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) |
(P) unclassified |
D00118 |
Naproxen (JP18/USP/INN); Naprosyn (TN) |
(P) unclassified |
D00120 |
Sulindac (JP18/USP/INN); Clinoril (TN) |
(P) unclassified |
D00126 |
Ibuprofen (JP18/USP/INN); Advil (TN); Motrin (TN) |
(P) unclassified |
D00127 |
Piroxicam (JP18/USP/INN); Feldene (TN) |
(P) unclassified |
D00129 |
Calcitriol (JAN/USP/INN); Rocaltrol (TN) |
(P) unclassified |
D00130 |
Diflunisal (JAN/USP/INN); Dolobid (TN) |
(P) unclassified |
D00132 |
Ketoprofen (JP18/USP/INN); Orudis (TN) |
(P) unclassified |
D00136 |
Haloperidol (JP18/USP/INN); Haldol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00140 |
Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) |
(P) unclassified |
D00141 |
Indomethacin (USP); Indometacin (JP18/INN); Aconip (TN); Indocin (TN) |
(P) unclassified |
D00142 |
Methotrexate (JP18/USP/INN); Otrexup (TN); Xatmep (TN) |
(P) unclassified |
D00151 |
Mefenamic acid (JP18/USP/INN); Ponstel (TN) |
(P) unclassified |
D00158 |
Tolmetin sodium (JAN/USP); Tolmetin sodium dihydrate; Tolectin (TN) |
(P) unclassified |
D00163 |
Chenodiol (USAN); Chenodeoxycholic acid (JP18/INN); Chenix (TN) |
(P) unclassified |
D00165 |
Hydrocortisone acetate (JP18/USP); Cortifoam (TN); U-cort (TN) |
(P) unclassified |
D00169 |
Meclofenamate sodium (USP); Meclofenamate sodium monohydrate; Meclomen (TN) |
(P) unclassified |
D00184 |
Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4 |
D00186 |
Ciprofloxacin (JP18/USP/INN); Cipro (TN); Otiprio (TN) |
(P) unclassified |
D00203 |
Amphotericin B (JP18/USP/INN); Ambisome (TN); Amphotec (TN); Fungizone (TN) |
(P) unclassified |
D00210 |
Norfloxacin (JP18/USP/INN); Noroxin (TN) |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
D00212 |
Vancomycin (USP); Vancocin (TN) |
(P) unclassified |
D00218 |
Acetazolamide (JP18/USP/INN); Diamox (TN) |
(P) unclassified |
D00224 |
Allopurinol (JP18/USP/INN); Zyloprim (TN) |
(P) unclassified |
D00235 |
Atenolol (JP18/USP/INN); Tenormin (TN) |
(P) unclassified |
D00238 |
Azathioprine (JP18/USP/INN); Azasan (TN); Imuran (TN); Jayempi (TN) |
(P) unclassified |
D00244 |
Betamethasone (JP18/USP/INN); Celestone (TN); Rinderon (TN) |
(P) unclassified |
D00246 |
Budesonide (JP18/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00251 |
Captopril (JP18/USP/INN); Apopril (TN); Capoten (TN) |
(P) unclassified |
D00252 |
Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00255 |
Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00276 |
Clarithromycin (JP18/USP/INN); Biaxin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00279 |
Clofibrate (JP18/USP/INN); Atromid-S (TN) |
(P) unclassified |
D00280 |
Clonazepam (JP18/USP/INN); Klonopin (TN) |
(P) unclassified |
D00282 |
Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) |
(P) CYP inhibition: CYP3A4 |
D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00285 |
Co-Trimoxazole (BAN); Sulfamethoxazole and trimethoprim; Bactrim (TN); Septra (TN) |
(P) unclassified |
D00289 |
Danazol (JP18/USP/INN); Danocrine (TN) |
(P) unclassified |
D00292 |
Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00293 |
Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00298 |
Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) Transporter inhibition: ABCB1 |
D00304 |
Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) |
(P) unclassified |
D00315 |
Etodolac (JP18/USP/INN); Lodine (TN) |
(P) unclassified |
D00319 |
Felodipine (JP18/USP/INN); Plendil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00322 |
Fluconazole (JP18/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
D00324 |
Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00325 |
Fluocinonide (JP18/USP/INN); Lidex (TN); Vanos (TN) |
(P) unclassified |
D00328 |
Flurandrenolide (USP); Fludroxycortide (JAN/INN); Cordran (TN) |
(P) unclassified |
D00330 |
Flurbiprofen (JP18/USP/INN); Ansaid (TN) |
(P) unclassified |
D00331 |
Furosemide (JP18/USP/INN); Frusemide; Lasix (TN) |
(P) unclassified |
D00333 |
Ganciclovir (JAN/USP/INN); Cytovene (TN); Vitrasert (TN); Zirgan (TN) |
(P) unclassified |
D00334 |
Gemfibrozil (JAN/USP/INN); Lopid (TN) |
(P) unclassified |
D00340 |
Hydrochlorothiazide (JP18/USP/INN); Esidrix (TN); Microzide (TN) |
(P) unclassified |
D00346 |
Isoniazid (JP18/USP/INN); Laniazid (TN) |
(P) unclassified |
D00349 |
Isradipine (USP/INN); Dynacirc (TN) |
(P) unclassified |
D00350 |
Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00351 |
Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00354 |
Lamotrigine (JAN/USP/INN); Lamictal (TN) |
(P) unclassified |
D00357 |
Losartan potassium (JP18/USP); Cozaar (TN) |
(P) unclassified |
D00359 |
Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00362 |
Lisinopril (USP); Lisinopril hydrate (JP18); Lisinopril dihydrate; Prinivil (TN); Zestril (TN) |
(P) unclassified |
D00369 |
Melphalan (JP18/USP/INN); Alkeran (TN) |
(P) unclassified |
D00371 |
Theophylline (JP18); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) |
(P) unclassified |
D00372 |
Thiabendazole (USP); Tiabendazole (JAN/INN); Mintezol (TN) |
(P) unclassified |
D00375 |
Mephenytoin (USP/INN); Mesantoin (TN) |
(P) unclassified |
D00377 |
Mesalamine (USP); Mesalazine (JP18/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) |
(P) unclassified |
D00378 |
Timolol (USAN); Timolol hemihydrate; Betimol (TN) |
(P) unclassified |
D00383 |
Trandolapril (JAN/USP/INN); Mavik (TN) |
(P) unclassified |
D00385 |
Triamcinolone (JP18/USP/INN); Aristocort (TN); Kenacort (TN) |
(P) unclassified |
D00386 |
Triamterene (JP18/USP/INN); Dyrenium (TN) |
(P) unclassified |
D00392 |
Trimethadione (JP18/INN); Tridione (TN) |
(P) unclassified |
D00399 |
Valproic acid (USP); Depakene (TN) |
(P) unclassified |
D00400 |
Valsartan (JP18/USP/INN); Diovan (TN) |
(P) unclassified |
D00404 |
Methsuximide (USP); Mesuximide (INN); Celontin (TN) |
(P) unclassified |
D00407 |
Methylprednisolone (JP18/USP/INN); Medrol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00409 |
Metronidazole (JP18/USP/INN); Flagyl (TN); Noritate (TN); Nuvessa (TN); Vandazole (TN) |
(P) unclassified |
D00416 |
Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) |
(P) unclassified |
D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
D00421 |
Ramipril (USP/INN); Altace (TN) |
(P) unclassified |
D00425 |
Nabumetone (JP18/USP/INN); Relafen (TN) |
(P) unclassified |
D00426 |
Risperidone (JP18/USP/INN); Risperdal (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
D00428 |
Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) |
(P) unclassified |
D00429 |
Saquinavir (JAN/USP/INN); Fortovase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D00432 |
Nadolol (JP18/USP/INN); Corgard (TN) |
(P) unclassified |
D00434 |
Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00437 |
Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00438 |
Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00442 |
Octreotide (USAN/INN) |
(P) unclassified |
D00443 |
Spironolactone (JP18/USP/INN); Aldactone (TN) |
(P) unclassified |
D00448 |
Sulfasalazine (USP/INN); Salazosulfapyridine (JP18); Azulfidine (TN) |
(P) unclassified |
D00452 |
Suprofen (JAN/USP/INN); Profenal (TN) |
(P) unclassified |
D00458 |
Quetiapine fumarate (JP18/USP); Seroquel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00459 |
Quinapril hydrochloride (JP18/USP); Accupril (TN) |
(P) unclassified |
D00463 |
Oxaprozin (JP18/USP/INN); Daypro (TN) |
(P) unclassified |
D00472 |
Prednisolone (JP18/USP/INN); Delta-cortef (TN) |
(P) unclassified |
D00473 |
Prednisone (USP); Prednisone monohydrate; Deltasone (TN); Meticorten (TN); Rayos (TN) |
(P) unclassified |
D00474 |
Primidone (JP18/USP/INN); Mysoline (TN) |
(P) unclassified |
D00476 |
Probucol (JP18/USP/INN); Lorelco (TN) |
(P) unclassified |
D00483 |
Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) |
(P) unclassified |
D00491 |
Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00495 |
Paramethadione (INN); Paradione (TN) |
(P) unclassified |
D00496 |
Penicillamine (JAN/USP/INN); Cuprimine (TN); Depen (TN) |
(P) unclassified |
D00504 |
Phenacemide (JAN/INN); Phenurone (TN) |
(P) unclassified |
D00506 |
Phenobarbital (JP18/USP/INN); Luminal (TN) |
(P) unclassified |
D00508 |
Phensuximide (USP/INN); Milontin (TN) |
(P) unclassified |
D00510 |
Phenylbutazone (JP18/USP/INN); Azolid (TN) |
(P) unclassified |
D00512 |
Phenytoin (JP18/USP/INN); Dilantin (TN) |
(P) unclassified |
D00513 |
Pindolol (JP18/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) |
(P) unclassified |
D00519 |
Chlorothiazide (JAN/USP/INN); Diuril (TN) |
(P) unclassified |
D00522 |
Candesartan (USAN/INN) |
(P) unclassified |
D00523 |
Irbesartan (JP18/USP/INN); Avapro (TN) |
(P) unclassified |
D00533 |
Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) |
(P) unclassified |
D00535 |
Vigabatrin (JAN/USP/INN); Sabril (TN) |
(P) unclassified |
D00536 |
Felbamate (USPINN); Felbatol (TN) |
(P) unclassified |
D00537 |
Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00538 |
Zonisamide (JP18/USP/INN); Excegran (TN) |
(P) unclassified |
D00539 |
Ethosuximide (JP18/USP/INN); Zarontin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00553 |
Prilocaine (USP/INN); Propitocaine (JAN) |
(P) unclassified |
D00554 |
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00556 |
Aminopyrine (JAN); Aminophenazone (INN) |
(P) unclassified |
D00563 |
Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00565 |
Fenofibrate (JP18/USP/INN); Antara (TN); Lipantil (TN); Lipofen (TN); Tricor (TN); Triglide (TN) |
(P) unclassified |
D00566 |
Sodium salicylate (JP18/USP); Salsonin (TN) |
(P) unclassified |
D00567 |
Celecoxib (JP18/USP/INN); Celebrex (TN); Onsenal (TN) |
(P) unclassified |
D00568 |
Rofecoxib (JAN/USAN/INN); Vioxx (TN) |
(P) unclassified |
D00570 |
Colchicine (JP18/USP); Colchicine (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D00578 |
Voriconazole (JP18/USP/INN); Vfend (TN) |
(P) unclassified |
D00579 |
Foscarnet sodium (USP/INN); Foscavir (TN) |
(P) unclassified |
D00594 |
Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) |
(P) unclassified |
D00597 |
Acebutolol hydrochloride (JP18/USP); Sectral (TN) |
(P) unclassified |
D00598 |
Betaxolol hydrochloride (JP18/USP); Betoptic (TN); Kerlone (TN) |
(P) unclassified |
D00599 |
Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) |
(P) unclassified |
D00601 |
Metoprolol tartrate (JP18/USP); Lopressor (TN) |
(P) unclassified |
D00602 |
Penbutolol sulfate (JP18/USP); Levatol (TN) |
(P) unclassified |
D00603 |
Timolol maleate (JP18/USP); Blocadren (TN); Istalol (TN); Timoptic (TN) |
(P) unclassified |
D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00615 |
Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00616 |
Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00617 |
Nicardipine hydrochloride (JP18/USAN); Cardene (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00618 |
Nisoldipine (JAN/USAN/INN); Sular (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00619 |
Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D00620 |
Benazepril hydrochloride (JAN/USP); Lotensin (TN) |
(P) unclassified |
D00621 |
Enalapril maleate (JP18/USP); Renivace (TN); Vasotec (TN) |
(P) unclassified |
D00622 |
Fosinopril sodium (USP); Monopril (TN) |
(P) unclassified |
D00623 |
Moexipril hydrochloride (USP); Univasc (TN) |
(P) unclassified |
D00624 |
Perindopril erbumine (JAN/USP); Aceon (TN) |
(P) unclassified |
D00626 |
Candesartan cilexetil (JP18/USP); Atacand (TN) |
(P) unclassified |
D00627 |
Telmisartan (JP18/USP/INN); Micardis (TN) |
(P) unclassified |
D00629 |
Nitrendipine (JP18/USAN/INN); Baypress (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00631 |
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00634 |
Bisoprolol fumarate (JP18/USP); Zebeta (TN) |
(P) unclassified |
D00635 |
Metoprolol succinate (USP); Toprol XL (TN) |
(P) unclassified |
D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00644 |
Esmolol hydrochloride (JAN/USP); Brevibloc (TN) |
(P) unclassified |
D00649 |
Amiloride hydrochloride (USP); Midamor (TN) |
(P) unclassified |
D00650 |
Bendroflumethiazide (JAN/USP/INN); Naturetin (TN) |
(P) unclassified |
D00651 |
Benzthiazide (JAN/INN); Exna (TN) |
(P) unclassified |
D00654 |
Hydroflumethiazide (JAN/USP/INN); Saluron (TN) |
(P) unclassified |
D00656 |
Methyclothiazide (JAN/USP/INN); Enduron (TN) |
(P) unclassified |
D00657 |
Polythiazide (JAN/USAN/INN); Renese (TN) |
(P) unclassified |
D00658 |
Trichlormethiazide (JP18/USP/INN); Naqua (TN) |
(P) unclassified |
D00661 |
