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Drug interaction list


Query:
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN)

Interactions: 536 hits    [ ATC classification | Therapeutic category ]

C07051  Indinavir (P) unclassified
D00059  Levodopa (JP18/USP/INN); Dopar (TN) (P) unclassified
D00079  Dinoprostone (JAN/USP/INN); Cervidil (TN); Prepidil (TN); Prostin E2 (TN) (P) unclassified
D00081  Dinoprost (JP18/USAN/INN); Prosmon (TN) (P) unclassified
D00106  Epoprostenol (USAN/INN); Prostaglandin I2; Prostacyclin; Epoprostenol (TN) (P) unclassified
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) (CI) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00118  Naproxen (JP18/USP/INN); Naprosyn (TN) (P) unclassified
D00136  Haloperidol (JP18/USP/INN); Haldol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00151  Mefenamic acid (JP18/USP/INN); Ponstel (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D00180  Alprostadil (JP18/USP/INN); Prostin VR pediatric (TN); Caverject (TN); Edex (TN); Muse (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (CI) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00218  Acetazolamide (JP18/USP/INN); Diamox (TN) (P) unclassified
D00228  Amoxapine (JP18/USP/INN); Asendin (TN) (P) unclassified
D00241  Baclofen (JP18/USP/INN); Kemstro (TN); Lioresal (TN) (P) unclassified
D00253  Carbidopa hydrate and levodopa; Parcopa (TN); Sinemet (TN) (P) unclassified
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00294  Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) (P) unclassified
D00296  Didanosine (JAN/USP/INN); Videx (TN) (P) unclassified
D00298  Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) (P) unclassified
D00302  Dipyridamole (JP18/USP/INN); Persantine (TN) (P) unclassified
D00304  Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) (P) unclassified
D00319  Felodipine (JP18/USP/INN); Plendil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP2C9 CYP3A4
D00331  Furosemide (JP18/USP/INN); Frusemide; Lasix (TN) (P) unclassified
D00336  Glyburide (USP); Glibenclamide (JP18/INN); Diabeta (TN); Glynase (TN); Micronase (TN) (CI) Enzyme: CYP2C9 CYP3A4 / CYP induction: CYP2C9 CYP3A4
D00346  Isoniazid (JP18/USP/INN); Laniazid (TN) (P) unclassified
D00349  Isradipine (USP/INN); Dynacirc (TN) (P) unclassified
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00353  Lamivudine (JAN/USP/INN); Epivir (TN) (P) unclassified
D00356  Latanoprost (JAN/USP/INN); Xalatan (TN) (P) unclassified
D00359  Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00382  Torsemide (USP); Torasemide (JAN/INN); Demadex (TN); Luprac (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D00383  Trandolapril (JAN/USP/INN); Mavik (TN) (P) unclassified
D00387  Triazolam (JP18/USP/INN); Halcion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00399  Valproic acid (USP); Depakene (TN) (P) unclassified
D00405  Methyldopa (USP); Methyldopa hydrate (JP18); Aldomet (TN) (P) unclassified
D00412  Zalcitabine (JAN/USP/INN); Hivid (TN) (P) unclassified
D00413  Zidovudine (JP18/USP/INN); Azidothymidine; Retrovir (TN) (P) unclassified
D00419  Misoprostol (JAN/USP/INN); Cytotec (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00426  Risperidone (JP18/USP/INN); Risperdal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) CYP induction: CYP2C9
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00432  Nadolol (JP18/USP/INN); Corgard (TN) (P) unclassified
D00434  Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00437  Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00438  Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00443  Spironolactone (JP18/USP/INN); Aldactone (TN) (P) unclassified
D00445  Stavudine (USAN/INN); Sanilvudine (JAN); Zerit (TN) (P) unclassified
D00458  Quetiapine fumarate (JP18/USP); Seroquel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00479  Prochlorperazine maleate (JP18/USP); Compazine (TN) (P) unclassified
D00480  Promethazine hydrochloride (JP18/USP); Phenergan (TN); Promethegan (TN) (P) unclassified
