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Drug interaction list


Query:
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN)

Interactions: 1275 hits    [ ATC classification | Therapeutic category ]

C00220  Methylene blue; Methylthioninium chloride (P) unclassified
C04931  Argatroban; (2R,4R)-4-Methyl-1[Nalpha-[(3-methyl-1,2,3,4-tetrahydro-8-quinolinyl)sulfonyl]-L-arginyl]-2-piperadinecarboxylic acid (P) unclassified
C06174  Codeine; (5alpha,6alpha)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol (P) unclassified
C07005  Flunisolide; Flunisolide anhydrous (P) unclassified
C07051  Indinavir (P) unclassified
C07547  Tubocurarine (P) unclassified
C07548  Atracurium (P) unclassified
C07551  Pancuronium (P) unclassified
C07553  Vecuronium (P) unclassified
D00066  Progesterone (JP18/USP/INN); Crinone (TN); Prometrium (TN) (P) unclassified
D00067  Estrone (JAN/USP/INN); Estrone (TN) (P) unclassified
D00088  Hydrocortisone (JP18/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) (P) CYP induction: CYP3A
D00094  Tretinoin (JAN/USP/INN); Avita (TN); Renova (TN); Retin A (TN); Tretinoin (TN) (P) unclassified
D00104  Chloramphenicol (JP18/USP/INN); Amphicol (TN); Chloromycetin (TN); Econochlor (TN) (P) unclassified
D00105  Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) (P) unclassified
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) (P) unclassified
D00109  Aspirin (JP18/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) (P) unclassified
D00118  Naproxen (JP18/USP/INN); Naprosyn (TN) (P) unclassified
D00123  Cyanamide (JP18); Cyanamide (TN) (P) unclassified
D00129  Calcitriol (JAN/USP/INN); Rocaltrol (TN) (P) unclassified
D00131  Disulfiram (JP18/USP/INN); Antabuse (TN) (P) unclassified
D00134  Albendazole (JAN/USP/INN); Albenza (TN) (P) unclassified
D00136  Haloperidol (JP18/USP/INN); Haldol (TN) (P) unclassified
D00140  Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) (P) CYP induction: CYP3A
D00142  Methotrexate (JP18/USP/INN); Otrexup (TN); Xatmep (TN) (P) unclassified
D00165  Hydrocortisone acetate (JP18/USP); Cortifoam (TN); U-cort (TN) (P) CYP induction: CYP3A
D00181  Argatroban (USP); Argatroban hydrate (JP18); Novastan (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) unclassified
D00186  Ciprofloxacin (JP18/USP/INN); Cipro (TN); Otiprio (TN) (P) unclassified
D00195  Codeine (USP); Codeine hydrate (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) unclassified
D00216  Acarbose (JAN/USAN/INN); Precose (TN) (P) unclassified
D00217  Acetaminophen (JP18/USP); Paracetamol (INN); Tylenol (TN) (P) unclassified
D00218  Acetazolamide (JP18/USP/INN); Diamox (TN) (P) unclassified
D00219  Acetohexamide (JP18/USP/INN); Dymelor (TN) (P) unclassified
D00224  Allopurinol (JP18/USP/INN); Zyloprim (TN) (P) unclassified
D00225  Alprazolam (JP18/USP/INN); Xanax (TN) (P) CYP induction: CYP3A
D00227  Aminophylline (USP/INN); Somophyllin (TN); Theophylline ethylenediamine (TN) (P) unclassified
D00228  Amoxapine (JP18/USP/INN); Asendin (TN) (P) unclassified
D00234  Astemizole (JAN/USP/INN); Hismanal (TN) (P) CYP induction: CYP3A
D00244  Betamethasone (JP18/USP/INN); Celestone (TN); Rinderon (TN) (P) unclassified
D00246  Budesonide (JP18/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) (P) unclassified
D00252  Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00255  Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) (P) Enzyme: CYP2C9
D00271  Chlorpropamide (JP18/USP/INN); Diabinese (TN) (P) unclassified
D00274  Cisapride (USP/INN) (P) CYP induction: CYP3A
D00275  Cisplatin (JP18/USP/INN); Platinol (TN) (P) unclassified
D00276  Clarithromycin (JP18/USP/INN); Biaxin (TN) (P) unclassified
D00280  Clonazepam (JP18/USP/INN); Klonopin (TN) (P) unclassified
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) unclassified
D00285  Co-Trimoxazole (BAN); Sulfamethoxazole and trimethoprim; Bactrim (TN); Septra (TN) (P) CYP inhibition: CYP2C9
D00287  Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) unclassified
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) unclassified
D00294  Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) (P) unclassified
D00295  Cimetidine (JP18/USP/INN); Tagamet (TN) (P) unclassified
D00297  Digitoxin (JAN/USP/INN); Crystodigin (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D00298  Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) (P) Transporter induction: ABCB1
D00302  Dipyridamole (JP18/USP/INN); Persantine (TN) (P) unclassified
D00303  Disopyramide (JP18/USAN/INN); Rythmodan P (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00304  Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) (P) unclassified
D00307  Doxycycline (USP); Doxycycline hydrate; Monodox (TN); Oracea (TN); Vibramycin (TN) (P) unclassified
D00311  Estazolam (JP18/USP/INN); ProSom (TN) (P) CYP induction: CYP3A
D00312  Estrone sodium sulfate; Sodium estrone sulfate (P) unclassified
D00316  Etretinate (JAN/USAN/INN); Tegison (TN) (P) unclassified
D00319  Felodipine (JP18/USP/INN); Plendil (TN) (P) unclassified
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) unclassified
D00321  Finasteride (JAN/USP/INN); Propecia (TN); Proscar (TN) (P) unclassified
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP2C9
D00324  Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) (P) unclassified
D00326  Fluoxetine (USAN/INN); Fluoxetine (TN) (P) Enzyme: CYP2C9
D00335  Glipizide (USP/INN); Glucotrol (TN) (P) unclassified
D00336  Glyburide (USP); Glibenclamide (JP18/INN); Diabeta (TN); Glynase (TN); Micronase (TN) (P) Enzyme: CYP2C9
D00343  Ifosfamide (JAN/USP/INN); Ifex (TN) (P) unclassified
D00346  Isoniazid (JP18/USP/INN); Laniazid (TN) (P) unclassified
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) unclassified
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) unclassified
D00354  Lamotrigine (JAN/USP/INN); Lamictal (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00355  Lansoprazole (JP18/USP/INN); Prevacid (TN) (P) unclassified
D00358  Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00359  Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) (P) unclassified
D00364  Loratadine (JAN/USP/INN); Claritin (TN) (P) unclassified
D00371  Theophylline (JP18); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) (P) unclassified
D00379  Tolazamide (JAN/USP/INN); Tolinase (TN) (P) unclassified
D00380  Tolbutamide (JP18/USP/INN); Orinase (TN) (P) unclassified
D00385  Triamcinolone (JP18/USP/INN); Aristocort (TN); Kenacort (TN) (P) unclassified
D00387  Triazolam (JP18/USP/INN); Halcion (TN) (P) unclassified
D00394  Trimipramine (USAN/INN) (P) unclassified
D00395  Troglitazone (JAN/USAN/INN); Rezulin (TN) (P) unclassified
D00399  Valproic acid (USP); Depakene (TN) (P) unclassified
D00407  Methylprednisolone (JP18/USP/INN); Medrol (TN) (P) unclassified
D00409  Metronidazole (JP18/USP/INN); Flagyl (TN); Noritate (TN); Nuvessa (TN); Vandazole (TN) (P) CYP inhibition: CYP2C9
D00413  Zidovudine (JP18/USP/INN); Azidothymidine; Retrovir (TN) (P) unclassified
D00416  Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) (P) CYP inhibition: CYP2C9
D00424  Rifabutin (JAN/USP/INN); Mycobutin (TN) (P) unclassified
D00426  Risperidone (JP18/USP/INN); Risperdal (TN) (P) unclassified
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) CYP induction: CYP2C9 CYP3A
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (P) Transporter induction: ABCB1
D00434  Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) (P) unclassified
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) CYP induction: CYP2B6
D00437  Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) unclassified
D00438  Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) (P) unclassified
D00446  Sucralfate (USP/INN); Sucralfate hydrate (JP18); Carafate (TN) (P) unclassified
D00453  Ofloxacin (JP18/USP/INN); Floxin (TN) (P) unclassified
D00455  Omeprazole (JP18/USP/INN); Prilosec (TN) (P) unclassified
D00456  Ondansetron (JAN/USP/INN); Zofran ODT (TN) (P) unclassified
D00457  Quazepam (JAN/USP/INN); Doral (TN) (P) Enzyme: CYP2C9
D00458  Quetiapine fumarate (JP18/USP); Seroquel (TN) (P) unclassified
D00465  Oxybutynin (USAN/INN); Anturol (TN); Oxytrol (TN) (P) unclassified
D00471  Praziquantel (JAN/USP/INN); Biltricide (TN) (P) unclassified
D00472  Prednisolone (JP18/USP/INN); Delta-cortef (TN) (P) CYP induction: CYP3A
D00484  Protriptyline hydrochloride (USP); Vivactil (TN) (P) unclassified
D00491  Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) (P) unclassified
D00492  Pancuronium bromide (JP18/USP/INN); Pavulon (TN) (P) unclassified
D00510  Phenylbutazone (JP18/USP/INN); Azolid (TN) (P) CYP inhibition: CYP2C9
D00521  Terfenadine (JAN/USAN/INN); Seldane (TN) (P) CYP induction: CYP3A
D00528  Caffeine (USP); Anhydrous caffeine (JP18); Anhydrous caffeine (TN); Respia (TN) (P) unclassified
D00529  Montelukast sodium (JP18/USP); Singulair (TN) (P) Enzyme: CYP2C9
D00530  Zaleplon (JAN/USP/INN); Sonata (TN) (P) unclassified
D00533  Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00535  Vigabatrin (JAN/USP/INN); Sabril (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00538  Zonisamide (JP18/USP/INN); Excegran (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A / CYP induction: CYP3A
D00539  Ethosuximide (JP18/USP/INN); Zarontin (TN) (P) unclassified
D00542  Halothane (JP18/USP/INN); Fluothane (TN) (P) unclassified
D00544  Methoxyflurane (USP/INN); Penthrane (TN) (P) unclassified
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) unclassified
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) unclassified
D00560  Pimozide (JP18/USP/INN); Orap (TN) (P) unclassified
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) unclassified
D00564  Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) (P) Enzyme: CYP2C9
D00570  Colchicine (JP18/USP); Colchicine (TN) (P) Transporter induction: ABCB1
D00578  Voriconazole (JP18/USP/INN); Vfend (TN) (P) unclassified
D00584  Fluorouracil (JP18/USP/INN); 5-FU (TN); Adrucil (TN); Carac (TN); Fluoroplex (TN) (P) unclassified
D00585  Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) (P) unclassified
D00592  Dapsone (USP); Diaphenylsulfone (JAN); Aczone (TN) (P) unclassified
D00593  Glimepiride (JP18/USP/INN); Amaryl (TN) (P) Enzyme: CYP2C9
D00594  Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) (P) unclassified
D00595  Buformin (USAN/INN) (P) unclassified
D00596  Rosiglitazone maleate (JAN/USP); Avandia (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) unclassified
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) (P) unclassified
D00616  Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) (P) unclassified
D00617  Nicardipine hydrochloride (JP18/USAN); Cardene (TN) (P) unclassified
D00618  Nisoldipine (JAN/USAN/INN); Sular (TN) (P) unclassified
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Transporter induction: ABCB1
D00625  Miglitol (JP18/USAN/INN); Glyset (TN) (P) unclassified
D00629  Nitrendipine (JP18/USAN/INN); Baypress (TN) (P) unclassified
D00631  Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) (P) Enzyme: CYP2C9
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00637  Disopyramide phosphate (JAN/USP); Norpace (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00638  Flecainide acetate (JP18/USP); Tambocor (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00639  Mexiletine hydrochloride (JP18/USP); Mexitil (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00640  Propafenone hydrochloride (JP18/USP); Rythmol (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00642  Quinidine gluconate (USP); Quinaglute (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00643  Quinidine polygalacturonate; Cardioquin (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D00646  Tolterodine (USAN/INN) (P) unclassified