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00670 |
Donepezil hydrochloride (JP18/USP); Aricept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00687 |
Salmeterol xinafoate (JAN/USP); Serevent (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00689 |
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18); Beclovent (TN); Qnasl (TN); Vanceril (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00690 |
Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) unclassified |
D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
D00708 |
Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) |
(P) unclassified |
D00709 |
Levetiracetam (JAN/USP/INN); Keppra (TN); E keppra (TN) |
(P) unclassified |
D00710 |
Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) |
(P) unclassified |
D00722 |
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18); Ditropan (TN); Gelnique (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00726 |
Metoclopramide (JP18/INN); Elieten (TN); Terperan (TN) |
(P) unclassified |
D00727 |
Olsalazine sodium (USAN); Dipentum (TN) |
(P) unclassified |
D00734 |
Ursodiol (USP); Ursodeoxycholic acid (JP18/INN); Actigall (TN); Urso (TN) |
(P) unclassified |
D00742 |
Etanercept (USAN/INN); Etanercept (genetical recombination) (JAN); Etanercept (genetical recombination) [Etanercept biosimilar 1] (JAN); Etanercept (genetical recombination) [Etanercept biosimilar 2] (JAN); Enbrel (TN) |
(P) unclassified |
D00749 |
Leflunomide (JAN/USP/INN); Arava (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00751 |
Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00752 |
Mycophenolate mofetil (JAN/USP); Cellcept (TN) |
(P) unclassified |
D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D00754 |
Thalidomide (JAN/USP/INN); Thalomid (TN); Thaled (TN) |
(P) unclassified |
D00780 |
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00809 |
Amitriptyline hydrochloride (JP18/USP); Elavil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00810 |
Choline salicylate (JAN/USAN/INN); Arthropan (TN) |
(P) unclassified |
D00813 |
Ketorolac tromethamine (USP); Acular (TN); Toradol (TN) |
(P) unclassified |
D00820 |
Trazodone hydrochloride (JAN/USP); Desyrel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00821 |
Venlafaxine hydrochloride (JAN/USP); Effexor (TN) |
(P) unclassified |
D00824 |
Fluvoxamine maleate (JP18/USP); Luvox (TN) |
(P) CYP inhibition: CYP3A4 |
D00827 |
Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) |
(P) unclassified |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
D00836 |
Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00851 |
Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) |
(P) unclassified |
D00854 |
Quinupristin and dalfopristin; Synercid (TN) |
(P) CYP inhibition: CYP3A4 |
D00865 |
Amikacin sulfate (JP18/USP); Amikin (TN) |
(P) unclassified |
D00866 |
Kanamycin sulfate (USP); Kanamycin monosulfate (JP18); Kantrex (TN) |
(P) unclassified |
D00867 |
Netilmicin sulfate (JAN/USP); Netromycin (TN) |
(P) unclassified |
D00868 |
Paromomycin sulfate (JAN/USP); Humatin (TN) |
(P) unclassified |
D00869 |
Spectinomycin hydrochloride (USP); Spectinomycin hydrochloride hydrate (JP18); Trobicin (TN) |
(P) unclassified |
D00880 |
Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) |
(P) unclassified |
D00881 |
Econazole nitrate (JAN/USP); Ecoza (TN); Spectazole (TN) |
(P) unclassified |
D00882 |
Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) |
(P) unclassified |
D00885 |
Oxiconazole nitrate (JAN/USAN); Oxistat (TN) |
(P) unclassified |
D00886 |
Sulconazole nitrate (JAN/USP); Exelderm (TN) |
(P) unclassified |
D00887 |
Atorvastatin calcium anhydorous; Lipitor (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D00888 |
Terconazole (USP/INN); Terazol 3 (TN) |
(P) unclassified |
D00889 |
Cerivastatin sodium (JAN/USAN); Baycol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00890 |
Tioconazole (JAN/USP/INN); Vagistat-1 (TN) |
(P) unclassified |
D00892 |
Fluvastatin sodium (JAN/USP); Lescol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00893 |
Pravastatin sodium (JP18/USP); CS-514; Pravachol (TN) |
(P) unclassified |
D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00903 |
Diclofenac potassium (USP); Cambia (TN); Cataflam (TN); Zipsor (TN) |
(P) unclassified |
D00904 |
Diclofenac sodium (JP18/USP); Solaraze (TN); Voltaren (TN) |
(P) unclassified |
D00926 |
Vancomycin hydrochloride (JP18/USP); Vancoled (TN); Vancocin (TN) |
(P) unclassified |
D00961 |
Bicalutamide (JP18/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
D00964 |
Letrozole (JAN/USP/INN); Femara (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00968 |
Fenoprofen calcium (JAN/USP); Nalfon (TN) |
(P) unclassified |
D00969 |
Meloxicam (JAN/USP/INN); Mobic (TN) |
(P) unclassified |
D00970 |
Naproxen sodium (USP); Anaprox (TN) |
(P) unclassified |
D00971 |
Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) |
(P) unclassified |
D00972 |
Betamethasone sodium phosphate (JP18/USP); Celestone (TN) |
(P) unclassified |
D00973 |
Cortisone acetate (JP18/USP); Cortone acetate (TN) |
(P) unclassified |
D00975 |
Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00976 |
Hydrocortisone cypionate |
(P) unclassified |
D00977 |
Hydrocortisone sodium phosphate (JP18/USP); Hydrocortone phosphate (TN) |
(P) unclassified |
D00978 |
Hydrocortisone sodium succinate (JP18/USP); A-hydrocort (TN); Solu-cortef (TN) |
(P) unclassified |
D00979 |
Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D00980 |
Prednisolone acetate (JP18/USP/INN); Econopred (TN); Pred forte (TN) |
(P) unclassified |
D00981 |
Prednisolone sodium phosphate (JP18/USP); Pediapred (TN) |
(P) unclassified |
D00982 |
Prednisolone tebutate (JAN/USP); Hydeltra-TBA (TN) |
(P) unclassified |
D00983 |
Triamcinolone acetonide (JP18/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) |
(P) unclassified |
D00984 |
Triamcinolone diacetate (JAN/USP); Aristocort (TN) |
(P) unclassified |
D00985 |
Triamcinolone hexacetonide (USP/INN); Aristospan (TN) |
(P) unclassified |
D00986 |
Fludrocortisone acetate (JP18/USP); Florinef acetate (TN) |
(P) unclassified |
D00992 |
Gold sodium thiomalate (USP); Sodium aurothiomalate (JP18); Myochrysine (TN) |
(P) unclassified |
D01025 |
Levobunolol hydrochloride (JAN/USP); Betagan (TN) |
(P) unclassified |
D01026 |
Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) |
(P) unclassified |
D01028 |
Ticlopidine hydrochloride (JP18/USP); Ticlid (TN) |
(P) unclassified |
D01037 |
1,4-Dimethyl-7-isopropylazulene (JAN); Guaiazulene; Azunol (TN) |
(P) unclassified |
D01049 |
Nimesulide (JAN/INN) |
(P) unclassified |
D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
D01063 |
Gentamicin sulfate (JP18/USP); Garamycin (TN); Gentacin (TN) |
(P) unclassified |
D01069 |
Cilazapril (USAN); Cilazapril hydrate (JP18); Inhibace (TN) |
(P) unclassified |
D01072 |
Chloramphenicol palmitate (JP18/USP); Chloromycetin palmitate (TN) |
(P) unclassified |
D01078 |
Telithromycin (JAN/USAN/INN); Ketek (TN) |
(P) unclassified |
D01087 |
Methyl salicylate (JP18/NF); Methyl salicylate (TN) |
(P) unclassified |
D01092 |
Lanoconazole (JP18/INN); Latoconazole; Astat (TN) |
(P) unclassified |
D01098 |
Maxacalcitol (JAN/USAN/INN); Oxarol (TN); Prezios (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01104 |
Barnidipine hydrochloride (JAN); Hypoca (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01115 |
Eplerenone (JP18/USAN/INN); Inspra (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01119 |
Temocapril hydrochloride (JP18/USAN); Acecol (TN) |
(P) unclassified |
D01122 |
Ibuprofen piconol (JP18/USAN); Staderm (TN) |
(P) unclassified |
D01125 |
Calcipotriene (USP); Calcipotriol (JAN); Dovonex (TN) |
(P) unclassified |
D01145 |
Azelnidipine (JP18/INN); Calblock (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01148 |
Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01154 |
Potassium acetate (JAN/USP); Potassium acetate (TN) |
(P) unclassified |
D01160 |
Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D01164 |
Aripiprazole (JAN/USP/INN); Abilify (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01173 |
Cilnidipine (JP18/INN); Atelec (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01176 |
Blonanserin (JAN/INN); AD 5423 |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01182 |
Alprenolol hydrochloride (JP18/USAN); Regletin (TN) |
(P) unclassified |
D01183 |
Tolfenamic acid (JAN/INN); Clotam (TN) |
(P) unclassified |
D01185 |
Protizinic acid (JAN/INN) |
(P) unclassified |
D01189 |
Metiazinic acid (JAN/INN) |
(P) unclassified |
D01190 |
Ethylphenacemide (JAN); Pheneturide (INN) |
(P) unclassified |
D01196 |
Acetazolamide sodium (JAN); Diamox (TN) |
(P) unclassified |
D01204 |
Olmesartan medoxomil (JP18/USP); Benicar (TN); Olmetec (TN) |
(P) Transporter inhibition: ABCB1 |
D01208 |
Aluminum clofibrate (JAN/INN); Alfibrate (TN) |
(P) unclassified |
D01212 |
Simfibrate (JAN/INN); Cholesolvin (TN) |
(P) unclassified |
D01213 |
Tolvaptan (JAN/USAN/INN); Samsca (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01229 |
Paramethasone acetate (JAN/USAN); Haldrone (TN) |
(P) unclassified |
D01235 |
Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01239 |
Prednisolone sodium succinate (JP18/USP); Kohakusanin (TN) |
(P) unclassified |
D01240 |
Deslanoside (JP18/USP/INN); Cedilanid-d (TN) |
(P) unclassified |
D01241 |
Penflutizide (JAN/INN) |
(P) unclassified |
D01243 |
Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) |
(P) unclassified |
D01246 |
Benzylhydrochlorothiazide (JAN); Behyd (TN) |
(P) unclassified |
D01247 |
Ethiazide (JAN/INN) |
(P) unclassified |
D01252 |
Alclofenac (JAN/USP/INN); Mervan (TN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01256 |
Cyclothiazide (JAN/USAN/INN); Anhydron (TN) |
(P) unclassified |
D01266 |
Difluprednate (JAN/USAN/INN); Durezol (TN) |
(P) unclassified |
D01267 |
Floctafenine (JAN/USAN/INN); Idarac (TN) |
(P) unclassified |
D01271 |
Bufexamac (JAN/INN); Anderm (TN) |
(P) unclassified |
D01272 |
Clobetasol propionate (JP18/USP); Clobex (TN); Cormax (TN); Olux (TN) |
(P) unclassified |
D01273 |
Clobetasone butyrate (JAN/USAN); Kindavate (TN) |
(P) unclassified |
D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01289 |
Suxibuzone (JAN/INN) |
(P) unclassified |
D01298 |
Potassium gluconate (JAN/USP); Gluconsan-K (TN) |
(P) unclassified |
D01300 |
Clinofibrate (JP18/INN); Lipoclin (TN) |
(P) unclassified |
D01303 |
Flunarizine hydrochloride (JAN/USAN) |
(P) unclassified |
D01305 |
Feprazone (JAN/INN) |
(P) unclassified |
D01308 |
Halcinonide (JAN/USP/INN); Halog (TN) |
(P) unclassified |
D01322 |
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01325 |
Tiaprofenic acid (JAN/INN); Surgam (TN) |
(P) unclassified |
D01327 |
Diflorasone diacetate (JP18/USP); Florone (TN); Psorcon (TN) |
(P) unclassified |
D01330 |
Clidanac (JAN/INN) |
(P) unclassified |
D01339 |
Midecamycin (JP18/INN); Medemycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01341 |
Tiaramide hydrochloride (JP18/USAN); Solantal (TN) |
(P) unclassified |
D01344 |
Fenbufen (JP18/USAN/INN) |
(P) unclassified |
D01350 |
Streptomycin sulfate (JP18/USP); Streptomycin sulfate (TN) |
(P) unclassified |
D01353 |
Emorfazone (JP18/INN); Pentoil (TN) |
(P) unclassified |
D01357 |
Betamethasone valerate (JP18/USP); Beta-Val (TN); Luxiq (TN); Rinderon-V (TN) |
(P) unclassified |
D01361 |
Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) |
(P) unclassified |
D01366 |
Bezafibrate (JP18/USAN/INN); Bezatol SR (TN) |
(P) unclassified |
D01367 |
Fluorometholone (JP18/USP/INN); NSC 33001; Fluor-op (TN); Fml (TN); Oxylone (TN) |
(P) unclassified |
D01370 |
Cladribine (JAN/USP/INN); Leustatin (TN); Mavenclad (TN) |
(P) unclassified |
D01372 |
Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01380 |
Isopropylantipyrine (JP18); Propyphenazone (INN); Yoshipyrin (TN) |
(P) unclassified |
D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) unclassified |
D01387 |
Amcinonide (JAN/USP/INN); Cyclocort (TN) |
(P) unclassified |
D01394 |
Epirizole (JP18/USAN); Mebron (TN) |
(P) unclassified |
D01397 |
Ampiroxicam (JP18/INN); Flucam (TN) |
(P) unclassified |
D01399 |
Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01402 |
Betamethasone acetate (JAN/USP) |
(P) unclassified |
D01410 |
Benzydamine hydrochloride (JAN/USAN); Tantum (TN) |
(P) unclassified |
D01418 |
Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01425 |
Lopinavir (JAN/USP/INN) |
(P) unclassified |
D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
D01434 |