D00503  Perphenazine (JP18/USP/INN); Trilafon (TN) (P) unclassified
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) CYP induction: CYP2C9
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D00515  Nitroglycerin (JP18/USP); Glyceryl trinitrate; Minitran (TN); Nitro-bid (TN); Nitro-dur (TN); Nitromist (TN); Transderm-nitro (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00538  Zonisamide (JP18/USP/INN); Excegran (TN) (P) unclassified
D00539  Ethosuximide (JP18/USP/INN); Zarontin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00547  Sevoflurane (JP18/USAN/INN); Ultane (TN) (P) unclassified
D00549  Propofol (JAN/USP/INN); Diprivan (TN) (P) unclassified
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00553  Prilocaine (USP/INN); Propitocaine (JAN) (P) unclassified
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00564  Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D00599  Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00608  Doxazosin mesylate (USP); Doxazosin mesilate (JP18); Cardura (TN) (P) unclassified
D00609  Prazosin hydrochloride (JP18/USP); Minipress (TN) (P) unclassified
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00616  Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00617  Nicardipine hydrochloride (JP18/USAN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00618  Nisoldipine (JAN/USAN/INN); Sular (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00629  Nitrendipine (JP18/USAN/INN); Baypress (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00631  Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP induction: CYP2C9 CYP3A4
D00634  Bisoprolol fumarate (JP18/USP); Zebeta (TN) (P) unclassified
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00658  Trichlormethiazide (JP18/USP/INN); Naqua (TN) (P) unclassified
D00678  Ondansetron hydrochloride hydrate (JAN/USP); Ondansetron hydrochloride; Zofran (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00682  Carboprost tromethamine (USP); Hemabate (TN) (P) unclassified
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) CYP induction: CYP2C9
D00710  Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) (P) unclassified
D00713  Thiamylal sodium (JP18); Surital (TN) (P) unclassified
D00714  Thiopental sodium (JP18/USP/INN); Pentothal (TN) (P) unclassified
D00762  Metyrosine (USP); Metirosine (JAN/INN); Demser (TN) (P) unclassified
D00776  Tizanidine hydrochloride (JP18/USP); Zanaflex (TN) (P) unclassified
D00789  Chlorpromazine hydrochloride (JP18/USP); Sonazine (TN) (P) unclassified
D00793  Fluphenazine decanoate (JAN/USP); Prolixin decanoate (TN) (P) unclassified
D00809  Amitriptyline hydrochloride (JP18/USP); Elavil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00811  Clomipramine hydrochloride (JP18/USP); Anafranil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00815  Imipramine hydrochloride (JP18/USP); Tofranil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00887  Atorvastatin calcium anhydorous; Lipitor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00889  Cerivastatin sodium (JAN/USAN); Baycol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00891  Abacavir sulfate (JAN/USP); Ziagen (TN) (P) unclassified
D00892  Fluvastatin sodium (JAN/USP); Lescol (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP inhibition: CYP2C9 / CYP induction: CYP2C9 CYP3A4
D00893  Pravastatin sodium (JP18/USP); CS-514; Pravachol (TN) (P) unclassified
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00895  Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) (P) unclassified
D00896  Efavirenz (JAN/USP/INN); Sustiva (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00904  Diclofenac sodium (JP18/USP); Solaraze (TN); Voltaren (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D00950  Levonorgestrel (JAN/USP/INN); Mirena (TN); Norplant (TN); Skyla (TN) (P) unclassified
D00961  Bicalutamide (JP18/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00969  Meloxicam (JAN/USP/INN); Mobic (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00987  Cabergoline (JP18/USP/INN); Cabaser (TN); Dostinex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01024  Tamsulosin hydrochloride (JP18/USP); Flomax (TN); Harnal (TN) (P) unclassified