D00653  Dorzolamide hydrochloride (JP18/USP); Trusopt (TN) (P) Enzyme: CYP2C9
D00661  Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) (P) unclassified
D00664  Cetirizine hydrochloride (JP18/USP); Zyrtec (TN) (P) Transporter induction: ABCB1
D00668  Dexchlorpheniramine maleate (USP); d-Chlorpheniramine maleate (JP18); Mylaramine (TN); Polaramine (TN) (P) CYP induction: CYP3A
D00670  Donepezil hydrochloride (JP18/USP); Aricept (TN) (P) unclassified
D00674  Naratriptan hydrochloride (JAN/USP); Amerge (TN) (P) Enzyme: CYP2C9
D00677  Granisetron hydrochloride (JAN/USP); Kytril (TN) (P) unclassified
D00678  Ondansetron hydrochloride hydrate (JAN/USP); Ondansetron hydrochloride; Zofran (TN) (P) unclassified
D00679  Ergotamine tartrate (JP18/USP); Ergomar (TN) (P) unclassified
D00680  Methylergonovine maleate (USP); Methylergometrine maleate (JP18); Methergine (TN) (P) unclassified
D00687  Salmeterol xinafoate (JAN/USP); Serevent (TN) (P) unclassified
D00689  Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18); Beclovent (TN); Qnasl (TN); Vanceril (TN) (P) unclassified
D00690  Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) (P) unclassified
D00696  Midazolam hydrochloride (USAN); Versed (TN) (P) unclassified
D00706  Zolpidem tartrate (JP18/USP); Ambien (TN); Intermezzo (TN) (P) unclassified
D00707  Fomepizole (JAN/USAN/INN); Antizol (TN) (P) CYP inhibition: CYP2C9
D00710  Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) (P) unclassified
D00722  Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18); Ditropan (TN); Gelnique (TN) (P) unclassified
D00724  Rabeprazole sodium (JP18/USP); Aciphex (TN); Pariet (TN) (P) unclassified
D00725  Dolasetron mesylate (USP); Anzemet (TN) (P) CYP induction: CYP3A
D00729  Loperamide hydrochloride (JAN/USP); Imodium (TN) (P) Transporter induction: ABCB1
D00746  Interferon beta-1b (USAN/INN); Interferon beta-1b (genetical recombination) (JAN); Betaseron (TN); Extavia (TN) (P) unclassified
D00749  Leflunomide (JAN/USP/INN); Arava (TN) (P) CYP inhibition: CYP2C9
D00751  Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) (P) unclassified
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (P) Transporter induction: ABCB1
D00758  Atracurium besylate (USP); Atracurium besilate (INN); Tracrium (TN) (P) unclassified
D00759  Cisatracurium besylate (USP); Cisatracurium besilate (INN); Nimbex (TN) (P) unclassified
D00760  Doxacurium chloride (USAN/INN); Nuromax (TN) (P) unclassified
D00763  Mivacurium chloride (USAN/INN); Mivacron (TN) (P) unclassified
D00764  Pipecuronium bromide (JAN/USAN/INN); Arduan (TN) (P) unclassified
D00765  Rocuronium bromide (JAN/USP/INN); Zemuron (TN) (P) unclassified
D00767  Vecuronium bromide (JAN/USP/INN); Norcuron (TN) (P) unclassified
D00769  Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18); Clopidogrel hydrogen sulphate; Isocover (TN); Plavix (TN) (P) CYP induction: CYP2B6
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) (P) unclassified
D00781  Entacapone (JP18/USP/INN); Comtan (TN) (P) CYP inhibition: CYP2C9
D00783  Botulinum toxin type A (JAN); Botox (TN); Dysport (TN) (P) unclassified
D00785  Selegiline hydrochloride (JAN/USP); Eldepryl (TN) (P) CYP induction: CYP2B6
D00794  Loxapine succinate (USP); Loxitane (TN) (P) unclassified
D00804  Ivermectin (JAN/USP/INN); Sklice (TN); Soolantra (TN); Stromectol (TN) (P) Transporter induction: ABCB1
D00809  Amitriptyline hydrochloride (JP18/USP); Elavil (TN) (P) unclassified
D00811  Clomipramine hydrochloride (JP18/USP); Anafranil (TN) (P) unclassified
D00812  Desipramine hydrochloride (JAN/USP); Norpramin (TN) (P) unclassified
D00814  Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) (P) Enzyme: CYP2C9
D00815  Imipramine hydrochloride (JP18/USP); Tofranil (TN) (P) unclassified
D00816  Nortriptyline hydrochloride (JP18/USP/INN); Pamelor (TN) (P) unclassified
D00818  Maprotiline hydrochloride (JP18/USP); Ludiomil (TN) (P) unclassified
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) unclassified
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) unclassified
D00822  Citalopram hydrobromide (USP); Celexa (TN) (P) Transporter induction: ABCB1
D00823  Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) (P) Enzyme: CYP2C9
D00824  Fluvoxamine maleate (JP18/USP); Luvox (TN) (P) unclassified
D00825  Sertraline hydrochloride (JAN/USP); Zoloft (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) CYP induction: CYP3A
D00836  Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) (P) unclassified
D00840  Levomethadyl acetate hydrochloride (USAN); Orlaam (TN) (P) unclassified
D00847  Oxycodone hydrochloride (USP); Oxecta (TN); Oxycontin (TN); Roxicodone (TN) (P) unclassified
D00851  Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) (P) CYP induction: CYP3A
D00882  Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) (P) CYP inhibition: CYP2C9
D00887  Atorvastatin calcium anhydorous; Lipitor (TN) (P) Transporter induction: ABCB1
D00889  Cerivastatin sodium (JAN/USAN); Baycol (TN) (P) unclassified
D00892  Fluvastatin sodium (JAN/USP); Lescol (TN) (P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) unclassified
D00895  Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) (P) CYP induction: CYP3A
D00896  Efavirenz (JAN/USP/INN); Sustiva (TN) (P) CYP induction: CYP2B6
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) unclassified
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) unclassified
D00944  Metformin hydrochloride (JP18/USP); Glucophage (TN) (P) unclassified
D00945  Pioglitazone hydrochloride (JP18/USP); Actos (TN) (P) unclassified
D00948  Estropipate (USP); Piperazine estrone sulfate; Ogen (TN) (P) unclassified
D00950  Levonorgestrel (JAN/USP/INN); Mirena (TN); Norplant (TN); Skyla (TN) (P) unclassified
D00960  Anastrozole (JP18/USP/INN); Arimidex (TN) (P) CYP inhibition: CYP2C9
D00963  Exemestane (JAN/USP/INN); Aromasin (TN) (P) unclassified
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) unclassified
D00966  Tamoxifen citrate (JP18/USP); Nolvadex (TN); Soltamox (TN) (P) unclassified
D00967  Toremifene citrate (JAN/USAN); Fareston (TN) (P) unclassified
D00969  Meloxicam (JAN/USP/INN); Mobic (TN) (P) Enzyme: CYP2C9
D00972  Betamethasone sodium phosphate (JP18/USP); Celestone (TN) (P) unclassified
D00973  Cortisone acetate (JP18/USP); Cortone acetate (TN) (P) unclassified
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) unclassified
D00976  Hydrocortisone cypionate (P) CYP induction: CYP3A
D00977  Hydrocortisone sodium phosphate (JP18/USP); Hydrocortone phosphate (TN) (P) CYP induction: CYP3A
D00978  Hydrocortisone sodium succinate (JP18/USP); A-hydrocort (TN); Solu-cortef (TN) (P) CYP induction: CYP3A
D00979  Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) (P) unclassified
D00981  Prednisolone sodium phosphate (JP18/USP); Pediapred (TN) (P) unclassified
D00983  Triamcinolone acetonide (JP18/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) (P) unclassified
D00986  Fludrocortisone acetate (JP18/USP); Florinef acetate (TN) (P) unclassified
D00987  Cabergoline (JP18/USP/INN); Cabaser (TN); Dostinex (TN) (P) unclassified
D01007  Propiverine hydrochloride (JP18); Bup-4 (TN); Mictonorm (TN) (P) unclassified
D01010  Levothyroxine sodium (USP); Levothyroxine sodium hydrate (JP18); Levothroid (TN); Levoxyl (TN); Synthroid (TN) (P) unclassified
D01011  Liothyronine sodium (JP18/USP); Cytomel (TN); Triostat (TN) (P) unclassified
D01012  Dried thyroid (JP18); Thyradin (TN) (P) unclassified
D01028  Ticlopidine hydrochloride (JP18/USP); Ticlid (TN) (P) unclassified
D01056  Benzbromarone (JP18/USAN/INN); Uroleap (TN) (P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01068  Vinblastine sulfate (JP18/USP); Exal (TN); Velban (TN) (P) unclassified
D01072  Chloramphenicol palmitate (JP18/USP); Chloromycetin palmitate (TN) (P) unclassified
D01078  Telithromycin (JAN/USAN/INN); Ketek (TN) (P) CYP induction: CYP3A
D01092  Lanoconazole (JP18/INN); Latoconazole; Astat (TN) (P) CYP inhibition: CYP2C9
D01098  Maxacalcitol (JAN/USAN/INN); Oxarol (TN); Prezios (TN) (P) unclassified
D01101  Bromperidol (JAN/USAN/INN); Impromen (TN) (P) unclassified
D01104  Barnidipine hydrochloride (JAN); Hypoca (TN) (P) unclassified
D01110  Melitracen hydrochloride (JAN/USAN) (P) unclassified
D01111  Nateglinide (JP18/USP/INN); Starsis (TN) (P) Enzyme: CYP2C9
D01115  Eplerenone (JP18/USAN/INN); Inspra (TN) (P) unclassified
D01121  Rebamipide (JP18/INN); Mucosta (TN) (P) unclassified
D01131  Lafutidine (JP18/INN); Protecadin (TN) (P) unclassified
D01145  Azelnidipine (JP18/INN); Calblock (TN) (P) unclassified
D01148  Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) (P) unclassified
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (P) Transporter induction: ABCB1
D01161  Fulvestrant (JAN/USP/INN); Faslodex (TN) (P) unclassified
D01163  Ergonovine maleate (USP); Ergometrine maleate (JP18); Ergometrine (TN) (P) unclassified
D01164  Aripiprazole (JAN/USP/INN); Abilify (TN) (P) unclassified
D01173  Cilnidipine (JP18/INN); Atelec (TN) (P) unclassified
D01176  Blonanserin (JAN/INN); AD 5423 (P) unclassified
D01196  Acetazolamide sodium (JAN); Diamox (TN) (P) unclassified
D01204  Olmesartan medoxomil (JP18/USP); Benicar (TN); Olmetec (TN) (P) Transporter induction: ABCB1
D01207  Omeprazole sodium (USAN); Losec sodium (TN) (P) unclassified
D01211  Leucovorin calcium (USP); Calcium folinate (JP18); Uzel (TN); Wellcovorin (TN) (P) unclassified
D01213  Tolvaptan (JAN/USAN/INN); Samsca (TN) (P) Transporter induction: ABCB1
D01215  Alcuronium chloride (JAN/USAN/INN); Alloferin (TN) (P) unclassified
D01217  Dydrogesterone (JP18/USP/INN); Duphaston (TN); Gynorest (TN) (P) unclassified
D01223  Capecitabine (JAN/USP/INN); Xeloda (TN) (P) Enzyme: CYP2C9
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D01236  Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) (P) CYP induction: CYP3A
D01239  Prednisolone sodium succinate (JP18/USP); Kohakusanin (TN) (P) unclassified
D01244  Tegafur (JP18/USAN/INN); Atillon (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) unclassified
D01269  Solifenacin succinate (JAN/USAN/INN); Vesicare (TN) (P) unclassified
D01280  Warfarin potassium (JP18); Athrombin-K (TN) (P) Enzyme: CYP2C9
D01285  Lofepramine hydrochloride (JAN/USAN); Amplit (TN) (P) unclassified
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D01293  Ethyl loflazepate (JP18/INN); Meilax (TN) (P) unclassified
D01296  Methylphenidate hydrochloride (JAN/USP); Concerta (TN); Metadate (TN); Quillivant xr (TN); Ritalin (TN) (P) unclassified
D01309  Doxifluridine (JP18/INN); Furtulon (TN) (P) unclassified
D01314  Dibenzepin hydrochloride (JAN/USAN) (P) unclassified
D01316  Mexazolam (JAN/INN); Melex (TN) (P) unclassified
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) unclassified
D01355  Tramadol hydrochloride (JP18/USP); Ultram (TN) (P) unclassified
D01356  Glymidine sodium (JAN/USAN/INN) (P) unclassified
D01358  Mianserin hydrochloride (JAN/USAN); Tetramide (TN) (P) unclassified
D01361  Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) (P) CYP induction: CYP3A
D01372  Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) (P) unclassified
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) unclassified