Deprodone propionate (JAN); Allomidon (TN) |
(P) unclassified |
D01437 |
Nifenazone (JAN/INN) |
(P) unclassified |
D01441 |
Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01442 |
Hydrocortisone succinate (JP18) |
(P) unclassified |
D01454 |
Bupranolol hydrochloride (JP18) |
(P) unclassified |
D01464 |
Flumethasone pivalate (USP); Flumetasone pivalate (JAN/BAN); Locorten (TN) |
(P) unclassified |
D01466 |
Ethenzamide (JP18/INN); Ethenzamide (TN) |
(P) unclassified |
D01471 |
Esatenolol (JAN/INN); (S)-Atenolol |
(P) unclassified |
D01472 |
Tacalcitol hydrate (JP18); Bonalfa high (TN); Curatoderm (TN) |
(P) unclassified |
D01475 |
Flurbiprofen axetil (JAN); FP 83; Ropion (TN) |
(P) unclassified |
D01480 |
Isoconazole nitrate (JAN); Adestan-G (TN) |
(P) unclassified |
D01492 |
Bucumolol hydrochloride (JP18) |
(P) unclassified |
D01504 |
Bufetolol hydrochloride (JP18); Adobiol (TN) |
(P) unclassified |
D01510 |
Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01512 |
Befunolol hydrochloride (JAN); Bentos (TN) |
(P) unclassified |
D01513 |
Alminoprofen (JP18/INN); Minalfen (TN) |
(P) unclassified |
D01518 |
Alfacalcidol (JAN/INN); Alsiodol (TN) |
(P) unclassified |
D01523 |
Arbekacin sulfate (JP18); Habekacin (TN) |
(P) unclassified |
D01545 |
Aceclofenac (JAN/INN); Aceclofenac (TN) |
(P) unclassified |
D01547 |
Zaltoprofen (JP18/INN); CN 100; Peon (TN) |
(P) unclassified |
D01549 |
Imidapril hydrochloride (JP18); Tanatril (TN) |
(P) unclassified |
D01553 |
Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01557 |
Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) |
(P) unclassified |
D01562 |
Aranidipine (JAN/INN); Sapresta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01565 |
Indometacin farnesil (JAN); Infree (TN) |
(P) unclassified |
D01566 |
Gusperimus trihydrochloride (USAN); Gusperimus hydrochloride (JAN); Spanidin (TN) |
(P) unclassified |
D01567 |
Ketophenylbutazone (JAN); Kebuzone (INN) |
(P) unclassified |
D01578 |
Pranoprofen (JP18/INN); Elicapric (TN) |
(P) unclassified |
D01581 |
Flufenamic acid (JAN/USAN/INN); Arlef (TN) |
(P) unclassified |
D01582 |
Acemetacin (JP18/INN); Rantudil (TN) |
(P) unclassified |
D01583 |
Pirfenidone (JAN/USAN/INN); Esbriet (TN) |
(P) unclassified |
D01594 |
Bendazac (JAN/USAN/INN); Iwazac (TN) |
(P) unclassified |
D01604 |
Efonidipine hydrochloride ethanolate (JAN); Efonidipine hydrochloride ethanol; Efonidipine hydrochloride; NZ 105 ethanolate; Landel (TN) |
(P) unclassified |
D01614 |
Acetylkitasamycin (JP18); Neo-leucomycin H (TN) |
(P) unclassified |
D01615 |
Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01618 |
Neomycin sulfate (USP); Fradiomycin sulfate (JP18); Mycifradin (TN); Neo-fradin (TN); Sofratulle (TN) |
(P) unclassified |
D01619 |
Hydrocortisone butyrate (JP18/USP); Locoid (TN) |
(P) unclassified |
D01620 |
Neticonazole hydrochloride (JAN); Atolant (TN) |
(P) unclassified |
D01632 |
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01636 |
Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01637 |
Betamethasone dipropionate (JP18/USP); Diprolene (TN); Rinderon-DP (TN); Sernivo (TN) |
(P) unclassified |
D01656 |
Brovincamine fumarate (JAN); Sabromin (TN) |
(P) unclassified |
D01661 |
Bucolome (JAN/INN); Paramidin (TN) |
(P) unclassified |
D01662 |
Falecalcitriol (JAN/INN); Hornel (TN) |
(P) unclassified |
D01664 |
Omoconazole nitrate (JAN/USAN) |
(P) unclassified |
D01667 |
Delapril hydrochloride (JAN/USAN); Adecut (TN) |
(P) unclassified |
D01675 |
Felbinac (JP18/USAN/INN); Dolinac (TN); Felbinac (TN) |
(P) unclassified |
D01689 |
Loteprednol etabonate (JAN/USAN); Lotemax (TN) |
(P) unclassified |
D01693 |
Dehydrocholic acid (JP18/USP/INN); Purified dehydrocholic acid (JP18); Decholin (TN) |
(P) unclassified |
D01703 |
Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01706 |
Migrenin (JP18); Migrenin (TN) |
(P) unclassified |
D01708 |
Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01709 |
Loxoprofen sodium hydrate (JP18); Lorfenamin (TN); Loxonin (TN) |
(P) unclassified |
D01710 |
Roxithromycin (JP18/USAN/INN); Rulide (TN) |
(P) unclassified |
D01712 |
Theophylline sodium acetate (JAN) |
(P) unclassified |
D01718 |
Mofezolac (JAN/INN); Mofezolac (TN) |
(P) unclassified |
D01741 |
Celiprolol hydrochloride (JAN/USAN); Selectol (TN) |
(P) unclassified |
D01744 |
Brotizolam (JP18/USAN/INN); Lendormin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01745 |
Domperidone (JP18/USAN/INN); Motilium (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01753 |
Dibekacin sulfate (JP18); Panimycin (TN) |
(P) unclassified |
D01762 |
Dipyrone (USAN); Sulpyrine hydrate (JP18); Metamizole sodium salt monohydrate; Sulpyrine (TN) |
(P) unclassified |
D01764 |
Diflucortolone valerate (JP18); Afusona (TN) |
(P) unclassified |
D01765 |
Proglumetacin maleate (JAN); Miridacin (TN) |
(P) unclassified |
D01767 |
Tenoxicam (JAN/USAN/INN); Tilcotil (TN) |
(P) unclassified |
D01775 |
Bifonazole (JP18/USAN/INN); Mycospor (TN) |
(P) unclassified |
D01776 |
Antipyrine (JP18/USP); Phenazone (INN) |
(P) unclassified |
D01787 |
Sulthiame (USAN); Sultiame (JP18); Ospolot (TN) |
(P) unclassified |
D01788 |
Amfenac sodium (USAN); Amfenac sodium hydrate (JAN); Fenazox (TN) |
(P) unclassified |
D01794 |
Bopindolol malonate (JAN); Sandonorm (TN) |
(P) unclassified |
D01795 |
Tilisolol hydrochloride (JAN); Selecal (TN) |
(P) unclassified |
D01806 |
Oxprenolol hydrochloride (JP18/USP); Okuspurecol (TN) |
(P) unclassified |
D01811 |
Salicylamide (JAN/USP/INN); Salicylamide (TN) |
(P) unclassified |
D01820 |
Alclometasone dipropionate (JAN/USP); Aclovate (TN) |
(P) unclassified |
D01821 |
Micronomicin sulfate (JP18); Sagamicin (TN); Santemycin (TN) |
(P) unclassified |
D01823 |
Ufenamate (JAN/INN); Flufenamic acid butyl ester; Combec (TN) |
(P) unclassified |
D01825 |
Fluocinolone acetonide (JP18/USP/INN); Fluocet (TN); Retisert (TN); Synalar (TN) |
(P) unclassified |
D01826 |
Isepamicin sulfate (JP18); Isepacin (TN) |
(P) unclassified |
D01832 |
Modafinil (JAN/USP/INN); Provigil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01841 |
Felbinac ethyl (JAN); LM 001 |
(P) unclassified |
D01847 |
Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN) |
(P) unclassified |
D01849 |
Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) |
(P) unclassified |
D01851 |
Mepranoprofen arbamel (JAN); Y-23023 |
(P) unclassified |
D01862 |
Pitavastatin calcium (JAN); NK 104; Livalo (TN) |
(CI,P) unclassified |
D01865 |
Pelubiprofen (JAN/INN) |
(P) unclassified |
D01866 |
Lornoxicam (JAN/USAN/INN); Lorcam (TN) |
(P) unclassified |
D01868 |
Bekanamycin sulfate (JP18); AKM; Kanendomycin (TN) |
(P) unclassified |
D01874 |
Vedaprofen (JAN/USAN/INN) |
(P) unclassified |
D01881 |
Astromicin sulfate (JAN/USAN); Fortimicin (TN) |
(P) unclassified |
D01886 |
Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) |
(P) unclassified |
D01896 |
Cilostazol (JP18/USP/INN); Pletal (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01897 |
Rokitamycin (JAN/INN); Ricamycin (TN) |
(P) unclassified |
D01898 |
Haloperidol decanoate (JAN/USP); Halomonth (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01900 |
Alacepril (JP18/INN); Cetapril (TN) |
(P) unclassified |
D01908 |
Nilvadipine (JP18/USAN/INN); Nivadil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D01915 |
Rosuvastatin calcium (JP18/USP); ZD 4522; Crestor (TN) |
(CI,P) unclassified |
D01922 |
Pratosartan (JAN/INN); KD 3-671 |
(P) unclassified |
D01933 |
Vatanidipine hydrochloride (JAN); AE 0047; Calbren (TN) |
(P) unclassified |
D01943 |
Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) |
(P) unclassified |
D01948 |
Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01958 |
Indenolol hydrochloride (JP18) |
(P) unclassified |
D01963 |
Ibufenac (JAN/USAN/INN); Dytransin (TN) |
(P) unclassified |
D01966 |
Ezetimibe (JAN/USP/INN); Zetia (TN) |
(P) unclassified |
D01969 |
Gallopamil hydrochloride (JAN) |
(P) unclassified |
D01974 |
Tilmacoxib (JAN/USAN/INN) |
(P) unclassified |
D01975 |
Fentiazac (JAN/USAN/INN) |
(P) unclassified |
D01977 |
Gefitinib (JP18/USAN/INN); Iressa (TN) |
(P) unclassified |
D01980 |
Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) |
(P) CYP inhibition: CYP3A4 |
D01998 |
Prednisolone farnesylate (JAN); PNF 21; Farnerate (TN) |
(P) unclassified |
D02000 |
Kitasamycin tartrate (JP18); Leucomycin tartrate (TN) |
(P) unclassified |
D02002 |
Isoniazid sodium methanesulfonate hydrate (JAN); Isoniazid sodium methanesulfonate monohydrate; Isoniazid sodium methanesulfonate; IHMS; Neoiscotin (TN) |
(P) unclassified |
D02008 |
Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02009 |
Erythromycin lactobionate (JP18/USP); Erythrocin (TN) |
(P) unclassified |
D02032 |
Betamethasone butyrate propionate (JAN); Antebate (TN) |
(P) unclassified |
D02045 |
Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02060 |
Potassium chloride (JP18/USP); K-dur (TN); KCL (TN); Kaon-Cl (TN); Klor-con (TN); Klotrix (TN) |
(P) unclassified |
D02061 |
Cyclopenthiazide (JAN/USAN/INN); Navidrex (TN) |
(P) unclassified |
D02075 |
Sodium gualenate (INN); Sodium guaiazulenesulfonate; Azunol ST (TN) |
(P) unclassified |
D02077 |
Potassium bicarbonate (USP); Potassium hydrogencarbonate; Potassium hydrogen carbonate; K-vescent (TN) |
(P) unclassified |
D02081 |
Metipranolol hydrochloride; Optipranolol (TN) |
(P) unclassified |
D02082 |
Eprosartan mesylate (USAN); Teveten (TN) |
(P) unclassified |
D02096 |
Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) |
(P) CYP induction: CYP3A4 |
D02097 |
Tiagabine hydrochloride (USP); Gabitril (TN) |
(P) unclassified |
D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
D02110 |
Indomethacin sodium (USP); Indometacin sodium hydrate (JAN); Indomethacin sodium trihydrate; Indometacin sodium; Indocin I.V. (TN) |
(P) unclassified |
D02112 |
Heparin sodium (JP18/USP/INN); Parnaparin sodium (INN); Liquemin sodium (TN) |
(P) unclassified |
D02114 |
Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02115 |
Methotrexate sodium; Trexall (TN); Rasuvo (TN) |
(P) unclassified |
D02134 |
Azithromycin hydrate (JP18); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) |
(P) Transporter inhibition: ABCB1 |
D02142 |
Teicoplanin (JP18/USAN/INN); Tagocid (TN) |
(P) unclassified |
D02156 |
Prednisolone hemisuccinate (USP); Prednisolone succinate (JP18) |
(P) unclassified |
D02165 |
Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02169 |
Croconazole hydrochloride (JP18); Pilzcin (TN) |
(P) unclassified |
D02174 |
Dexamethasone acetate (JAN/USP); Decadronal (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02181 |
Sisomicin sulfate (JAN/USP); Siseptin (TN) |
(P) unclassified |
D02184 |
Erythromycin stearate (JP18/USP); Bristamycin (TN) |
(P) unclassified |
D02185 |
Chloramphenicol sodium succinate (JP18/USP); Chloromycetin succinate (TN) |
(P) unclassified |
D02186 |
Oleandomycin phosphate (JAN); Matromycin (TN) |
(P) unclassified |
D02209 |
Ribostamycin sulfate (JP18); Vistamycin (TN) |
(P) unclassified |
D02213 |
Metoclopramide hydrochloride (JAN); Metoclopramide dihydrochloride monohydrate; Primperan (TN); Reglan (TN) |
(P) unclassified |
D02216 |
Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP18); Ciloxan (TN); Cipro (TN); Proquin XR (TN) |
(P) unclassified |
D02219 |
Terbinafine hydrochloride (JP18/USP); Lamisil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02229 |
Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02250 |
Octreotide acetate (JAN); Octreotide diacetate; Sandostatin (TN) |
(P) unclassified |
D02258 |
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D02264 |
Dipotassium glycyrrhizinate (JAN); Glycyrrhizinate dipotassium; Neubormitin (TN) |
(P) unclassified |
D02267 |
Foscarnet sodium hydrate (JAN); Foscarnet sodium hexahydrate; Trisodium phosphonoformate hexahydrate; Foscavir (TN) |
(P) unclassified |
D02269 |
Kitasamycin (JP18/USAN); Leucomycin (TN) |
(P) unclassified |
D02286 |
Betamethasone benzoate (USP); Uticort (TN) |
(P) unclassified |
D02287 |
Clocortolone pivalate (USP); Cloderm (TN) |
(P) unclassified |
D02288 |
Hydrocortisone valerate (USP); Westcort (TN) |
(P) unclassified |
D02289 |
Medrysone (USAN); HMS (TN) |
(P) unclassified |
D02290 |
Flurbiprofen sodium (USP); Ocufen (TN) |
(P) unclassified |
D02322 |
Apramycin (USAN/INN) |
(P) unclassified |
D02338 |
Acebutolol (USAN/INN) |
(P) unclassified |
D02341 |
Meclofenamic acid (USAN/INN) |
(P) unclassified |
D02342 |
Bisoprolol (JAN/USAN/INN) |
(P) unclassified |
D02350 |
Fenoprofen (USAN/INN) |
(P) unclassified |
D02355 |