D01055  Emivirine (USAN/INN); Coactinon (TN) (P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01104  Barnidipine hydrochloride (JAN); Hypoca (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01107  Milnacipran hydrochloride (JAN/USAN); Savella (TN); Toledomin (TN) (P) unclassified
D01115  Eplerenone (JP18/USAN/INN); Inspra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01145  Azelnidipine (JP18/INN); Calblock (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01164  Aripiprazole (JAN/USP/INN); Abilify (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01173  Cilnidipine (JP18/INN); Atelec (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01176  Blonanserin (JAN/INN); AD 5423 (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01179  Duloxetine hydrochloride (JAN/USP); Cymbalta (TN); Yentreve (TN) (P) unclassified
D01188  Pimilprost (JAN/INN) (P) unclassified
D01196  Acetazolamide sodium (JAN); Diamox (TN) (P) unclassified
D01199  Emtricitabine (JAN/USAN/INN); Emtriva (TN) (P) unclassified
D01213  Tolvaptan (JAN/USAN/INN); Samsca (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01240  Deslanoside (JP18/USP/INN); Cedilanid-d (TN) (P) unclassified
D01243  Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01280  Warfarin potassium (JP18); Athrombin-K (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D01302  Hydralazine hydrochloride (JP18/USP); Apresoline (TN) (P) unclassified
D01303  Flunarizine hydrochloride (JAN/USAN) (P) unclassified
D01321  Zotepine (JAN/INN); Setous (TN) (P) unclassified
D01323  Azosemide (JP18/USAN/INN); Diart (TN) (P) unclassified
D01333  Urapidil (JP18/INN); Ebrantil (TN) (P) unclassified
D01337  Epoprostenol sodium (JAN/USAN); Flolan (TN); Veletri (TN) (P) unclassified
D01352  Dinoprost tromethamine (JAN/USP); Prostin F2 alpha (TN) (P) unclassified
D01358  Mianserin hydrochloride (JAN/USAN); Tetramide (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01372  Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01425  Lopinavir (JAN/USP/INN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP2C9 CYP3A4
D01452  Isopropyl unoprostone (JAN); Unoprostone isopropyl; Rescula (TN) (P) unclassified
D01469  Amosulalol hydrochloride (JP18); Lowgan (TN) (P) unclassified
D01485  Propericiazine (JAN); Periciazine; Neuleptil (TN) (P) unclassified
D01520  Levomepromazine hydrochloride (JAN/USAN); Nozinan (TN) (P) unclassified
D01546  Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Dosulepin (TN) (P) unclassified
D01549  Imidapril hydrochloride (JP18); Tanatril (TN) (P) unclassified
D01551  Beraprost sodium (JP18/USAN); Procylin (TN) (P) unclassified
D01553  Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01562  Aranidipine (JAN/INN); Sapresta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01578  Pranoprofen (JP18/INN); Elicapric (TN) (P) unclassified
D01604  Efonidipine hydrochloride ethanolate (JAN); Efonidipine hydrochloride ethanol; Efonidipine hydrochloride; NZ 105 ethanolate; Landel (TN) (P) unclassified
D01656  Brovincamine fumarate (JAN); Sabromin (TN) (P) unclassified
D01674  Naftopidil (JP18/INN); Flivas (TN) (P) unclassified
D01691  Nipradilol (JAN/INN); Hypadil (TN) (P) unclassified
D01709  Loxoprofen sodium hydrate (JP18); Lorfenamin (TN); Loxonin (TN) (P) unclassified
D01741  Celiprolol hydrochloride (JAN/USAN); Selectol (TN) (P) unclassified
D01744  Brotizolam (JP18/USAN/INN); Lendormin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01849  Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) (P) unclassified
D01862  Pitavastatin calcium (JAN); NK 104; Livalo (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D01869  Ornoprostil (JAN/INN); Ronok (TN) (P) unclassified
D01877  Mefruside (JP18/USAN/INN); Baycaron (TN) (P) unclassified
D01887  Bunazosin hydrochloride (JP18); Detantol (TN) (P) unclassified
D01891  Enprostil (JAN/USAN/INN); Camleed (TN) (P) unclassified
D01895  Tripamide (JAN/USAN/INN); Normonal (TN) (P) unclassified