D01413  Estradiol valerate (JAN/USP/INN); Deladumone (TN) (P) unclassified
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) unclassified
D01425  Lopinavir (JAN/USP/INN) (P) CYP induction: CYP3A
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP2C9
D01441  Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) (P) unclassified
D01442  Hydrocortisone succinate (JP18) (P) CYP induction: CYP3A
D01450  Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D01453  Caffeine hydrate (JP18); Caffeine monohydrate; Caffeine (TN) (P) unclassified
D01455  Cifenline succinate (USAN); Cibenzoline succinate (JP18); Cibenol (TN); Cipralan (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D01468  Nemonapride (JAN/INN); Emilace (TN) (P) unclassified
D01477  Opipramol hydrochloride (JAN/USAN); Insidon (TN) (P) unclassified
D01478  Ebastine (JP18/USAN/INN); Kestine (TN) (P) unclassified
D01481  Dihydrocodeine phosphate (JP18); Dihydro (TN) (P) unclassified
D01501  Isoniazid calcium pyruvinate (JAN); Pyruvic acid calcium isoniazid (P) unclassified
D01510  Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) (P) unclassified
D01514  Etizolam (JP18/INN); Sedekopan (TN) (P) Enzyme: CYP2C9
D01546  Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Dosulepin (TN) (P) unclassified
D01553  Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) (P) unclassified
D01562  Aranidipine (JAN/INN); Sapresta (TN) (P) unclassified
D01564  Rilmazafone hydrochloride hydrate (JP18); Rilmazafone hydrochloride dihydrate; Rilmazafone hydrochloride; Rhythmy (TN) (P) unclassified
D01599  Gliclazide (JP18/INN); Glimicron (TN) (P) unclassified
D01615  Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) (P) unclassified
D01617  Estradiol dipropionate (JAN); Ovahormon (TN) (P) unclassified
D01619  Hydrocortisone butyrate (JP18/USP); Locoid (TN) (P) CYP induction: CYP3A
D01624  Sarpogrelate hydrochloride (JP18); Anplag (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D01632  Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) (P) unclassified
D01643  Aluminoparaaminosalicylate calcium hydrate (JAN); Aluminoparaaminosalicylate calcium pentahydrate; Aluminoparaaminosalicylate calcium; Alumino nippas calcium (TN) (P) unclassified
D01656  Brovincamine fumarate (JAN); Sabromin (TN) (P) unclassified
D01663  Quinine ethylcarbonate (JP18); Quinine ethylcarbonate (TN) (P) Transporter induction: ABCB1
D01665  Voglibose (JP18/USAN/INN); Basen (TN) (P) unclassified
D01692  Alfuzosin hydrochloride (JAN/USAN); Uroxatral (TN) (P) unclassified
D01697  Colforsin daropate hydrochloride (JAN); Nkh 477; Adehl (TN) (P) CYP induction: CYP3A
D01699  Darifenacin hydrobromide (JAN/USAN); Enablex (TN) (P) unclassified
D01703  Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) (P) unclassified
D01708  Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) (P) unclassified
D01710  Roxithromycin (JP18/USAN/INN); Rulide (TN) (P) CYP induction: CYP3A
D01712  Theophylline sodium acetate (JAN) (P) unclassified
D01744  Brotizolam (JP18/USAN/INN); Lendormin (TN) (P) unclassified
D01745  Domperidone (JP18/USAN/INN); Motilium (TN) (P) unclassified
D01769  Vindesine sulfate (JAN/USAN); Fildesin (TN) (P) CYP induction: CYP3A
D01784  Carmofur (JP18/INN); Mifurol (TN) (P) unclassified
D01787  Sulthiame (USAN); Sultiame (JP18); Ospolot (TN) (P) unclassified
D01799  Glyclopyramide (JAN/INN); Deamelin-S (TN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) CYP inhibition: CYP2C9
D01849  Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) (P) CYP induction: CYP3A
D01854  Mitiglinide calcium hydrate (JP18); Mitiglinide calcium dihydrate; Glufast (TN) (P) unclassified
D01855  Mozavaptane hydrochloride (JAN) (P) unclassified
D01872  Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18); Dopram (TN) (P) unclassified
D01886  Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) (P) CYP induction: CYP3A
D01896  Cilostazol (JP18/USP/INN); Pletal (TN) (P) unclassified
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) unclassified
D01908  Nilvadipine (JP18/USAN/INN); Nivadil (TN) (P) unclassified
D01935  Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) (P) unclassified
D01948  Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) (P) unclassified
D01953  Estradiol benzoate (JP18/USP); Ovahormon (TN) (P) unclassified
D01965  Silodosin (JP18/INN); KMD 3213; Rapaflo (TN); Urief (TN) (P) unclassified
D01973  Eletriptan hydrobromide (JAN/USAN); Relpax (TN) (P) unclassified
D01977  Gefitinib (JP18/USAN/INN); Iressa (TN) (P) unclassified
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) unclassified
D01984  Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN); Esomeprazole magnesium trihydrate; Nexium (TN) (P) unclassified
D01994  Mosapride citrate hydrate (JP18); Mosapride citrate dihydrate; Gasmotin (TN) (P) unclassified
D02002  Isoniazid sodium methanesulfonate hydrate (JAN); Isoniazid sodium methanesulfonate monohydrate; Isoniazid sodium methanesulfonate; IHMS; Neoiscotin (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) unclassified
D02009  Erythromycin lactobionate (JP18/USP); Erythrocin (TN) (P) CYP induction: CYP3A
D02034  Setiptiline maleate (JAN); Tecipul (TN) (P) unclassified
D02045  Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) (P) unclassified
D02086  Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D02092  Cisapride (JAN); Cisapride monohydrate; Propulsid (TN) (P) CYP induction: CYP3A
D02101  Codeine phosphate (USP); Codeine phosphate hydrate (JP18); Codeine (TN) (P) unclassified
D02102  Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6 / Transporter induction: ABCB1
D02114  Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) (P) unclassified
D02129  Doxycycline hyclate (USP); Doxycycline hydrochloride hydrate (JP18); Doryx (TN); Lymepak (TN); Periostat (TN); Vibra-tabs (TN) (P) unclassified
D02131  Tegafur and uracil; Uftoral (TN) (P) unclassified
D02134  Azithromycin hydrate (JP18); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) (P) Transporter induction: ABCB1
D02165  Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) (P) unclassified
D02168  Topotecan hydrochloride (USAN); Nogitecan hydrochloride (JAN); Hycamtin (TN); Potactasol (TN) (P) Transporter induction: ABCB1
D02173  Galantamine hydrobromide (JAN/USP); Razadyne (TN); Reminyl (TN) (P) unclassified
D02174  Dexamethasone acetate (JAN/USP); Decadronal (TN) (P) unclassified
D02175  Compound oxycodone (JP18); Pavinal (TN) (P) unclassified
D02184  Erythromycin stearate (JP18/USP); Bristamycin (TN) (P) CYP induction: CYP3A
D02185  Chloramphenicol sodium succinate (JP18/USP); Chloromycetin succinate (TN) (P) unclassified
D02197  Vincristine sulfate (JP18/USP); VCR; Marqibo (TN); Oncovin (TN); Vincasar (TN); Vincrex (TN) (P) CYP induction: CYP3A
D02204  Hexamethonium bromide (JAN/INN); Hexamethonium bromide (TN) (P) unclassified
D02205  Ethylmorphine hydrochloride hydrate (JP18); Ethylmorphine hydrochloride dihydrate; Ethylmorphine hydrochloride (TN) (P) unclassified
D02206  Buformin hydrochloride (JP18); Dibetos-B (TN) (P) unclassified
D02207  Tubocurarine chloride (USP); Tubocurarine chloride hydrate (JAN); Tubocurarine chloride (TN) (P) unclassified
D02211  Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18); Migranal (TN); Trudhesa (TN) (P) unclassified
D02216  Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP18); Ciloxan (TN); Cipro (TN); Proquin XR (TN) (P) unclassified
D02219  Terbinafine hydrochloride (JP18/USP); Lamisil (TN) (P) Enzyme: CYP2C9
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) unclassified
D02258  Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) (P) Transporter induction: ABCB1
D02260  Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18); Paxil (TN) (P) unclassified
D02261  Quinine hydrochloride hydrate (JP18); Quinine hydrochloride dihydrate; Quinine hydrochloride (TN) (P) Transporter induction: ABCB1
D02262  Quinine sulfate (USP); Quinine sulfate hydrate (JP18); Quinine hydrogen sulfate; Coco-quinine (TN) (P) Transporter induction: ABCB1
D02268  Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18); Circanol (TN); Hydergine (TN); Inorter (TN) (P) unclassified
D02272  Quinidine sulfate (USP); Quinidine sulfate hydrate (JP18); Quinidex (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D02274  Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18); Dantrium (TN); Ryanodex (TN) (P) CYP induction: CYP3A
D02288  Hydrocortisone valerate (USP); Westcort (TN) (P) CYP induction: CYP3A
D02292  Gallamine triethiodide (USP); Flaxedil (TN) (P) unclassified
D02312  Methylene blue (USP); Methylthioninium chloride; Methylthioninium chloride proveblue (TN) (P) CYP inhibition: CYP2C9
D02340  Loxapine (USAN/INN); Adasuve (TN) (P) unclassified
D02347  Dantrolene (USAN/INN) (P) CYP induction: CYP3A
D02356  Verapamil (USAN/INN) (P) Transporter induction: ABCB1
D02360  Sertraline (INN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D02362  Paroxetine (USP/INN); Paroxetine (TN) (P) unclassified
D02375  Terbinafine (USAN/INN); Lamasil (TN) (P) Enzyme: CYP2C9
D02404  Procaterol hydrochloride (USAN); Pro-Air (TN) (P) unclassified
D02408  Trimipramine maleate (JAN/USP); Surmontil (TN) (P) unclassified
D02416  Aluminum hydroxide (USP); Aluminum hydroxide, dried (USP); Dried aluminum hydroxide gel (JP18); ALterna GEL (TN); Dialume (TN) (P) unclassified
D02425  Carbutamide (INN); Invenol (TN) (P) unclassified
D02427  Glibornuride (USAN/INN); Glutril (TN) (P) unclassified
D02430  Gliquidone (INN); Glurenorm (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (CI,P) CYP induction: CYP3A
D02497  Fosamprenavir (INN) (P) unclassified
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) CYP induction: CYP3A
D02501  Caspofungin acetate (JAN/USAN); Cancidas (TN) (P) unclassified
D02523  Erythromycin acistrate (USAN); Erasis (TN) (P) CYP induction: CYP3A
D02524  Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) (P) CYP induction: CYP3A
D02525  Erythromycin propionate (USAN) (P) CYP induction: CYP3A
D02537  Dronedarone (INN) (P) CYP induction: CYP3A
D02554  Rifaximin (JAN/USAN/INN); Xifaxan (TN) (P) Transporter induction: ABCB1
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) Transporter induction: ABCB1
D02561  Moclobemide (USAN/INN); Aurorix (TN) (P) unclassified
D02562  Rasagiline mesylate (USAN); Rasagiline mesilate (JAN); Azilect (TN) (P) unclassified
D02565  Dimetacrine (INN) (P) unclassified
D02566  Maprotiline (USAN) (P) unclassified
D02567  Escitalopram oxalate (JAN/USP); Lexapro (TN) (P) unclassified
D02570  Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) (P) unclassified
D02577  Flibanserin (USAN/INN); Addyi (TN) (P) unclassified
D02587  Metildigoxin (JP18); Lanirapid (TN) (P) Transporter induction: ABCB1
D02591  Dexamethasone acefurate (USAN/INN) (P) unclassified
D02592  Dexamethasone beloxil (USAN) (P) unclassified
D02593  Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN); Protonix (TN) (P) unclassified
D02615  Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital; Vegetamin (TN) (P) CYP induction: CYP3A
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) unclassified
D02626  Bromperidol decanoate (USAN) (P) unclassified
D02666  Iloperidone (USAN/INN); Fanapt (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02704  Tampramine fumarate (USAN) (P) unclassified
D02714  Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) (P) Transporter induction: ABCB1
D02731  Vardenafil dihydrochoride (USAN); Levitra (TN) (P) unclassified