Tolmetin (USAN/INN) |
(P) unclassified |
D02356 |
Verapamil (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D02358 |
Metoprolol (USAN/INN) |
(P) unclassified |
D02372 |
Perospirone hydrochloride hydrate (JAN); Lullan (TN) |
(P) unclassified |
D02374 |
Metipranolol (USAN/INN) |
(P) unclassified |
D02375 |
Terbinafine (USAN/INN); Lamasil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02389 |
Primidolol (USAN/INN) |
(P) unclassified |
D02420 |
Acetylspiramycin (JP18); Spiramycin II; Acetylspiramycin (TN) |
(P) unclassified |
D02453 |
Flumethiazide (INN); Ademol (TN) |
(P) unclassified |
D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
D02490 |
Tylosin (USP/INN); TS; Tylan (TN) |
(P) unclassified |
D02492 |
Tilmicosin (USP/INN); TMS; Micotil (TN) |
(P) unclassified |
D02493 |
Tilmicosin phosphate (USAN); TP |
(P) unclassified |
D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) unclassified |
D02501 |
Caspofungin acetate (JAN/USAN); Cancidas (TN) |
(P) unclassified |
D02512 |
Dihydrostreptomycin sulfate (USP) |
(P) unclassified |
D02523 |
Erythromycin acistrate (USAN); Erasis (TN) |
(P) unclassified |
D02524 |
Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) |
(P) unclassified |
D02525 |
Erythromycin propionate (USAN) |
(P) unclassified |
D02537 |
Dronedarone (INN) |
(P) unclassified |
D02542 |
Tobramycin sulfate (USP); Nebcin (TN) |
(P) unclassified |
D02543 |
Amikacin (USP/INN) |
(P) unclassified |
D02544 |
Sisomicin (USAN/INN) |
(P) unclassified |
D02545 |
Isepamicin (USAN/INN) |
(P) unclassified |
D02554 |
Rifaximin (JAN/USAN/INN); Xifaxan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 / Transporter inhibition: ABCB1 |
D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D02556 |
Ravuconazole (prop.INN) |
(P) unclassified |
D02557 |
Chlormidazole (INN) |
(P) unclassified |
D02582 |
Fenticonazole (INN) |
(P) unclassified |
D02583 |
Fenticonazole nitrate (USAN); Lomexin (TN) |
(P) unclassified |
D02584 |
Aliconazole (INN) |
(P) unclassified |
D02585 |
Vibunazole; Bay N-7133 |
(P) unclassified |
D02586 |
Alteconazole (INN) |
(P) unclassified |
D02587 |
Metildigoxin (JP18); Lanirapid (TN) |
(P) Transporter inhibition: ABCB1 |
D02591 |
Dexamethasone acefurate (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02592 |
Dexamethasone beloxil (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02596 |
Tocilizumab (USAN/INN); Tocilizumab (genetical recombination) (JAN); Actemra (TN) |
(P) unclassified |
D02597 |
Adalimumab (USAN/INN); Adalimumab (genetical recombination) (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 1] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 2] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 3] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 4] (JAN); Adalimumab-adaz; Adalimumab-adbm; Adalimumab-afzb; Adalimumab-atto; Adalimumab-bwwd; Adalimumab-fkjp; Adalimumab-aaty; Adalimumab-aacf; Adalimumab-aqvh; Humira (TN); Abrilada (TN); Amjevita (TN); Cyltezo (TN); Hadlima (TN); Hyrimoz (TN) |
(P) unclassified |
D02598 |
Infliximab (USAN/INN); Infliximab (genetical recombination) (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 1] (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 2] (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 3] (JAN); Infliximab-dyyb; Infliximab-abda; Infliximab-axxq; Remicade (TN); Inflectra (TN); Renflexis (TN); Avsola (TN) |
(P) unclassified |
D02624 |
Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02629 |
Fluspirilene (USAN/INN); Imap (TN) |
(P) unclassified |
D02630 |
Penfluridol (USAN/INN); Semap (TN) |
(P) unclassified |
D02633 |
Lomerizine hydrochloride (JAN); Terranas (TN) |
(P) unclassified |
D02689 |
Ramelteon (JAN/USAN/INN); Rozerem (TN) |
(P) unclassified |
D02690 |
Cholestyramine resin (USP); Colestyramine (JAN/INN); Questran (TN) |
(P) unclassified |
D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
D02706 |
Sodium gualenate hydrate (JAN); Azulene sulfonate sodium hydrate; Sodium guaiazulene sulfonate; Azunol (TN) |
(P) unclassified |
D02709 |
Valdecoxib (USAN/INN); Bextra (TN) |
(P) unclassified |
D02714 |
Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D02715 |
Balsalazide disodium (USP); Colazide (TN) |
(P) unclassified |
D02732 |
Pranlukast hydrate (JP18); Onon (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02765 |
Adaprolol maleate (USAN) |
(P) unclassified |
D02766 |
Valpromide (INN); Depamide (TN) |
(P) unclassified |
D02800 |
Alefacept (USAN/INN); Amevive (TN) |
(P) unclassified |
D02802 |
Alemtuzumab (USAN/INN); Alemtuzumab (genetical recombination) (JAN); Campath (TN); Lemtrada (TN) |
(P) unclassified |
D02834 |
Alprenoxime hydrochloride (USAN) |
(P) unclassified |
D02838 |
Althiazide (USAN); Altizide (INN) |
(P) unclassified |
D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02910 |
Amiodarone (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02914 |
Amlodipine maleate (USAN); Amvaz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D02934 |
Anakinra (USAN/INN); Kineret (TN) |
(P) unclassified |
D02944 |
Anirolac (USAN/INN) |
(P) unclassified |
D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02980 |
Adomiparin sodium (USAN); Ardeparin sodium (USAN/INN); Semuloparin sodium (USAN/INN); Normiflo (TN) |
(P) unclassified |
D02994 |
Rituximab (USAN/INN); Rituximab (genetical recombination) (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 1] (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 2] (JAN); Rituximab-abbs; Rituximab-pvvr; Rituximab-arrx; Rituxan (TN); Riabni (TN); Truximab (TN) |
(P) unclassified |
D03023 |
Azaconazole (USAN/INN) |
(P) unclassified |
D03033 |
Azathioprine sodium (USP); Imuran (TN) |
(P) unclassified |
D03058 |
Basiliximab (USAN/INN); Basiliximab (genetical recombination) (JAN); Simulect (TN) |
(P) unclassified |
D03063 |
BCG vaccine (USP); Freeze-dried BCG vaccine (for percutaneous use) (JP18); BCG vaccine (TN) |
(CI) unclassified |
D03067 |
Belfosdil (USAN/INN) |
(P) unclassified |
D03068 |
Belimumab (USAN); Belimumab (genetical recombination) (JAN); Benlysta (TN); LymphoStat-B (TN) |
(P) unclassified |
D03077 |
Benazeprilat (USAN/INN) |
(P) unclassified |
D03080 |
Benoxaprofen (USAN/INN); Oraflex (TN) |
(P) unclassified |
D03098 |
Berythromycin (USAN/INN); Erythromycin B |
(P) unclassified |
D03104 |
Betamicin sulfate (USAN) |
(P) unclassified |
D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
D03150 |
Bortezomib (JAN/USAN/INN); Velcade (TN) |
(P) unclassified |
D03163 |
Bromfenac sodium (USAN); Bromfenac sodium hydrate (JP18); Bromfenac sodium sesquihydrate; Bromday (TN); Prolensa (TN); Xibrom (TN); Yellox (TN) |
(P) unclassified |
D03165 |
Bromocriptine (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03170 |
Bucindolol hydrochloride (USAN) |
(P) unclassified |
D03177 |
Bunolol hydrochloride (USAN) |
(P) unclassified |
D03189 |
Buthiazide (USAN); Butizide (INN) |
(P) unclassified |
D03190 |
Butikacin (USAN/INN) |
(P) unclassified |
D03198 |
Butoxamine hydrochloride (USAN) |
(P) unclassified |
D03203 |
Abatacept (USAN/INN); Abatacept (genetical recombination) (JAN); Orencia (TN) |
(P) unclassified |
D03204 |
Abetimus sodium (USAN) |
(P) unclassified |
D03208 |
Aliskiren (USAN/INN); Rasilez (TN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D03218 |
Axitinib (JAN/USAN); Inlyta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03222 |
Belatacept (USAN/INN); Nulojix (TN) |
(P) unclassified |
D03253 |
Brecanavir (USAN) |
(P) unclassified |
D03254 |
Flufenamate aluminum (JAN); Flufenamic acid aluminum; Opyrin (TN) |
(P) unclassified |
D03256 |
Valganciclovir hydrochloride (JAN/USP); Valcyte (TN) |
(P) unclassified |
D03260 |
Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03262 |
Kanamycin sulfate (JP18); Kanamycin sulfate (TN) |
(P) unclassified |
D03301 |
Prednisolone valerate acetate (JAN); PDL; Spirazon (TN) |
(P) unclassified |
D03325 |
Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03337 |
Reviparin sodium (JAN); Clivarine (TN) |
(P) unclassified |
D03353 |
Dalteparin sodium (JAN/USP/INN); Ardeparin sodium; Fragmin (TN) |
(P) unclassified |
D03363 |
Canrenone (USAN) |
(P) unclassified |
D03385 |
Carbaspirin calcium (USAN); Carbasalate calcium (INN) |
(P) unclassified |
D03410 |
Carprofen (USP/INN); Rimadyl (TN) |
(P) unclassified |
D03415 |
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03440 |
Ceronapril (USAN/INN) |
(P) unclassified |
D03441 |
Certolizumab pegol (USAN/INN); Certolizumab pegol (genetical recombination) (JAN); Cimzia (TN) |
(P) unclassified |
D03449 |
Cetamolol hydrochloride (USAN) |
(P) unclassified |
D03461 |
Chloramphenicol pantothenate complex (USAN/INN); Pantofenicol (TN) |
(P) unclassified |
D03471 |
Chlorothiazide sodium (USP); Diuril (TN) |
(P) unclassified |
D03489 |
Cicloprofen (USAN/INN) |
(P) unclassified |
D03490 |
Cicloprolol hydrochloride (USAN) |
(P) unclassified |
D03521 |
Ciprofibrate (USAN/INN) |
(P) unclassified |
D03526 |
Cisconazole (USAN/INN) |
(P) unclassified |
D03536 |
Clentiazem maleate (JAN/USAN) |
(P) unclassified |
D03540 |
Cliprofen (USAN/INN) |
(P) unclassified |
D03541 |
Clocortolone acetate (USAN) |
(P) unclassified |
D03560 |
Clopirac (USAN/INN) |
(P) unclassified |
D03561 |
Cloprednol (USAN/INN); Cloradryn (TN) |
(P) unclassified |
D03594 |
Cortivazol (USAN) |
(P) unclassified |
D03601 |
Crilvastatin (USAN/INN) |
(P) unclassified |
D03639 |
Daclizumab (USAN/INN); Zenapax (TN); Zinbryta (TN) |
(P) unclassified |
D03643 |
Dalvastatin (USAN/INN) |
(P) unclassified |
D03652 |
Darbufelone mesylate (USAN) |
(P) unclassified |
D03655 |
Darodipine (USAN/INN) |
(P) unclassified |
D03656 |
Darunavir (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
D03671 |
Deflazacort (USAN/INN); Emflaza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D03673 |
Deligoparin sodium (USAN/INN) |
(P) unclassified |
D03674 |
Enoxaparin sodium (JAN/USP/INN); Lovenox (TN) |
(P) unclassified |
D03689 |
Deracoxib (USAN) |
(P) unclassified |
D03696 |
Desonide (USP/INN); Desowen (TN); Verdeso (TN) |
(P) unclassified |
D03697 |
Desoximetasone (USP/INN); Topicort (TN) |
(P) unclassified |
D03710 |
Etoricoxib (USAN/INN) |
(P) unclassified |
D03712 |
Firocoxib (USAN/INN); Equioxx (TN) [veterinary] |
(P) unclassified |
D03714 |
Lumiracoxib (USAN/INN) |
(P) unclassified |
D03715 |
Dexibuprofen (USAN/INN) |
(P) unclassified |
D03716 |
Parecoxib (USAN/INN) |
(P) unclassified |
D03717 |
Parecoxib sodium (USAN); Dynastat (TN) |
(P) unclassified |
D03718 |
Dexibuprofen lysine (USAN); Dexibuprofen lysine monohydrate; Doctrin (TN) |
(P) unclassified |
D03727 |
Dexpemedolac (USAN/INN) |
(P) unclassified |
D03729 |
Dexpropranolol hydrochloride (USAN) |
(P) unclassified |
D03752 |
Quinapril (INN) |
(P) unclassified |
D03753 |
Perindopril (USAN/INN) |
(P) unclassified |
D03756 |
Indolapril hydrochloride (USAN) |
(P) unclassified |
D03758 |
Libenzapril (USAN/INN) |
(P) unclassified |
D03759 |
Diacetolol hydrochloride (USAN) |
(P) unclassified |
D03760 |
Pentopril (USAN/INN) |
(P) unclassified |
D03763 |
Pivopril (USAN/INN) |
(P) unclassified |
D03765 |
Spirapril hydrochloride (USAN); Renormax (TN) |
(P) unclassified |
D03767 |
Zofenopril calcium (USAN); Zoprace (TN) |
(P) unclassified |
D03769 |
Enalaprilat (USP); Enalaprilat dihydrate; Vasotec (TN) |
(P) unclassified |
D03772 |
Fosinoprilat (USAN/INN) |
(P) unclassified |
D03773 |
Quinaprilat (USAN/INN) |
(P) unclassified |
D03775 |
Spiraprilat (USAN/INN) |
(P) unclassified |
D03776 |
Zofenoprilat arginine (USAN) |
(P) unclassified |
D03799 |
Dienogest (JAN/USAN/INN); Endometrion (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03812 |
Diflucortolone (USAN) |
(P) unclassified |
D03813 |
Diflucortolone pivalate (USAN) |
(P) unclassified |
D03816 |
Tenivastatin calcium (USAN) |
(P) unclassified |
D03820 |
Dutasteride (JAN/USP/INN); Avodart (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03830 |
Diltiazem malate (USAN); Tiamate (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D03839 |
Droxinavir hydrochloride (USAN) |
(P) unclassified |
D03840 |
Palinavir (USAN/INN) |
(P) unclassified |
D03842 |
Telinavir (USAN/INN) |
(P) unclassified |
D03843 |
Tipranavir disodium (USAN) |
(P) unclassified |
D03844 |
Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) |
(P) unclassified |
D03846 |
Dimethyl fumarate (JAN/USAN); Tecfidera (TN) |
(P) unclassified |
D03865 |
Dirithromycin (USP/INN); Dynabac (TN) |
(P) unclassified |
D03883 |
Doconazole (USAN/INN) |
(P) unclassified |
D03914 |
Dronedarone hydrochloride (USP); Multaq (TN) |
(P) unclassified |
D03936 |