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01902  Fonazine mesylate (USAN); Dimetotiazine mesilate (JAN); Banistyl (TN) (P) unclassified
D01908  Nilvadipine (JP18/USAN/INN); Nivadil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01915  Rosuvastatin calcium (JP18/USP); ZD 4522; Crestor (TN) (P) unclassified
D01933  Vatanidipine hydrochloride (JAN); AE 0047; Calbren (TN) (P) unclassified
D01943  Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) (P) unclassified
D01964  Travoprost (JAN/USP/INN); Travatan (TN) (P) unclassified
D01965  Silodosin (JP18/INN); KMD 3213; Rapaflo (TN); Urief (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01969  Gallopamil hydrochloride (JAN) (P) unclassified
D01977  Gefitinib (JP18/USAN/INN); Iressa (TN) (P) unclassified
D01982  Tenofovir disoproxil fumarate (JAN/USAN); Viread (TN) (P) unclassified
D02002  Isoniazid sodium methanesulfonate hydrate (JAN); Isoniazid sodium methanesulfonate monohydrate; Isoniazid sodium methanesulfonate; IHMS; Neoiscotin (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02022  Prochlorperazine mesilate (JAN); Prochlorperazine dimethanesulfonate; Novamin (TN) (P) unclassified
D02034  Setiptiline maleate (JAN); Tecipul (TN) (P) unclassified
D02037  Perphenazine maleate (JP18); PZC (TN) (P) unclassified
D02045  Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02048  Clinprost (JAN/INN); TEI 9090; Arteron (TN) (P) unclassified
D02073  Gemeprost (JAN/USAN/INN); Preglandin (TN) (P) unclassified
D02076  Brimonidine tartrate (JAN/USAN); Alphagan (TN) (P) unclassified
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D02135  Levodopa and benserazide hydrochloride; Madopar (TN) (P) unclassified
D02163  Fluphenazine maleate (JAN); Flumezin (TN) (P) unclassified
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02245  Trimeprazine tartrate (USP); Alimemazine tartrate (JP18); Alimezine (TN) (P) unclassified
D02248  Levomepromazine maleate (JP18/USAN); Hirnamin (TN) (P) unclassified
D02258  Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02297  Emtricitabine and tenofovir disoproxil; Truvada (TN) (P) unclassified
D02342  Bisoprolol (JAN/USAN/INN) (P) unclassified
D02343  Carboprost (USAN/INN) (P) unclassified
D02356  Verapamil (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02372  Perospirone hydrochloride hydrate (JAN); Lullan (TN) (P) unclassified
D02408  Trimipramine maleate (JAN/USP); Surmontil (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) unclassified
D02499  Enfuvirtide (USAN/INN); Fuzeon (TN) (P) unclassified
D02537  Dronedarone (INN) (P) unclassified
D02540  Garenoxacin mesylate (USAN); Garenoxacin mesilate hydrate (JAN) (P) unclassified
D02587  Metildigoxin (JP18); Lanirapid (TN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02629  Fluspirilene (USAN/INN); Imap (TN) (P) unclassified
D02630  Penfluridol (USAN/INN); Semap (TN) (P) unclassified
D02633  Lomerizine hydrochloride (JAN); Terranas (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02705  Alprostadil alfadex (JP18); Tandetron (TN); Caverject (TN) (P) unclassified
D02719  Rosaprostol (INN) (P) unclassified
D02720  Beraprost (USAN) (P) unclassified
D02721  Iloprost (USAN/INN); Ventavis (TN) (P) unclassified
D02722  Limaprost (INN) (P) unclassified
D02723  Ecraprost (USAN/INN) (P) unclassified
D02724  Bimatoprost (JAN/USAN/INN); Lumigan (TN); Latisse (TN) (P) unclassified
D02725  Sulprostone (USAN/INN) (P) unclassified
D02731  Vardenafil dihydrochoride (USAN); Levitra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02734  Abacavir succinate (USAN) (P) unclassified
D02802  Alemtuzumab (USAN/INN); Alemtuzumab (genetical recombination) (JAN); Campath (TN); Lemtrada (TN) (P) unclassified
D02860  Limaprost alfadex (JP18); Opalmon (TN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02890  Amdoxovir (USAN/INN) (P) unclassified
D02914  Amlodipine maleate (USAN); Amvaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 CYP2C9