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) unclassified
D02735  Rimabotulinumtoxin B (USAN); Botulinum toxin type B (JAN); Myobloc (TN) (P) unclassified
D02740  Lidocaine and prilocaine; Lidocaine and propitocaine; Emla (TN); Oraqix (TN); Lidocaine and prilocaine (TN) (P) unclassified
D02824  Almotriptan (USAN) (P) unclassified
D02825  Almotriptan malate (USP); Axert (TN) (P) unclassified
D02829  Alosetron hydrochloride (USAN); Lotrpnex (TN) (P) Enzyme: CYP2C9
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) unclassified
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (P) unclassified
D02910  Amiodarone (USAN/INN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D02914  Amlodipine maleate (USAN); Amvaz (TN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) CYP induction: CYP2C9
D02972  Aptazapine maleate (USAN) (P) unclassified
D03038  Azipramine hydrochloride (USAN) (P) unclassified
D03071  Beloxepin (USAN/INN) (P) unclassified
D03098  Berythromycin (USAN/INN); Erythromycin B (P) CYP induction: CYP3A
D03164  Bromindione (USAN/INN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) unclassified
D03199  Butriptyline hydrochloride (USAN) (P) unclassified
D03208  Aliskiren (USAN/INN); Rasilez (TN) (P) Transporter induction: ABCB1
D03213  Apixaban (JAN/USAN/INN); Eliquis (TN) (P) Transporter induction: ABCB1
D03215  Armodafinil (USAN/INN); Nuvigil (TN) (P) unclassified
D03217  Avanafil (USAN/INN); Stendra (TN); Spedra (TN) (P) unclassified
D03218  Axitinib (JAN/USAN); Inlyta (TN) (P) unclassified
D03230  Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) (P) unclassified
D03250  Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) (P) unclassified
D03252  Bosutinib (USAN) (P) unclassified
D03259  Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN); Mylotarg (TN) (P) unclassified
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (P) unclassified
D03325  Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) (P) unclassified
D03368  Calcium para-aminosalicylate (JP18); Nippas calcium (TN) (P) unclassified
D03415  Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) (P) Enzyme: CYP2C9
D03461  Chloramphenicol pantothenate complex (USAN/INN); Pantofenicol (TN) (P) unclassified
D03491  Cidoxepin hydrochloride (USAN) (P) unclassified
D03492  Cifenline (USAN); Cibenzoline (INN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D03503  Cimetidine hydrochloride (USP); Cimetidine hydrochloride (TN) (P) unclassified
D03504  Cinacalcet (USAN) (P) unclassified
D03505  Cinacalcet hydrochloride (JAN/USAN); Sensipar (TN); Mimpara (TN) (P) unclassified
D03579  Codeine polistirex (USAN) (P) unclassified
D03580  Codeine sulfate (USP); Codeine sulfate trihydrate; Codeine sulfate (TN) (P) unclassified
D03584  Colforsin (USAN/INN) (P) CYP induction: CYP3A
D03654  Darifenacin (USAN/INN) (P) unclassified
D03656  Darunavir (USAN/INN) (P) unclassified
D03657  Dasantafil (USAN/INN) (P) unclassified
D03658  Dasatinib (JAN/INN) (P) unclassified
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) unclassified
D03671  Deflazacort (USAN/INN); Emflaza (TN) (P) Transporter induction: ABCB1
D03725  Hydrocodone bitartrate (USP); Hydrocodone bitartrate hemipentahydrate; Dicodid (TN) (P) CYP induction: CYP2B6
D03730  Dexrazoxane (JAN/USAN/INN) (P) unclassified
D03731  Selegiline (USAN/INN); Emsam (TN) (P) CYP induction: CYP2B6
D03783  Oxycodone terephthalate (USP) (P) unclassified
D03798  Dicumarol (USAN); Dicoumarol (INN); Dicumarol (TN) (P) unclassified
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) unclassified
D03820  Dutasteride (JAN/USP/INN); Avodart (TN) (P) unclassified
D03825  Dihydrocodeine bitartrate (USP) (P) unclassified
D03830  Diltiazem malate (USAN); Tiamate (TN) (P) unclassified
D03833  Indinavir (USAN); Indinavir hydrate (P) unclassified
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) unclassified
D03837  Fosamprenavir sodium (USAN) (P) unclassified
D03844  Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP3A CYP2B6
D03852  Droperidol and fentanyl citrate; Innovar (TN) (P) unclassified
D03903  Doxycycline calcium (USP) (P) unclassified
D03904  Doxycycline fosfatex (USAN) (P) unclassified
D03914  Dronedarone hydrochloride (USP); Multaq (TN) (P) CYP induction: CYP3A
D03917  Drospirenone (JAN/USP/INN); Slynd (TN) (P) unclassified
D03960  Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (P) unclassified
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Transporter induction: ABCB1
D04048  Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D04052  Epinephrine and lidocaine hydrochloride; Adrenaline and lidocaine hydrochloride; Xylocaine (TN) (P) unclassified
D04054  Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate (P) CYP induction: CYP3A
D04056  Esomeprazole sodium (USAN); Nexium IV (TN) (P) unclassified
D04061  Estradiol acetate (USAN); Femring (TN) (P) unclassified
D04063  Estradiol cypionate (USP); Depo-estradiol (TN) (P) unclassified
D04064  Estradiol enanthate (USAN) (P) unclassified
D04065  Estradiol undecylate (USAN/INN); Delestrec (TN) (P) unclassified
D04070  Estrogens, conjugated (JAN/USP); Conjugated estrogens; Premarin (TN) (P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9
D04121  Exenatide (JAN/USAN/INN); Byetta (TN) (P) unclassified
D04148  Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) (P) CYP induction: CYP2B6
D04197  Floxuridine (USP/INN); FUDR (TN) (P) unclassified
D04214  Flunisolide acetate (USAN) (P) unclassified
D04292  Galantamine (USAN/INN); Reminyl (TN) (P) unclassified
D04300  Ganaxolone (USAN/INN); Ztalmy (TN) (P) CYP induction: CYP2B6
D04313  Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate; Huscode (TN) (P) unclassified
D04314  Gepirone hydrochloride (USAN); Exxua (TN) (P) unclassified
D04338  Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride; Sekicode (TN) (P) unclassified
D04340  Dextromethorphan hydrobromide and potassium cresolsulfonate; Medicon (TN) (P) unclassified
D04370  Granisetron (JAN/USAN/INN); Sancuso (TN) (P) unclassified
D04403  Guar gum (NF) (P) unclassified
D04435  Hexafluorenium bromide (USAN); Hexafluronium bromide (INN); Mylaxen (TN) (P) unclassified
D04446  Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) (P) unclassified
D04447  Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) (P) unclassified
D04461  Hydrocodone polistirex (USAN) (P) CYP induction: CYP2B6
D04463  Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) (P) Enzyme: CYP2C9
D04467  Hydrocortisone hemisuccinate (USP) (P) CYP induction: CYP3A
D04475  Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) (P) unclassified
D04477  Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) (P) unclassified
D04482  Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) (P) unclassified
D04483  Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) (P) unclassified
D04484  Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) (P) unclassified
D04539  Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) (P) unclassified
D04540  Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) (P) unclassified
D04541  Insulin human, isophane (USP) (P) unclassified
D04542  Insulin human zinc (USP) (P) unclassified
D04543  Insulin human zinc, extended (USP) (P) unclassified
D04547  Insulin, isophane (USP); Isophane insulin human (genetical recombination) injectable aqueous suspension (JP18); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) (P) unclassified
D04550  Insulin zinc, prompt (USP); Semilente iletin (TN) (P) unclassified
D04551  Insulin zinc (USP); Lente iletin (TN) (P) unclassified
D04554  Interferon beta-1a (USAN); Interferon beta-1a (genetical recombination) (JAN); Avonex (TN); Rebif (TN) (P) unclassified
D04556  Intriptyline hydrochloride (USAN) (P) unclassified
D04605  Iprindole (USAN/INN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) unclassified
D04645  Ixabepilone (JAN/USAN/INN); Ixempra (TN) (P) unclassified
D04652  Ketipramine fumarate (USAN) (P) unclassified
D04716  Levomethadyl acetate (USAN); Levacetylmethadol (INN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (P) unclassified
D04813  Lidocaine hydrochloride and epinephrine bitartrate; Lidocaine hydrochloride and adrenaline bitartrate; Ora (TN); Lidosite (TN) (P) unclassified
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) unclassified
D04859  Maribavir (JAN/USAN/INN); Camvia (TN); Livtencity (TN) (P) unclassified
D04895  Mefloquine (USAN/INN) (P) CYP induction: CYP3A
D04966  Metformin (USAN/INN) (P) unclassified
D04999  Methylphenidate (USAN/INN); Daytrana (TN) (P) unclassified
D05000  Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18) (P) unclassified
D05001  Methylprednisolone sodium phosphate (USAN) (P) unclassified
D05002  Methylprednisolone suleptanate (USAN/INN) (P) unclassified
D05016  Metronidazole hydrochloride (USAN); Flagyl I.V. (TN) (P) CYP inhibition: CYP2C9
D05017  Metronidazole phosphate (USAN) (P) CYP inhibition: CYP2C9
D05028  Midazolam maleate (USAN) (P) unclassified
D05029  Midostaurin (JAN/USAN/INN); Rydapt (TN) (P) unclassified
D05143  Nepafenac (JAN/USAN/INN); Nevanac (TN) (P) unclassified
D05152  Netupitant (USAN/INN) (P) CYP induction: CYP3A
D05177  Nitisinone (JAN/USAN/INN); Orfadin (TN) (P) CYP inhibition: CYP2C9
D05231  Octriptyline phosphate (USAN) (P) unclassified
D05246  Olmesartan (USAN/INN) (P) Transporter induction: ABCB1
D05259  Omeprazole magnesium (USP); Prilosec OTC (TN) (P) unclassified
D05261  Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) (P) unclassified
D05284  Oxaprotiline hydrochloride (USAN) (P) unclassified
D05312  Oxycodone (USAN/INN) (P) unclassified
D05333  Paclitaxel poliglumex (USAN/INN) (P) unclassified
D05343  Palonosetron hydrochloride (JAN/USP); Aloxi (TN) (P) unclassified
D05353  Pantoprazole (USAN/INN) (P) unclassified
D05366  Procaterol hydrochloride hydrate (JP18); Meptin (TN) (P) unclassified
D05374  Paroxetine hydrochloride (USP); Paxil (TN) (P) unclassified
D05375  Paroxetine mesylate (USAN); Brisdelle (TN); Pexeva (TN) (P) unclassified
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (P) unclassified
D05429  Aminophylline hydrate (JP18) (P) unclassified
D05457  Phenprocoumon (USAN/INN); Liquamar (TN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP18) (P) unclassified
D05594  Pramlintide (USAN/INN) (P) unclassified
D05595  Pramlintide acetate (USAN); Symlin (TN) (P) unclassified
D05622  Proinsulin human (USAN) (P) unclassified
D05681  Quinine ascorbate (USAN); Quinine biascorbate (P) Transporter induction: ABCB1
D05700  Ranolazine (USAN/INN); Ranexa (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D05701  Ranolazine hydrochloride (USAN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D05703  Rapacuronium bromide (USAN/INN); Raplon (TN) (P) unclassified
D05744  Roflumilast (JAN/USAN/INN); Daliresp (TN); Zoryve (TN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D05792  Salmeterol (USAN/INN) (P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) CYP inhibition: CYP2C9
D05932  Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) (P) unclassified
D05987  Synthetic conjugated estrogens, B (USAN); Enjuvia (TN) (P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (P) unclassified
D06103  Theophylline (USP); Theophylline monohydrate; Accurbron (TN) (P) unclassified
D06104  Theophylline sodium glycinate (USP); Asbron (TN) (P) unclassified
D06177  Tolbutamide sodium, sterile; Orinase diagnostic (TN) (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (P) unclassified