Econazole (USAN/INN) |
(P) unclassified |
D03940 |
Eculizumab (USAN/INN); Eculizumab (genetical recombination) (JAN); Soliris (TN) |
(P) unclassified |
D03959 |
Efalizumab (USAN/INN); Raptiva (TN) |
(P) unclassified |
D03960 |
Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) |
(P) unclassified |
D03978 |
Eltrombopag olamine (JAN/USAN); Promacta (TN) |
(P) unclassified |
D03997 |
Enilconazole (USAN/INN) |
(P) unclassified |
D04003 |
Enolicam sodium (USAN); Enolicam sodium monohydrate |
(P) unclassified |
D04023 |
Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D04033 |
Epithiazide (USAN); Epitizide (INN) |
(P) unclassified |
D04040 |
Eprosartan (USAN/INN) |
(P) unclassified |
D04054 |
Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate |
(P) unclassified |
D04059 |
Mepenzolate bromide and phenobarbital; Trancolon P (TN) |
(P) unclassified |
D04102 |
Etofenamate (USAN/INN) |
(P) unclassified |
D04112 |
Etravirine (JAN/USAN/INN); Intelence (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D04126 |
Saralasin acetate (USAN); Sarenin (TN) |
(P) unclassified |
D04142 |
Fenclofenac (USAN/INN) |
(P) unclassified |
D04144 |
Fenclorac (USAN/INN) |
(P) unclassified |
D04145 |
Fendosal (USAN/INN); Alnovin (TN) |
(P) unclassified |
D04148 |
Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04187 |
Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) |
(P) unclassified |
D04190 |
Flestolol sulfate (USAN) |
(P) unclassified |
D04193 |
Flordipine (USAN/INN) |
(P) unclassified |
D04201 |
Flucloronide (USAN); Fluclorolone acetonide (INN) |
(P) unclassified |
D04206 |
Flufenisal (USAN/INN) |
(P) unclassified |
D04208 |
Flumethasone (USAN); Flumetasone (INN) |
(P) unclassified |
D04214 |
Flunisolide acetate (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04217 |
Fluocortin butyl (USAN) |
(P) unclassified |
D04218 |
Fluocortolone (USAN/INN) |
(P) unclassified |
D04219 |
Fluocortolone caproate (USAN) |
(P) unclassified |
D04221 |
Fluorometholone acetate (USP); Fluorometholone 17-acetate; Flarex (TN) |
(P) unclassified |
D04225 |
Fluperolone acetate (USAN); Methral (TN) |
(P) unclassified |
D04243 |
Forasartan (USAN/INN) |
(P) unclassified |
D04244 |
Formocortal (USAN/INN); Deflamene (TN) |
(P) unclassified |
D04260 |
Fostedil (USAN/INN) |
(P) unclassified |
D04273 |
Furaprofen (USAN/INN) |
(P) unclassified |
D04277 |
Furobufen (USAN/INN) |
(P) unclassified |
D04300 |
Ganaxolone (USAN/INN); Ztalmy (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04301 |
Ganciclovir sodium (USAN); Cytovene IV (TN) |
(P) unclassified |
D04358 |
Golimumab (USAN/INN); Golimumab (genetical recombination) (JAN); Simponi (TN) |
(P) unclassified |
D04409 |
Halobetasol propionate (USP); Ulobetasol propionate; Ultravate (TN) |
(P) unclassified |
D04411 |
Halofenate (USAN/INN) |
(P) unclassified |
D04427 |
Heparin calcium (JP18); Nadroparin calcium (INN); Calciparin; Calciparine (TN) |
(P) unclassified |
D04446 |
Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04447 |
Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04463 |
Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04467 |
Hydrocortisone hemisuccinate (USP) |
(P) unclassified |
D04482 |
Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) |
(P) unclassified |
D04483 |
Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) |
(P) unclassified |
D04484 |
Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) |
(P) unclassified |
D04489 |
Ibritumomab tiuxetan (USAN/INN); Ibritumomab tiuxetan (genetical recombination) (JAN); Zevalin (TN) |
(P) unclassified |
D04490 |
Ibuprofen aluminum (USAN) |
(P) unclassified |
D04530 |
Indoprofen (USAN/INN) |
(P) unclassified |
D04536 |
Influenza virus vaccine (USP); FluShield (TN); Fluarix quadrivalent (TN) |
(P) unclassified |
D04624 |
Isoconazole (USAN/INN) |
(P) unclassified |
D04638 |
Isoxepac (USAN/INN); Artil (TN) |
(P) unclassified |
D04639 |
Isoxicam (USAN/INN); Maxicam (TN) |
(P) unclassified |
D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04657 |
Lacidipine (USAN/INN); Motens (TN) |
(P) unclassified |
D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
D04687 |
Lenalidomide (JAN/USAN/INN); Revlimid (TN) |
(P) unclassified |
D04710 |
Levobetaxolol hydrochloride (USAN); Betaxon (TN) |
(P) unclassified |
D04725 |
Lexithromycin (USAN/INN) |
(P) unclassified |
D04733 |
Lidoflazine (USAN/INN); Angex (TN) |
(P) unclassified |
D04736 |
Lifibrate (USAN/INN) |
(P) unclassified |
D04737 |
Lifibrol (USAN/INN) |
(P) unclassified |
D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(CI,P) unclassified |
D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D04863 |
Mavacoxib (USAN) |
(P) unclassified |
D04866 |
Freeze-dried live attenuated measles vaccine (JP18) |
(CI) unclassified |
D04888 |
Medroxalol (USAN/INN) |
(P) unclassified |
D04889 |
Medroxalol hydrochloride (USAN) |
(P) unclassified |
D04896 |
Megalomicin potassium phosphate (USAN) |
(P) unclassified |
D04948 |
Potassium L-aspartate (JAN); Potassium aspartate; L-Aspartate potassium; Aspara K (TN) |
(P) unclassified |
D04952 |
Potassium aspartate and magnesium aspartate (JAN/USAN); Aspara (TN) |
(P) unclassified |
D04976 |
Methalthiazide (USAN) |
(P) unclassified |
D04977 |
Parnaparin sodium (JP18); Lowhepa (TN) |
(P) unclassified |
D05000 |
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D05001 |
Methylprednisolone sodium phosphate (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D05002 |
Methylprednisolone suleptanate (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D05008 |
Metoclopramide hydrochloride (USP); Metoclopramide monohydrochloride monohydrate; Clopra (TN); Reglan (TN) |
(P) unclassified |
D05011 |
Metoprolol fumarate (USP); Lopressor (TN) |
(P) unclassified |
D05016 |
Metronidazole hydrochloride (USAN); Flagyl I.V. (TN) |
(P) unclassified |
D05017 |
Metronidazole phosphate (USAN) |
(P) unclassified |
D05024 |
Mibefradil dihydrochloride (USAN); Posicor (TN) |
(P) unclassified |
D05089 |
Freeze-dried live attenuated mumps vaccine (JP18); Freeze-dried live attenuated mumps vaccine (TN) |
(CI) unclassified |
D05092 |
Muromonab-CD3 (JAN/USAN/INN); Orthoclone okt3 (TN) |
(P) unclassified |
D05094 |
Mycophenolate mofetil hydrochloride (USAN); Cellcept (TN) |
(P) unclassified |
D05095 |
Mycophenolate sodium (USP); Myfortic (TN) |
(P) unclassified |
D05096 |
Mycophenolic acid (USAN/INN); Mycophenolic acid (TN) |
(P) unclassified |
D05102 |
Nafenopin (USAN/INN) |
(P) unclassified |
D05121 |
Naproxol (USAN/INN) |
(P) unclassified |
D05127 |
Nebivolol (USAN/INN) |
(P) unclassified |
D05128 |
Nebramycin (USAN) |
(P) unclassified |
D05140 |
Framycetin (INN); Fradiomycin B; Neomycin B; FRM |
(P) unclassified |
D05141 |
Neomycin palmitate (USAN) |
(P) unclassified |
D05142 |
Neomycin undecylenate (USAN) |
(P) unclassified |
D05143 |
Nepafenac (JAN/USAN/INN); Nevanac (TN) |
(P) unclassified |
D05153 |
Neutramycin (USAN) |
(P) unclassified |
D05181 |
Aspirin aluminum (JP18) |
(P) unclassified |
D05182 |
Influenza HA vaccine (JP18) |
(P) unclassified |
D05218 |
Ocrelizumab (USAN); Ocrelizumab (genetical recombination) (JAN); Ocrevus (TN) |
(P) unclassified |
D05230 |
Octreotide pamoate (USAN) |
(P) unclassified |
D05246 |
Olmesartan (USAN/INN) |
(P) Transporter inhibition: ABCB1 |
D05248 |
Freeze-dried inactivated tissue culture ravies vaccine (JP18) |
(P) unclassified |
D05268 |
Orconazole nitrate (USAN) |
(P) unclassified |
D05319 |
Oxyphenbutazone hydrate; Tandearil (TN) |
(P) unclassified |
D05345 |
Pamatolol sulfate (USAN) |
(P) unclassified |
D05351 |
Josamycin propionate (JP18); Josamy (TN) |
(P) CYP inhibition: CYP3A4 |
D05367 |
Parconazole hydrochloride (USAN) |
(P) unclassified |
D05380 |
Pazopanib hydrochloride (JAN/USAN); Votrient (TN) |
(P) unclassified |
D05404 |
Pemedolac (USAN/INN) |
(P) unclassified |
D05425 |
Pentisomicin (USAN/INN) |
(P) unclassified |
D05429 |
Aminophylline hydrate (JP18) |
(P) unclassified |
D05442 |
Perhexiline maleate (USAN) |
(P) unclassified |
D05451 |
Phenbutazone sodium glycerate (USAN) |
(P) unclassified |
D05462 |
Oxycodone hydrochloride hydrate (JP18) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D05511 |
Piroxicam betadex (USAN) |
(P) unclassified |
D05512 |
Piroxicam cinnamate (USAN) |
(P) unclassified |
D05513 |
Piroxicam olamine (USAN) |
(P) unclassified |
D05515 |
Pirprofen (USAN/INN) |
(P) unclassified |
D05538 |
Mozenavir (INN) |
(P) unclassified |
D05544 |
Live oral polimyelitis vaccine (JAN); Poliovirus vaccine live oral; Orimune (TN) |
(CI) unclassified |
D05587 |
Practolol (USAN) |
(P) unclassified |
D05598 |
Pravadoline maleate (USAN) |
(P) unclassified |
D05601 |
Prednicarbate (USP/INN); Dermatop (TN) |
(P) unclassified |
D05619 |
Prodolic acid (USAN/INN) |
(P) unclassified |
D05621 |
Progabide (USAN/INN); Gabren (TN) |
(P) unclassified |
D05629 |
Propikacin (USAN) |
(P) unclassified |
D05640 |
Prorenoate potassium (USAN/INN) |
(P) unclassified |
D05713 |
Relomycin (USAN/INN) |
(P) unclassified |
D05717 |
Repromicin (USAN/INN) |
(P) unclassified |
D05719 |
Resocortol butyrate (USAN) |
(P) unclassified |
D05729 |
Rimexolone (USP/INN); Vexol (TN) |
(P) unclassified |
D05757 |
Rosaramicin (USAN/INN) |
(P) unclassified |
D05758 |
Rosaramicin butyrate (USAN) |
(P) unclassified |
D05759 |
Rosaramicin propionate (USAN) |
(P) unclassified |
D05760 |
Rosaramicin sodium phosphate (USAN) |
(P) unclassified |
D05761 |
Rosaramicin stearate (USAN) |
(P) unclassified |
D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
D05788 |
Salcolex (USAN); Salcolex tetrahydrate |
(P) unclassified |
D05789 |
Salethamide maleate (USAN) |
(P) unclassified |
D05791 |
Salicylate meglumine (USAN) |
(P) unclassified |
D05793 |
Salnacedin (USAN/INN) |
(P) unclassified |
D05800 |
Saperconazole (USAN/INN) |
(P) unclassified |
D05801 |
Saprisartan potassium (USAN) |
(P) unclassified |
D05811 |
Sedecamycin (USAN/INN) |
(P) unclassified |
D05830 |
Sermetacin (USAN/INN) |
(P) unclassified |
D05908 |
Spiramycin (JAN/USAN/INN); Rovamycin (TN) |
(P) unclassified |
D05912 |
Spiroxasone (USAN/INN) |
(P) unclassified |
D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D05937 |
Sudoxicam (USAN/INN) |
(P) unclassified |
D05995 |
Talmetacin (USAN/INN) |
(P) unclassified |
D05998 |
Talosalate (USAN/INN) |
(P) unclassified |
D06010 |
Tasosartan (USAN/INN) |
(P) unclassified |
D06060 |
Teludipine hydrochloride (USAN) |
(P) unclassified |
D06068 |
Temsirolimus (JAN/USAN/INN); Torisel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06076 |
Teprotide (USAN/INN) |
(P) unclassified |
D06082 |
Tesicam (USAN) |
(P) unclassified |
D06102 |
Theofibrate (USAN); Etofylline clofibrate (INN); Duolip (TN) |
(P) unclassified |
D06103 |
Theophylline (USP); Theophylline monohydrate; Accurbron (TN) |
(P) unclassified |
D06104 |
Theophylline sodium glycinate (USP); Asbron (TN) |
(P) unclassified |
D06133 |
Tibric acid (USAN/INN) |
(P) unclassified |
D06143 |
Tifurac sodium (USAN) |
(P) unclassified |
D06156 |
Tiopinac (USAN/INN) |
(P) unclassified |
D06171 |
Tixocortol pivalate (USAN) |
(P) unclassified |
D06199 |
Trabectedin (JAN/USAN/INN); Yondelis (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06209 |
Treloxinate (USAN/INN) |
(P) unclassified |
D06216 |
Triamcinolone acetonide sodium phosphate (USAN) |
(P) unclassified |
D06254 |
Trospectomycin sulfate (USAN) |
(P) unclassified |
D06258 |
Tulathromycin (JAN/USAN/INN) |
(P) unclassified |
D06273 |
Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06315 |
Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06347 |
Yellow fever vaccine (USP); YF-Vax (TN) |
(CI) unclassified |
D06363 |
Ziconotide (USAN/INN); Prialt (TN) |
(P) unclassified |
D06364 |
Zidometacin (USAN/INN) |
(P) unclassified |
D06373 |
Zinoconazole hydrochloride (USAN) |
(P) unclassified |
D06382 |
Zomepirac sodium (USAN); Zomepirac sodium dihydrate |
(P) unclassified |
D06390 |
Azithromycin (USP); Zmax (TN) |
(P) Transporter inhibition: ABCB1 |
D06398 |
Tinzaparin sodium (USAN); Innohep (TN) |
(P) unclassified |
D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06405 |
Nalfurafine hydrochloride (JAN/USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06412 |
Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06466 |
Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) |
(CI) unclassified |
D06475 |
Adsorbed hepatitis B vaccine (JP18); Bimmugen (TN) |
(P) unclassified |
D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D06495 |
Octreotide acetate (USP); Sandostatin (TN) |
(P) unclassified |
D06511 |
Freeze-dried smallpox vaccine prepared in cell culture (JP18) |