D02994  Rituximab (USAN/INN); Rituximab (genetical recombination) (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 1] (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 2] (JAN); Rituximab-abbs; Rituximab-pvvr; Rituximab-arrx; Rituxan (TN); Riabni (TN); Truximab (TN) (P) unclassified
D02995  Asenapine maleate (JAN/USAN); Saphris (TN) (P) unclassified
D03001  Atevirdine mesylate (USAN) (P) unclassified
D03067  Belfosdil (USAN/INN) (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03150  Bortezomib (JAN/USAN/INN); Velcade (TN) (P) unclassified
D03187  Butaprost (USAN/INN) (P) unclassified
D03217  Avanafil (USAN/INN); Stendra (TN); Spedra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03218  Axitinib (JAN/USAN); Inlyta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03253  Brecanavir (USAN) (P) unclassified
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03269  Dinoprostone betadex (JAN); Prostarmon E (TN) (P) unclassified
D03290  Promethazine methylenedisalicylate (JAN); Pyrethia (TN) (P) unclassified
D03371  Capravirine (USAN/INN) (P) unclassified
D03399  Carboprost methyl (USAN) (P) unclassified
D03522  Ciprostene calcium (USAN) (P) unclassified
D03536  Clentiazem maleate (JAN/USAN) (P) unclassified
D03601  Crilvastatin (USAN/INN) (P) unclassified
D03643  Dalvastatin (USAN/INN) (P) unclassified
D03655  Darodipine (USAN/INN) (P) unclassified
D03656  Darunavir (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03657  Dasantafil (USAN/INN) (P) unclassified
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP induction: CYP3A4
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03816  Tenivastatin calcium (USAN) (P) unclassified
D03830  Diltiazem malate (USAN); Tiamate (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03839  Droxinavir hydrochloride (USAN) (P) unclassified
D03840  Palinavir (USAN/INN) (P) unclassified
D03842  Telinavir (USAN/INN) (P) unclassified
D03843  Tipranavir disodium (USAN) (P) unclassified
D03914  Dronedarone hydrochloride (USP); Multaq (TN) (P) unclassified
D03981  Elvucitabine (USAN/INN) (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04034  Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) (P) unclassified
D04038  Perphenazine fendizoate (JAN); PZC (TN) (P) unclassified
D04046  Salicylamide, acetaminophen, anhydrous caffeine and promethazine methylenedisalicylate; PL (TN) (P) unclassified
D04059  Mepenzolate bromide and phenobarbital; Trancolon P (TN) (P) unclassified
D04104  Etonogestrel (USAN/INN); Implanon (TN); Nexplanon (TN) (P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP inhibition: CYP2C9 / CYP induction: CYP2C9 CYP3A4
D04193  Flordipine (USAN/INN) (P) unclassified
D04260  Fostedil (USAN/INN) (P) unclassified
D04460  Ethinylestradiol and ethynodiol diacetate; Edulen (TN); Zovia (TN) (P) unclassified
D04463  Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP induction: CYP2C9 CYP3A4
D04482  Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) (P) unclassified
D04483  Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) (P) unclassified
D04484  Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D04657  Lacidipine (USAN/INN); Motens (TN) (P) unclassified
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04733  Lidoflazine (USAN/INN); Angex (TN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (P) unclassified
D04786  Loviride (USAN/INN) (P) unclassified
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04965  Perphenazine hydrochloride; Perphenazine dihydrochloride; PZC intramuscular injection (TN) (P) unclassified
D05024  Mibefradil dihydrochloride (USAN); Posicor (TN) (P) unclassified
D05177  Nitisinone (JAN/USAN/INN); Orfadin (TN) (P) CYP inhibition: CYP2C9
D05339  Paliperidone (JAN/USP/INN); Invega (TN) (P) unclassified
D05340  Paliperidone palmitate (JAN/USAN); Xeplion (TN); Trevicta (TN); Invega sustenna (TN); Invega trinza (TN) (P) unclassified
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (P) unclassified
D05442  Perhexiline maleate (USAN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP18) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05538  Mozenavir (INN) (P) unclassified
D05732  Rioprostil (USAN/INN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D06060  Teludipine hydrochloride (USAN) (P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06074  Tenofovir (USAN); Tenofovir hydrate (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06213  Treprostinil (JAN/USAN/INN); Remodulin (TN) (P) unclassified
D06272  Sorafenib tosylate (USAN); Sorafenib tosilate (JAN); Nexavar (TN) (P) unclassified
D06274  Tafluprost (JAN/USAN/INN); Zioptan (TN) (P) unclassified
D06363  Ziconotide (USAN/INN); Prialt (TN) (P) unclassified
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06407  Vandetanib (JAN/USAN/INN); Caprelsa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06580  Dexelvucitabine (USAN/INN); Reverset (TN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 CYP2C9
D06670  Maraviroc (JAN/INN); Selzentry (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06676  Raltegravir (INN); MK-0518 (P) unclassified
D06677  Elvitegravir (JAN/USAN); Vitekta (TN) (P) unclassified
D07057  Abacavir (INN) (P) unclassified
D07132  Buprenorphine (JAN/INN); Temgesic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07133  Raltegravir potassium (JAN/USAN); Isentress (TN) (P) unclassified
D07185  Fendiline (INN) (P) unclassified
D07450  Amlodipine (USP/INN); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07474  Atorvastatin (INN); Lipitor (TN); Sortis (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07494  Barnidipine (INN); Vasexten (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07507  Zidovudine and lamivudine; Combivir (TN); Lamivudine zidovudine (TN) (P) unclassified
D07509  Benidipine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07520  Bepridil (INN); Bepadin (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP induction: CYP2C9 CYP3A4
D07545  Brovincamine (INN); Sarbromin (TN) (P) unclassified
D07569  Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9 CYP3A4
D07661  Cerivastatin (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07782  Delavirdine (INN) (P) unclassified
D07845  Diltiazem (INN); Surazem (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07886  Efonidipine (INN) (P) unclassified
D07943  Fendiline hydrochloride; Sensit (TN) (P) unclassified
D07971  Flunarizine (INN); Sibelium (TN) (P) unclassified
D07983  Fluvastatin (INN); Fluvas (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP inhibition: CYP2C9 / CYP induction: CYP2C9 CYP3A4
D08009  Gallopamil (INN) (P) unclassified
D08065  Iloprost tromethamine; Iloprost trometamol; Ventavis (TN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08111  Lercanidipine (INN); Lercanil (TN) (P) unclassified
D08155  Manidipine (INN); Manidipine 6300; Artedil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08217  Mibefradil (INN) (P) unclassified
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D08270  Nicardipine (INN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08340  Perhexiline (INN) (P) unclassified
D08410  Pravastatin (INN); Pravator (TN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) CYP induction: CYP3A4
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08492  Rosuvastatin (INN); Creston (TN) (P) unclassified
D08514  Sildenafil (INN); Aphrodil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08556  Tacrolimus (INN); Prograf (TN) (CI) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08575  Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) (P) unclassified
D08591  Tiaprost (INN); Iliren [veterinary] (TN) (P) unclassified
D08605  Tipranavir (INN); Aptivus (TN) (P) unclassified
D08628  Treprostinil monosodium salt; Treprostinil sodium; Trepulmix (TN) (P) unclassified
D08661  Unoprostone (INN); Rescula (TN) (P) unclassified
D08667  Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) (P) unclassified
D08668  Vardenafil (USAN/INN); Levitra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08682  Warfarin (INN); Warfarine; Choice (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D08686  Ziconotide acetate; Prialt (TN) (P) unclassified
D08768  Promethazine hibenzate; Hiberna (TN) (P) unclassified
D08775  Abacavir sulfate and lamivudine; Epzicom (TN) (P) unclassified
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08860  Apremilast (JAN/USAN); Otezla (TN) (P) unclassified
D08892  Clevidipine (USAN/INN); Clevidipine butyrate; Cleviprex (TN) (P) unclassified
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) unclassified
D09321  Obinutuzumab (USAN/INN); Obinutuzumab (genetical recombination) (JAN); Gazyva (TN) (P) unclassified
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) unclassified
D09594  Olmesartan medoxomil and azelnidipine; Rezaltas (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09621  Gisadenafil (USAN/INN) (P) unclassified
D09622  Gisadenafil besylate (USAN) (P) unclassified
D09634  Lersivirine (USAN/INN) (P) unclassified
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09687  Ulipristal acetate (JAN/USAN); Ella (TN) (P) unclassified
D09701  Abiraterone acetate (JAN/USP); Zytiga (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09720  Rilpivirine (JAN/USAN/INN); Rekambys (TN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09741  Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09743  Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09789  Kirenidipine hydrochloride (JAN) (P) unclassified
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09873  Bedaquiline fumarate (JAN/USAN); Sirturo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (P) unclassified
D09906  Fosdevirine (USAN/INN) (P) unclassified
D09920  Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) (P) unclassified
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (P) unclassified
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (P) unclassified
D09958  Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) (P) unclassified
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09989  Vardenafil hydrochloride (USP) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP inhibition: CYP2C9 / CYP induction: CYP3A4
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10019  Panobinostat lactate (JAN); Farydak (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (P) Enzyme: CYP2C9 CYP3A4 / CYP induction: CYP2C9 CYP3A4
D10027  Udenafil (USAN/INN) (P) unclassified
D10066  Dolutegravir (USAN); Tivicay (TN) (P) unclassified
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4 CYP2C9
D10113  Dolutegravir sodium (JAN/USAN); Tivicay (TN) (P) unclassified
D10131  Ixazomib citrate (JAN/USAN); Ninlaro (TN) (P) unclassified
D10135  Macitentan (JAN/USAN); Opsumit (TN) (CI,P) Enzyme: CYP3A4 / Target: EDNRA EDNRB / CYP induction: CYP3A4
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10185  Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (P) unclassified
D10243  Irbesartan and amlodipine besilate (JP18); Aimix (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10293  Carbidopa, levodopa and entacapone; Stalevo (TN) (P) CYP inhibition: CYP2C9
D10298  Brimonidine tartrate and timolol maleate; Combigan (TN); Aibeta (TN) (P) unclassified
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10428  Tenofovir alafenamide (USAN/INN) (P) unclassified
D10430  Treprostinil diolamine (USAN); Orenitram (TN) (P) unclassified
D10441  Latanoprostene bunod (USAN/INN); Vyzulta (TN) (P) unclassified
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (P) unclassified
D10461  Dienogest and estradiol valerate; Natazia (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10480  Irbesartan and trichlormethiazide; Irtra (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10548  Cabotegravir (JAN/USAN/INN); Vocabria (TN); Apretude (TN) (P) unclassified
D10549  Cabotegravir sodium (JAN/USAN); Vocabria (TN) (P) unclassified
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) CYP inhibition: CYP2C9
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10568  Pitavastatin calcium hydrate (JP18); Livalo (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D10571  Rilpivirine hydrochloride, tenofovir disoproxil fumarate and emtricitabine; Complera (TN); Eviplera (TN) (P) unclassified
D10600  Dolutegravir, abacavir and lamivudine; Triumeq (TN) (P) unclassified
D10605  Tenofovir alafenamide fumarate (JAN/USAN); Vemlidy (TN) (P) unclassified
D10624  Doravirine (JAN/USAN/INN); Pifeltro (TN) (P) unclassified
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (P) unclassified
D10711  Pemafibrate (JAN); Parmodia (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D10753  Atazanavir and cobicistat; Evotaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10754  Lamivudine and raltegravir; Lamivudine and raltegravir potassium; Dutrebis (TN) (P) unclassified
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (P) unclassified
D10756  Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10766  Osimertinib mesylate (USAN); Osimertinib mesilate (JAN); Tagrisso (TN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) CYP induction: CYP2C9
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (P) unclassified
D10834  Tenofovir disoproxil phosphate (P) unclassified
D10835  Emtricitabine and tenofovir alafenamide; Descovy (TN) (P) unclassified
D10836  Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) (P) unclassified
D10838  Abacavir, lamivudine and zidovudine; Trizivir (TN) (P) unclassified
D10851  Efavirenz, emtricitabine and tenofovir disoproxil; Atripla (TN) (P) unclassified
D10854  Brinzolamide and brimonidine tartrate; Simbrinza (TN); Ailamide (TN) (P) unclassified
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10892  Esaxerenone (JAN/INN) (P) unclassified
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (P) unclassified
D10909  Bictegravir (USAN/INN) (P) unclassified
D10910  Bictegravir sodium (JAN/USAN) (P) unclassified
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11039  Bictegravir, emtricitabine and tenofovir alafenamide; Biktarvy (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11045  Darolutamide (JAN/USAN/INN); Nebeqa (TN) (P) unclassified
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D11092  Pitavastatin magnesium; Zypitamag (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11095  Atorvastatin calcium propylene glycol solvate (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11190  Vosoritide (USAN/INN); Vosoritide (genetical recombination) (JAN); Voxzogo (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11246  Dapivirine (USAN/INN) (P) unclassified
D11282  Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (P) unclassified
D11391  Tenofovir disoproxil maleate (P) unclassified
D11392  Efavirenz, lamivudine and tenofovir disoproxil fumarate; Symfi (TN) (P) unclassified
D11395  Lamivudine and tenofovir disoproxil; Cimduo (TN); Temixys (TN) (P) unclassified
D11396  Doravirine, lamivudine and tenofovir disoproxil; Delstrigo (TN) (P) unclassified
D11400  Abrocitinib (JAN/USAN); Cibinqo (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D11404  Asciminib hydrochloride (JAN/USAN); Scemblix (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11521  Lamivudine, nevirapine and zidovudine (P) unclassified
D11522  Dolutegravir and lamivudine; Dovato (TN) (P) unclassified
D11659  Tolvaptan sodium phosphate (JAN); Samtasu (TN) (P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (P) unclassified
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11881  Amlodipine benzoate; Katerzia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) unclassified
D12005  Treprostinil palmitil (USAN/INN) (P) unclassified
D12015  St. John's wort; SJW (P) unclassified
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12311  Bortezomib hydrate (JAN) (P) unclassified
D12353  Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) (P) unclassified
D12437  Ripasudil hydrochloride and brimonidine tartrate; Gla-alpha (TN) (P) unclassified
D12494  Foslevodopa and foscarbidopa; Vyalev (TN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (CI,P) unclassified
D12599  Bimatoprost grenod (USAN) (P) unclassified
D12617  Sepetaprost (JAN/INN) (P) unclassified
D12629  Treprostinil phosphate (USAN); Treprostinil biphosphate (P) unclassified
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4