D06272  Sorafenib tosylate (USAN); Sorafenib tosilate (JAN); Nexavar (TN) (P) unclassified
D06273  Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) (P) unclassified
D06304  Vindesine (USAN/INN) (P) CYP induction: CYP3A
D06305  Vinepidine sulfate (USAN) (P) unclassified
D06306  Vinglycinate sulfate (USAN) (P) unclassified
D06307  Vinleurosine sulfate (USAN) (P) unclassified
D06308  Vinrosidine sulfate (USAN) (P) unclassified
D06309  Vinzolidine sulfate (USAN) (P) unclassified
D06315  Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) (P) unclassified
D06390  Azithromycin (USP); Zmax (TN) (P) Transporter induction: ABCB1
D06399  Tegafur, gimeracil and oteracil potassium; Ts-1 (TN); Teysuno (TN) (P) unclassified
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (P) unclassified
D06404  Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) (P) unclassified
D06405  Nalfurafine hydrochloride (JAN/USAN) (P) unclassified
D06407  Vandetanib (JAN/USAN/INN); Caprelsa (TN) (P) unclassified
D06412  Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) (P) Transporter induction: ABCB1
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Transporter induction: ABCB1
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) unclassified
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) unclassified
D06482  Thyroid (USP); Thyradin (TN) (P) unclassified
D06553  Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) CYP induction: CYP2C9
D06637  Romidepsin (JAN/USAN/INN); Istodax (TN) (P) CYP induction: CYP3A
D06645  Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP18); Sitagliptin phosphate monohydrate; Januvia (TN) (P) unclassified
D06670  Maraviroc (JAN/INN); Selzentry (TN) (P) unclassified
D06676  Raltegravir (INN); MK-0518 (P) unclassified
D06876  Hydrocortisone aceponate (INN); Efficort (TN) (P) CYP induction: CYP3A
D07064  Acenocoumarol (INN); Acenocoumarin; Mini-sintrom (TN) (P) unclassified
D07073  Dexamethasone cipecilate (JAN/INN) (P) unclassified
D07080  Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) (P) unclassified
D07082  Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) (P) Transporter induction: ABCB1
D07086  Rivaroxaban (JAN/USAN/INN); Xarelto (TN) (P) Transporter induction: ABCB1
D07106  Albendazole oxide (INN) (P) unclassified
D07113  Loperamide oxide (INN) (P) Transporter induction: ABCB1
D07117  Metahexamide (INN) (P) unclassified
D07118  Glisoxepide (INN) (P) unclassified
D07124  Alfuzosin (INN); Xatral (TN) (P) unclassified
D07129  Alosetron (INN) (P) Enzyme: CYP2C9
D07131  Ethyl biscoumacetate (INN) (P) unclassified
D07132  Buprenorphine (JAN/INN); Temgesic (TN) (P) unclassified
D07133  Raltegravir potassium (JAN/USAN); Isentress (TN) (P) unclassified
D07135  Clorindione (INN); G-25766 (P) unclassified
D07136  Diphenadione (INN) (P) unclassified
D07137  Tioclomarol (INN) (P) unclassified
D07139  Cloricromen (INN) (P) unclassified
D07144  Dabigatran etexilate (USAN/INN); Pradaxa (TN) (P) Transporter induction: ABCB1
D07165  Ivabradine (USAN/INN) (P) unclassified
D07175  Palonosetron (INN); Aloxi (TN) (P) unclassified
D07192  Benfluorex (INN/BAN); Mediaxal (TN) (P) unclassified
D07203  Methylprednisolone aceponate (INN); Advantan (TN) (P) unclassified
D07214  Tiratricol (INN); Tiracana (TN) (P) unclassified
D07226  Fesoterodine (INN) (P) unclassified
D07283  Esketamine (USAN/INN) (P) CYP induction: CYP2B6
D07299  Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) (P) Enzyme: CYP2C9 / Target: SCN10A SCN3A SCN9A
D07334  Imipraminoxide (INN) (P) unclassified
D07335  Amineptine (INN); Survector (TN) (P) unclassified
D07336  Quinupramine (INN) (P) unclassified
D07402  Levocetirizine (USAN/INN); Xazal (TN) (P) unclassified
D07407  Rupatadine (INN) (P) unclassified
D07448  Amitriptyline (INN); Laroxyl (TN) (P) unclassified
D07450  Amlodipine (USP/INN); Norvasc (TN) (P) unclassified
D07457  Anisindione (INN); Miradon (TN) (P) unclassified
D07474  Atorvastatin (INN); Lipitor (TN); Sortis (TN) (P) Transporter induction: ABCB1
D07486  Azithromycin (INN); Azasite (TN); Azithromycin (TN) (P) Transporter induction: ABCB1
D07494  Barnidipine (INN); Vasexten (TN) (P) unclassified
D07507  Zidovudine and lamivudine; Combivir (TN); Lamivudine zidovudine (TN) (P) unclassified
D07508  Benfluorex hydrochloride; Mediator (TN) (P) unclassified
D07509  Benidipine (INN) (P) unclassified
D07520  Bepridil (INN); Bepadin (TN) (P) Enzyme: CYP2C9
D07523  Betaine (JAN); Cystadane (TN) (P) unclassified
D07538  Bosentan (INN) (P) Enzyme: CYP2C9 / CYP induction: CYP2C9
D07545  Brovincamine (INN); Sarbromin (TN) (P) unclassified
D07552  Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D07564  Allopurinol sodium; Aloprim (TN) (P) unclassified
D07569  Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) (P) unclassified
D07585  Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine; Cleamine A (TN) (P) unclassified
D07601  Butriptyline (INN); Evadyne (TN) (P) unclassified
D07603  Caffeine citrate (USP); Cafcit (TN) (P) unclassified
D07626  Caspofungin (INN); Cancidas (TN) (P) unclassified
D07661  Cerivastatin (INN) (P) unclassified
D07662  Cetirizine (INN); Cetiderm (TN) (P) Transporter induction: ABCB1
D07667  Cevimeline (INN) (P) unclassified
D07674  Chloramphenicol stearate; Quemicetina (TN) (P) unclassified
D07675  Chloramphenicol succinate; Chloramphenicol ICN (TN) (P) unclassified
D07702  Ciprofloxacin lactate; Ciproxin (TN) (P) unclassified
D07704  Citalopram (USP/INN); Citadur (TN) (P) Transporter induction: ABCB1
D07705  Citalopram hydrochloride; Seropram (TN) (P) Transporter induction: ABCB1
D07710  Clarithromycin lactobionate; Klacid (TN) (P) unclassified
D07727  Clomipramine (INN); Anafranil (TN) (P) unclassified
D07729  Clopidogrel (USP/INN); Clopidogrel (TN); Plavix (TN) (P) CYP induction: CYP2B6
D07736  Cloricromen hydrohloride; Proendotel (TN) (P) unclassified
D07740  Codeine hydrochloride; Bisoltus (TN) (P) unclassified
D07748  Conivaptan (INN) (P) CYP induction: CYP3A
D07760  Cyclophosphamide (INN); Cyclophosphamide (TN); Cytoxan (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D07782  Delavirdine (INN) (P) CYP induction: CYP3A
D07791  Desipramine (INN) (P) unclassified
D07793  Desvenlafaxine (INN); Khedezla (TN) (P) unclassified
D07796  Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) (P) unclassified
D07797  Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) (P) unclassified
D07798  Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) (P) unclassified
D07799  Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) (P) unclassified
D07800  Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) (P) unclassified
D07801  Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) (P) unclassified
D07802  Dexamethasone phosphate; Decadron-phosphate (TN) (P) unclassified
D07803  Dexchlorpheniramine (INN); d-Chloropheniramine; Dapriton (TN) (P) CYP induction: CYP3A
D07812  Dibenzepin (INN) (P) unclassified
D07831  Dihydrocodeine (INN); Remedacen (TN) (P) unclassified
D07832  Dihydrocodeine thiocyanate; Paracodin (TN) (P) unclassified
D07837  Dihydroergotamine (INN); Neomigran (TN) (P) unclassified
D07838  Dihydroergotamine tartrate; Divegal (TN) (P) unclassified
D07839  Dihydroergotoxine; Co-Dergocrin (TN) (P) unclassified
D07845  Diltiazem (INN); Surazem (TN) (P) unclassified
D07866  Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) (P) unclassified
D07867  Dolasetron (INN) (P) CYP induction: CYP3A
D07868  Domperidone maleate; Domperidone (TN) (P) unclassified
D07869  Donepezil (JAN/INN); Donaz (TN); Allydone (TN) (P) unclassified
D07871  Dorzolamide (INN); Trusopt (TN) (P) Enzyme: CYP2C9
D07872  Dosulepin (INN); Dothiepin; Dothep (TN) (P) unclassified
D07873  Doxapram (INN); Docatone (TN) (P) unclassified
D07875  Doxepin (INN); Sinequan (TN) (P) Enzyme: CYP2C9
D07876  Doxycycline (INN); Doxychel (TN); Doxycycline (TN) (P) unclassified
D07877  Doxycycline hydrochloride; Vibramycin (TN) (P) unclassified
D07887  Eletriptan (INN) (P) unclassified
D07905  Ergometrine (INN) (P) unclassified
D07906  Ergotamine (INN) (P) unclassified
D07907  Erlotinib (INN) (P) unclassified
D07909  Erythromycin thiocyanate; Erythrocin (TN) (P) CYP induction: CYP3A
D07910  Erythromycin stinoprate (INN); Erysec (TN) (P) CYP induction: CYP3A
D07913  Escitalopram (INN); Esertia (TN) (P) unclassified
D07917  Esomeprazole (INN); Inexium paranova (TN) (P) unclassified
D07918  Estradiol hemihydrate; Estrasorb (TN); Vagifem (TN) (P) unclassified
D07919  Estradiol 17 beta-hemisuccinate; 17beta-Estradiol hemisuccinate; Eutocol (TN) (P) unclassified
D07928  Ethinylestradiol propanesulfonate; Turisteron (TN) (P) unclassified
D07929  Ethylmorphine (BAN) (P) unclassified
D07945  Fenfluramine (INN); Ponderax (TN) (P) CYP induction: CYP2B6
D07962  Flecainide (INN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D07969  Fluindione (INN); Previsccan (TN) (P) unclassified
D07974  Fluorouracil sodium salt; Fluorouracil (TN) (P) unclassified
D07981  Fluticasone (INN); Fluticaps (TN) (P) unclassified
D07983  Fluvastatin (INN); Fluvas (TN) (P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9
D07984  Fluvoxamine (INN) (P) unclassified
D08031  Guanfacine (INN); Estulic (TN) (P) unclassified
D08035  Haloperidol lactate; Haldol (TN) (P) unclassified
D08045  Hydrocodone (INN); Dihydrocodeinone (P) CYP induction: CYP2B6
D08046  Hydrocodone hydrochloride; Dihydrocodeinone hydrochloride; Dicodid (TN) (P) CYP induction: CYP2B6
D08050  Hydroxychloroquine (INN); Polirreumin (TN) (P) unclassified
D08066  Imatinib (INN); Glamox (TN) (P) unclassified
D08070  Imipramine (INN); Tofranil (TN) (P) unclassified
D08071  Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) (P) unclassified
D08072  Imipraminoxide hydrochloride; Elepsin (TN) (P) unclassified
D08080  Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP18); Insulin Humacart (TN) (P) unclassified
D08086  Irinotecan (INN); Biotecan (TN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) unclassified
D08108  Lapatinib (INN) (P) Transporter induction: ABCB1
D08111  Lercanidipine (INN); Lercanil (TN) (P) CYP induction: CYP3A
D08116  Levobupivacaine (INN); Novabupi (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08118  Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN); Xyzal (TN) (P) unclassified
D08125  Levothyroxine (BAN); Forthyron (TN) (P) unclassified
D08127  Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08128  Liothyronine (INN); Thyrolar (TN) (P) unclassified
D08129  Liothyronine hydrochloride; Thyrotradin (TN) (P) unclassified
D08140  Lofepramine (INN) (P) unclassified
D08144  Loperamide (INN); Diamide (TN) (P) Transporter induction: ABCB1
D08148  Loxapine hydrochloride; Desconex (TN) (P) unclassified
D08155  Manidipine (INN); Manidipine 6300; Artedil (TN) (P) unclassified
D08171  Melitracen (INN); Adelax (TN) (P) unclassified
D08195  Methadone (BAN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6 / Transporter induction: ABCB1
D08207  Methylergometrine (INN); Ergotyl (TN) (P) unclassified
D08214  Metronidazole benzoate (USP); Elyzol (TN) (P) CYP inhibition: CYP2C9
D08215  Mexiletine (INN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08216  Mianserin (INN); Tolvon (TN) (P) unclassified
D08227  Mometasone (INN) (P) unclassified
D08229  Montelukast (INN); Brondilat (TN) (P) Enzyme: CYP2C9
D08236  Mosapride (INN); Mosart (TN) (P) unclassified
D08255  Naratriptan (INN); Naramig (TN) (P) Enzyme: CYP2C9
D08259  Nelfinavir (INN); Viracept (TN) (P) unclassified
D08270  Nicardipine (INN); Cardene (TN) (P) unclassified