(CI) unclassified |
D06512 |
Freeze-dried live attenuated rubella vaccine (JP18) |
(CI) unclassified |
D06573 |
Carisbamate (USAN) |
(P) unclassified |
D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D06598 |
Gamithromycin (USAN/INN) |
(P) unclassified |
D06606 |
Ibuprofen lysine (USAN); Ibuprofen L-lysine (JAN); Solufenum; Neoprofen (TN) |
(P) unclassified |
D06622 |
Nebivolol hydrochloride (USAN); Bystolic (TN) |
(P) unclassified |
D06630 |
Pramiconazole (USAN/INN) |
(P) unclassified |
D06635 |
Rilonacept (USAN/INN); Arcalyst (TN) |
(P) unclassified |
D06637 |
Romidepsin (JAN/USAN/INN); Istodax (TN) |
(P) unclassified |
D06646 |
Epanolol (USAN/INN) |
(P) unclassified |
D06673 |
Meprednisone (USP/INN) |
(P) unclassified |
D06876 |
Hydrocortisone aceponate (INN); Efficort (TN) |
(P) unclassified |
D06883 |
Sertaconazole (INN) |
(P) unclassified |
D06886 |
Natalizumab (USAN/INN); Natalizumab (genetical recombination) (JAN); Tysabri (TN) |
(P) unclassified |
D07073 |
Dexamethasone cipecilate (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07077 |
Ambrisentan (JAN/INN); Letairis (TN); Volibris (TN) |
(P) unclassified |
D07082 |
Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) |
(CI,P) Transporter inhibition: ABCB1 |
D07116 |
Alclometasone (INN) |
(P) unclassified |
D07141 |
Indobufen (INN) |
(P) unclassified |
D07144 |
Dabigatran etexilate (USAN/INN); Pradaxa (TN) |
(P) Transporter inhibition: ABCB1 |
D07156 |
Alprenolol (INN) |
(P) unclassified |
D07172 |
Mebutizide (INN) |
(P) unclassified |
D07181 |
Mepindolol (INN) |
(P) unclassified |
D07182 |
Tertatolol (INN) |
(P) unclassified |
D07183 |
Cloranolol (INN) |
(P) unclassified |
D07184 |
Talinolol (INN) |
(P) unclassified |
D07185 |
Fendiline (INN) |
(P) unclassified |
D07186 |
Ronifibrate (INN) |
(P) unclassified |
D07187 |
Etofibrate (INN) |
(P) unclassified |
D07188 |
Clofibride (INN) |
(P) unclassified |
D07193 |
Flutrimazole (INN) |
(P) unclassified |
D07201 |
Fluprednidene (INN) |
(P) unclassified |
D07202 |
Halometasone (INN) |
(P) unclassified |
D07203 |
Methylprednisolone aceponate (INN); Advantan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07219 |
Flunoxaprofen (INN) |
(P) unclassified |
D07230 |
Prednylidene (INN) |
(P) unclassified |
D07242 |
Flurithromycin (INN) |
(P) unclassified |
D07262 |
Mofebutazone (INN); Monazone (TN) |
(P) unclassified |
D07263 |
Clofezone (JAN/INN); Clofezone dihydrate |
(P) unclassified |
D07264 |
Bumadizone (INN) |
(P) unclassified |
D07265 |
Lonazolac (INN) |
(P) unclassified |
D07266 |
Oxametacin (INN) |
(P) unclassified |
D07267 |
Droxicam (INN) |
(P) unclassified |
D07268 |
Ibuproxam (INN); Ibudros (TN) |
(P) unclassified |
D07269 |
Dexketoprofen (INN) |
(P) unclassified |
D07290 |
Dipyrocetyl (INN) |
(P) unclassified |
D07291 |
Benorilate (INN); Benorylate |
(P) unclassified |
D07292 |
Guacetisal (INN); Prontomucil (TN) |
(P) unclassified |
D07293 |
Imidazole salicylate (INN); Selezen (TN) |
(P) unclassified |
D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) unclassified |
D07299 |
Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07300 |
Beclamide (INN) |
(P) unclassified |
D07421 |
Aloxiprin (INN); Superpyrin (TN) |
(P) unclassified |
D07432 |
Streptoduocin (BAN); Streptomycin sulfate and dihydrostreptomycin sulfate |
(P) unclassified |
D07436 |
Afelimomab (INN) |
(P) unclassified |
D07443 |
Amfenac (INN) |
(P) unclassified |
D07447 |
Amiloride (INN); Amiclaran (TN) |
(P) unclassified |
D07450 |
Amlodipine (USP/INN); Norvasc (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07453 |
Amtolmetin guacil (INN); Artromed (TN) |
(P) unclassified |
D07462 |
Arbekacin (INN) |
(P) unclassified |
D07464 |
Paramethasone (INN); Dillar (TN) |
(P) unclassified |
D07467 |
Paromomycin (INN); Paromomycin (TN) |
(P) unclassified |
D07470 |
Astromicin (INN) |
(P) unclassified |
D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
D07474 |
Atorvastatin (INN); Lipitor (TN); Sortis (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D07486 |
Azithromycin (INN); Azasite (TN); Azithromycin (TN) |
(P) Transporter inhibition: ABCB1 |
D07488 |
Balsalazide (INN) |
(P) unclassified |
D07494 |
Barnidipine (INN); Vasexten (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07495 |
Beclometasone (INN); Beclometason (TN) |
(P) unclassified |
D07496 |
Befunolol (INN) |
(P) unclassified |
D07497 |
Bekanamycin (INN); Kanamycin B |
(P) unclassified |
D07499 |
Benazepril (INN); Benazepril Sandoz (TN); Forteekor [veterinary] (TN) |
(P) unclassified |
D07503 |
Bendazac lysine (BAN); Bendalina (TN) |
(P) unclassified |
D07509 |
Benidipine (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07510 |
Adomiparin (USAN); Semuloparin (USAN); Heparin (BAN); Enoxaparin; Bemiparin; Parnaparin; Nadroparin; Heparin (TN) |
(P) unclassified |
D07516 |
Benzydamine (INN); Apo-Benzydamine (TN) |
(P) unclassified |
D07517 |
Benzydamine salicylate; Fulgium (TN) |
(P) unclassified |
D07520 |
Bepridil (INN); Bepadin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07526 |
Betaxolol (INN); Betaxolol (TN) |
(P) unclassified |
D07529 |
Binifibrate (INN); Biniwas (TN) |
(P) unclassified |
D07537 |
Bopindolol (INN); Sandonorm (TN) |
(P) unclassified |
D07538 |
Bosentan (INN) |
(CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07541 |
Bromfenac (INN) |
(P) unclassified |
D07545 |
Brovincamine (INN); Sarbromin (TN) |
(P) unclassified |
D07549 |
Bumadizone calcium salt hemihydrate; Desflam (TN); Eumotol (TN) |
(P) unclassified |
D07564 |
Allopurinol sodium; Aloprim (TN) |
(P) unclassified |
D07569 |
Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07578 |
Eldecalcitol (JAN/INN); Edirol (TN) |
(P) unclassified |
D07579 |
Aspirin calcium salt; Notras (TN) |
(P) unclassified |
D07580 |
Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) |
(P) unclassified |
D07581 |
Aspirin magnesium salt; Mobidin (TN) |
(P) unclassified |
D07582 |
Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) |
(P) unclassified |
D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
D07590 |
Bupranolol (INN) |
(P) unclassified |
D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
D07598 |
Butoconazole (INN); Gynofort (TN) |
(P) unclassified |
D07608 |
Carazolol (INN); Conducton (TN); Suacron [veterinary] (TN) |
(P) unclassified |
D07612 |
Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) |
(P) unclassified |
D07624 |
Carteolol (INN) |
(P) unclassified |
D07626 |
Caspofungin (INN); Cancidas (TN) |
(P) unclassified |
D07660 |
Celiprolol (INN); Celiprolol PCH (TN) |
(P) unclassified |
D07661 |
Cerivastatin (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07674 |
Chloramphenicol stearate; Quemicetina (TN) |
(P) unclassified |
D07675 |
Chloramphenicol succinate; Chloramphenicol ICN (TN) |
(P) unclassified |
D07676 |
Chlormidazole hydrochloride; Unfungicid (TN) |
(P) unclassified |
D07682 |
Clazosentan sodium (JAN/USAN); Pivlaz (TN) |
(P) unclassified |
D07699 |
Cilazapril (INN); Inhibace (TN) |
(P) unclassified |
D07702 |
Ciprofloxacin lactate; Ciproxin (TN) |
(P) unclassified |
D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07715 |
Clobetasol (INN); Clobecort Amex (TN) |
(P) unclassified |
D07717 |
Clobetasone (INN) |
(P) unclassified |
D07719 |
Clocortolone (INN) |
(P) unclassified |
D07723 |
Clofibric acid (INN) |
(P) unclassified |
D07724 |
Magnesium clofibrate (INN); Clofibric acid magnesium salt; Clofibrate Magnesico Chobet (TN) |
(P) unclassified |
D07749 |
Cortisone (INN); Cortisone (TN) |
(P) unclassified |
D07752 |
Croconazole (INN) |
(P) unclassified |
D07781 |
Delapril (INN); Delaket (TN) |
(P) unclassified |
D07796 |
Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07797 |
Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07798 |
Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07799 |
Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07800 |
Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07801 |
Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07802 |
Dexamethasone phosphate; Decadron-phosphate (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07811 |
Dibekacin (INN) |
(P) unclassified |
D07816 |
Diclofenac (USAN/INN); Solaraze (TN); Zorvolex (TN) |
(P) unclassified |
D07817 |
Diclofenac diethylamine; Voltaren Emulgel (TN) |
(P) unclassified |
D07818 |
Diclofenac epolamine; Diclofenac hydroxyethylpyrrolidine; Flector (TN) |
(P) unclassified |
D07819 |
Diclofenac calcium; Voltaren Actingo Extra (TN) |
(P) unclassified |
D07824 |
Diethylamine salicylate; Algesal (TN) |
(P) unclassified |
D07827 |
Diflorasone (INN); Murode (TN) |
(P) unclassified |
D07840 |
Dihydrostreptomycin (INN) |
(P) unclassified |
D07845 |
Diltiazem (INN); Surazem (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07866 |
Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07869 |
Donepezil (JAN/INN); Donaz (TN); Allydone (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07882 |
Eberconazole (INN) |
(P) unclassified |
D07884 |
Eberconazole nitrate; Ebernet (TN) |
(P) unclassified |
D07886 |
Efonidipine (INN) |
(P) unclassified |
D07888 |
Eltenac (INN); Telzenac (TN) |
(P) unclassified |
D07892 |
Enalapril (INN); Enalapril (TN) |
(P) unclassified |
D07909 |
Erythromycin thiocyanate; Erythrocin (TN) |
(P) unclassified |
D07910 |
Erythromycin stinoprate (INN); Erysec (TN) |
(P) unclassified |
D07916 |
Esmolol (INN) |
(P) unclassified |
D07943 |
Fendiline hydrochloride; Sensit (TN) |
(P) unclassified |
D07945 |
Fenfluramine (INN); Ponderax (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07967 |
Fludrocortisone (INN); Astonin-H (TN) |
(P) unclassified |
D07971 |
Flunarizine (INN); Sibelium (TN) |
(P) unclassified |
D07972 |
Fluocortin (INN) |
(P) unclassified |
D07973 |
Fluocortolone 21-pivalate; Fluocortolone pivalate; Ultradil (TN) |
(P) unclassified |
D07980 |
Fluprednidene acetate; Fluprednidene 21-acetate; Decoderm (TN) |
(P) unclassified |
D07981 |
Fluticasone (INN); Fluticaps (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07983 |
Fluvastatin (INN); Fluvas (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D07984 |
Fluvoxamine (INN) |
(P) CYP inhibition: CYP3A4 |
D07991 |
Fosfosal (INN); Aydolid (TN) |
(P) unclassified |
D07992 |
Fosinopril (INN); Monopril (TN) |
(P) unclassified |
D07993 |
Fosphenytoin (INN) |
(P) CYP induction: CYP3A4 |
D07994 |
Framycetin sulfate; Neomycin B sulfate; Isofra (TN) |
(P) unclassified |
D07999 |
Sodium furosemide; Frosemide sodium; Lasix (TN) |
(P) unclassified |
D08001 |
Furosemide diolamine; Furosemide diethanolamine salt; Nuriban (TN) |
(P) unclassified |
D08009 |
Gallopamil (INN) |
(P) unclassified |
D08013 |
Gentamicin (BAN); Gentamicin (TN) |
(P) unclassified |
D08021 |
Glucametacin (INN); Glucametan (TN) |
(P) unclassified |
D08032 |
Gusperimus (INN); 15-Deoxyspergualin |
(P) unclassified |
D08050 |
Hydroxychloroquine (INN); Polirreumin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08058 |
Ibuprofen arginine salt; Zafen (TN) |
(P) unclassified |
D08059 |
Ibuprofen sodium; Ibuprofen sodium anhydrous; Esprenit (TN) |
(P) unclassified |
D08066 |
Imatinib (INN); Glamox (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08067 |
Azilsartan medoxomil (USAN) |
(P) unclassified |
D08068 |
Imidapril (INN); Hipertene (TN) |
(P) unclassified |
D08074 |
Penbutolol (INN) |
(P) unclassified |
D08078 |
Indenolol (INN) |
(P) unclassified |
D08083 |
Vedolizumab (USAN); Vedolizumab (genetical recombination) (JAN); Entyvio (TN) |
(P) unclassified |
D08095 |
Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08102 |
Ketoprofen lysine; Artrosilene (TN) |
(P) unclassified |
D08103 |
Ketoprofen sodium; Orudis (TN) |
(P) unclassified |
D08104 |
Ketorolac (INN); Toradol (TN) |
(P) unclassified |
D08111 |
Lercanidipine (INN); Lercanil (TN) |
(P) unclassified |
D08115 |
Levobunolol (INN) |
(P) unclassified |
D08131 |
Lisinopril (INN); Zestril (TN) |
(P) unclassified |
D08142 |
Lonazolac calcium salt; Argun (TN) |
(P) unclassified |
D08146 |
Losartan (INN); Losartic (TN) |
(P) unclassified |
D08147 |
Loteprednol (INN) |
(P) unclassified |
D08149 |
Loxoprofen (INN) |
(P) unclassified |
D08153 |
Mabuprofen (INN); Aldospray analgesico (TN) |
(P) unclassified |
D08155 |
Manidipine (INN); Manidipine 6300; Artedil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08162 |
Meclofenamate sodium; Meclomen (TN) |
(P) unclassified |
D08190 |
Dipyrone (BAN); Metamizole sodium; Vetalgin (TN) |
(P) unclassified |
D08214 |
Metronidazole benzoate (USP); Elyzol (TN) |
(P) unclassified |
D08217 |
Mibefradil (INN) |