D08283  Nordazepam (INN); Calmday (TN) (P) unclassified
D08288  Nortriptyline (INN); Nortrilen (TN) (P) unclassified
D08291  Ofloxacin hydrochloride; Tarivid (TN) (P) unclassified
D08297  Opipramol (INN); Opipramol dura (TN) (P) unclassified
D08351  Phenformin (BAN) (P) unclassified
D08352  Phenformin hydrochloride; Debei (TN) (P) unclassified
D08354  Phenindione (INN); Hedulin (TN) (P) unclassified
D08363  Phenylbutazone calcium; Peralgin (TN) (P) CYP inhibition: CYP2C9
D08364  Phenylbutazone sodium; Ambene (TN) (P) CYP inhibition: CYP2C9
D08378  Pioglitazone (INN); Actos (TN) (P) unclassified
D08408  Pranlukast (INN); Azlaire (TN) (P) unclassified
D08424  Procaterol (INN); Meptin (TN) (P) unclassified
D08435  Propafenone (INN); Propafenon hexal (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08441  Propiverine (INN) (P) unclassified
D08447  Protriptyline (INN) (P) unclassified
D08456  Quetiapine (INN); Norsic (TN) (P) unclassified
D08458  Quinidine (BAN); Kinidin (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08459  Quinidine phenylethylbarbiturate; Quinidine 5-ethyl 5-phenyl barbiturate; Natisedine (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08460  Quinine (BAN); Kinder Quinina (TN) (P) Transporter induction: ABCB1
D08461  Quinine dihydrochloride; Quinine (TN) (P) Transporter induction: ABCB1
D08463  Rabeprazole (INN); Eraloc (TN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) unclassified
D08481  Rilmazafone (INN) (P) unclassified
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) unclassified
D08490  Ropivacaine (INN); Naropin (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D08491  Rosiglitazone (INN); Gaudil (TN) (P) unclassified
D08493  Dorzolamide hydrochloride and timolol maleate (JP18); Cosopt (TN) (P) Enzyme: CYP2C9
D08497  Rupatadine fumarate (JAN); Rinialer (TN); Rupafin (TN) (P) unclassified
D08508  Sarpogrelate (INN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D08511  Setiptiline (INN) (P) unclassified
D08514  Sildenafil (INN); Aphrodil (TN) (P) unclassified
D08516  Sitagliptin (USAN/INN) (P) unclassified
D08522  Solifenacin (INN) (P) unclassified
D08552  Sunitinib (INN) (P) unclassified
D08553  Suxethonium chloride (INN); Curacit (TN) (P) unclassified
D08556  Tacrolimus (INN); Prograf (TN) (P) unclassified
D08559  Tamoxifen (INN); Tamoxifen (TN); Tamoplex (TN) (P) unclassified
D08575  Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) (P) unclassified
D08594  Ticlopidine (INN); Ticlopidin-Puren (TN) (P) unclassified
D08616  Teneligliptin (INN) (P) unclassified
D08618  Topotecan (BAN); Hycamtin (TN) (P) Transporter induction: ABCB1
D08620  Toremifene (INN); Fareston (TN) (P) unclassified
D08623  Tramadol (INN); Amanda (TN) (P) unclassified
D08626  Trazodone (INN); Trittico (TN) (P) unclassified
D08655  Tubocurarine chloride (INN); Tubaine (TN); Tubocurarine Chloride (TN) (P) unclassified
D08667  Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) (P) unclassified
D08668  Vardenafil (USAN/INN); Levitra (TN) (P) unclassified
D08670  Venlafaxine (INN); Efectin (TN) (P) unclassified
D08675  Vinblastine (INN); Vinblastina (TN) (P) unclassified
D08676  Vinburnine (INN); Cervoxan (TN) (P) unclassified
D08677  Vincamine (INN); Cetal retard (TN) (P) unclassified
D08678  Vincamine hydrochloride; Vadicate (TN) (P) unclassified
D08679  Vincristine (INN); Tecnocris (TN) (P) CYP induction: CYP3A
D08680  Vinorelbine (INN); Navelbine (TN) (P) unclassified
D08682  Warfarin (INN); Warfarine; Choice (TN) (P) Enzyme: CYP2C9
D08690  Zolpidem (INN); Sanval (TN) (P) unclassified
D08695  dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea; Coughcode N (TN) (P) unclassified
D08697  Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate; Opisezol codeine (TN) (P) unclassified
D08699  Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) (P) unclassified
D08774  Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) (P) unclassified
D08843  Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) (P) unclassified
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) unclassified
D08860  Apremilast (JAN/USAN); Otezla (TN) (P) unclassified
D08870  Belinostat (USAN/INN); Beleodaq (TN) (P) Enzyme: CYP2C9
D08897  Dapagliflozin (JAN/USAN/INN); Forxiga (TN) (P) unclassified
D08903  Dexlansoprazole (INN/USAN); Dexilant (TN) (P) unclassified
D08914  Eribulin mesylate (USAN); Eribulin mesilate (JAN); Halaven (TN) (P) unclassified
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) unclassified
D08950  Neratinib (USAN/INN) (P) unclassified
D08953  Nilotinib (USAN/INN) (P) Transporter induction: ABCB1
D08964  Perampanel (USAN); Fycompa (TN) (P) CYP induction: CYP3A
D08969  Pimavanserin tartrate (USAN); Nuplazide (TN) (P) unclassified
D08976  Pomalidomide (JAN/USAN/INN); Pomalyst (TN) (P) unclassified
D08988  Rolapitant hydrochloride (USAN); Varubi (TN) (P) unclassified
D08996  Saxagliptin (USAN/INN) (P) unclassified
D09012  Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) (P) unclassified
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) CYP induction: CYP3A / Transporter induction: ABCB1
D09032  Vinflunine ditartrate (USAN); Javlor (TN) (P) unclassified
D09033  Voclosporin (JAN/USAN/INN); Lupkynis (TN) (P) unclassified
D09187  Estradiol and levonorgestrel; Wellnara (TN); Climara pro (TN) (P) unclassified
D09188  Estradiol and norethindrone; Menoaid (TN); Activella (TN); Combipatch (TN); Estradiol and norethindrone acetate (TN) (P) unclassified
D09215  Eslicarbazepine (USAN/INN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D09318  Indacaterol (USAN/INN) (P) Transporter induction: ABCB1
D09319  Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) (P) Transporter induction: ABCB1
D09339  Esomeprazole potassium (USAN) (P) unclassified
D09347  Fostamatinib (USAN) (P) unclassified
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) unclassified
D09365  Palovarotene (JAN/USAN/INN); Sohonos (TN) (P) unclassified
D09388  Tasimelteon (USAN/INN); Hetlioz (TN) (P) unclassified
D09394  Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) (P) CYP inhibition: CYP2C9
D09535  Mirabegron (JAN/USAN/INN); Myrbetriq (TN) (P) unclassified
D09544  Ozenoxacin (JAN/USAN/INN); Xepi (TN) (P) unclassified
D09546  Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) (P) Transporter induction: ABCB1
D09566  Linagliptin (JAN/USAN/INN); Tradjenta (TN) (P) unclassified
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D09592  Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) (P) Transporter induction: ABCB1
D09594  Olmesartan medoxomil and azelnidipine; Rezaltas (TN) (P) unclassified
D09595  Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) (P) unclassified
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A
D09621  Gisadenafil (USAN/INN) (P) unclassified
D09622  Gisadenafil besylate (USAN) (P) unclassified
D09637  Lomitapide (USAN/INN) (P) unclassified
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) unclassified
D09666  Selumetinib (USAN/INN) (P) Enzyme: CYP2C9
D09676  Tecarfarin (USAN/INN) (P) unclassified
D09677  Tecarfarin sodium (USAN) (P) unclassified
D09683  Tivozanib (USAN/INN) (P) unclassified
D09698  Vilazodone (USAN/INN) (P) unclassified
D09699  Vilazodone hydrochloride (USAN); Viibryd (TN) (P) unclassified
D09701  Abiraterone acetate (JAN/USP); Zytiga (TN) (P) unclassified
D09707  Dabigatran (USAN/INN) (P) Transporter induction: ABCB1
D09710  Edoxaban (USAN/INN) (P) Transporter induction: ABCB1
D09720  Rilpivirine (JAN/USAN/INN); Rekambys (TN) (CI,P) CYP induction: CYP3A
D09724  Afatinib (USAN/INN) (P) Transporter induction: ABCB1
D09727  Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (P) unclassified
D09729  Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) (P) unclassified
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (P) CYP induction: CYP3A
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) unclassified
D09733  Afatinib dimaleate (USAN); Afatinib maleate (JAN); Gilotrif (TN); Giotrif (TN) (P) Transporter induction: ABCB1
D09741  Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) (P) unclassified
D09742  Lansoprazole, amoxicillin hydrate and metronidazole; Lampion (TN) (P) unclassified
D09743  Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) unclassified
D09744  Pioglitazone hydrochloride and metformin hydrochloride (JP18); Pioglitazone and metformin; Metact (TN) (P) unclassified
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) unclassified
D09753  Saxagliptin hydrate (JAN); Onglyza (TN) (P) unclassified
D09755  Cabazitaxel (USAN/INN); Jevtana (TN) (P) CYP induction: CYP3A
D09756  Teneligliptin hydrobromide hydrate (JAN) (P) unclassified
D09763  Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JAN); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) (P) unclassified
D09765  Vorapaxar (USAN/INN) (P) unclassified
D09766  Vorapaxar sulfate (JAN/USAN); Zontivity (TN) (P) unclassified
D09773  Isoniazid glucuronate sodium (JAN) (P) unclassified
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) unclassified
D09785  Delamanid (JAN/USAN); Deltyba (TN) (P) unclassified
D09796  Hydrocortisone caproate (JAN) (P) CYP induction: CYP3A
D09807  Difethiarol (JAN); Difethialone (P) unclassified
D09847  Metildigoxin (INN); Medigoxin (BAN) (P) Transporter induction: ABCB1
D09848  Pioglitazone hydrochloride and glimepiride tablets (JP18); Pioglitazone and glimepiride; Duetact; Sonias (TN) (P) Enzyme: CYP2C9
D09872  Bedaquiline (USAN/INN) (P) unclassified
D09873  Bedaquiline fumarate (JAN/USAN); Sirturo (TN) (P) unclassified
D09876  Cariprazine hydrochloride (JAN/USAN); Vraylar (TN) (P) unclassified
D09881  Cobicistat (JAN/USAN/INN); Tybost (TN) (P) CYP induction: CYP3A
D09889  Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) (P) unclassified
D09893  Eliglustat (USAN/INN) (P) Transporter induction: ABCB1
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (P) Transporter induction: ABCB1
D09919  Lenvatinib (USAN/INN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D09920  Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D09950  Ponatinib (USAN/INN) (P) CYP induction: CYP3A
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (P) CYP induction: CYP3A
D09955  Quizartinib (USAN/INN) (P) CYP induction: CYP3A
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (P) CYP induction: CYP3A
D09958  Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) (CI,P) CYP induction: CYP3A
D09959  Ruxolitinib (USAN/INN) (P) unclassified
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (P) unclassified
D09970  Tofacitinib (USAN); Tasocitinib (P) unclassified
D09987  Vaniprevir (JAN/USAN/INN); Vanihep (TN) (P) CYP induction: CYP3A
D09989  Vardenafil hydrochloride (USP) (P) unclassified
D09994  Selexipag (JAN/USAN/INN); Uptravi (TN) (P) unclassified
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP inhibition: CYP2C9
D09997  Cariprazine (USAN/INN) (P) unclassified
D09999  Tramadol hydrochloride and acetaminophen; Tramcet (TN) (P) unclassified
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) unclassified
D10019  Panobinostat lactate (JAN); Farydak (TN) (P) unclassified
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (P) Enzyme: CYP2C9
D10025  Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) (P) unclassified
D10027  Udenafil (USAN/INN) (P) unclassified
D10064  Dabrafenib (USAN) (P) CYP induction: CYP2C9
D10065  Daclatasvir (USAN) (P) Transporter induction: ABCB1
D10066  Dolutegravir (USAN); Tivicay (TN) (P) unclassified