(P) unclassified |
D08219 |
Micronomicin (DCF) |
(P) unclassified |
D08225 |
Moexipril (INN) |
(P) unclassified |
D08227 |
Mometasone (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08260 |
Neomycin (INN); Fradiomycin; Neomycin; Kaomycine (TN) |
(P) unclassified |
D08268 |
Netilmicin (INN); Netira (TN) |
(P) unclassified |
D08270 |
Nicardipine (INN); Cardene (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08275 |
Niflumic acid (INN); Niflugel (TN) |
(P) unclassified |
D08287 |
Norfloxacin nicotinate; Quinabic soluble powder (TN) [veterinary] |
(P) unclassified |
D08295 |
Olsalazine (INN) |
(P) unclassified |
D08296 |
Omoconazole (INN) |
(P) unclassified |
D08313 |
Oxiconazole (INN) |
(P) unclassified |
D08318 |
Oxprenolol (INN); Oxprenolol (TN) |
(P) unclassified |
D08324 |
Oxyphenbutazone (INN); Reozon (TN); Oxyphenbutazone (TN) |
(P) unclassified |
D08340 |
Perhexiline (INN) |
(P) unclassified |
D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) unclassified |
D08363 |
Phenylbutazone calcium; Peralgin (TN) |
(P) unclassified |
D08364 |
Phenylbutazone sodium; Ambene (TN) |
(P) unclassified |
D08374 |
Piketoprofen (INN); Calmatel (TN) |
(P) unclassified |
D08375 |
Piketoprofen hydrochloride; Triparsean (TN) |
(P) unclassified |
D08410 |
Pravastatin (INN); Pravator (TN) |
(P) unclassified |
D08412 |
Prednisolone pivalate; Prednisolone 21-pivalate; Ultracortenol (TN) |
(P) unclassified |
D08413 |
Prednisolone sodium metazoate (USAN); Prednisolone metasulfobenzoate sodium; Prednisolone 21-(sodium 3-sulfobenzoate); Predenema (TN) |
(P) unclassified |
D08414 |
Prednisolone 21-(sodium tetrahydrophthalate); Prednisolone sodium tetrahydrophthalate; Fenicort (TN) |
(P) unclassified |
D08415 |
Prednisolone steaglate (BAN); Prednisolone 21-steaglate; Sintisone (TN) |
(P) unclassified |
D08416 |
Prednisone acetate; Prednisone 21-acetate |
(P) unclassified |
D08427 |
Proglumetacin (INN); Bruxel (TN) |
(P) unclassified |
D08443 |
Propranolol (INN); Propranolol (TN) |
(P) unclassified |
D08476 |
Resocortol (INN) |
(P) unclassified |
D08478 |
Ribostamycin (INN) |
(P) unclassified |
D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
D08488 |
Amlodipine besilate and atorvastatin calcium; Caduet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08492 |
Rosuvastatin (INN); Creston (TN) |
(CI,P) unclassified |
D08497 |
Rupatadine fumarate (JAN); Rinialer (TN); Rupafin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08501 |
Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) |
(P) unclassified |
D08510 |
Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) |
(P) unclassified |
D08525 |
Sotalol (INN); Darob mite (TN) |
(P) unclassified |
D08526 |
Spectinomycin (INN); Adspec (TN); Prospec (TN) |
(P) unclassified |
D08527 |
Spiramycin adipate; Rovamycina (TN); Spiramaicina (TN) |
(P) unclassified |
D08528 |
Spiramycin embonate; Cofamix STS (TN) |
(P) unclassified |
D08529 |
Spirapril (INN) |
(P) unclassified |
D08531 |
Streptomycin (INN); Streptomycin (TN) |
(P) unclassified |
D08535 |
Sulconazole (INN) |
(P) unclassified |
D08554 |
Tacalcitol (INN); Bonalfa (TN) |
(P) unclassified |
D08556 |
Tacrolimus (INN); Prograf (TN) |
(CI,P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4 |
D08566 |
Temocapril (INN) |
(P) unclassified |
D08572 |
Tertatolol hydrochloride; Artex (TN) |
(P) unclassified |
D08586 |
Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) |
(P) unclassified |
D08588 |
Tiagabine (INN); Gabitril (TN) |
(P) unclassified |
D08592 |
Tiaramide (INN) |
(P) unclassified |
D08594 |
Ticlopidine (INN); Ticlopidin-Puren (TN) |
(P) unclassified |
D08598 |
Tilisolol (INN) |
(P) unclassified |
D08600 |
Timolol (INN); Timolol (TN); Betimol (TN) |
(P) unclassified |
D08605 |
Tipranavir (INN); Aptivus (TN) |
(P) unclassified |
D08610 |
Tixocortol (INN) |
(P) unclassified |
D08630 |
Tribuzone (prop.INN); Benetazon (TN) |
(P) unclassified |
D08657 |
Apricoxib (USAN/INN) |
(P) unclassified |
D08660 |
Ulobetasol (INN); Halobetasol |
(P) unclassified |
D08667 |
Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) |
(P) unclassified |
D08686 |
Ziconotide acetate; Prialt (TN) |
(P) unclassified |
D08688 |
Zofenopril (INN); Zofenil (TN) |
(P) unclassified |
D08699 |
Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08776 |
Pneumococcal vaccine polyvalent; Pneumococcus vaccine; Pneumovax 23 (TN) |
(P) unclassified |
D08777 |
Freeze-dried live attenuated varicella vaccine |
(CI) unclassified |
D08804 |
Freeze-dried live attenuated measles-rubella combined vaccine; Mearubik (TN) |
(CI) unclassified |
D08808 |
Anti-human thymocyte immunoglobulin, equine (JAN); Atgam (TN); Lymphoglobuline (TN) |
(P) unclassified |
D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08860 |
Apremilast (JAN/USAN); Otezla (TN) |
(P) unclassified |
D08864 |
Azilsartan (JAN/USAN/INN); Azilva (TN) |
(P) unclassified |
D08865 |
Azilsartan kamedoxomil (USAN); Edarbi (TN) |
(P) unclassified |
D08879 |
Brivaracetam (JAN/USAN/INN); Briviact (TN) |
(P) unclassified |
D08890 |
Choline fenofibrate (USAN/INN); Trilipix (TN) |
(P) unclassified |
D08892 |
Clevidipine (USAN/INN); Clevidipine butyrate; Cleviprex (TN) |
(P) unclassified |
D08923 |
Fesoterodine fumarate (JAN/USAN); Toviaz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D08964 |
Perampanel (USAN); Fycompa (TN) |
(P) unclassified |
D08976 |
Pomalidomide (JAN/USAN/INN); Pomalyst (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09012 |
Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(CI,P) Transporter inhibition: ABCB1 |
D09033 |
Voclosporin (JAN/USAN/INN); Lupkynis (TN) |
(P) Enzyme: CYP3A4 / Target: CHP1 CHP2 PPP3CA PPP3CB PPP3CC PPP3R1 PPP3R2 / CYP inhibition: CYP3A4 |
D09190 |
Anti-human thymocyte immunoglobulin, rabbit (JAN); Thymoglobuline (TN) |
(P) unclassified |
D09197 |
Valsartan and hydrochlorothiazide (JP18); Co-dio (TN) |
(P) unclassified |
D09208 |
Cetilistat (JAN/USAN/INN); Oblean (TN) |
(P) unclassified |
D09214 |
Ustekinumab (USAN/INN); Ustekinumab (genetical recombination) (JAN); Ustekinumab (genetical recombination) [Ustekinumab biosimilar 1] (JAN); Stelara (TN) |
(P) unclassified |
D09215 |
Eslicarbazepine (USAN/INN) |
(P) CYP induction: CYP3A4 |
D09314 |
Ofatumumab (USAN/INN); Ofatumumab (genetical recombination) (JAN); Arzerra (TN); Kesimpta (TN) |
(P) unclassified |
D09315 |
Canakinumab (USAN/INN); Canakinumab (genetical recombination) (JAN); Ilaris (TN) |
(P) unclassified |
D09319 |
Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09360 |
Obeticholic acid (JAN/USAN/INN); Ocaliva (TN) |
(P) unclassified |
D09394 |
Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) |
(P) CYP inhibition: CYP3A4 |
D09546 |
Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) |
(P) Transporter inhibition: ABCB1 |
D09568 |
Naproxcinod (USAN/INN) |
(P) unclassified |
D09569 |
Ezogabine (USAN); Retigabine (INN); Potiga (TN) |
(P) unclassified |
D09572 |
Riociguat (JAN/USAN/INN); Adempas (TN) |
(P) Transporter inhibition: ABCB1 |
D09587 |
Brentuximab vedotin (USAN/INN); Brentuximab vedotin (genetical recombination) (JAN); Adcetris (TN) |
(P) unclassified |
D09588 |
Briakinumab (USAN/INN) |
(P) unclassified |
D09594 |
Olmesartan medoxomil and azelnidipine; Rezaltas (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09595 |
Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09612 |
Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) |
(P) CYP induction: CYP3A4 |
D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09642 |
Modithromycin (USAN/INN) |
(P) unclassified |
D09669 |
Siltuximab (USAN/INN); Sylvant (TN) |
(P) unclassified |
D09680 |
Teprotumumab (USAN/INN); Teprotumumab (genetical recombination) (JAN); Teprotumumab-trbw; Tepezza (TN) |
(P) unclassified |
D09702 |
Albaconazole (USAN/INN) |
(P) unclassified |
D09707 |
Dabigatran (USAN/INN) |
(P) Transporter inhibition: ABCB1 |
D09710 |
Edoxaban (USAN/INN) |
(P) Transporter inhibition: ABCB1 |
D09725 |
Emulsified influenza HA vaccine (A/H1N1); Arepanrix (H1N1) (TN) |
(P) unclassified |
D09728 |
Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09730 |
Olaparib (JAN/USAN/INN); Lynparza (TN) |
(P) unclassified |
D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09733 |
Afatinib dimaleate (USAN); Afatinib maleate (JAN); Gilotrif (TN); Giotrif (TN) |
(P) Transporter inhibition: ABCB1 |
D09741 |
Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09743 |
Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09745 |
Valsartan and amlodipine besilate; Exforge (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09753 |
Saxagliptin hydrate (JAN); Onglyza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09760 |
Ibuprofen sodium (USAN); Ibuprofen sodium hydrate |
(P) unclassified |
D09783 |
Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09789 |
Kirenidipine hydrochloride (JAN) |
(P) unclassified |
D09796 |
Hydrocortisone caproate (JAN) |
(P) unclassified |
D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
D09809 |
Tylosin acetate isovalerte (JAN) |
(P) unclassified |
D09813 |
Lenalidomide hydrate (JAN); Revlimid (TN) |
(P) unclassified |
D09843 |
Beradilol monoethyl maleate (JAN); TZC-5665 |
(P) unclassified |
D09881 |
Cobicistat (JAN/USAN/INN); Tybost (TN) |
(P) Enzyme-Target: CYP3A4 |
D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(CI,P) Transporter inhibition: ABCB1 |
D09919 |
Lenvatinib (USAN/INN) |
(P) Transporter inhibition: ABCB1 |
D09920 |
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) |
(P) Transporter inhibition: ABCB1 |
D09951 |
Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) |
(P) unclassified |
D09956 |
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) |
(P) unclassified |
D09960 |
Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09967 |
Secukinumab (USAN/INN); Secukinumab (genetical recombination) (JAN); Cosentyx (TN) |
(P) unclassified |
D09970 |
Tofacitinib (USAN); Tasocitinib |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D09987 |
Vaniprevir (JAN/USAN/INN); Vanihep (TN) |
(CI) unclassified |
D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
D10001 |
Fingolimod (INN); Gilenya (TN) |
(P) unclassified |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
D10017 |
Naproxen etemesil (USAN) |
(P) unclassified |
D10019 |
Panobinostat lactate (JAN); Farydak (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10021 |
Efinaconazole (JAN/USAN/INN); Clenafin (TN); Jublia (TN) |
(P) unclassified |
D10024 |
Selumetinib sulfate (JAN/USAN); Koselugo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10032 |
Tylvalosin (USAN/INN) |
(P) unclassified |
D10033 |
Tylosin tartrate (USP) |
(P) unclassified |
D10034 |
Tylvalosin tartrate (USAN); Aiviosin [veterinary] (TN) |
(P) unclassified |
D10061 |
Brodalumab (USAN); Brodalumab (genetical recombination) (JAN); Siliq (TN) |
(P) unclassified |
D10071 |
Ixekizumab (USAN); Ixekizumab (genetical recombination) (JAN); Taltz (TN) |
(P) unclassified |
D10080 |
Sirukumab (USAN); Sirukumab (genetical recombination) (JAN) |
(P) unclassified |
D10081 |
Simeprevir (JAN/USAN) |
(P) Transporter inhibition: ABCB1 |
D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) unclassified |
D10093 |
Asunaprevir (JAN/USAN); Sunvepra (TN) |
(CI) CYP induction: CYP3A4 / Transporter inhibition: ABCB1 |
D10095 |
Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) |
(P) unclassified |
D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D10135 |
Macitentan (JAN/USAN); Opsumit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10137 |
Regorafenib hydrate (JAN); Stivarga (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D10147 |
Pasireotide (USAN) |
(P) unclassified |
D10151 |
Plazomicin (USAN) |
(P) unclassified |
D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
D10172 |
Teriflunomide (USAN); Aubagio (TN) |
(P) unclassified |
D10192 |
Recombinant adsorbed quadrivalent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil (TN); Silgard (TN) |
(P) unclassified |
D10198 |
Calcipotriol hydrate (JAN); Calcipotriol monohydrate; Calcipotriene hydrate; Dovonex (TN) |
(P) unclassified |
D10212 |
Recombinant adsorbed bivalent human papillomavirus-like particle vaccine (derived from Trichoplusia ni cells); Cervarix (TN) |
(P) unclassified |
D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
D10223 |
Ibrutinib (JAN/USAN); Imbruvica (TN) |
(P) unclassified |
D10226 |
Sacubitril valsartan sodium hydrate (JAN); Sacubitril mixture with valsartan; Entresto (TN) |
(P) unclassified |
D10243 |
Irbesartan and amlodipine besilate (JP18); Aimix (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10254 |