D10081  Simeprevir (JAN/USAN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) CYP induction: CYP3A
D10093  Asunaprevir (JAN/USAN); Sunvepra (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) CYP induction: CYP2C9
D10105  Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) (P) Transporter induction: ABCB1
D10113  Dolutegravir sodium (JAN/USAN); Tivicay (TN) (P) unclassified
D10119  Sonidegib (USAN/INN); Erismodegib (P) CYP induction: CYP3A
D10120  Esomeprazole strontium (USAN); Esomeprazole strontium tetrahydrate; Esomeprazole strontium (TN) (P) unclassified
D10131  Ixazomib citrate (JAN/USAN); Ninlaro (TN) (P) unclassified
D10135  Macitentan (JAN/USAN); Opsumit (TN) (CI,P) unclassified
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (P) Transporter induction: ABCB1
D10138  Regorafenib (USAN/INN); Stivarga (TN) (P) Transporter induction: ABCB1
D10158  Safinamide (USAN/INN) (P) unclassified
D10159  Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) (P) unclassified
D10160  Mitiglinide calcium hydrate and voglibose; Glubes (TN) (P) unclassified
D10184  Vortioxetine (USAN); Brintellix (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D10185  Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D10188  Naldemedine (USAN/INN) (P) unclassified
D10190  Tivozanib hydrochloride (USAN); Tivozanib hydrochloride monohydrate; Fotivda (TN) (P) unclassified
D10191  Safinamide mesylate (USAN); Safinamide mesilate (JAN); Safinamide methanesulfonate; Xadago (TN); Equfina (TN) (P) unclassified
D10195  Luseogliflozin hydrate (JAN); Lusefi (TN) (P) unclassified
D10196  Ipragliflozin (INN) (P) unclassified
D10200  Ipragliflozin L-proline (JAN); Suglat (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (P) CYP induction: CYP3A
D10243  Irbesartan and amlodipine besilate (JP18); Aimix (TN) (P) unclassified
D10244  Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) (P) unclassified
D10246  Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) (P) unclassified
D10251  Glimepiride and rosiglitazone maleate; Avandaryl (TN) (P) unclassified
D10253  Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) (P) unclassified
D10258  Simvastatin and sitagliptin phosphate; Juvisync (TN) (P) unclassified
D10261  Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) (P) unclassified
D10262  Saxagliptin hydrochloride; Onglyza (TN) (P) unclassified
D10263  Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) (P) unclassified
D10264  Linagliptin and metformin hydrochloride; Jentaduet (TN) (P) Transporter induction: ABCB1
D10265  Glipizide and metformin hydrochloride; Metaglip (TN) (P) unclassified
D10266  Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) (P) unclassified
D10293  Carbidopa, levodopa and entacapone; Stalevo (TN) (P) CYP inhibition: CYP2C9
D10306  Avatrombopag (USAN/INN) (P) Enzyme: CYP2C9
D10307  Avatrombopag maleate (JAN/USAN); Doptelet (TN) (P) Enzyme: CYP2C9
D10308  Baricitinib (JAN/USAN/INN); Olumiant (TN) (P) Transporter induction: ABCB1
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) unclassified
D10313  Ertugliflozin (USAN/INN) (P) unclassified
D10315  Momelotinib (USAN/INN) (P) Enzyme: CYP2C9
D10319  Panobinostat (USAN/INN); Farydak (TN) (P) unclassified
D10355  Aripiprazole cavoxil (USAN) (P) unclassified
D10358  Momelotinib dihydrochloride (USAN) (P) Enzyme: CYP2C9
D10364  Aripiprazole lauroxil (USAN); Aristada (TN) (P) unclassified
D10366  Sofosbuvir (JAN/USAN/INN); Sovaldi (TN) (CI,P) Transporter induction: ABCB1
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10375  Naloxegol oxalate (USAN); Movantik (TN); Moventig (TN) (P) CYP induction: CYP3A
D10385  Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) (P) unclassified
D10396  Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN); Ofev (TN) (P) Transporter induction: ABCB1
D10428  Tenofovir alafenamide (USAN/INN) (P) Transporter induction: ABCB1
D10433  Vibegron (JAN/USAN/INN); Beova (TN); Gemtesa (TN) (P) Transporter induction: ABCB1
D10434  Vintafolide (USAN/INN) (P) unclassified
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (P) unclassified
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (P) CYP induction: CYP3A
D10459  Empagliflozin (JAN/USAN/INN); Jardiance (TN) (P) Transporter induction: ABCB1
D10461  Dienogest and estradiol valerate; Natazia (TN) (P) CYP induction: CYP3A
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) unclassified
D10469  Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) unclassified
D10479  Naloxegol (USAN/INN) (P) CYP induction: CYP3A
D10481  Nintedanib (USAN/INN); Ofev (TN) (P) Transporter induction: ABCB1
D10500  Metformin hydrochloride and repaglinide; Prandimet (TN) (P) unclassified
D10501  Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) (P) unclassified
D10502  Gemigliptin (INN) (P) unclassified
D10505  Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) (P) Transporter induction: ABCB1
D10506  Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) (P) unclassified
D10512  Brinzolamide and timolol maleate; Azorga (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D10513  Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) (P) CYP induction: CYP2B6
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) unclassified
D10519  Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) (P) unclassified
D10520  Rabeprazole, amoxicillin and metronidazole; Rabefine (TN) (P) unclassified
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) unclassified
D10525  Valsartan and cilnidipine; Atedio (TN) (P) unclassified
D10527  Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) (P) unclassified
D10533  Umeclidinium bromide and vilanterol; Anoro (TN) (P) unclassified
D10537  Methylthioninium chloride hydrate (JAN); Methylene blue (TN) (P) CYP inhibition: CYP2C9
D10542  Alectinib (USAN/INN) (P) unclassified
D10548  Cabotegravir (JAN/USAN/INN); Vocabria (TN); Apretude (TN) (CI) unclassified
D10549  Cabotegravir sodium (JAN/USAN); Vocabria (TN) (CI) unclassified
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) CYP inhibition: CYP2C9 / CYP induction: CYP3A
D10560  Idelalisib (JAN/USAN/INN); Zydelig (TN) (P) CYP induction: CYP3A
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) CYP induction: CYP3A
D10570  Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) (P) unclassified
D10571  Rilpivirine hydrochloride, tenofovir disoproxil fumarate and emtricitabine; Complera (TN); Eviplera (TN) (P) CYP induction: CYP3A
D10572  Fosnetupitant and palonosetron hydrochloride; Netupitant and palonosetron hydrochloride; Akynzeo (TN) (P) unclassified
D10578  Ledipasvir and sofosbuvir; Harvoni (TN) (CI,P) Transporter induction: ABCB1
D10582  Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10586  Dapagliflozin and metformin; Xigduo xr (TN) (P) unclassified
D10587  Canagliflozin and metformin; Invokamet (TN) (P) unclassified
D10588  Empagliflozin and linagliptin; Glyxambi (TN) (P) Transporter induction: ABCB1
D10600  Dolutegravir, abacavir and lamivudine; Triumeq (TN) (P) unclassified
D10605  Tenofovir alafenamide fumarate (JAN/USAN); Vemlidy (TN) (P) Transporter induction: ABCB1
D10612  Benzhydrocodone (USAN/INN) (P) unclassified
D10624  Doravirine (JAN/USAN/INN); Pifeltro (TN) (CI,P) CYP induction: CYP3A
D10625  Elbasvir (JAN/USAN/INN); Erelsa (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10627  Esketamine hydrochloride (JAN/USAN); Spravato (TN) (P) CYP induction: CYP2B6
D10630  Fedratinib (USAN/INN) (P) unclassified
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) unclassified
D10639  Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10642  Irinotecan sucrosofate (USAN) (P) unclassified
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (CI,P) CYP induction: CYP3A
D10644  Isavuconazonium (USAN) (CI,P) CYP induction: CYP3A
D10662  Rimegepant (USAN/INN) (P) unclassified
D10663  Rimegepant sulfate (USAN); Nurtec odt (TN); Vydura (TN) (P) unclassified
D10669  Sotagliflozin (USAN/INN); Inpefa (TN) (P) unclassified
D10673  Ubrogepant (USAN/INN); Ubrelvy (TN) (P) unclassified
D10675  Valbenazine (USAN/INN) (P) unclassified
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (P) CYP induction: CYP3A
D10692  Benzhydrocodone hydrochloride (USAN) (P) unclassified
D10696  Capmatinib (USAN/INN) (P) unclassified
D10707  Fostemsavir (USAN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10708  Fostemsavir tromethamine (USAN); Fostemsavir trometamol; Rukobia (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10709  Gilteritinib (USAN/INN) (P) Transporter induction: ABCB1
D10711  Pemafibrate (JAN); Parmodia (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP3A
D10729  Sonidegib phosphate (USAN); Sonidegib diphosphate; Odomzo (TN) (P) CYP induction: CYP3A
D10734  Temsavir (USAN/INN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10742  Rolapitant (USAN/INN); Varubi (TN) (P) unclassified
D10743  Vildagliptin and metformin hydrochloride (P) unclassified
D10745  Ombitasvir, paritaprevir and ritonavir; Technivie (TN) (P) Transporter induction: ABCB1
D10749  Pitolisant (USAN/INN); Wakix (TN); Ozawade (TN) (P) unclassified
D10752  Empagliflozin and metformin; Synjardy (TN) (P) unclassified
D10753  Atazanavir and cobicistat; Evotaz (TN) (P) unclassified
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (CI) unclassified
D10756  Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) (P) CYP induction: CYP3A
D10761  Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) (P) CYP induction: CYP3A
D10766  Osimertinib mesylate (USAN); Osimertinib mesilate (JAN); Tagrisso (TN) (P) CYP induction: CYP3A
D10772  Lascufloxacin hydrochloride (JAN); Lasvic (TN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) unclassified
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) unclassified
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) CYP induction: CYP3A
D10797  Copanlisib hydrochloride (USAN) (P) CYP induction: CYP3A
D10798  Copanlisib hydrochloride hydrate (JAN); Aliqopa (TN) (P) CYP induction: CYP3A
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (P) Transporter induction: ABCB1
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) CYP induction: CYP2C9
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) unclassified
D10811  Fentanyl hydrochloride (JAN); Ionsys (TN) (P) unclassified
D10822  Ciprofloxacin hydrate (JAN); Ciprofloxacin hemiheptahydrate (P) unclassified
D10823  Clopidogrel hydrochloride; Clopidogrel (TN) (P) CYP induction: CYP2B6
D10824  Clopidogrel besilate; Clopidogrel besylate; Clopidogrel (TN) (P) CYP induction: CYP2B6
D10826  Saxagliptin and dapagliflozin; Qtern (TN) (P) unclassified
D10827  Sofosbuvir and velpatasvir; Epclusa (TN) (CI,P) CYP induction: CYP2B6 / Transporter induction: ABCB1
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (CI) unclassified
D10835  Emtricitabine and tenofovir alafenamide; Descovy (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10836  Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) (CI,P) CYP induction: CYP3A / Transporter induction: ABCB1
D10865  Bexagliflozin (USAN); Brenzavvy (TN) (P) unclassified
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (P) unclassified
D10867  Copanlisib (USAN/INN) (P) CYP induction: CYP3A
D10882  Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D10883  Ribociclib (USAN/INN) (P) unclassified
D10888  Relugolix (JAN/USAN/INN); Orgovyx (TN) (P) Transporter induction: ABCB1
D10889  Momelotinib hydrochloride hydrate (JAN); Momelotinib dihydrochloride monohydrate; Ojjaara (TN); Omjjara (TN) (P) Enzyme: CYP2C9
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) unclassified
D10892  Esaxerenone (JAN/INN) (P) CYP induction: CYP3A
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (P) CYP induction: CYP3A
D10895  Fosaprepitant (INN) (P) CYP induction: CYP2C9
D10897  Teneligliptin and canagliflozin; Teneligliptin and canagliflozin; Canalia (TN) (P) Transporter induction: ABCB1
D10898  Neratinib maleate; Nerlynx (TN) (P) unclassified
D10915  Cannabidiol (USAN/INN); CBD; Epidiolex (TN) (P) Transporter induction: ABCB1
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) unclassified
D10927  Erdafitinib (JAN/USAN/INN); Balversa (TN) (P) Enzyme: CYP2C9 / Transporter induction: ABCB1
D10930  Etrasimod (USAN) (P) Enzyme: CYP2C9
D10931  Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) (P) Enzyme: CYP2C9
D10954  Mirvetuximab soravtansine (USAN/INN); Mirvetuximab soravtansine-gynx; Elahere (TN) (P) unclassified
D10960  Nirogacestat (USAN/INN) (P) Enzyme: CYP2C9
D10964  Omaveloxolone (USAN/INN); Skyclarys (TN) (P) CYP induction: CYP3A
D10979  Ribociclib succinate (USAN); Kisqali (TN) (P) unclassified
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D10994  Upadacitinib (USAN/INN) (P) unclassified
D10995  Upadacitinib tartrate (USAN) (P) unclassified
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) unclassified
D11000  Vamorolone (USAN/INN); Agamree (TN) (P) unclassified
D11009  Indacaterol acetate (JAN) (P) Transporter induction: ABCB1
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) CYP induction: CYP3A
D11014  Glecaprevir and pibrentasvir; Mavyret (TN) (P) Transporter induction: ABCB1
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) unclassified
D11023  Evogliptin (INN) (P) unclassified
D11034  Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) (P) unclassified
D11039  Bictegravir, emtricitabine and tenofovir alafenamide; Biktarvy (TN) (CI) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) unclassified
D11043  Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) (P) unclassified
D11045  Darolutamide (JAN/USAN/INN); Nebeqa (TN) (P) unclassified
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) unclassified
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (P) unclassified
D11056  Mirtazapine hydrate (JAN) (P) unclassified
D11061  Osilodrostat (USAN/INN) (P) CYP induction: CYP2B6
D11062  Osilodrostat phosphate (JAN/USAN); Isturisa (TN) (P) CYP induction: CYP2B6
D11066  Ertugliflozin and sitagliptin; Steglujan (TN) (P) unclassified
D11067  Ertugliflozin and metformin; Segluromet (TN) (P) unclassified
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) Enzyme: CYP2C9
D11073  Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN); Tepmetko (TN) (P) unclassified
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) unclassified
D11095  Atorvastatin calcium propylene glycol solvate (P) Transporter induction: ABCB1
D11113  Levothyroxine sodium (INN); Levothyroxine sodium anhydrous (P) unclassified
D11114  Esomeprazole magnesium dihydrate (P) unclassified
D11137  Larotrectinib (USAN/INN) (P) CYP induction: CYP3A
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) CYP induction: CYP3A
D11141  Tucatinib (USAN/INN); Tukysa (TN) (P) unclassified
D11150  Cenobamate (USAN/INN); Xcopri (TN) (P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A / CYP induction: CYP2B6
D11158  Leniolisib (USAN/INN) (P) unclassified
D11159  Leniolisib phosphate (USAN); Joenja (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11222  Selinexor (USAN/INN); Xpovio (TN) (P) unclassified
D11252  Fexinidazole (USAN/INN); Fexinidazole (TN) (P) unclassified
D11270  Pexidartinib (USAN/INN) (P) unclassified
D11271  Pexidartinib hydrochloride (JAN/USAN); Turalio (TN) (P) unclassified
D11282  Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) (CI,P) CYP induction: CYP3A
D11296  Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) (P) unclassified
D11313  Atogepant (USAN); Qulipta (TN); Aquipta (TN) (P) unclassified
D11330  Voxelotor (USAN); Oxbryta (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D11342  Dorzagliatin (USAN) (P) unclassified
D11360  Tirzepatide (JAN/USAN); Mounjaro (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11371  Capivasertib (JAN/USAN); Truqap (TN) (P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (CI) unclassified
D11389  Dutasteride and tamsulosin; Jalyn (TN) (P) unclassified
D11396  Doravirine, lamivudine and tenofovir disoproxil; Delstrigo (TN) (P) CYP induction: CYP3A
D11403  Asciminib (USAN/INN) (P) unclassified
D11404  Asciminib hydrochloride (JAN/USAN); Scemblix (TN) (P) unclassified
D11405  Prabotulinumtoxin A (USAN); PrabotulinumtoxinA-xvfs; Jeuveau (TN) (P) unclassified
D11406  Risdiplam (JAN/USAN/INN); Evrysdi (TN) (P) unclassified
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (P) unclassified
D11422  Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) (P) CYP induction: CYP3A
D11444  Tazemetostat (USAN/INN) (P) Transporter induction: ABCB1
D11453  Nirogacestat hydrobromide (USAN); Ogsiveo (TN) (P) Enzyme: CYP2C9
D11454  Repotrectinib (JAN/USAN); Augtyro (TN) (P) unclassified
D11460  Siponimod (USAN/INN) (P) Enzyme: CYP2C9
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) Transporter induction: ABCB1
D11490  Pitolisant hydrochloride (USAN); Wakix (TN) (P) unclassified
D11521  Lamivudine, nevirapine and zidovudine (P) CYP induction: CYP3A CYP2B6
D11522  Dolutegravir and lamivudine; Dovato (TN) (P) unclassified
D11553  Lidocaine and tetracaine; Pliaglis (TN); Synera (TN) (P) unclassified
D11555  Calcium levofolinate hydrate (JP18); Levoleucovorin calcium pentahydrate; Calcium levofolinate pentahydrate; Isovorin (TN) (P) unclassified
D11565  Grazoprevir (USAN/INN); Grazoprevir anhydrous (P) CYP induction: CYP3A / Transporter induction: ABCB1
D11567  Insulin degludec and liraglutide; Xultophy (TN) (P) unclassified
D11568  Edoxaban tosylate (USAN) (P) Transporter induction: ABCB1
D11572  Beclomethasone dipropionate monohydrate; Beconase aq (TN) (P) unclassified
D11573  Oxycodone and ibuprofen (P) unclassified
D11576  Naproxen and esomeprazole magnesium; Vimovo (TN) (P) Enzyme: CYP2C9
D11616  Aspirin and omeprazole; Yosprala (TN) (P) unclassified
D11617  Eletriptan hydrobromide monohydrate (P) unclassified
D11619  Desvenlafaxine succinate anhydrous; Desvenlafaxine succinate (TN) (P) unclassified
D11628  Benzhydrocodone and acetaminophen; Apadaz (TN) (P) unclassified
D11630  Aminophylline dihydrate (P) unclassified
D11631  Lefamulin (USAN/INN) (P) unclassified
D11632  Lefamulin acetate (USAN); Xenleta (TN) (P) unclassified
D11652  Tenapanor (USAN/INN) (P) unclassified
D11653  Tenapanor hydrochloride (JAN/USAN); Ibsrela (TN); Phozevel (TN); Xphozah (TN) (P) unclassified
D11656  Azelastine hydrochloride and fluticasone propionate; Dymista (TN) (P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11671  Elacestrant (USAN/INN) (P) Enzyme: CYP2C9
D11672  Elacestrant hydrochloride (USAN); Elacestrant dihydrochloride; Orserdu (TN) (P) Enzyme: CYP2C9
D11673  Berotralstat (USAN/INN) (P) Transporter induction: ABCB1
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) Transporter induction: ABCB1
D11700  Elexacaftor, ivacaftor and tezacaftor; Trikafta (TN); Kaftrio (TN) (P) CYP induction: CYP3A
D11706  Omeprazole and sodium bicarbonate; Zegerid (TN) (P) unclassified
D11710  Phentermine and topiramate; Qsymia (TN) (P) unclassified
D11711  Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) (P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) unclassified
D11716  Odevixibat (USAN); Bylvay (TN) (P) Transporter induction: ABCB1
D11717  Tepotinib (USAN/INN) (P) unclassified
D11720  Acalabrutinib maleate (USAN) (P) CYP induction: CYP3A
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (P) unclassified
D11768  Pacritinib (USAN/INN); Vonjo (TN) (P) unclassified
D11776  Sparsentan (USAN/INN); Filspari (TN) (P) CYP induction: CYP3A
D11784  Vonoprazan (USAN/INN) (P) unclassified
D11793  Zuranolone (JAN/USAN/INN); Zurzuvae (TN) (P) unclassified
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11807  Imeglimin hydrochloride (JAN); Twymeeg (TN) (P) unclassified
D11816  Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) (P) unclassified
D11851  Butalbital, acetaminophen, caffeine and codeine phosphate (P) unclassified
D11856  Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) (P) unclassified
D11858  Omeprazole magnesium, amoxicillin and rifabutin; Talicia (TN) (P) CYP induction: CYP3A
D11860  Butalbital, aspirin, caffeine and codeine; Fiorinal with codeine (TN) (P) unclassified
D11881  Amlodipine benzoate; Katerzia (TN) (P) unclassified
D11886  Daridorexant (USAN/INN) (P) unclassified
D11923  Lobeglitazone (INN) (P) unclassified
D11924  Beinaglutide (INN) (P) unclassified
D11954  Belzutifan (JAN/USAN/INN); Welireg (TN) (P) unclassified
D11966  Cabotegravir and rilpivirine; Cabenuva (TN) (P) CYP induction: CYP3A
D11968  Teneligliptin hydrobromide (JAN) (P) unclassified
D11969  Mobocertinib succinate (JAN); Exkivity (TN) (P) CYP induction: CYP3A
D11977  Fruquintinib (JAN/USAN); Fruzaqla (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP3A
D12001  Mobocertinib (USAN/INN) (P) CYP induction: CYP3A
D12015  St. John's wort; SJW (P) unclassified
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) CYP induction: CYP3A
D12130  Drospirenone, ethinyl estradiol and levomefolate calcium; Beyaz (TN); Safyral (TN); Tydemy (TN) (P) unclassified
D12137  Elagolix, estradiol and norethisterone; Oriahnn (TN) (P) CYP induction: CYP3A
D12161  Lenacapavir (USAN/INN) (P) CYP induction: CYP3A / Transporter induction: ABCB1
D12162  Lenacapavir sodium (JAN/USAN); Sunlenca (TN) (CI,P) CYP induction: CYP3A / Transporter induction: ABCB1
D12265  Mavacamten (JAN/USAN/INN); Camzyos (TN) (P) Enzyme: CYP2C9
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (CI,P) unclassified
D12294  Sitagliptin phosphate (JAN) (P) unclassified
D12301  Adagrasib (USAN/INN); Krazati (TN) (P) unclassified
D12312  Codeine phosphate and chlorpheniramine maleate; Tuxarin (TN) (P) unclassified
D12313  Chlorpheniramine polistirex and codeine polistirex; Tuzistra (TN) (P) unclassified
D12353  Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) (CI,P) CYP induction: CYP3A
D12388  Fosifloxuridine nafalbenamide (P) unclassified
D12403  Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) (P) unclassified
D12442  Tucatinib ethanolate (JAN); Tucatinib hemiethanolate (P) unclassified
D12444  Nilotinib hydrochloride dihydrate (JAN) (P) Transporter induction: ABCB1
D12483  Olutasidenib (USAN/INN); Rezlidhia (TN) (P) unclassified
D12484  Carfloglitazar (INN) (P) unclassified
D12486  Finasteride and tadalafil; Entadfi (TN) (P) unclassified
D12497  Drospirenone and estradiol; Angeliq (TN) (P) unclassified
D12544  Vortioxetine hemihydrobromide (USAN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D12586  Mifepristone and misoprostol; Mefeego (TN) (CI,P) CYP induction: CYP3A
D12609  Dasatinib laurylsulfate (USAN) (P) unclassified
D12619  Ensitrelvir (USAN/INN) (P) CYP induction: CYP3A
D12637  Darunavir hydrate (P) unclassified
D12703  Linagliptin hydrate (JAN); Linagliptin hemihydrate (P) unclassified
D12704  Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate (P) CYP induction: CYP3A
D12752  Darunavir propylene glycolate (P) unclassified
D12756  Vonoprazan and amoxicillin; Voquezna (TN) (P) Enzyme: CYP2C9 / CYP induction: CYP2B6
D12816  Dexlansoprazole sesquihydrate (P) unclassified
D12854  Nilotinib laurylsulfate (USAN) (P) Transporter induction: ABCB1