Esflurbiprofen (JAN) |
(P) unclassified |
D10308 |
Baricitinib (JAN/USAN/INN); Olumiant (TN) |
(P) Transporter inhibition: ABCB1 |
D10309 |
Brexpiprazole (JAN/USAN/INN); Rexulti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
D10385 |
Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10396 |
Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN); Ofev (TN) |
(P) Transporter inhibition: ABCB1 |
D10400 |
Tildrakizumab (USAN); Tildrakizumab (genetical recombination) (JAN); Tildrakizumab-asmn; Ilumya (TN) |
(P) unclassified |
D10438 |
Guselkumab (USAN/INN); Guselkumab (genetical recombination) (JAN); Tremfya (TN) |
(P) unclassified |
D10450 |
Alectinib hydrochloride (JAN); Alecensa (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10452 |
Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) |
(P) unclassified |
D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10469 |
Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) |
(P) Transporter inhibition: ABCB1 |
D10478 |
Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10492 |
Tildipirosin (USAN/INN); Zuprevo [veterinary] (TN) |
(P) unclassified |
D10497 |
Pasireotide diaspartate; Signifor (TN) |
(P) unclassified |
D10501 |
Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10505 |
Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D10506 |
Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10513 |
Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10516 |
Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10520 |
Rabeprazole, amoxicillin and metronidazole; Rabefine (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10524 |
Azilsartan and amlodipine besilate; Zacras (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10525 |
Valsartan and cilnidipine; Atedio (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10527 |
Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10528 |
Aldosterone (INN) |
(P) unclassified |
D10533 |
Umeclidinium bromide and vilanterol; Anoro (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10534 |
Calcipotriene and betamethasone dipropionate; Calcipotriol and betamethasone dipropionate; Dovobet (TN); Enstilar (TN); Taclonex (TN) |
(P) unclassified |
D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
D10556 |
Fimasartan (INN) |
(P) unclassified |
D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
D10568 |
Pitavastatin calcium hydrate (JP18); Livalo (TN) |
(CI,P) unclassified |
D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10639 |
Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) |
(CI) Transporter inhibition: ABCB1 |
D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
D10653 |
Peficitinib (USAN/INN) |
(P) unclassified |
D10655 |
Plazomicin sulfate (USAN); Zemdri (TN) |
(P) unclassified |
D10656 |
Polmacoxib (USAN/INN) |
(P) unclassified |
D10679 |
Venetoclax (JAN/USAN/INN); Venclexta (TN) |
(CI,P) unclassified |
D10688 |
Abemaciclib (JAN/USAN/INN); Verzenio (TN) |
(P) unclassified |
D10699 |
Cholic acid (JAN/USAN); Cholbam (TN) |
(P) unclassified |
D10711 |
Pemafibrate (JAN); Parmodia (TN) |
(CI,P) unclassified |
D10721 |
Peficitinib hydrobromide (JAN/USAN); Smyraf (TN) |
(P) unclassified |
D10733 |
Talazoparib tosylate (USAN); Talazoparib tosilate (JAN); Talzenna (TN) |
(P) unclassified |
D10745 |
Ombitasvir, paritaprevir and ritonavir; Technivie (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D10750 |
Isavuconazole (INN); Cresemba (TN) |
(P) unclassified |
D10753 |
Atazanavir and cobicistat; Evotaz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
D10756 |
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) |
(P) unclassified |
D10761 |
Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) |
(P) unclassified |
D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10780 |
Perampanel hydrate (JAN); Fycompa (TN) |
(P) unclassified |
D10800 |
Gilteritinib fumarate (JAN/USAN); Xospata (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
D10805 |
Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10822 |
Ciprofloxacin hydrate (JAN); Ciprofloxacin hemiheptahydrate |
(P) unclassified |
D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
D10866 |
Brigatinib (JAN/USAN); Alunbrig (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10871 |
Filgotinib (USAN/INN) |
(P) unclassified |
D10872 |
Filgotinib hydrochloride (USAN) |
(P) unclassified |
D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10892 |
Esaxerenone (JAN/INN) |
(P) unclassified |
D10893 |
Acalabrutinib (JAN/USAN/INN); Calquence (TN) |
(P) unclassified |
D10915 |
Cannabidiol (USAN/INN); CBD; Epidiolex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10930 |
Etrasimod (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10931 |
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10944 |
Itacitinib (USAN/INN) |
(P) unclassified |
D10945 |
Itacitinib adipate (JAN/USAN) |
(P) unclassified |
D10967 |
Ozanimod hydrochloride (JAN/USAN); Zeposia (TN) |
(P) unclassified |
D10968 |
Ozanimod (USAN/INN) |
(P) unclassified |
D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
D10993 |
Tucidinostat (JAN/USAN/INN); Hiyasta (TN) |
(P) unclassified |
D10994 |
Upadacitinib (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10995 |
Upadacitinib tartrate (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D10999 |
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11000 |
Vamorolone (USAN/INN); Agamree (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
D11014 |
Glecaprevir and pibrentasvir; Mavyret (TN) |
(P) Transporter inhibition: ABCB1 |
D11022 |
Lemborexant (JAN/USAN/INN); Dayvigo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11035 |
Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) |
(P) unclassified |
D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D11048 |
Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11052 |
Risankizumab (USAN/INN); Risankizumab (genetical recombination) (JAN); Risankizumab-rzaa; Skyrizi (TN) |
(P) unclassified |
D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11054 |
Ravulizumab (USAN/INN); Ravulizumab (genetical recombination) (JAN); Ultomiris (TN) |
(P) unclassified |
D11070 |
Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) |
(P) unclassified |
D11072 |
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) |
(P) unclassified |
D11079 |
Satralizumab (USAN/INN); Satralizumab (genetical recombination) (JAN); satralizumab-mwge; Enspryng (TN) |
(P) unclassified |
D11082 |
Anifrolumab (USAN); Anifrolumab (genetical recombination) (JAN); Anifrolumab-fnia; Saphnelo (TN) |
(P) unclassified |
D11092 |
Pitavastatin magnesium; Zypitamag (TN) |
(CI,P) unclassified |
D11093 |
Avacopan (JAN/USAN/INN); Tavneos (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11095 |
Atorvastatin calcium propylene glycol solvate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D11106 |
Filgotinib maleate (JAN/USAN); Jyseleca (TN) |
(P) unclassified |
D11120 |
Emapalumab (USAN/INN); Emapalumab (genetical recombination) (JAN); Emapalumab-lzsg; Gamifant (TN) |
(P) unclassified |
D11123 |
Mirikizumab (USAN/INN); Mirikizumab (genetical recombination) (JAN); Mirikizumab-mrkz; Omvoh (TN) |
(P) unclassified |
D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
D11150 |
Cenobamate (USAN/INN); Xcopri (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11154 |
Diroximel fumarate (JAN/USAN/INN); Vumerity (TN) |
(P) unclassified |
D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
D11204 |
Octreotide hydrochloride (USAN) |
(P) unclassified |
D11215 |
Ponesimod (USAN/INN); Ponvory (TN) |
(P) unclassified |
D11243 |
Ublituximab (USAN/INN); Briumvi (TN) |
(P) unclassified |
D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
D11397 |
Darvadstrocel (INN); Alofisel (TN) |
(P) unclassified |
D11417 |
Pemigatinib (JAN/USAN/INN); Pemazyre (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11460 |
Siponimod (USAN/INN) |
(P) unclassified |
D11470 |
Imlifidase (USAN/INN); Idefirix (TN) |
(P) unclassified |
D11472 |
Remdesivir (JAN/USAN); Veklury (TN) |
(P) unclassified |
D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) Transporter inhibition: ABCB1 |
D11520 |
Ezetimibe and rosuvastatin; Roszet (TN); Rosuzet (TN) |
(CI) unclassified |
D11525 |
Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) |
(P) unclassified |
D11530 |
Sutimlimab (USAN/INN); Sutimlimab (genetical recombination) (JAN); Sutimlimab-jome; Enjaymo (TN) |
(P) unclassified |
D11550 |
Bimekizumab (USAN/INN); Bimekizumab (genetical recombination) (JAN); Bimzelx (TN) |
(P) unclassified |
D11565 |
Grazoprevir (USAN/INN); Grazoprevir anhydrous |
(CI) Transporter inhibition: ABCB1 |
D11568 |
Edoxaban tosylate (USAN) |
(P) Transporter inhibition: ABCB1 |
D11572 |
Beclomethasone dipropionate monohydrate; Beconase aq (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11580 |
Perindopril arginine |
(P) unclassified |
D11584 |
Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) |
(P) unclassified |
D11613 |
Pegcetacoplan (JAN/USAN/INN); Empaveli (TN) |
(P) unclassified |
D11641 |
Danicopan (JAN/USAN/INN); Voydeya (TN) |
(P) unclassified |
D11659 |
Tolvaptan sodium phosphate (JAN); Samtasu (TN) |
(P) unclassified |
D11662 |
Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) |
(P) unclassified |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 / Transporter inhibition: ABCB1 |
D11696 |
Crovalimab (USAN/INN); Crovalimab (genetical recombination) (JAN); Piasky (TN) |
(P) unclassified |
D11703 |
Opinercept (INN) |
(P) unclassified |
D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11725 |
Futibatinib (JAN/USAN/INN); Lytgobi (TN) |
(P) unclassified |
D11757 |
Inebilizumab (USAN/INN); Inebilizumab (genetical recombination) (JAN); Inebilizumab-cdon; Uplizna (TN) |
(P) unclassified |
D11785 |
Oteseconazole (USAN/INN); Vivijoa (TN) |
(P) unclassified |
D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
D11815 |
Belumosudil (USAN) |
(P) unclassified |
D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) unclassified |
D11817 |
Deucravacitinib (JAN/USAN); Sotyktu (TN) |
(P) unclassified |
D11861 |
Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) |
(P) unclassified |
D11862 |
Indacaterol and mometasone furoate; Atectura (TN) |
(P) unclassified |
D11863 |
Human papillomavirus 9-valent vaccine, recombinant; Recombinant adsorbed 9-valent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil 9 (TN); Silgard 9 (TN) |
(P) unclassified |
D11876 |
Efgartigimod alfa (USAN/INN); Efgartigimod alfa (genetical recombination) (JAN); Efgartigimod alfa-fcab; Vyvgart (TN) |
(P) unclassified |
D11881 |
Amlodipine benzoate; Katerzia (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
D12015 |
St. John's wort; SJW |
(P) unclassified |
D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
D12066 |
Spesolimab (USAN/INN); Spesolimab (genetical recombination) (JAN); Spesolimab-sbzo; Spevigo (TN) |
(P) unclassified |
D12182 |
Rozanolixizumab (USAN/INN); Rozanolixizumab (genetical recombination) (JAN); rozanolixizumab-noli; Rystiggo (TN) |
(P) unclassified |
D12251 |
Iptacopan (USAN/INN) |
(P) unclassified |
D12252 |
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) |
(P) unclassified |
D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D12311 |
Bortezomib hydrate (JAN) |
(P) unclassified |
D12326 |
Opelconazole (USAN/INN) |
(P) unclassified |
D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(P) unclassified |
D12356 |
Zilucoplan sodium (JAN); Zilbrysq (TN) |
(P) unclassified |
D12357 |
Zilucoplan (USAN/INN) |
(P) unclassified |
D12410 |
Landiolol (USAN/INN) |
(P) unclassified |
D12438 |
Pitavastatin calcium and ezetimibe; Livazebe (TN) |
(CI) unclassified |
D12487 |
Olokizumab (INN) |
(P) unclassified |
D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |
D12595 |
Aspirin trelamine (USAN) |
(P) unclassified |
D12596 |
Aspirin trelamine hydrochloride (USAN) |
(P) unclassified |
D12597 |
Ibuprofen trelamine (USAN); Ibuprofen diethylaminoethyl ester |
(P) unclassified |
D12598 |
Ibuprofen trelamine hydrochloride (USAN) |
(P) unclassified |
D12609 |
Dasatinib laurylsulfate (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
D12684 |
Efgartigimod alfa and hyaluronidase; Efgartigimod alfa (genetical recombination) and vorhyaluronidase alfa (genetical recombination); Efgartigimod alfa and hyaluronidase-qvfc; Vyvgard hytrulo (TN); Vyvdura (TN) |
(P) unclassified |
D12747 |
Divozilimab (INN) |
(P) unclassified |
D12748 |
Levilimab (INN) |
(P) unclassified |
D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |