C00220 |
Methylene blue; Methylthioninium chloride |
(P) unclassified |
C04931 |
Argatroban; (2R,4R)-4-Methyl-1[Nalpha-[(3-methyl-1,2,3,4-tetrahydro-8-quinolinyl)sulfonyl]-L-arginyl]-2-piperadinecarboxylic acid |
(P) unclassified |
C06174 |
Codeine; (5alpha,6alpha)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol |
(P) unclassified |
C07005 |
Flunisolide; Flunisolide anhydrous |
(P) unclassified |
C07051 |
Indinavir |
(P) unclassified |
C07547 |
Tubocurarine |
(P) unclassified |
C07548 |
Atracurium |
(P) unclassified |
C07551 |
Pancuronium |
(P) unclassified |
C07553 |
Vecuronium |
(P) unclassified |
D00066 |
Progesterone (JP18/USP/INN); Crinone (TN); Prometrium (TN) |
(P) unclassified |
D00067 |
Estrone (JAN/USP/INN); Estrone (TN) |
(P) unclassified |
D00088 |
Hydrocortisone (JP18/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) |
(P) CYP induction: CYP3A |
D00094 |
Tretinoin (JAN/USP/INN); Avita (TN); Renova (TN); Retin A (TN); Tretinoin (TN) |
(P) unclassified |
D00104 |
Chloramphenicol (JP18/USP/INN); Amphicol (TN); Chloromycetin (TN); Econochlor (TN) |
(P) unclassified |
D00105 |
Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) |
(P) unclassified |
D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) |
(P) unclassified |
D00109 |
Aspirin (JP18/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) |
(P) unclassified |
D00118 |
Naproxen (JP18/USP/INN); Naprosyn (TN) |
(P) unclassified |
D00123 |
Cyanamide (JP18); Cyanamide (TN) |
(P) unclassified |
D00129 |
Calcitriol (JAN/USP/INN); Rocaltrol (TN) |
(P) unclassified |
D00131 |
Disulfiram (JP18/USP/INN); Antabuse (TN) |
(P) unclassified |
D00134 |
Albendazole (JAN/USP/INN); Albenza (TN) |
(P) unclassified |
D00136 |
Haloperidol (JP18/USP/INN); Haldol (TN) |
(P) unclassified |
D00140 |
Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) |
(P) CYP induction: CYP3A |
D00142 |
Methotrexate (JP18/USP/INN); Otrexup (TN); Xatmep (TN) |
(P) unclassified |
D00165 |
Hydrocortisone acetate (JP18/USP); Cortifoam (TN); U-cort (TN) |
(P) CYP induction: CYP3A |
D00181 |
Argatroban (USP); Argatroban hydrate (JP18); Novastan (TN) |
(P) unclassified |
D00184 |
Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) unclassified |
D00186 |
Ciprofloxacin (JP18/USP/INN); Cipro (TN); Otiprio (TN) |
(P) unclassified |
D00195 |
Codeine (USP); Codeine hydrate |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) unclassified |
D00216 |
Acarbose (JAN/USAN/INN); Precose (TN) |
(P) unclassified |
D00217 |
Acetaminophen (JP18/USP); Paracetamol (INN); Tylenol (TN) |
(P) unclassified |
D00218 |
Acetazolamide (JP18/USP/INN); Diamox (TN) |
(P) unclassified |
D00219 |
Acetohexamide (JP18/USP/INN); Dymelor (TN) |
(P) unclassified |
D00224 |
Allopurinol (JP18/USP/INN); Zyloprim (TN) |
(P) unclassified |
D00225 |
Alprazolam (JP18/USP/INN); Xanax (TN) |
(P) CYP induction: CYP3A |
D00227 |
Aminophylline (USP/INN); Somophyllin (TN); Theophylline ethylenediamine (TN) |
(P) unclassified |
D00228 |
Amoxapine (JP18/USP/INN); Asendin (TN) |
(P) unclassified |
D00234 |
Astemizole (JAN/USP/INN); Hismanal (TN) |
(P) CYP induction: CYP3A |
D00244 |
Betamethasone (JP18/USP/INN); Celestone (TN); Rinderon (TN) |
(P) unclassified |
D00246 |
Budesonide (JP18/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) |
(P) unclassified |
D00252 |
Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00255 |
Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) |
(P) Enzyme: CYP2C9 |
D00271 |
Chlorpropamide (JP18/USP/INN); Diabinese (TN) |
(P) unclassified |
D00274 |
Cisapride (USP/INN) |
(P) CYP induction: CYP3A |
D00275 |
Cisplatin (JP18/USP/INN); Platinol (TN) |
(P) unclassified |
D00276 |
Clarithromycin (JP18/USP/INN); Biaxin (TN) |
(P) unclassified |
D00280 |
Clonazepam (JP18/USP/INN); Klonopin (TN) |
(P) unclassified |
D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) unclassified |
D00285 |
Co-Trimoxazole (BAN); Sulfamethoxazole and trimethoprim; Bactrim (TN); Septra (TN) |
(P) CYP inhibition: CYP2C9 |
D00287 |
Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D00292 |
Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) |
(P) unclassified |
D00293 |
Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) |
(P) unclassified |
D00294 |
Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) |
(P) unclassified |
D00295 |
Cimetidine (JP18/USP/INN); Tagamet (TN) |
(P) unclassified |
D00297 |
Digitoxin (JAN/USP/INN); Crystodigin (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D00298 |
Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) Transporter induction: ABCB1 |
D00302 |
Dipyridamole (JP18/USP/INN); Persantine (TN) |
(P) unclassified |
D00303 |
Disopyramide (JP18/USAN/INN); Rythmodan P (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00304 |
Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) |
(P) unclassified |
D00307 |
Doxycycline (USP); Doxycycline hydrate; Monodox (TN); Oracea (TN); Vibramycin (TN) |
(P) unclassified |
D00311 |
Estazolam (JP18/USP/INN); ProSom (TN) |
(P) CYP induction: CYP3A |
D00312 |
Estrone sodium sulfate; Sodium estrone sulfate |
(P) unclassified |
D00316 |
Etretinate (JAN/USAN/INN); Tegison (TN) |
(P) unclassified |
D00319 |
Felodipine (JP18/USP/INN); Plendil (TN) |
(P) unclassified |
D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) unclassified |
D00321 |
Finasteride (JAN/USP/INN); Propecia (TN); Proscar (TN) |
(P) unclassified |
D00322 |
Fluconazole (JP18/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP2C9 |
D00324 |
Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) |
(P) unclassified |
D00326 |
Fluoxetine (USAN/INN); Fluoxetine (TN) |
(P) Enzyme: CYP2C9 |
D00335 |
Glipizide (USP/INN); Glucotrol (TN) |
(P) unclassified |
D00336 |
Glyburide (USP); Glibenclamide (JP18/INN); Diabeta (TN); Glynase (TN); Micronase (TN) |
(P) Enzyme: CYP2C9 |
D00343 |
Ifosfamide (JAN/USP/INN); Ifex (TN) |
(P) unclassified |
D00346 |
Isoniazid (JP18/USP/INN); Laniazid (TN) |
(P) unclassified |
D00350 |
Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) |
(P) unclassified |
D00351 |
Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) |
(P) unclassified |
D00354 |
Lamotrigine (JAN/USP/INN); Lamictal (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00355 |
Lansoprazole (JP18/USP/INN); Prevacid (TN) |
(P) unclassified |
D00358 |
Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00359 |
Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) |
(P) unclassified |
D00364 |
Loratadine (JAN/USP/INN); Claritin (TN) |
(P) unclassified |
D00371 |
Theophylline (JP18); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) |
(P) unclassified |
D00379 |
Tolazamide (JAN/USP/INN); Tolinase (TN) |
(P) unclassified |
D00380 |
Tolbutamide (JP18/USP/INN); Orinase (TN) |
(P) unclassified |
D00385 |
Triamcinolone (JP18/USP/INN); Aristocort (TN); Kenacort (TN) |
(P) unclassified |
D00387 |
Triazolam (JP18/USP/INN); Halcion (TN) |
(P) unclassified |
D00394 |
Trimipramine (USAN/INN) |
(P) unclassified |
D00395 |
Troglitazone (JAN/USAN/INN); Rezulin (TN) |
(P) unclassified |
D00399 |
Valproic acid (USP); Depakene (TN) |
(P) unclassified |
D00407 |
Methylprednisolone (JP18/USP/INN); Medrol (TN) |
(P) unclassified |
D00409 |
Metronidazole (JP18/USP/INN); Flagyl (TN); Noritate (TN); Nuvessa (TN); Vandazole (TN) |
(P) CYP inhibition: CYP2C9 |
D00413 |
Zidovudine (JP18/USP/INN); Azidothymidine; Retrovir (TN) |
(P) unclassified |
D00416 |
Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) |
(P) CYP inhibition: CYP2C9 |
D00424 |
Rifabutin (JAN/USP/INN); Mycobutin (TN) |
(P) unclassified |
D00426 |
Risperidone (JP18/USP/INN); Risperdal (TN) |
(P) unclassified |
D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) CYP induction: CYP2C9 CYP3A |
D00429 |
Saquinavir (JAN/USP/INN); Fortovase (TN) |
(P) Transporter induction: ABCB1 |
D00434 |
Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) |
(P) unclassified |
D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) CYP induction: CYP2B6 |
D00437 |
Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) |
(P) unclassified |
D00438 |
Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) |
(P) unclassified |
D00446 |
Sucralfate (USP/INN); Sucralfate hydrate (JP18); Carafate (TN) |
(P) unclassified |
D00453 |
Ofloxacin (JP18/USP/INN); Floxin (TN) |
(P) unclassified |
D00455 |
Omeprazole (JP18/USP/INN); Prilosec (TN) |
(P) unclassified |
D00456 |
Ondansetron (JAN/USP/INN); Zofran ODT (TN) |
(P) unclassified |
D00457 |
Quazepam (JAN/USP/INN); Doral (TN) |
(P) Enzyme: CYP2C9 |
D00458 |
Quetiapine fumarate (JP18/USP); Seroquel (TN) |
(P) unclassified |
D00465 |
Oxybutynin (USAN/INN); Anturol (TN); Oxytrol (TN) |
(P) unclassified |
D00471 |
Praziquantel (JAN/USP/INN); Biltricide (TN) |
(P) unclassified |
D00472 |
Prednisolone (JP18/USP/INN); Delta-cortef (TN) |
(P) CYP induction: CYP3A |
D00484 |
Protriptyline hydrochloride (USP); Vivactil (TN) |
(P) unclassified |
D00491 |
Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) |
(P) unclassified |
D00492 |
Pancuronium bromide (JP18/USP/INN); Pavulon (TN) |
(P) unclassified |
D00510 |
Phenylbutazone (JP18/USP/INN); Azolid (TN) |
(P) CYP inhibition: CYP2C9 |
D00521 |
Terfenadine (JAN/USAN/INN); Seldane (TN) |
(P) CYP induction: CYP3A |
D00528 |
Caffeine (USP); Anhydrous caffeine (JP18); Anhydrous caffeine (TN); Respia (TN) |
(P) unclassified |
D00529 |
Montelukast sodium (JP18/USP); Singulair (TN) |
(P) Enzyme: CYP2C9 |
D00530 |
Zaleplon (JAN/USP/INN); Sonata (TN) |
(P) unclassified |
D00533 |
Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00535 |
Vigabatrin (JAN/USP/INN); Sabril (TN) |
(P) unclassified |
D00537 |
Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00538 |
Zonisamide (JP18/USP/INN); Excegran (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A / CYP induction: CYP3A |
D00539 |
Ethosuximide (JP18/USP/INN); Zarontin (TN) |
(P) unclassified |
D00542 |
Halothane (JP18/USP/INN); Fluothane (TN) |
(P) unclassified |
D00544 |
Methoxyflurane (USP/INN); Penthrane (TN) |
(P) unclassified |
D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) unclassified |
D00554 |
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) |
(P) unclassified |
D00560 |
Pimozide (JP18/USP/INN); Orap (TN) |
(P) unclassified |
D00563 |
Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) |
(P) unclassified |
D00564 |
Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) |
(P) Enzyme: CYP2C9 |
D00570 |
Colchicine (JP18/USP); Colchicine (TN) |
(P) Transporter induction: ABCB1 |
D00578 |
Voriconazole (JP18/USP/INN); Vfend (TN) |
(P) unclassified |
D00584 |
Fluorouracil (JP18/USP/INN); 5-FU (TN); Adrucil (TN); Carac (TN); Fluoroplex (TN) |
(P) unclassified |
D00585 |
Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) |
(P) unclassified |
D00592 |
Dapsone (USP); Diaphenylsulfone (JAN); Aczone (TN) |
(P) unclassified |
D00593 |
Glimepiride (JP18/USP/INN); Amaryl (TN) |
(P) Enzyme: CYP2C9 |
D00594 |
Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) |
(P) unclassified |
D00595 |
Buformin (USAN/INN) |
(P) unclassified |
D00596 |
Rosiglitazone maleate (JAN/USP); Avandia (TN) |
(P) unclassified |
D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) unclassified |
D00615 |
Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) |
(P) unclassified |
D00616 |
Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) |
(P) unclassified |
D00617 |
Nicardipine hydrochloride (JP18/USAN); Cardene (TN) |
(P) unclassified |
D00618 |
Nisoldipine (JAN/USAN/INN); Sular (TN) |
(P) unclassified |
D00619 |
Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Transporter induction: ABCB1 |
D00625 |
Miglitol (JP18/USAN/INN); Glyset (TN) |
(P) unclassified |
D00629 |
Nitrendipine (JP18/USAN/INN); Baypress (TN) |
(P) unclassified |
D00631 |
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) |
(P) Enzyme: CYP2C9 |
D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00637 |
Disopyramide phosphate (JAN/USP); Norpace (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00638 |
Flecainide acetate (JP18/USP); Tambocor (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00639 |
Mexiletine hydrochloride (JP18/USP); Mexitil (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00640 |
Propafenone hydrochloride (JP18/USP); Rythmol (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00642 |
Quinidine gluconate (USP); Quinaglute (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00643 |
Quinidine polygalacturonate; Cardioquin (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D00646 |
Tolterodine (USAN/INN) |
(P) unclassified |
D00653 |
Dorzolamide hydrochloride (JP18/USP); Trusopt (TN) |
(P) Enzyme: CYP2C9 |
D00661 |
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) |
(P) unclassified |
D00664 |
Cetirizine hydrochloride (JP18/USP); Zyrtec (TN) |
(P) Transporter induction: ABCB1 |
D00668 |
Dexchlorpheniramine maleate (USP); d-Chlorpheniramine maleate (JP18); Mylaramine (TN); Polaramine (TN) |
(P) CYP induction: CYP3A |
D00670 |
Donepezil hydrochloride (JP18/USP); Aricept (TN) |
(P) unclassified |
D00674 |
Naratriptan hydrochloride (JAN/USP); Amerge (TN) |
(P) Enzyme: CYP2C9 |
D00677 |
Granisetron hydrochloride (JAN/USP); Kytril (TN) |
(P) unclassified |
D00678 |
Ondansetron hydrochloride hydrate (JAN/USP); Ondansetron hydrochloride; Zofran (TN) |
(P) unclassified |
D00679 |
Ergotamine tartrate (JP18/USP); Ergomar (TN) |
(P) unclassified |
D00680 |
Methylergonovine maleate (USP); Methylergometrine maleate (JP18); Methergine (TN) |
(P) unclassified |
D00687 |
Salmeterol xinafoate (JAN/USP); Serevent (TN) |
(P) unclassified |
D00689 |
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18); Beclovent (TN); Qnasl (TN); Vanceril (TN) |
(P) unclassified |
D00690 |
Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) |
(P) unclassified |
D00696 |
Midazolam hydrochloride (USAN); Versed (TN) |
(P) unclassified |
D00706 |
Zolpidem tartrate (JP18/USP); Ambien (TN); Intermezzo (TN) |
(P) unclassified |
D00707 |
Fomepizole (JAN/USAN/INN); Antizol (TN) |
(P) CYP inhibition: CYP2C9 |
D00710 |
Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) |
(P) unclassified |
D00722 |
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18); Ditropan (TN); Gelnique (TN) |
(P) unclassified |
D00724 |
Rabeprazole sodium (JP18/USP); Aciphex (TN); Pariet (TN) |
(P) unclassified |
D00725 |
Dolasetron mesylate (USP); Anzemet (TN) |
(P) CYP induction: CYP3A |
D00729 |
Loperamide hydrochloride (JAN/USP); Imodium (TN) |
(P) Transporter induction: ABCB1 |
D00746 |
Interferon beta-1b (USAN/INN); Interferon beta-1b (genetical recombination) (JAN); Betaseron (TN); Extavia (TN) |
(P) unclassified |
D00749 |
Leflunomide (JAN/USP/INN); Arava (TN) |
(P) CYP inhibition: CYP2C9 |
D00751 |
Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) |
(P) unclassified |
D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Transporter induction: ABCB1 |
D00758 |
Atracurium besylate (USP); Atracurium besilate (INN); Tracrium (TN) |
(P) unclassified |
D00759 |
Cisatracurium besylate (USP); Cisatracurium besilate (INN); Nimbex (TN) |
(P) unclassified |
D00760 |
Doxacurium chloride (USAN/INN); Nuromax (TN) |
(P) unclassified |
D00763 |
Mivacurium chloride (USAN/INN); Mivacron (TN) |
(P) unclassified |
D00764 |
Pipecuronium bromide (JAN/USAN/INN); Arduan (TN) |
(P) unclassified |
D00765 |
Rocuronium bromide (JAN/USP/INN); Zemuron (TN) |
(P) unclassified |
D00767 |
Vecuronium bromide (JAN/USP/INN); Norcuron (TN) |
(P) unclassified |
D00769 |
Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18); Clopidogrel hydrogen sulphate; Isocover (TN); Plavix (TN) |
(P) CYP induction: CYP2B6 |
D00780 |
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) |
(P) unclassified |
D00781 |
Entacapone (JP18/USP/INN); Comtan (TN) |
(P) CYP inhibition: CYP2C9 |
D00783 |
Botulinum toxin type A (JAN); Botox (TN); Dysport (TN) |
(P) unclassified |
D00785 |
Selegiline hydrochloride (JAN/USP); Eldepryl (TN) |
(P) CYP induction: CYP2B6 |
D00794 |
Loxapine succinate (USP); Loxitane (TN) |
(P) unclassified |
D00804 |
Ivermectin (JAN/USP/INN); Sklice (TN); Soolantra (TN); Stromectol (TN) |
(P) Transporter induction: ABCB1 |
D00809 |
Amitriptyline hydrochloride (JP18/USP); Elavil (TN) |
(P) unclassified |
D00811 |
Clomipramine hydrochloride (JP18/USP); Anafranil (TN) |
(P) unclassified |
D00812 |
Desipramine hydrochloride (JAN/USP); Norpramin (TN) |
(P) unclassified |
D00814 |
Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) |
(P) Enzyme: CYP2C9 |
D00815 |
Imipramine hydrochloride (JP18/USP); Tofranil (TN) |
(P) unclassified |
D00816 |
Nortriptyline hydrochloride (JP18/USP/INN); Pamelor (TN) |
(P) unclassified |
D00818 |
Maprotiline hydrochloride (JP18/USP); Ludiomil (TN) |
(P) unclassified |
D00820 |
Trazodone hydrochloride (JAN/USP); Desyrel (TN) |
(P) unclassified |
D00821 |
Venlafaxine hydrochloride (JAN/USP); Effexor (TN) |
(P) unclassified |
D00822 |
Citalopram hydrobromide (USP); Celexa (TN) |
(P) Transporter induction: ABCB1 |
D00823 |
Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) |
(P) Enzyme: CYP2C9 |
D00824 |
Fluvoxamine maleate (JP18/USP); Luvox (TN) |
(P) unclassified |
D00825 |
Sertraline hydrochloride (JAN/USP); Zoloft (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) CYP induction: CYP3A |
D00836 |
Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) |
(P) unclassified |
D00840 |
Levomethadyl acetate hydrochloride (USAN); Orlaam (TN) |
(P) unclassified |
D00847 |
Oxycodone hydrochloride (USP); Oxecta (TN); Oxycontin (TN); Roxicodone (TN) |
(P) unclassified |
D00851 |
Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) |
(P) CYP induction: CYP3A |
D00882 |
Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) |
(P) CYP inhibition: CYP2C9 |
D00887 |
Atorvastatin calcium anhydorous; Lipitor (TN) |
(P) Transporter induction: ABCB1 |
D00889 |
Cerivastatin sodium (JAN/USAN); Baycol (TN) |
(P) unclassified |
D00892 |
Fluvastatin sodium (JAN/USP); Lescol (TN) |
(P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9 |
D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) unclassified |
D00895 |
Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) |
(P) CYP induction: CYP3A |
D00896 |
Efavirenz (JAN/USP/INN); Sustiva (TN) |
(P) CYP induction: CYP2B6 |
D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) unclassified |
D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) unclassified |
D00944 |
Metformin hydrochloride (JP18/USP); Glucophage (TN) |
(P) unclassified |
D00945 |
Pioglitazone hydrochloride (JP18/USP); Actos (TN) |
(P) unclassified |
D00948 |
Estropipate (USP); Piperazine estrone sulfate; Ogen (TN) |
(P) unclassified |
D00950 |
Levonorgestrel (JAN/USP/INN); Mirena (TN); Norplant (TN); Skyla (TN) |
(P) unclassified |
D00960 |
Anastrozole (JP18/USP/INN); Arimidex (TN) |
(P) CYP inhibition: CYP2C9 |
D00963 |
Exemestane (JAN/USP/INN); Aromasin (TN) |
(P) unclassified |
D00964 |
Letrozole (JAN/USP/INN); Femara (TN) |
(P) unclassified |
D00966 |
Tamoxifen citrate (JP18/USP); Nolvadex (TN); Soltamox (TN) |
(P) unclassified |
D00967 |
Toremifene citrate (JAN/USAN); Fareston (TN) |
(P) unclassified |
D00969 |
Meloxicam (JAN/USP/INN); Mobic (TN) |
(P) Enzyme: CYP2C9 |
D00972 |
Betamethasone sodium phosphate (JP18/USP); Celestone (TN) |
(P) unclassified |
D00973 |
Cortisone acetate (JP18/USP); Cortone acetate (TN) |
(P) unclassified |
D00975 |
Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) |
(P) unclassified |
D00976 |
Hydrocortisone cypionate |
(P) CYP induction: CYP3A |
D00977 |
Hydrocortisone sodium phosphate (JP18/USP); Hydrocortone phosphate (TN) |
(P) CYP induction: CYP3A |
D00978 |
Hydrocortisone sodium succinate (JP18/USP); A-hydrocort (TN); Solu-cortef (TN) |
(P) CYP induction: CYP3A |
D00979 |
Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) |
(P) unclassified |
D00981 |
Prednisolone sodium phosphate (JP18/USP); Pediapred (TN) |
(P) unclassified |
D00983 |
Triamcinolone acetonide (JP18/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) |
(P) unclassified |
D00986 |
Fludrocortisone acetate (JP18/USP); Florinef acetate (TN) |
(P) unclassified |
D00987 |
Cabergoline (JP18/USP/INN); Cabaser (TN); Dostinex (TN) |
(P) unclassified |
D01007 |
Propiverine hydrochloride (JP18); Bup-4 (TN); Mictonorm (TN) |
(P) unclassified |
D01010 |
Levothyroxine sodium (USP); Levothyroxine sodium hydrate (JP18); Levothroid (TN); Levoxyl (TN); Synthroid (TN) |
(P) unclassified |
D01011 |
Liothyronine sodium (JP18/USP); Cytomel (TN); Triostat (TN) |
(P) unclassified |
D01012 |
Dried thyroid (JP18); Thyradin (TN) |
(P) unclassified |
D01028 |
Ticlopidine hydrochloride (JP18/USP); Ticlid (TN) |
(P) unclassified |
D01056 |
Benzbromarone (JP18/USAN/INN); Uroleap (TN) |
(P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9 |
D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
D01068 |
Vinblastine sulfate (JP18/USP); Exal (TN); Velban (TN) |
(P) unclassified |
D01072 |
Chloramphenicol palmitate (JP18/USP); Chloromycetin palmitate (TN) |
(P) unclassified |
D01078 |
Telithromycin (JAN/USAN/INN); Ketek (TN) |
(P) CYP induction: CYP3A |
D01092 |
Lanoconazole (JP18/INN); Latoconazole; Astat (TN) |
(P) CYP inhibition: CYP2C9 |
D01098 |
Maxacalcitol (JAN/USAN/INN); Oxarol (TN); Prezios (TN) |
(P) unclassified |
D01101 |
Bromperidol (JAN/USAN/INN); Impromen (TN) |
(P) unclassified |
D01104 |
Barnidipine hydrochloride (JAN); Hypoca (TN) |
(P) unclassified |
D01110 |
Melitracen hydrochloride (JAN/USAN) |
(P) unclassified |
D01111 |
Nateglinide (JP18/USP/INN); Starsis (TN) |
(P) Enzyme: CYP2C9 |
D01115 |
Eplerenone (JP18/USAN/INN); Inspra (TN) |
(P) unclassified |
D01121 |
Rebamipide (JP18/INN); Mucosta (TN) |
(P) unclassified |
D01131 |
Lafutidine (JP18/INN); Protecadin (TN) |
(P) unclassified |
D01145 |
Azelnidipine (JP18/INN); Calblock (TN) |
(P) unclassified |
D01148 |
Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) |
(P) unclassified |
D01160 |
Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) |
(P) Transporter induction: ABCB1 |
D01161 |
Fulvestrant (JAN/USP/INN); Faslodex (TN) |
(P) unclassified |
D01163 |
Ergonovine maleate (USP); Ergometrine maleate (JP18); Ergometrine (TN) |
(P) unclassified |
D01164 |
Aripiprazole (JAN/USP/INN); Abilify (TN) |
(P) unclassified |
D01173 |
Cilnidipine (JP18/INN); Atelec (TN) |
(P) unclassified |
D01176 |
Blonanserin (JAN/INN); AD 5423 |
(P) unclassified |
D01196 |
Acetazolamide sodium (JAN); Diamox (TN) |
(P) unclassified |
D01204 |
Olmesartan medoxomil (JP18/USP); Benicar (TN); Olmetec (TN) |
(P) Transporter induction: ABCB1 |
D01207 |
Omeprazole sodium (USAN); Losec sodium (TN) |
(P) unclassified |
D01211 |
Leucovorin calcium (USP); Calcium folinate (JP18); Uzel (TN); Wellcovorin (TN) |
(P) unclassified |
D01213 |
Tolvaptan (JAN/USAN/INN); Samsca (TN) |
(P) Transporter induction: ABCB1 |
D01215 |
Alcuronium chloride (JAN/USAN/INN); Alloferin (TN) |
(P) unclassified |
D01217 |
Dydrogesterone (JP18/USP/INN); Duphaston (TN); Gynorest (TN) |
(P) unclassified |
D01223 |
Capecitabine (JAN/USP/INN); Xeloda (TN) |
(P) Enzyme: CYP2C9 |
D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2C9 |
D01236 |
Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) |
(P) CYP induction: CYP3A |
D01239 |
Prednisolone sodium succinate (JP18/USP); Kohakusanin (TN) |
(P) unclassified |
D01244 |
Tegafur (JP18/USAN/INN); Atillon (TN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) unclassified |
D01269 |
Solifenacin succinate (JAN/USAN/INN); Vesicare (TN) |
(P) unclassified |
D01280 |
Warfarin potassium (JP18); Athrombin-K (TN) |
(P) Enzyme: CYP2C9 |
D01285 |
Lofepramine hydrochloride (JAN/USAN); Amplit (TN) |
(P) unclassified |
D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D01293 |
Ethyl loflazepate (JP18/INN); Meilax (TN) |
(P) unclassified |
D01296 |
Methylphenidate hydrochloride (JAN/USP); Concerta (TN); Metadate (TN); Quillivant xr (TN); Ritalin (TN) |
(P) unclassified |
D01309 |
Doxifluridine (JP18/INN); Furtulon (TN) |
(P) unclassified |
D01314 |
Dibenzepin hydrochloride (JAN/USAN) |
(P) unclassified |
D01316 |
Mexazolam (JAN/INN); Melex (TN) |
(P) unclassified |
D01322 |
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) |
(P) unclassified |
D01355 |
Tramadol hydrochloride (JP18/USP); Ultram (TN) |
(P) unclassified |
D01356 |
Glymidine sodium (JAN/USAN/INN) |
(P) unclassified |
D01358 |
Mianserin hydrochloride (JAN/USAN); Tetramide (TN) |
(P) unclassified |
D01361 |
Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) |
(P) CYP induction: CYP3A |
D01372 |
Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) |
(P) unclassified |
D01399 |
Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) unclassified |
D01413 |
Estradiol valerate (JAN/USP/INN); Deladumone (TN) |
(P) unclassified |
D01418 |
Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) |
(P) unclassified |
D01425 |
Lopinavir (JAN/USP/INN) |
(P) CYP induction: CYP3A |
D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP2C9 |
D01441 |
Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) |
(P) unclassified |
D01442 |
Hydrocortisone succinate (JP18) |
(P) CYP induction: CYP3A |
D01450 |
Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D01453 |
Caffeine hydrate (JP18); Caffeine monohydrate; Caffeine (TN) |
(P) unclassified |
D01455 |
Cifenline succinate (USAN); Cibenzoline succinate (JP18); Cibenol (TN); Cipralan (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D01468 |
Nemonapride (JAN/INN); Emilace (TN) |
(P) unclassified |
D01477 |
Opipramol hydrochloride (JAN/USAN); Insidon (TN) |
(P) unclassified |
D01478 |
Ebastine (JP18/USAN/INN); Kestine (TN) |
(P) unclassified |
D01481 |
Dihydrocodeine phosphate (JP18); Dihydro (TN) |
(P) unclassified |
D01501 |
Isoniazid calcium pyruvinate (JAN); Pyruvic acid calcium isoniazid |
(P) unclassified |
D01510 |
Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) |
(P) unclassified |
D01514 |
Etizolam (JP18/INN); Sedekopan (TN) |
(P) Enzyme: CYP2C9 |
D01546 |
Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Dosulepin (TN) |
(P) unclassified |
D01553 |
Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) |
(P) unclassified |
D01562 |
Aranidipine (JAN/INN); Sapresta (TN) |
(P) unclassified |
D01564 |
Rilmazafone hydrochloride hydrate (JP18); Rilmazafone hydrochloride dihydrate; Rilmazafone hydrochloride; Rhythmy (TN) |
(P) unclassified |
D01599 |
Gliclazide (JP18/INN); Glimicron (TN) |
(P) unclassified |
D01615 |
Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) |
(P) unclassified |
D01617 |
Estradiol dipropionate (JAN); Ovahormon (TN) |
(P) unclassified |
D01619 |
Hydrocortisone butyrate (JP18/USP); Locoid (TN) |
(P) CYP induction: CYP3A |
D01624 |
Sarpogrelate hydrochloride (JP18); Anplag (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D01632 |
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) |
(P) unclassified |
D01643 |
Aluminoparaaminosalicylate calcium hydrate (JAN); Aluminoparaaminosalicylate calcium pentahydrate; Aluminoparaaminosalicylate calcium; Alumino nippas calcium (TN) |
(P) unclassified |
D01656 |
Brovincamine fumarate (JAN); Sabromin (TN) |
(P) unclassified |
D01663 |
Quinine ethylcarbonate (JP18); Quinine ethylcarbonate (TN) |
(P) Transporter induction: ABCB1 |
D01665 |
Voglibose (JP18/USAN/INN); Basen (TN) |
(P) unclassified |
D01692 |
Alfuzosin hydrochloride (JAN/USAN); Uroxatral (TN) |
(P) unclassified |
D01697 |
Colforsin daropate hydrochloride (JAN); Nkh 477; Adehl (TN) |
(P) CYP induction: CYP3A |
D01699 |
Darifenacin hydrobromide (JAN/USAN); Enablex (TN) |
(P) unclassified |
D01703 |
Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) |
(P) unclassified |
D01708 |
Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) |
(P) unclassified |
D01710 |
Roxithromycin (JP18/USAN/INN); Rulide (TN) |
(P) CYP induction: CYP3A |
D01712 |
Theophylline sodium acetate (JAN) |
(P) unclassified |
D01744 |
Brotizolam (JP18/USAN/INN); Lendormin (TN) |
(P) unclassified |
D01745 |
Domperidone (JP18/USAN/INN); Motilium (TN) |
(P) unclassified |
D01769 |
Vindesine sulfate (JAN/USAN); Fildesin (TN) |
(P) CYP induction: CYP3A |
D01784 |
Carmofur (JP18/INN); Mifurol (TN) |
(P) unclassified |
D01787 |
Sulthiame (USAN); Sultiame (JP18); Ospolot (TN) |
(P) unclassified |
D01799 |
Glyclopyramide (JAN/INN); Deamelin-S (TN) |
(P) unclassified |
D01832 |
Modafinil (JAN/USP/INN); Provigil (TN) |
(P) CYP inhibition: CYP2C9 |
D01849 |
Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) |
(P) CYP induction: CYP3A |
D01854 |
Mitiglinide calcium hydrate (JP18); Mitiglinide calcium dihydrate; Glufast (TN) |
(P) unclassified |
D01855 |
Mozavaptane hydrochloride (JAN) |
(P) unclassified |
D01872 |
Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18); Dopram (TN) |
(P) unclassified |
D01886 |
Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) |
(P) CYP induction: CYP3A |
D01896 |
Cilostazol (JP18/USP/INN); Pletal (TN) |
(P) unclassified |
D01898 |
Haloperidol decanoate (JAN/USP); Halomonth (TN) |
(P) unclassified |
D01908 |
Nilvadipine (JP18/USAN/INN); Nivadil (TN) |
(P) unclassified |
D01935 |
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) |
(P) unclassified |
D01948 |
Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) |
(P) unclassified |
D01953 |
Estradiol benzoate (JP18/USP); Ovahormon (TN) |
(P) unclassified |
D01965 |
Silodosin (JP18/INN); KMD 3213; Rapaflo (TN); Urief (TN) |
(P) unclassified |
D01973 |
Eletriptan hydrobromide (JAN/USAN); Relpax (TN) |
(P) unclassified |
D01977 |
Gefitinib (JP18/USAN/INN); Iressa (TN) |
(P) unclassified |
D01980 |
Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) |
(P) unclassified |
D01984 |
Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN); Esomeprazole magnesium trihydrate; Nexium (TN) |
(P) unclassified |
D01994 |
Mosapride citrate hydrate (JP18); Mosapride citrate dihydrate; Gasmotin (TN) |
(P) unclassified |
D02002 |
Isoniazid sodium methanesulfonate hydrate (JAN); Isoniazid sodium methanesulfonate monohydrate; Isoniazid sodium methanesulfonate; IHMS; Neoiscotin (TN) |
(P) unclassified |
D02008 |
Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) |
(CI,P) unclassified |
D02009 |
Erythromycin lactobionate (JP18/USP); Erythrocin (TN) |
(P) CYP induction: CYP3A |
D02034 |
Setiptiline maleate (JAN); Tecipul (TN) |
(P) unclassified |
D02045 |
Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) |
(P) unclassified |
D02086 |
Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D02092 |
Cisapride (JAN); Cisapride monohydrate; Propulsid (TN) |
(P) CYP induction: CYP3A |
D02101 |
Codeine phosphate (USP); Codeine phosphate hydrate (JP18); Codeine (TN) |
(P) unclassified |
D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 / Transporter induction: ABCB1 |
D02114 |
Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) |
(P) unclassified |
D02129 |
Doxycycline hyclate (USP); Doxycycline hydrochloride hydrate (JP18); Doryx (TN); Lymepak (TN); Periostat (TN); Vibra-tabs (TN) |
(P) unclassified |
D02131 |
Tegafur and uracil; Uftoral (TN) |
(P) unclassified |
D02134 |
Azithromycin hydrate (JP18); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) |
(P) Transporter induction: ABCB1 |
D02165 |
Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) |
(P) unclassified |
D02168 |
Topotecan hydrochloride (USAN); Nogitecan hydrochloride (JAN); Hycamtin (TN); Potactasol (TN) |
(P) Transporter induction: ABCB1 |
D02173 |
Galantamine hydrobromide (JAN/USP); Razadyne (TN); Reminyl (TN) |
(P) unclassified |
D02174 |
Dexamethasone acetate (JAN/USP); Decadronal (TN) |
(P) unclassified |
D02175 |
Compound oxycodone (JP18); Pavinal (TN) |
(P) unclassified |
D02184 |
Erythromycin stearate (JP18/USP); Bristamycin (TN) |
(P) CYP induction: CYP3A |
D02185 |
Chloramphenicol sodium succinate (JP18/USP); Chloromycetin succinate (TN) |
(P) unclassified |
D02197 |
Vincristine sulfate (JP18/USP); VCR; Marqibo (TN); Oncovin (TN); Vincasar (TN); Vincrex (TN) |
(P) CYP induction: CYP3A |
D02204 |
Hexamethonium bromide (JAN/INN); Hexamethonium bromide (TN) |
(P) unclassified |
D02205 |
Ethylmorphine hydrochloride hydrate (JP18); Ethylmorphine hydrochloride dihydrate; Ethylmorphine hydrochloride (TN) |
(P) unclassified |
D02206 |
Buformin hydrochloride (JP18); Dibetos-B (TN) |
(P) unclassified |
D02207 |
Tubocurarine chloride (USP); Tubocurarine chloride hydrate (JAN); Tubocurarine chloride (TN) |
(P) unclassified |
D02211 |
Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18); Migranal (TN); Trudhesa (TN) |
(P) unclassified |
D02216 |
Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP18); Ciloxan (TN); Cipro (TN); Proquin XR (TN) |
(P) unclassified |
D02219 |
Terbinafine hydrochloride (JP18/USP); Lamisil (TN) |
(P) Enzyme: CYP2C9 |
D02229 |
Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) |
(P) unclassified |
D02258 |
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) |
(P) Transporter induction: ABCB1 |
D02260 |
Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18); Paxil (TN) |
(P) unclassified |
D02261 |
Quinine hydrochloride hydrate (JP18); Quinine hydrochloride dihydrate; Quinine hydrochloride (TN) |
(P) Transporter induction: ABCB1 |
D02262 |
Quinine sulfate (USP); Quinine sulfate hydrate (JP18); Quinine hydrogen sulfate; Coco-quinine (TN) |
(P) Transporter induction: ABCB1 |
D02268 |
Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18); Circanol (TN); Hydergine (TN); Inorter (TN) |
(P) unclassified |
D02272 |
Quinidine sulfate (USP); Quinidine sulfate hydrate (JP18); Quinidex (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D02274 |
Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18); Dantrium (TN); Ryanodex (TN) |
(P) CYP induction: CYP3A |
D02288 |
Hydrocortisone valerate (USP); Westcort (TN) |
(P) CYP induction: CYP3A |
D02292 |
Gallamine triethiodide (USP); Flaxedil (TN) |
(P) unclassified |
D02312 |
Methylene blue (USP); Methylthioninium chloride; Methylthioninium chloride proveblue (TN) |
(P) CYP inhibition: CYP2C9 |
D02340 |
Loxapine (USAN/INN); Adasuve (TN) |
(P) unclassified |
D02347 |
Dantrolene (USAN/INN) |
(P) CYP induction: CYP3A |
D02356 |
Verapamil (USAN/INN) |
(P) Transporter induction: ABCB1 |
D02360 |
Sertraline (INN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D02362 |
Paroxetine (USP/INN); Paroxetine (TN) |
(P) unclassified |
D02375 |
Terbinafine (USAN/INN); Lamasil (TN) |
(P) Enzyme: CYP2C9 |
D02404 |
Procaterol hydrochloride (USAN); Pro-Air (TN) |
(P) unclassified |
D02408 |
Trimipramine maleate (JAN/USP); Surmontil (TN) |
(P) unclassified |
D02416 |
Aluminum hydroxide (USP); Aluminum hydroxide, dried (USP); Dried aluminum hydroxide gel (JP18); ALterna GEL (TN); Dialume (TN) |
(P) unclassified |
D02425 |
Carbutamide (INN); Invenol (TN) |
(P) unclassified |
D02427 |
Glibornuride (USAN/INN); Glutril (TN) |
(P) unclassified |
D02430 |
Gliquidone (INN); Glurenorm (TN) |
(P) unclassified |
D02484 |
Artemether and lumefantrine; Coartem (TN) |
(CI,P) CYP induction: CYP3A |
D02497 |
Fosamprenavir (INN) |
(P) unclassified |
D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) CYP induction: CYP3A |
D02501 |
Caspofungin acetate (JAN/USAN); Cancidas (TN) |
(P) unclassified |
D02523 |
Erythromycin acistrate (USAN); Erasis (TN) |
(P) CYP induction: CYP3A |
D02524 |
Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) |
(P) CYP induction: CYP3A |
D02525 |
Erythromycin propionate (USAN) |
(P) CYP induction: CYP3A |
D02537 |
Dronedarone (INN) |
(P) CYP induction: CYP3A |
D02554 |
Rifaximin (JAN/USAN/INN); Xifaxan (TN) |
(P) Transporter induction: ABCB1 |
D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) Transporter induction: ABCB1 |
D02561 |
Moclobemide (USAN/INN); Aurorix (TN) |
(P) unclassified |
D02562 |
Rasagiline mesylate (USAN); Rasagiline mesilate (JAN); Azilect (TN) |
(P) unclassified |
D02565 |
Dimetacrine (INN) |
(P) unclassified |
D02566 |
Maprotiline (USAN) |
(P) unclassified |
D02567 |
Escitalopram oxalate (JAN/USP); Lexapro (TN) |
(P) unclassified |
D02570 |
Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) |
(P) unclassified |
D02577 |
Flibanserin (USAN/INN); Addyi (TN) |
(P) unclassified |
D02587 |
Metildigoxin (JP18); Lanirapid (TN) |
(P) Transporter induction: ABCB1 |
D02591 |
Dexamethasone acefurate (USAN/INN) |
(P) unclassified |
D02592 |
Dexamethasone beloxil (USAN) |
(P) unclassified |
D02593 |
Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN); Protonix (TN) |
(P) unclassified |
D02615 |
Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital; Vegetamin (TN) |
(P) CYP induction: CYP3A |
D02624 |
Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) |
(P) unclassified |
D02626 |
Bromperidol decanoate (USAN) |
(P) unclassified |
D02666 |
Iloperidone (USAN/INN); Fanapt (TN) |
(P) unclassified |
D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
D02704 |
Tampramine fumarate (USAN) |
(P) unclassified |
D02714 |
Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) |
(P) Transporter induction: ABCB1 |
D02731 |
Vardenafil dihydrochoride (USAN); Levitra (TN) |
(P) unclassified |
D02732 |
Pranlukast hydrate (JP18); Onon (TN) |
(P) unclassified |
D02735 |
Rimabotulinumtoxin B (USAN); Botulinum toxin type B (JAN); Myobloc (TN) |
(P) unclassified |
D02740 |
Lidocaine and prilocaine; Lidocaine and propitocaine; Emla (TN); Oraqix (TN); Lidocaine and prilocaine (TN) |
(P) unclassified |
D02824 |
Almotriptan (USAN) |
(P) unclassified |
D02825 |
Almotriptan malate (USP); Axert (TN) |
(P) unclassified |
D02829 |
Alosetron hydrochloride (USAN); Lotrpnex (TN) |
(P) Enzyme: CYP2C9 |
D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) unclassified |
D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) unclassified |
D02910 |
Amiodarone (USAN/INN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D02914 |
Amlodipine maleate (USAN); Amvaz (TN) |
(P) unclassified |
D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) CYP induction: CYP2C9 |
D02972 |
Aptazapine maleate (USAN) |
(P) unclassified |
D03038 |
Azipramine hydrochloride (USAN) |
(P) unclassified |
D03071 |
Beloxepin (USAN/INN) |
(P) unclassified |
D03098 |
Berythromycin (USAN/INN); Erythromycin B |
(P) CYP induction: CYP3A |
D03164 |
Bromindione (USAN/INN) |
(P) unclassified |
D03165 |
Bromocriptine (USAN/INN) |
(P) unclassified |
D03199 |
Butriptyline hydrochloride (USAN) |
(P) unclassified |
D03208 |
Aliskiren (USAN/INN); Rasilez (TN) |
(P) Transporter induction: ABCB1 |
D03213 |
Apixaban (JAN/USAN/INN); Eliquis (TN) |
(P) Transporter induction: ABCB1 |
D03215 |
Armodafinil (USAN/INN); Nuvigil (TN) |
(P) unclassified |
D03217 |
Avanafil (USAN/INN); Stendra (TN); Spedra (TN) |
(P) unclassified |
D03218 |
Axitinib (JAN/USAN); Inlyta (TN) |
(P) unclassified |
D03230 |
Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) |
(P) unclassified |
D03250 |
Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) |
(P) unclassified |
D03252 |
Bosutinib (USAN) |
(P) unclassified |
D03259 |
Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN); Mylotarg (TN) |
(P) unclassified |
D03260 |
Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) |
(P) unclassified |
D03325 |
Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) |
(P) unclassified |
D03368 |
Calcium para-aminosalicylate (JP18); Nippas calcium (TN) |
(P) unclassified |
D03415 |
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) |
(P) Enzyme: CYP2C9 |
D03461 |
Chloramphenicol pantothenate complex (USAN/INN); Pantofenicol (TN) |
(P) unclassified |
D03491 |
Cidoxepin hydrochloride (USAN) |
(P) unclassified |
D03492 |
Cifenline (USAN); Cibenzoline (INN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D03503 |
Cimetidine hydrochloride (USP); Cimetidine hydrochloride (TN) |
(P) unclassified |
D03504 |
Cinacalcet (USAN) |
(P) unclassified |
D03505 |
Cinacalcet hydrochloride (JAN/USAN); Sensipar (TN); Mimpara (TN) |
(P) unclassified |
D03579 |
Codeine polistirex (USAN) |
(P) unclassified |
D03580 |
Codeine sulfate (USP); Codeine sulfate trihydrate; Codeine sulfate (TN) |
(P) unclassified |
D03584 |
Colforsin (USAN/INN) |
(P) CYP induction: CYP3A |
D03654 |
Darifenacin (USAN/INN) |
(P) unclassified |
D03656 |
Darunavir (USAN/INN) |
(P) unclassified |
D03657 |
Dasantafil (USAN/INN) |
(P) unclassified |
D03658 |
Dasatinib (JAN/INN) |
(P) unclassified |
D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) unclassified |
D03671 |
Deflazacort (USAN/INN); Emflaza (TN) |
(P) Transporter induction: ABCB1 |
D03725 |
Hydrocodone bitartrate (USP); Hydrocodone bitartrate hemipentahydrate; Dicodid (TN) |
(P) CYP induction: CYP2B6 |
D03730 |
Dexrazoxane (JAN/USAN/INN) |
(P) unclassified |
D03731 |
Selegiline (USAN/INN); Emsam (TN) |
(P) CYP induction: CYP2B6 |
D03783 |
Oxycodone terephthalate (USP) |
(P) unclassified |
D03798 |
Dicumarol (USAN); Dicoumarol (INN); Dicumarol (TN) |
(P) unclassified |
D03799 |
Dienogest (JAN/USAN/INN); Endometrion (TN) |
(P) unclassified |
D03820 |
Dutasteride (JAN/USP/INN); Avodart (TN) |
(P) unclassified |
D03825 |
Dihydrocodeine bitartrate (USP) |
(P) unclassified |
D03830 |
Diltiazem malate (USAN); Tiamate (TN) |
(P) unclassified |
D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) unclassified |
D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) unclassified |
D03837 |
Fosamprenavir sodium (USAN) |
(P) unclassified |
D03844 |
Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP3A CYP2B6 |
D03852 |
Droperidol and fentanyl citrate; Innovar (TN) |
(P) unclassified |
D03903 |
Doxycycline calcium (USP) |
(P) unclassified |
D03904 |
Doxycycline fosfatex (USAN) |
(P) unclassified |
D03914 |
Dronedarone hydrochloride (USP); Multaq (TN) |
(P) CYP induction: CYP3A |
D03917 |
Drospirenone (JAN/USP/INN); Slynd (TN) |
(P) unclassified |
D03960 |
Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) |
(P) unclassified |
D04023 |
Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) |
(P) unclassified |
D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Transporter induction: ABCB1 |
D04048 |
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D04052 |
Epinephrine and lidocaine hydrochloride; Adrenaline and lidocaine hydrochloride; Xylocaine (TN) |
(P) unclassified |
D04054 |
Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate |
(P) CYP induction: CYP3A |
D04056 |
Esomeprazole sodium (USAN); Nexium IV (TN) |
(P) unclassified |
D04061 |
Estradiol acetate (USAN); Femring (TN) |
(P) unclassified |
D04063 |
Estradiol cypionate (USP); Depo-estradiol (TN) |
(P) unclassified |
D04064 |
Estradiol enanthate (USAN) |
(P) unclassified |
D04065 |
Estradiol undecylate (USAN/INN); Delestrec (TN) |
(P) unclassified |
D04070 |
Estrogens, conjugated (JAN/USP); Conjugated estrogens; Premarin (TN) |
(P) unclassified |
D04112 |
Etravirine (JAN/USAN/INN); Intelence (TN) |
(P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9 |
D04121 |
Exenatide (JAN/USAN/INN); Byetta (TN) |
(P) unclassified |
D04148 |
Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) |
(P) CYP induction: CYP2B6 |
D04197 |
Floxuridine (USP/INN); FUDR (TN) |
(P) unclassified |
D04214 |
Flunisolide acetate (USAN) |
(P) unclassified |
D04292 |
Galantamine (USAN/INN); Reminyl (TN) |
(P) unclassified |
D04300 |
Ganaxolone (USAN/INN); Ztalmy (TN) |
(P) CYP induction: CYP2B6 |
D04313 |
Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate; Huscode (TN) |
(P) unclassified |
D04314 |
Gepirone hydrochloride (USAN); Exxua (TN) |
(P) unclassified |
D04338 |
Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride; Sekicode (TN) |
(P) unclassified |
D04340 |
Dextromethorphan hydrobromide and potassium cresolsulfonate; Medicon (TN) |
(P) unclassified |
D04370 |
Granisetron (JAN/USAN/INN); Sancuso (TN) |
(P) unclassified |
D04403 |
Guar gum (NF) |
(P) unclassified |
D04435 |
Hexafluorenium bromide (USAN); Hexafluronium bromide (INN); Mylaxen (TN) |
(P) unclassified |
D04446 |
Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) |
(P) unclassified |
D04447 |
Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) |
(P) unclassified |
D04461 |
Hydrocodone polistirex (USAN) |
(P) CYP induction: CYP2B6 |
D04463 |
Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) |
(P) Enzyme: CYP2C9 |
D04467 |
Hydrocortisone hemisuccinate (USP) |
(P) CYP induction: CYP3A |
D04475 |
Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) |
(P) unclassified |
D04477 |
Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) |
(P) unclassified |
D04482 |
Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) |
(P) unclassified |
D04483 |
Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) |
(P) unclassified |
D04484 |
Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) |
(P) unclassified |
D04539 |
Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) |
(P) unclassified |
D04540 |
Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) |
(P) unclassified |
D04541 |
Insulin human, isophane (USP) |
(P) unclassified |
D04542 |
Insulin human zinc (USP) |
(P) unclassified |
D04543 |
Insulin human zinc, extended (USP) |
(P) unclassified |
D04547 |
Insulin, isophane (USP); Isophane insulin human (genetical recombination) injectable aqueous suspension (JP18); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) |
(P) unclassified |
D04550 |
Insulin zinc, prompt (USP); Semilente iletin (TN) |
(P) unclassified |
D04551 |
Insulin zinc (USP); Lente iletin (TN) |
(P) unclassified |
D04554 |
Interferon beta-1a (USAN); Interferon beta-1a (genetical recombination) (JAN); Avonex (TN); Rebif (TN) |
(P) unclassified |
D04556 |
Intriptyline hydrochloride (USAN) |
(P) unclassified |
D04605 |
Iprindole (USAN/INN) |
(P) unclassified |
D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) unclassified |
D04645 |
Ixabepilone (JAN/USAN/INN); Ixempra (TN) |
(P) unclassified |
D04652 |
Ketipramine fumarate (USAN) |
(P) unclassified |
D04716 |
Levomethadyl acetate (USAN); Levacetylmethadol (INN) |
(P) unclassified |
D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(P) unclassified |
D04813 |
Lidocaine hydrochloride and epinephrine bitartrate; Lidocaine hydrochloride and adrenaline bitartrate; Ora (TN); Lidosite (TN) |
(P) unclassified |
D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(CI,P) unclassified |
D04859 |
Maribavir (JAN/USAN/INN); Camvia (TN); Livtencity (TN) |
(P) unclassified |
D04895 |
Mefloquine (USAN/INN) |
(P) CYP induction: CYP3A |
D04966 |
Metformin (USAN/INN) |
(P) unclassified |
D04999 |
Methylphenidate (USAN/INN); Daytrana (TN) |
(P) unclassified |
D05000 |
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18) |
(P) unclassified |
D05001 |
Methylprednisolone sodium phosphate (USAN) |
(P) unclassified |
D05002 |
Methylprednisolone suleptanate (USAN/INN) |
(P) unclassified |
D05016 |
Metronidazole hydrochloride (USAN); Flagyl I.V. (TN) |
(P) CYP inhibition: CYP2C9 |
D05017 |
Metronidazole phosphate (USAN) |
(P) CYP inhibition: CYP2C9 |
D05028 |
Midazolam maleate (USAN) |
(P) unclassified |
D05029 |
Midostaurin (JAN/USAN/INN); Rydapt (TN) |
(P) unclassified |
D05143 |
Nepafenac (JAN/USAN/INN); Nevanac (TN) |
(P) unclassified |
D05152 |
Netupitant (USAN/INN) |
(P) CYP induction: CYP3A |
D05177 |
Nitisinone (JAN/USAN/INN); Orfadin (TN) |
(P) CYP inhibition: CYP2C9 |
D05231 |
Octriptyline phosphate (USAN) |
(P) unclassified |
D05246 |
Olmesartan (USAN/INN) |
(P) Transporter induction: ABCB1 |
D05259 |
Omeprazole magnesium (USP); Prilosec OTC (TN) |
(P) unclassified |
D05261 |
Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) |
(P) unclassified |
D05284 |
Oxaprotiline hydrochloride (USAN) |
(P) unclassified |
D05312 |
Oxycodone (USAN/INN) |
(P) unclassified |
D05333 |
Paclitaxel poliglumex (USAN/INN) |
(P) unclassified |
D05343 |
Palonosetron hydrochloride (JAN/USP); Aloxi (TN) |
(P) unclassified |
D05353 |
Pantoprazole (USAN/INN) |
(P) unclassified |
D05366 |
Procaterol hydrochloride hydrate (JP18); Meptin (TN) |
(P) unclassified |
D05374 |
Paroxetine hydrochloride (USP); Paxil (TN) |
(P) unclassified |
D05375 |
Paroxetine mesylate (USAN); Brisdelle (TN); Pexeva (TN) |
(P) unclassified |
D05380 |
Pazopanib hydrochloride (JAN/USAN); Votrient (TN) |
(P) unclassified |
D05429 |
Aminophylline hydrate (JP18) |
(P) unclassified |
D05457 |
Phenprocoumon (USAN/INN); Liquamar (TN) |
(P) unclassified |
D05462 |
Oxycodone hydrochloride hydrate (JP18) |
(P) unclassified |
D05594 |
Pramlintide (USAN/INN) |
(P) unclassified |
D05595 |
Pramlintide acetate (USAN); Symlin (TN) |
(P) unclassified |
D05622 |
Proinsulin human (USAN) |
(P) unclassified |
D05681 |
Quinine ascorbate (USAN); Quinine biascorbate |
(P) Transporter induction: ABCB1 |
D05700 |
Ranolazine (USAN/INN); Ranexa (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D05701 |
Ranolazine hydrochloride (USAN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D05703 |
Rapacuronium bromide (USAN/INN); Raplon (TN) |
(P) unclassified |
D05744 |
Roflumilast (JAN/USAN/INN); Daliresp (TN); Zoryve (TN) |
(P) unclassified |
D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D05792 |
Salmeterol (USAN/INN) |
(P) unclassified |
D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) CYP inhibition: CYP2C9 |
D05932 |
Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) |
(P) unclassified |
D05987 |
Synthetic conjugated estrogens, B (USAN); Enjuvia (TN) |
(P) unclassified |
D06068 |
Temsirolimus (JAN/USAN/INN); Torisel (TN) |
(P) unclassified |
D06103 |
Theophylline (USP); Theophylline monohydrate; Accurbron (TN) |
(P) unclassified |
D06104 |
Theophylline sodium glycinate (USP); Asbron (TN) |
(P) unclassified |
D06177 |
Tolbutamide sodium, sterile; Orinase diagnostic (TN) |
(P) unclassified |
D06199 |
Trabectedin (JAN/USAN/INN); Yondelis (TN) |
(P) unclassified |
D06272 |
Sorafenib tosylate (USAN); Sorafenib tosilate (JAN); Nexavar (TN) |
(P) unclassified |
D06273 |
Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) |
(P) unclassified |
D06304 |
Vindesine (USAN/INN) |
(P) CYP induction: CYP3A |
D06305 |
Vinepidine sulfate (USAN) |
(P) unclassified |
D06306 |
Vinglycinate sulfate (USAN) |
(P) unclassified |
D06307 |
Vinleurosine sulfate (USAN) |
(P) unclassified |
D06308 |
Vinrosidine sulfate (USAN) |
(P) unclassified |
D06309 |
Vinzolidine sulfate (USAN) |
(P) unclassified |
D06315 |
Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) |
(P) unclassified |
D06390 |
Azithromycin (USP); Zmax (TN) |
(P) Transporter induction: ABCB1 |
D06399 |
Tegafur, gimeracil and oteracil potassium; Ts-1 (TN); Teysuno (TN) |
(P) unclassified |
D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) unclassified |
D06404 |
Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) |
(P) unclassified |
D06405 |
Nalfurafine hydrochloride (JAN/USAN) |
(P) unclassified |
D06407 |
Vandetanib (JAN/USAN/INN); Caprelsa (TN) |
(P) unclassified |
D06412 |
Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) |
(P) Transporter induction: ABCB1 |
D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Transporter induction: ABCB1 |
D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) unclassified |
D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) unclassified |
D06482 |
Thyroid (USP); Thyradin (TN) |
(P) unclassified |
D06553 |
Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) |
(P) unclassified |
D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) CYP induction: CYP2C9 |
D06637 |
Romidepsin (JAN/USAN/INN); Istodax (TN) |
(P) CYP induction: CYP3A |
D06645 |
Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP18); Sitagliptin phosphate monohydrate; Januvia (TN) |
(P) unclassified |
D06670 |
Maraviroc (JAN/INN); Selzentry (TN) |
(P) unclassified |
D06676 |
Raltegravir (INN); MK-0518 |
(P) unclassified |
D06876 |
Hydrocortisone aceponate (INN); Efficort (TN) |
(P) CYP induction: CYP3A |
D07064 |
Acenocoumarol (INN); Acenocoumarin; Mini-sintrom (TN) |
(P) unclassified |
D07073 |
Dexamethasone cipecilate (JAN/INN) |
(P) unclassified |
D07080 |
Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) |
(P) unclassified |
D07082 |
Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) |
(P) Transporter induction: ABCB1 |
D07086 |
Rivaroxaban (JAN/USAN/INN); Xarelto (TN) |
(P) Transporter induction: ABCB1 |
D07106 |
Albendazole oxide (INN) |
(P) unclassified |
D07113 |
Loperamide oxide (INN) |
(P) Transporter induction: ABCB1 |
D07117 |
Metahexamide (INN) |
(P) unclassified |
D07118 |
Glisoxepide (INN) |
(P) unclassified |
D07124 |
Alfuzosin (INN); Xatral (TN) |
(P) unclassified |
D07129 |
Alosetron (INN) |
(P) Enzyme: CYP2C9 |
D07131 |
Ethyl biscoumacetate (INN) |
(P) unclassified |
D07132 |
Buprenorphine (JAN/INN); Temgesic (TN) |
(P) unclassified |
D07133 |
Raltegravir potassium (JAN/USAN); Isentress (TN) |
(P) unclassified |
D07135 |
Clorindione (INN); G-25766 |
(P) unclassified |
D07136 |
Diphenadione (INN) |
(P) unclassified |
D07137 |
Tioclomarol (INN) |
(P) unclassified |
D07139 |
Cloricromen (INN) |
(P) unclassified |
D07144 |
Dabigatran etexilate (USAN/INN); Pradaxa (TN) |
(P) Transporter induction: ABCB1 |
D07165 |
Ivabradine (USAN/INN) |
(P) unclassified |
D07175 |
Palonosetron (INN); Aloxi (TN) |
(P) unclassified |
D07192 |
Benfluorex (INN/BAN); Mediaxal (TN) |
(P) unclassified |
D07203 |
Methylprednisolone aceponate (INN); Advantan (TN) |
(P) unclassified |
D07214 |
Tiratricol (INN); Tiracana (TN) |
(P) unclassified |
D07226 |
Fesoterodine (INN) |
(P) unclassified |
D07283 |
Esketamine (USAN/INN) |
(P) CYP induction: CYP2B6 |
D07299 |
Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) |
(P) Enzyme: CYP2C9 / Target: SCN10A SCN3A SCN9A |
D07334 |
Imipraminoxide (INN) |
(P) unclassified |
D07335 |
Amineptine (INN); Survector (TN) |
(P) unclassified |
D07336 |
Quinupramine (INN) |
(P) unclassified |
D07402 |
Levocetirizine (USAN/INN); Xazal (TN) |
(P) unclassified |
D07407 |
Rupatadine (INN) |
(P) unclassified |
D07448 |
Amitriptyline (INN); Laroxyl (TN) |
(P) unclassified |
D07450 |
Amlodipine (USP/INN); Norvasc (TN) |
(P) unclassified |
D07457 |
Anisindione (INN); Miradon (TN) |
(P) unclassified |
D07474 |
Atorvastatin (INN); Lipitor (TN); Sortis (TN) |
(P) Transporter induction: ABCB1 |
D07486 |
Azithromycin (INN); Azasite (TN); Azithromycin (TN) |
(P) Transporter induction: ABCB1 |
D07494 |
Barnidipine (INN); Vasexten (TN) |
(P) unclassified |
D07507 |
Zidovudine and lamivudine; Combivir (TN); Lamivudine zidovudine (TN) |
(P) unclassified |
D07508 |
Benfluorex hydrochloride; Mediator (TN) |
(P) unclassified |
D07509 |
Benidipine (INN) |
(P) unclassified |
D07520 |
Bepridil (INN); Bepadin (TN) |
(P) Enzyme: CYP2C9 |
D07523 |
Betaine (JAN); Cystadane (TN) |
(P) unclassified |
D07538 |
Bosentan (INN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2C9 |
D07545 |
Brovincamine (INN); Sarbromin (TN) |
(P) unclassified |
D07552 |
Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D07564 |
Allopurinol sodium; Aloprim (TN) |
(P) unclassified |
D07569 |
Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) |
(P) unclassified |
D07585 |
Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine; Cleamine A (TN) |
(P) unclassified |
D07601 |
Butriptyline (INN); Evadyne (TN) |
(P) unclassified |
D07603 |
Caffeine citrate (USP); Cafcit (TN) |
(P) unclassified |
D07626 |
Caspofungin (INN); Cancidas (TN) |
(P) unclassified |
D07661 |
Cerivastatin (INN) |
(P) unclassified |
D07662 |
Cetirizine (INN); Cetiderm (TN) |
(P) Transporter induction: ABCB1 |
D07667 |
Cevimeline (INN) |
(P) unclassified |
D07674 |
Chloramphenicol stearate; Quemicetina (TN) |
(P) unclassified |
D07675 |
Chloramphenicol succinate; Chloramphenicol ICN (TN) |
(P) unclassified |
D07702 |
Ciprofloxacin lactate; Ciproxin (TN) |
(P) unclassified |
D07704 |
Citalopram (USP/INN); Citadur (TN) |
(P) Transporter induction: ABCB1 |
D07705 |
Citalopram hydrochloride; Seropram (TN) |
(P) Transporter induction: ABCB1 |
D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(P) unclassified |
D07727 |
Clomipramine (INN); Anafranil (TN) |
(P) unclassified |
D07729 |
Clopidogrel (USP/INN); Clopidogrel (TN); Plavix (TN) |
(P) CYP induction: CYP2B6 |
D07736 |
Cloricromen hydrohloride; Proendotel (TN) |
(P) unclassified |
D07740 |
Codeine hydrochloride; Bisoltus (TN) |
(P) unclassified |
D07748 |
Conivaptan (INN) |
(P) CYP induction: CYP3A |
D07760 |
Cyclophosphamide (INN); Cyclophosphamide (TN); Cytoxan (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D07782 |
Delavirdine (INN) |
(P) CYP induction: CYP3A |
D07791 |
Desipramine (INN) |
(P) unclassified |
D07793 |
Desvenlafaxine (INN); Khedezla (TN) |
(P) unclassified |
D07796 |
Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) |
(P) unclassified |
D07797 |
Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) |
(P) unclassified |
D07798 |
Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) |
(P) unclassified |
D07799 |
Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) |
(P) unclassified |
D07800 |
Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) |
(P) unclassified |
D07801 |
Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) |
(P) unclassified |
D07802 |
Dexamethasone phosphate; Decadron-phosphate (TN) |
(P) unclassified |
D07803 |
Dexchlorpheniramine (INN); d-Chloropheniramine; Dapriton (TN) |
(P) CYP induction: CYP3A |
D07812 |
Dibenzepin (INN) |
(P) unclassified |
D07831 |
Dihydrocodeine (INN); Remedacen (TN) |
(P) unclassified |
D07832 |
Dihydrocodeine thiocyanate; Paracodin (TN) |
(P) unclassified |
D07837 |
Dihydroergotamine (INN); Neomigran (TN) |
(P) unclassified |
D07838 |
Dihydroergotamine tartrate; Divegal (TN) |
(P) unclassified |
D07839 |
Dihydroergotoxine; Co-Dergocrin (TN) |
(P) unclassified |
D07845 |
Diltiazem (INN); Surazem (TN) |
(P) unclassified |
D07866 |
Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) |
(P) unclassified |
D07867 |
Dolasetron (INN) |
(P) CYP induction: CYP3A |
D07868 |
Domperidone maleate; Domperidone (TN) |
(P) unclassified |
D07869 |
Donepezil (JAN/INN); Donaz (TN); Allydone (TN) |
(P) unclassified |
D07871 |
Dorzolamide (INN); Trusopt (TN) |
(P) Enzyme: CYP2C9 |
D07872 |
Dosulepin (INN); Dothiepin; Dothep (TN) |
(P) unclassified |
D07873 |
Doxapram (INN); Docatone (TN) |
(P) unclassified |
D07875 |
Doxepin (INN); Sinequan (TN) |
(P) Enzyme: CYP2C9 |
D07876 |
Doxycycline (INN); Doxychel (TN); Doxycycline (TN) |
(P) unclassified |
D07877 |
Doxycycline hydrochloride; Vibramycin (TN) |
(P) unclassified |
D07887 |
Eletriptan (INN) |
(P) unclassified |
D07905 |
Ergometrine (INN) |
(P) unclassified |
D07906 |
Ergotamine (INN) |
(P) unclassified |
D07907 |
Erlotinib (INN) |
(P) unclassified |
D07909 |
Erythromycin thiocyanate; Erythrocin (TN) |
(P) CYP induction: CYP3A |
D07910 |
Erythromycin stinoprate (INN); Erysec (TN) |
(P) CYP induction: CYP3A |
D07913 |
Escitalopram (INN); Esertia (TN) |
(P) unclassified |
D07917 |
Esomeprazole (INN); Inexium paranova (TN) |
(P) unclassified |
D07918 |
Estradiol hemihydrate; Estrasorb (TN); Vagifem (TN) |
(P) unclassified |
D07919 |
Estradiol 17 beta-hemisuccinate; 17beta-Estradiol hemisuccinate; Eutocol (TN) |
(P) unclassified |
D07928 |
Ethinylestradiol propanesulfonate; Turisteron (TN) |
(P) unclassified |
D07929 |
Ethylmorphine (BAN) |
(P) unclassified |
D07945 |
Fenfluramine (INN); Ponderax (TN) |
(P) CYP induction: CYP2B6 |
D07962 |
Flecainide (INN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D07969 |
Fluindione (INN); Previsccan (TN) |
(P) unclassified |
D07974 |
Fluorouracil sodium salt; Fluorouracil (TN) |
(P) unclassified |
D07981 |
Fluticasone (INN); Fluticaps (TN) |
(P) unclassified |
D07983 |
Fluvastatin (INN); Fluvas (TN) |
(P) Enzyme: CYP2C9 / CYP inhibition: CYP2C9 |
D07984 |
Fluvoxamine (INN) |
(P) unclassified |
D08031 |
Guanfacine (INN); Estulic (TN) |
(P) unclassified |
D08035 |
Haloperidol lactate; Haldol (TN) |
(P) unclassified |
D08045 |
Hydrocodone (INN); Dihydrocodeinone |
(P) CYP induction: CYP2B6 |
D08046 |
Hydrocodone hydrochloride; Dihydrocodeinone hydrochloride; Dicodid (TN) |
(P) CYP induction: CYP2B6 |
D08050 |
Hydroxychloroquine (INN); Polirreumin (TN) |
(P) unclassified |
D08066 |
Imatinib (INN); Glamox (TN) |
(P) unclassified |
D08070 |
Imipramine (INN); Tofranil (TN) |
(P) unclassified |
D08071 |
Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) |
(P) unclassified |
D08072 |
Imipraminoxide hydrochloride; Elepsin (TN) |
(P) unclassified |
D08080 |
Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP18); Insulin Humacart (TN) |
(P) unclassified |
D08086 |
Irinotecan (INN); Biotecan (TN) |
(P) unclassified |
D08095 |
Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) |
(P) unclassified |
D08108 |
Lapatinib (INN) |
(P) Transporter induction: ABCB1 |
D08111 |
Lercanidipine (INN); Lercanil (TN) |
(P) CYP induction: CYP3A |
D08116 |
Levobupivacaine (INN); Novabupi (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08118 |
Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN); Xyzal (TN) |
(P) unclassified |
D08125 |
Levothyroxine (BAN); Forthyron (TN) |
(P) unclassified |
D08127 |
Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08128 |
Liothyronine (INN); Thyrolar (TN) |
(P) unclassified |
D08129 |
Liothyronine hydrochloride; Thyrotradin (TN) |
(P) unclassified |
D08140 |
Lofepramine (INN) |
(P) unclassified |
D08144 |
Loperamide (INN); Diamide (TN) |
(P) Transporter induction: ABCB1 |
D08148 |
Loxapine hydrochloride; Desconex (TN) |
(P) unclassified |
D08155 |
Manidipine (INN); Manidipine 6300; Artedil (TN) |
(P) unclassified |
D08171 |
Melitracen (INN); Adelax (TN) |
(P) unclassified |
D08195 |
Methadone (BAN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 / Transporter induction: ABCB1 |
D08207 |
Methylergometrine (INN); Ergotyl (TN) |
(P) unclassified |
D08214 |
Metronidazole benzoate (USP); Elyzol (TN) |
(P) CYP inhibition: CYP2C9 |
D08215 |
Mexiletine (INN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08216 |
Mianserin (INN); Tolvon (TN) |
(P) unclassified |
D08227 |
Mometasone (INN) |
(P) unclassified |
D08229 |
Montelukast (INN); Brondilat (TN) |
(P) Enzyme: CYP2C9 |
D08236 |
Mosapride (INN); Mosart (TN) |
(P) unclassified |
D08255 |
Naratriptan (INN); Naramig (TN) |
(P) Enzyme: CYP2C9 |
D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) unclassified |
D08270 |
Nicardipine (INN); Cardene (TN) |
(P) unclassified |
D08283 |
Nordazepam (INN); Calmday (TN) |
(P) unclassified |
D08288 |
Nortriptyline (INN); Nortrilen (TN) |
(P) unclassified |
D08291 |
Ofloxacin hydrochloride; Tarivid (TN) |
(P) unclassified |
D08297 |
Opipramol (INN); Opipramol dura (TN) |
(P) unclassified |
D08351 |
Phenformin (BAN) |
(P) unclassified |
D08352 |
Phenformin hydrochloride; Debei (TN) |
(P) unclassified |
D08354 |
Phenindione (INN); Hedulin (TN) |
(P) unclassified |
D08363 |
Phenylbutazone calcium; Peralgin (TN) |
(P) CYP inhibition: CYP2C9 |
D08364 |
Phenylbutazone sodium; Ambene (TN) |
(P) CYP inhibition: CYP2C9 |
D08378 |
Pioglitazone (INN); Actos (TN) |
(P) unclassified |
D08408 |
Pranlukast (INN); Azlaire (TN) |
(P) unclassified |
D08424 |
Procaterol (INN); Meptin (TN) |
(P) unclassified |
D08435 |
Propafenone (INN); Propafenon hexal (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08441 |
Propiverine (INN) |
(P) unclassified |
D08447 |
Protriptyline (INN) |
(P) unclassified |
D08456 |
Quetiapine (INN); Norsic (TN) |
(P) unclassified |
D08458 |
Quinidine (BAN); Kinidin (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08459 |
Quinidine phenylethylbarbiturate; Quinidine 5-ethyl 5-phenyl barbiturate; Natisedine (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08460 |
Quinine (BAN); Kinder Quinina (TN) |
(P) Transporter induction: ABCB1 |
D08461 |
Quinine dihydrochloride; Quinine (TN) |
(P) Transporter induction: ABCB1 |
D08463 |
Rabeprazole (INN); Eraloc (TN) |
(P) unclassified |
D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) unclassified |
D08481 |
Rilmazafone (INN) |
(P) unclassified |
D08488 |
Amlodipine besilate and atorvastatin calcium; Caduet (TN) |
(P) unclassified |
D08490 |
Ropivacaine (INN); Naropin (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D08491 |
Rosiglitazone (INN); Gaudil (TN) |
(P) unclassified |
D08493 |
Dorzolamide hydrochloride and timolol maleate (JP18); Cosopt (TN) |
(P) Enzyme: CYP2C9 |
D08497 |
Rupatadine fumarate (JAN); Rinialer (TN); Rupafin (TN) |
(P) unclassified |
D08508 |
Sarpogrelate (INN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D08511 |
Setiptiline (INN) |
(P) unclassified |
D08514 |
Sildenafil (INN); Aphrodil (TN) |
(P) unclassified |
D08516 |
Sitagliptin (USAN/INN) |
(P) unclassified |
D08522 |
Solifenacin (INN) |
(P) unclassified |
D08552 |
Sunitinib (INN) |
(P) unclassified |
D08553 |
Suxethonium chloride (INN); Curacit (TN) |
(P) unclassified |
D08556 |
Tacrolimus (INN); Prograf (TN) |
(P) unclassified |
D08559 |
Tamoxifen (INN); Tamoxifen (TN); Tamoplex (TN) |
(P) unclassified |
D08575 |
Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) |
(P) unclassified |
D08594 |
Ticlopidine (INN); Ticlopidin-Puren (TN) |
(P) unclassified |
D08616 |
Teneligliptin (INN) |
(P) unclassified |
D08618 |
Topotecan (BAN); Hycamtin (TN) |
(P) Transporter induction: ABCB1 |
D08620 |
Toremifene (INN); Fareston (TN) |
(P) unclassified |
D08623 |
Tramadol (INN); Amanda (TN) |
(P) unclassified |
D08626 |
Trazodone (INN); Trittico (TN) |
(P) unclassified |
D08655 |
Tubocurarine chloride (INN); Tubaine (TN); Tubocurarine Chloride (TN) |
(P) unclassified |
D08667 |
Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) |
(P) unclassified |
D08668 |
Vardenafil (USAN/INN); Levitra (TN) |
(P) unclassified |
D08670 |
Venlafaxine (INN); Efectin (TN) |
(P) unclassified |
D08675 |
Vinblastine (INN); Vinblastina (TN) |
(P) unclassified |
D08676 |
Vinburnine (INN); Cervoxan (TN) |
(P) unclassified |
D08677 |
Vincamine (INN); Cetal retard (TN) |
(P) unclassified |
D08678 |
Vincamine hydrochloride; Vadicate (TN) |
(P) unclassified |
D08679 |
Vincristine (INN); Tecnocris (TN) |
(P) CYP induction: CYP3A |
D08680 |
Vinorelbine (INN); Navelbine (TN) |
(P) unclassified |
D08682 |
Warfarin (INN); Warfarine; Choice (TN) |
(P) Enzyme: CYP2C9 |
D08690 |
Zolpidem (INN); Sanval (TN) |
(P) unclassified |
D08695 |
dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea; Coughcode N (TN) |
(P) unclassified |
D08697 |
Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate; Opisezol codeine (TN) |
(P) unclassified |
D08699 |
Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) |
(P) unclassified |
D08774 |
Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) |
(P) unclassified |
D08843 |
Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) |
(P) unclassified |
D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) unclassified |
D08860 |
Apremilast (JAN/USAN); Otezla (TN) |
(P) unclassified |
D08870 |
Belinostat (USAN/INN); Beleodaq (TN) |
(P) Enzyme: CYP2C9 |
D08897 |
Dapagliflozin (JAN/USAN/INN); Forxiga (TN) |
(P) unclassified |
D08903 |
Dexlansoprazole (INN/USAN); Dexilant (TN) |
(P) unclassified |
D08914 |
Eribulin mesylate (USAN); Eribulin mesilate (JAN); Halaven (TN) |
(P) unclassified |
D08923 |
Fesoterodine fumarate (JAN/USAN); Toviaz (TN) |
(P) unclassified |
D08950 |
Neratinib (USAN/INN) |
(P) unclassified |
D08953 |
Nilotinib (USAN/INN) |
(P) Transporter induction: ABCB1 |
D08964 |
Perampanel (USAN); Fycompa (TN) |
(P) CYP induction: CYP3A |
D08969 |
Pimavanserin tartrate (USAN); Nuplazide (TN) |
(P) unclassified |
D08976 |
Pomalidomide (JAN/USAN/INN); Pomalyst (TN) |
(P) unclassified |
D08988 |
Rolapitant hydrochloride (USAN); Varubi (TN) |
(P) unclassified |
D08996 |
Saxagliptin (USAN/INN) |
(P) unclassified |
D09012 |
Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) |
(P) unclassified |
D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(CI,P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D09032 |
Vinflunine ditartrate (USAN); Javlor (TN) |
(P) unclassified |
D09033 |
Voclosporin (JAN/USAN/INN); Lupkynis (TN) |
(P) unclassified |
D09187 |
Estradiol and levonorgestrel; Wellnara (TN); Climara pro (TN) |
(P) unclassified |
D09188 |
Estradiol and norethindrone; Menoaid (TN); Activella (TN); Combipatch (TN); Estradiol and norethindrone acetate (TN) |
(P) unclassified |
D09215 |
Eslicarbazepine (USAN/INN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D09318 |
Indacaterol (USAN/INN) |
(P) Transporter induction: ABCB1 |
D09319 |
Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) |
(P) Transporter induction: ABCB1 |
D09339 |
Esomeprazole potassium (USAN) |
(P) unclassified |
D09347 |
Fostamatinib (USAN) |
(P) unclassified |
D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) unclassified |
D09365 |
Palovarotene (JAN/USAN/INN); Sohonos (TN) |
(P) unclassified |
D09388 |
Tasimelteon (USAN/INN); Hetlioz (TN) |
(P) unclassified |
D09394 |
Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) |
(P) CYP inhibition: CYP2C9 |
D09535 |
Mirabegron (JAN/USAN/INN); Myrbetriq (TN) |
(P) unclassified |
D09544 |
Ozenoxacin (JAN/USAN/INN); Xepi (TN) |
(P) unclassified |
D09546 |
Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) |
(P) Transporter induction: ABCB1 |
D09566 |
Linagliptin (JAN/USAN/INN); Tradjenta (TN) |
(P) unclassified |
D09572 |
Riociguat (JAN/USAN/INN); Adempas (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D09592 |
Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) |
(P) Transporter induction: ABCB1 |
D09594 |
Olmesartan medoxomil and azelnidipine; Rezaltas (TN) |
(P) unclassified |
D09595 |
Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) |
(P) unclassified |
D09612 |
Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A |
D09621 |
Gisadenafil (USAN/INN) |
(P) unclassified |
D09622 |
Gisadenafil besylate (USAN) |
(P) unclassified |
D09637 |
Lomitapide (USAN/INN) |
(P) unclassified |
D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(P) unclassified |
D09666 |
Selumetinib (USAN/INN) |
(P) Enzyme: CYP2C9 |
D09676 |
Tecarfarin (USAN/INN) |
(P) unclassified |
D09677 |
Tecarfarin sodium (USAN) |
(P) unclassified |
D09683 |
Tivozanib (USAN/INN) |
(P) unclassified |
D09698 |
Vilazodone (USAN/INN) |
(P) unclassified |
D09699 |
Vilazodone hydrochloride (USAN); Viibryd (TN) |
(P) unclassified |
D09701 |
Abiraterone acetate (JAN/USP); Zytiga (TN) |
(P) unclassified |
D09707 |
Dabigatran (USAN/INN) |
(P) Transporter induction: ABCB1 |
D09710 |
Edoxaban (USAN/INN) |
(P) Transporter induction: ABCB1 |
D09720 |
Rilpivirine (JAN/USAN/INN); Rekambys (TN) |
(CI,P) CYP induction: CYP3A |
D09724 |
Afatinib (USAN/INN) |
(P) Transporter induction: ABCB1 |
D09727 |
Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) |
(P) unclassified |
D09728 |
Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) |
(P) unclassified |
D09729 |
Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) |
(P) unclassified |
D09730 |
Olaparib (JAN/USAN/INN); Lynparza (TN) |
(P) CYP induction: CYP3A |
D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) unclassified |
D09733 |
Afatinib dimaleate (USAN); Afatinib maleate (JAN); Gilotrif (TN); Giotrif (TN) |
(P) Transporter induction: ABCB1 |
D09741 |
Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) |
(P) unclassified |
D09742 |
Lansoprazole, amoxicillin hydrate and metronidazole; Lampion (TN) |
(P) unclassified |
D09743 |
Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) |
(P) unclassified |
D09744 |
Pioglitazone hydrochloride and metformin hydrochloride (JP18); Pioglitazone and metformin; Metact (TN) |
(P) unclassified |
D09745 |
Valsartan and amlodipine besilate; Exforge (TN) |
(P) unclassified |
D09753 |
Saxagliptin hydrate (JAN); Onglyza (TN) |
(P) unclassified |
D09755 |
Cabazitaxel (USAN/INN); Jevtana (TN) |
(P) CYP induction: CYP3A |
D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) unclassified |
D09763 |
Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JAN); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) |
(P) unclassified |
D09765 |
Vorapaxar (USAN/INN) |
(P) unclassified |
D09766 |
Vorapaxar sulfate (JAN/USAN); Zontivity (TN) |
(P) unclassified |
D09773 |
Isoniazid glucuronate sodium (JAN) |
(P) unclassified |
D09783 |
Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) |
(P) unclassified |
D09785 |
Delamanid (JAN/USAN); Deltyba (TN) |
(P) unclassified |
D09796 |
Hydrocortisone caproate (JAN) |
(P) CYP induction: CYP3A |
D09807 |
Difethiarol (JAN); Difethialone |
(P) unclassified |
D09847 |
Metildigoxin (INN); Medigoxin (BAN) |
(P) Transporter induction: ABCB1 |
D09848 |
Pioglitazone hydrochloride and glimepiride tablets (JP18); Pioglitazone and glimepiride; Duetact; Sonias (TN) |
(P) Enzyme: CYP2C9 |
D09872 |
Bedaquiline (USAN/INN) |
(P) unclassified |
D09873 |
Bedaquiline fumarate (JAN/USAN); Sirturo (TN) |
(P) unclassified |
D09876 |
Cariprazine hydrochloride (JAN/USAN); Vraylar (TN) |
(P) unclassified |
D09881 |
Cobicistat (JAN/USAN/INN); Tybost (TN) |
(P) CYP induction: CYP3A |
D09889 |
Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) |
(P) unclassified |
D09893 |
Eliglustat (USAN/INN) |
(P) Transporter induction: ABCB1 |
D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(P) Transporter induction: ABCB1 |
D09919 |
Lenvatinib (USAN/INN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D09920 |
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D09950 |
Ponatinib (USAN/INN) |
(P) CYP induction: CYP3A |
D09951 |
Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) |
(P) CYP induction: CYP3A |
D09955 |
Quizartinib (USAN/INN) |
(P) CYP induction: CYP3A |
D09956 |
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) |
(P) CYP induction: CYP3A |
D09958 |
Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) |
(CI,P) CYP induction: CYP3A |
D09959 |
Ruxolitinib (USAN/INN) |
(P) unclassified |
D09960 |
Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) |
(P) unclassified |
D09970 |
Tofacitinib (USAN); Tasocitinib |
(P) unclassified |
D09987 |
Vaniprevir (JAN/USAN/INN); Vanihep (TN) |
(P) CYP induction: CYP3A |
D09989 |
Vardenafil hydrochloride (USP) |
(P) unclassified |
D09994 |
Selexipag (JAN/USAN/INN); Uptravi (TN) |
(P) unclassified |
D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP inhibition: CYP2C9 |
D09997 |
Cariprazine (USAN/INN) |
(P) unclassified |
D09999 |
Tramadol hydrochloride and acetaminophen; Tramcet (TN) |
(P) unclassified |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) unclassified |
D10019 |
Panobinostat lactate (JAN); Farydak (TN) |
(P) unclassified |
D10024 |
Selumetinib sulfate (JAN/USAN); Koselugo (TN) |
(P) Enzyme: CYP2C9 |
D10025 |
Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) |
(P) unclassified |
D10027 |
Udenafil (USAN/INN) |
(P) unclassified |
D10064 |
Dabrafenib (USAN) |
(P) CYP induction: CYP2C9 |
D10065 |
Daclatasvir (USAN) |
(P) Transporter induction: ABCB1 |
D10066 |
Dolutegravir (USAN); Tivicay (TN) |
(P) unclassified |
D10081 |
Simeprevir (JAN/USAN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) CYP induction: CYP3A |
D10093 |
Asunaprevir (JAN/USAN); Sunvepra (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10095 |
Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) |
(P) unclassified |
D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) CYP induction: CYP2C9 |
D10105 |
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) |
(P) Transporter induction: ABCB1 |
D10113 |
Dolutegravir sodium (JAN/USAN); Tivicay (TN) |
(P) unclassified |
D10119 |
Sonidegib (USAN/INN); Erismodegib |
(P) CYP induction: CYP3A |
D10120 |
Esomeprazole strontium (USAN); Esomeprazole strontium tetrahydrate; Esomeprazole strontium (TN) |
(P) unclassified |
D10131 |
Ixazomib citrate (JAN/USAN); Ninlaro (TN) |
(P) unclassified |
D10135 |
Macitentan (JAN/USAN); Opsumit (TN) |
(CI,P) unclassified |
D10137 |
Regorafenib hydrate (JAN); Stivarga (TN) |
(P) Transporter induction: ABCB1 |
D10138 |
Regorafenib (USAN/INN); Stivarga (TN) |
(P) Transporter induction: ABCB1 |
D10158 |
Safinamide (USAN/INN) |
(P) unclassified |
D10159 |
Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) |
(P) unclassified |
D10160 |
Mitiglinide calcium hydrate and voglibose; Glubes (TN) |
(P) unclassified |
D10184 |
Vortioxetine (USAN); Brintellix (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D10185 |
Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D10188 |
Naldemedine (USAN/INN) |
(P) unclassified |
D10190 |
Tivozanib hydrochloride (USAN); Tivozanib hydrochloride monohydrate; Fotivda (TN) |
(P) unclassified |
D10191 |
Safinamide mesylate (USAN); Safinamide mesilate (JAN); Safinamide methanesulfonate; Xadago (TN); Equfina (TN) |
(P) unclassified |
D10195 |
Luseogliflozin hydrate (JAN); Lusefi (TN) |
(P) unclassified |
D10196 |
Ipragliflozin (INN) |
(P) unclassified |
D10200 |
Ipragliflozin L-proline (JAN); Suglat (TN) |
(P) unclassified |
D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
D10223 |
Ibrutinib (JAN/USAN); Imbruvica (TN) |
(P) CYP induction: CYP3A |
D10243 |
Irbesartan and amlodipine besilate (JP18); Aimix (TN) |
(P) unclassified |
D10244 |
Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) |
(P) unclassified |
D10246 |
Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) |
(P) unclassified |
D10251 |
Glimepiride and rosiglitazone maleate; Avandaryl (TN) |
(P) unclassified |
D10253 |
Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) |
(P) unclassified |
D10258 |
Simvastatin and sitagliptin phosphate; Juvisync (TN) |
(P) unclassified |
D10261 |
Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) |
(P) unclassified |
D10262 |
Saxagliptin hydrochloride; Onglyza (TN) |
(P) unclassified |
D10263 |
Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) |
(P) unclassified |
D10264 |
Linagliptin and metformin hydrochloride; Jentaduet (TN) |
(P) Transporter induction: ABCB1 |
D10265 |
Glipizide and metformin hydrochloride; Metaglip (TN) |
(P) unclassified |
D10266 |
Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) |
(P) unclassified |
D10293 |
Carbidopa, levodopa and entacapone; Stalevo (TN) |
(P) CYP inhibition: CYP2C9 |
D10306 |
Avatrombopag (USAN/INN) |
(P) Enzyme: CYP2C9 |
D10307 |
Avatrombopag maleate (JAN/USAN); Doptelet (TN) |
(P) Enzyme: CYP2C9 |
D10308 |
Baricitinib (JAN/USAN/INN); Olumiant (TN) |
(P) Transporter induction: ABCB1 |
D10309 |
Brexpiprazole (JAN/USAN/INN); Rexulti (TN) |
(P) unclassified |
D10313 |
Ertugliflozin (USAN/INN) |
(P) unclassified |
D10315 |
Momelotinib (USAN/INN) |
(P) Enzyme: CYP2C9 |
D10319 |
Panobinostat (USAN/INN); Farydak (TN) |
(P) unclassified |
D10355 |
Aripiprazole cavoxil (USAN) |
(P) unclassified |
D10358 |
Momelotinib dihydrochloride (USAN) |
(P) Enzyme: CYP2C9 |
D10364 |
Aripiprazole lauroxil (USAN); Aristada (TN) |
(P) unclassified |
D10366 |
Sofosbuvir (JAN/USAN/INN); Sovaldi (TN) |
(CI,P) Transporter induction: ABCB1 |
D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
D10375 |
Naloxegol oxalate (USAN); Movantik (TN); Moventig (TN) |
(P) CYP induction: CYP3A |
D10385 |
Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) |
(P) unclassified |
D10396 |
Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN); Ofev (TN) |
(P) Transporter induction: ABCB1 |
D10428 |
Tenofovir alafenamide (USAN/INN) |
(P) Transporter induction: ABCB1 |
D10433 |
Vibegron (JAN/USAN/INN); Beova (TN); Gemtesa (TN) |
(P) Transporter induction: ABCB1 |
D10434 |
Vintafolide (USAN/INN) |
(P) unclassified |
D10450 |
Alectinib hydrochloride (JAN); Alecensa (TN) |
(P) unclassified |
D10452 |
Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) |
(P) CYP induction: CYP3A |
D10459 |
Empagliflozin (JAN/USAN/INN); Jardiance (TN) |
(P) Transporter induction: ABCB1 |
D10461 |
Dienogest and estradiol valerate; Natazia (TN) |
(P) CYP induction: CYP3A |
D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) unclassified |
D10469 |
Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10478 |
Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) |
(P) unclassified |
D10479 |
Naloxegol (USAN/INN) |
(P) CYP induction: CYP3A |
D10481 |
Nintedanib (USAN/INN); Ofev (TN) |
(P) Transporter induction: ABCB1 |
D10500 |
Metformin hydrochloride and repaglinide; Prandimet (TN) |
(P) unclassified |
D10501 |
Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) |
(P) unclassified |
D10502 |
Gemigliptin (INN) |
(P) unclassified |
D10505 |
Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) |
(P) Transporter induction: ABCB1 |
D10506 |
Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) |
(P) unclassified |
D10512 |
Brinzolamide and timolol maleate; Azorga (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D10513 |
Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) |
(P) CYP induction: CYP2B6 |
D10516 |
Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) |
(P) unclassified |
D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) unclassified |
D10520 |
Rabeprazole, amoxicillin and metronidazole; Rabefine (TN) |
(P) unclassified |
D10524 |
Azilsartan and amlodipine besilate; Zacras (TN) |
(P) unclassified |
D10525 |
Valsartan and cilnidipine; Atedio (TN) |
(P) unclassified |
D10527 |
Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) |
(P) unclassified |
D10533 |
Umeclidinium bromide and vilanterol; Anoro (TN) |
(P) unclassified |
D10537 |
Methylthioninium chloride hydrate (JAN); Methylene blue (TN) |
(P) CYP inhibition: CYP2C9 |
D10542 |
Alectinib (USAN/INN) |
(P) unclassified |
D10548 |
Cabotegravir (JAN/USAN/INN); Vocabria (TN); Apretude (TN) |
(CI) unclassified |
D10549 |
Cabotegravir sodium (JAN/USAN); Vocabria (TN) |
(CI) unclassified |
D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) CYP inhibition: CYP2C9 / CYP induction: CYP3A |
D10560 |
Idelalisib (JAN/USAN/INN); Zydelig (TN) |
(P) CYP induction: CYP3A |
D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) CYP induction: CYP3A |
D10570 |
Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) |
(P) unclassified |
D10571 |
Rilpivirine hydrochloride, tenofovir disoproxil fumarate and emtricitabine; Complera (TN); Eviplera (TN) |
(P) CYP induction: CYP3A |
D10572 |
Fosnetupitant and palonosetron hydrochloride; Netupitant and palonosetron hydrochloride; Akynzeo (TN) |
(P) unclassified |
D10578 |
Ledipasvir and sofosbuvir; Harvoni (TN) |
(CI,P) Transporter induction: ABCB1 |
D10582 |
Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10586 |
Dapagliflozin and metformin; Xigduo xr (TN) |
(P) unclassified |
D10587 |
Canagliflozin and metformin; Invokamet (TN) |
(P) unclassified |
D10588 |
Empagliflozin and linagliptin; Glyxambi (TN) |
(P) Transporter induction: ABCB1 |
D10600 |
Dolutegravir, abacavir and lamivudine; Triumeq (TN) |
(P) unclassified |
D10605 |
Tenofovir alafenamide fumarate (JAN/USAN); Vemlidy (TN) |
(P) Transporter induction: ABCB1 |
D10612 |
Benzhydrocodone (USAN/INN) |
(P) unclassified |
D10624 |
Doravirine (JAN/USAN/INN); Pifeltro (TN) |
(CI,P) CYP induction: CYP3A |
D10625 |
Elbasvir (JAN/USAN/INN); Erelsa (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10627 |
Esketamine hydrochloride (JAN/USAN); Spravato (TN) |
(P) CYP induction: CYP2B6 |
D10630 |
Fedratinib (USAN/INN) |
(P) unclassified |
D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) unclassified |
D10639 |
Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10642 |
Irinotecan sucrosofate (USAN) |
(P) unclassified |
D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(CI,P) CYP induction: CYP3A |
D10644 |
Isavuconazonium (USAN) |
(CI,P) CYP induction: CYP3A |
D10662 |
Rimegepant (USAN/INN) |
(P) unclassified |
D10663 |
Rimegepant sulfate (USAN); Nurtec odt (TN); Vydura (TN) |
(P) unclassified |
D10669 |
Sotagliflozin (USAN/INN); Inpefa (TN) |
(P) unclassified |
D10673 |
Ubrogepant (USAN/INN); Ubrelvy (TN) |
(P) unclassified |
D10675 |
Valbenazine (USAN/INN) |
(P) unclassified |
D10679 |
Venetoclax (JAN/USAN/INN); Venclexta (TN) |
(P) unclassified |
D10688 |
Abemaciclib (JAN/USAN/INN); Verzenio (TN) |
(P) CYP induction: CYP3A |
D10692 |
Benzhydrocodone hydrochloride (USAN) |
(P) unclassified |
D10696 |
Capmatinib (USAN/INN) |
(P) unclassified |
D10707 |
Fostemsavir (USAN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10708 |
Fostemsavir tromethamine (USAN); Fostemsavir trometamol; Rukobia (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10709 |
Gilteritinib (USAN/INN) |
(P) Transporter induction: ABCB1 |
D10711 |
Pemafibrate (JAN); Parmodia (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP3A |
D10729 |
Sonidegib phosphate (USAN); Sonidegib diphosphate; Odomzo (TN) |
(P) CYP induction: CYP3A |
D10734 |
Temsavir (USAN/INN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10742 |
Rolapitant (USAN/INN); Varubi (TN) |
(P) unclassified |
D10743 |
Vildagliptin and metformin hydrochloride |
(P) unclassified |
D10745 |
Ombitasvir, paritaprevir and ritonavir; Technivie (TN) |
(P) Transporter induction: ABCB1 |
D10749 |
Pitolisant (USAN/INN); Wakix (TN); Ozawade (TN) |
(P) unclassified |
D10752 |
Empagliflozin and metformin; Synjardy (TN) |
(P) unclassified |
D10753 |
Atazanavir and cobicistat; Evotaz (TN) |
(P) unclassified |
D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(CI) unclassified |
D10756 |
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) |
(P) CYP induction: CYP3A |
D10761 |
Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) |
(P) CYP induction: CYP3A |
D10766 |
Osimertinib mesylate (USAN); Osimertinib mesilate (JAN); Tagrisso (TN) |
(P) CYP induction: CYP3A |
D10772 |
Lascufloxacin hydrochloride (JAN); Lasvic (TN) |
(P) unclassified |
D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) unclassified |
D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) unclassified |
D10780 |
Perampanel hydrate (JAN); Fycompa (TN) |
(P) CYP induction: CYP3A |
D10797 |
Copanlisib hydrochloride (USAN) |
(P) CYP induction: CYP3A |
D10798 |
Copanlisib hydrochloride hydrate (JAN); Aliqopa (TN) |
(P) CYP induction: CYP3A |
D10800 |
Gilteritinib fumarate (JAN/USAN); Xospata (TN) |
(P) Transporter induction: ABCB1 |
D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) CYP induction: CYP2C9 |
D10805 |
Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) |
(P) unclassified |
D10811 |
Fentanyl hydrochloride (JAN); Ionsys (TN) |
(P) unclassified |
D10822 |
Ciprofloxacin hydrate (JAN); Ciprofloxacin hemiheptahydrate |
(P) unclassified |
D10823 |
Clopidogrel hydrochloride; Clopidogrel (TN) |
(P) CYP induction: CYP2B6 |
D10824 |
Clopidogrel besilate; Clopidogrel besylate; Clopidogrel (TN) |
(P) CYP induction: CYP2B6 |
D10826 |
Saxagliptin and dapagliflozin; Qtern (TN) |
(P) unclassified |
D10827 |
Sofosbuvir and velpatasvir; Epclusa (TN) |
(CI,P) CYP induction: CYP2B6 / Transporter induction: ABCB1 |
D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(CI) unclassified |
D10835 |
Emtricitabine and tenofovir alafenamide; Descovy (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10836 |
Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) |
(CI,P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10865 |
Bexagliflozin (USAN); Brenzavvy (TN) |
(P) unclassified |
D10866 |
Brigatinib (JAN/USAN); Alunbrig (TN) |
(P) unclassified |
D10867 |
Copanlisib (USAN/INN) |
(P) CYP induction: CYP3A |
D10882 |
Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D10883 |
Ribociclib (USAN/INN) |
(P) unclassified |
D10888 |
Relugolix (JAN/USAN/INN); Orgovyx (TN) |
(P) Transporter induction: ABCB1 |
D10889 |
Momelotinib hydrochloride hydrate (JAN); Momelotinib dihydrochloride monohydrate; Ojjaara (TN); Omjjara (TN) |
(P) Enzyme: CYP2C9 |
D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) unclassified |
D10892 |
Esaxerenone (JAN/INN) |
(P) CYP induction: CYP3A |
D10893 |
Acalabrutinib (JAN/USAN/INN); Calquence (TN) |
(P) CYP induction: CYP3A |
D10895 |
Fosaprepitant (INN) |
(P) CYP induction: CYP2C9 |
D10897 |
Teneligliptin and canagliflozin; Teneligliptin and canagliflozin; Canalia (TN) |
(P) Transporter induction: ABCB1 |
D10898 |
Neratinib maleate; Nerlynx (TN) |
(P) unclassified |
D10915 |
Cannabidiol (USAN/INN); CBD; Epidiolex (TN) |
(P) Transporter induction: ABCB1 |
D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) unclassified |
D10927 |
Erdafitinib (JAN/USAN/INN); Balversa (TN) |
(P) Enzyme: CYP2C9 / Transporter induction: ABCB1 |
D10930 |
Etrasimod (USAN) |
(P) Enzyme: CYP2C9 |
D10931 |
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) |
(P) Enzyme: CYP2C9 |
D10954 |
Mirvetuximab soravtansine (USAN/INN); Mirvetuximab soravtansine-gynx; Elahere (TN) |
(P) unclassified |
D10960 |
Nirogacestat (USAN/INN) |
(P) Enzyme: CYP2C9 |
D10964 |
Omaveloxolone (USAN/INN); Skyclarys (TN) |
(P) CYP induction: CYP3A |
D10979 |
Ribociclib succinate (USAN); Kisqali (TN) |
(P) unclassified |
D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
D10994 |
Upadacitinib (USAN/INN) |
(P) unclassified |
D10995 |
Upadacitinib tartrate (USAN) |
(P) unclassified |
D10999 |
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) |
(P) unclassified |
D11000 |
Vamorolone (USAN/INN); Agamree (TN) |
(P) unclassified |
D11009 |
Indacaterol acetate (JAN) |
(P) Transporter induction: ABCB1 |
D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) CYP induction: CYP3A |
D11014 |
Glecaprevir and pibrentasvir; Mavyret (TN) |
(P) Transporter induction: ABCB1 |
D11022 |
Lemborexant (JAN/USAN/INN); Dayvigo (TN) |
(P) unclassified |
D11023 |
Evogliptin (INN) |
(P) unclassified |
D11034 |
Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) |
(P) unclassified |
D11039 |
Bictegravir, emtricitabine and tenofovir alafenamide; Biktarvy (TN) |
(CI) unclassified |
D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) unclassified |
D11043 |
Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) |
(P) unclassified |
D11045 |
Darolutamide (JAN/USAN/INN); Nebeqa (TN) |
(P) unclassified |
D11048 |
Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) |
(P) unclassified |
D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) unclassified |
D11056 |
Mirtazapine hydrate (JAN) |
(P) unclassified |
D11061 |
Osilodrostat (USAN/INN) |
(P) CYP induction: CYP2B6 |
D11062 |
Osilodrostat phosphate (JAN/USAN); Isturisa (TN) |
(P) CYP induction: CYP2B6 |
D11066 |
Ertugliflozin and sitagliptin; Steglujan (TN) |
(P) unclassified |
D11067 |
Ertugliflozin and metformin; Segluromet (TN) |
(P) unclassified |
D11070 |
Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) |
(P) unclassified |
D11072 |
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) |
(P) Enzyme: CYP2C9 |
D11073 |
Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN); Tepmetko (TN) |
(P) unclassified |
D11093 |
Avacopan (JAN/USAN/INN); Tavneos (TN) |
(P) unclassified |
D11095 |
Atorvastatin calcium propylene glycol solvate |
(P) Transporter induction: ABCB1 |
D11113 |
Levothyroxine sodium (INN); Levothyroxine sodium anhydrous |
(P) unclassified |
D11114 |
Esomeprazole magnesium dihydrate |
(P) unclassified |
D11137 |
Larotrectinib (USAN/INN) |
(P) CYP induction: CYP3A |
D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) CYP induction: CYP3A |
D11141 |
Tucatinib (USAN/INN); Tukysa (TN) |
(P) unclassified |
D11150 |
Cenobamate (USAN/INN); Xcopri (TN) |
(P) Target: SCN10A SCN11A SCN1A SCN2A SCN3A SCN4A SCN5A SCN8A SCN9A / CYP induction: CYP2B6 |
D11158 |
Leniolisib (USAN/INN) |
(P) unclassified |
D11159 |
Leniolisib phosphate (USAN); Joenja (TN) |
(P) unclassified |
D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
D11222 |
Selinexor (USAN/INN); Xpovio (TN) |
(P) unclassified |
D11252 |
Fexinidazole (USAN/INN); Fexinidazole (TN) |
(P) unclassified |
D11270 |
Pexidartinib (USAN/INN) |
(P) unclassified |
D11271 |
Pexidartinib hydrochloride (JAN/USAN); Turalio (TN) |
(P) unclassified |
D11282 |
Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) |
(CI,P) CYP induction: CYP3A |
D11296 |
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) |
(P) unclassified |
D11313 |
Atogepant (USAN); Qulipta (TN); Aquipta (TN) |
(P) unclassified |
D11330 |
Voxelotor (USAN); Oxbryta (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D11342 |
Dorzagliatin (USAN) |
(P) unclassified |
D11360 |
Tirzepatide (JAN/USAN); Mounjaro (TN) |
(P) unclassified |
D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) unclassified |
D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(CI) unclassified |
D11389 |
Dutasteride and tamsulosin; Jalyn (TN) |
(P) unclassified |
D11396 |
Doravirine, lamivudine and tenofovir disoproxil; Delstrigo (TN) |
(P) CYP induction: CYP3A |
D11403 |
Asciminib (USAN/INN) |
(P) unclassified |
D11404 |
Asciminib hydrochloride (JAN/USAN); Scemblix (TN) |
(P) unclassified |
D11405 |
Prabotulinumtoxin A (USAN); PrabotulinumtoxinA-xvfs; Jeuveau (TN) |
(P) unclassified |
D11406 |
Risdiplam (JAN/USAN/INN); Evrysdi (TN) |
(P) unclassified |
D11417 |
Pemigatinib (JAN/USAN/INN); Pemazyre (TN) |
(P) unclassified |
D11422 |
Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) |
(P) CYP induction: CYP3A |
D11444 |
Tazemetostat (USAN/INN) |
(P) Transporter induction: ABCB1 |
D11453 |
Nirogacestat hydrobromide (USAN); Ogsiveo (TN) |
(P) Enzyme: CYP2C9 |
D11454 |
Repotrectinib (JAN/USAN); Augtyro (TN) |
(P) unclassified |
D11460 |
Siponimod (USAN/INN) |
(P) Enzyme: CYP2C9 |
D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) Transporter induction: ABCB1 |
D11490 |
Pitolisant hydrochloride (USAN); Wakix (TN) |
(P) unclassified |
D11521 |
Lamivudine, nevirapine and zidovudine |
(P) CYP induction: CYP3A CYP2B6 |
D11522 |
Dolutegravir and lamivudine; Dovato (TN) |
(P) unclassified |
D11553 |
Lidocaine and tetracaine; Pliaglis (TN); Synera (TN) |
(P) unclassified |
D11555 |
Calcium levofolinate hydrate (JP18); Levoleucovorin calcium pentahydrate; Calcium levofolinate pentahydrate; Isovorin (TN) |
(P) unclassified |
D11565 |
Grazoprevir (USAN/INN); Grazoprevir anhydrous |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D11567 |
Insulin degludec and liraglutide; Xultophy (TN) |
(P) unclassified |
D11568 |
Edoxaban tosylate (USAN) |
(P) Transporter induction: ABCB1 |
D11572 |
Beclomethasone dipropionate monohydrate; Beconase aq (TN) |
(P) unclassified |
D11573 |
Oxycodone and ibuprofen |
(P) unclassified |
D11576 |
Naproxen and esomeprazole magnesium; Vimovo (TN) |
(P) Enzyme: CYP2C9 |
D11616 |
Aspirin and omeprazole; Yosprala (TN) |
(P) unclassified |
D11617 |
Eletriptan hydrobromide monohydrate |
(P) unclassified |
D11619 |
Desvenlafaxine succinate anhydrous; Desvenlafaxine succinate (TN) |
(P) unclassified |
D11628 |
Benzhydrocodone and acetaminophen; Apadaz (TN) |
(P) unclassified |
D11630 |
Aminophylline dihydrate |
(P) unclassified |
D11631 |
Lefamulin (USAN/INN) |
(P) unclassified |
D11632 |
Lefamulin acetate (USAN); Xenleta (TN) |
(P) unclassified |
D11652 |
Tenapanor (USAN/INN) |
(P) unclassified |
D11653 |
Tenapanor hydrochloride (JAN/USAN); Ibsrela (TN); Phozevel (TN); Xphozah (TN) |
(P) unclassified |
D11656 |
Azelastine hydrochloride and fluticasone propionate; Dymista (TN) |
(P) unclassified |
D11662 |
Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) |
(P) unclassified |
D11671 |
Elacestrant (USAN/INN) |
(P) Enzyme: CYP2C9 |
D11672 |
Elacestrant hydrochloride (USAN); Elacestrant dihydrochloride; Orserdu (TN) |
(P) Enzyme: CYP2C9 |
D11673 |
Berotralstat (USAN/INN) |
(P) Transporter induction: ABCB1 |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) Transporter induction: ABCB1 |
D11700 |
Elexacaftor, ivacaftor and tezacaftor; Trikafta (TN); Kaftrio (TN) |
(P) CYP induction: CYP3A |
D11706 |
Omeprazole and sodium bicarbonate; Zegerid (TN) |
(P) unclassified |
D11710 |
Phentermine and topiramate; Qsymia (TN) |
(P) unclassified |
D11711 |
Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) |
(P) unclassified |
D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) unclassified |
D11716 |
Odevixibat (USAN); Bylvay (TN) |
(P) Transporter induction: ABCB1 |
D11717 |
Tepotinib (USAN/INN) |
(P) unclassified |
D11720 |
Acalabrutinib maleate (USAN) |
(P) CYP induction: CYP3A |
D11725 |
Futibatinib (JAN/USAN/INN); Lytgobi (TN) |
(P) unclassified |
D11768 |
Pacritinib (USAN/INN); Vonjo (TN) |
(P) unclassified |
D11776 |
Sparsentan (USAN/INN); Filspari (TN) |
(P) CYP induction: CYP3A |
D11784 |
Vonoprazan (USAN/INN) |
(P) unclassified |
D11793 |
Zuranolone (JAN/USAN/INN); Zurzuvae (TN) |
(P) unclassified |
D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
D11807 |
Imeglimin hydrochloride (JAN); Twymeeg (TN) |
(P) unclassified |
D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) unclassified |
D11851 |
Butalbital, acetaminophen, caffeine and codeine phosphate |
(P) unclassified |
D11856 |
Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) |
(P) unclassified |
D11858 |
Omeprazole magnesium, amoxicillin and rifabutin; Talicia (TN) |
(P) CYP induction: CYP3A |
D11860 |
Butalbital, aspirin, caffeine and codeine; Fiorinal with codeine (TN) |
(P) unclassified |
D11881 |
Amlodipine benzoate; Katerzia (TN) |
(P) unclassified |
D11886 |
Daridorexant (USAN/INN) |
(P) unclassified |
D11923 |
Lobeglitazone (INN) |
(P) unclassified |
D11924 |
Beinaglutide (INN) |
(P) unclassified |
D11954 |
Belzutifan (JAN/USAN/INN); Welireg (TN) |
(P) unclassified |
D11966 |
Cabotegravir and rilpivirine; Cabenuva (TN) |
(P) CYP induction: CYP3A |
D11968 |
Teneligliptin hydrobromide (JAN) |
(P) unclassified |
D11969 |
Mobocertinib succinate (JAN); Exkivity (TN) |
(P) CYP induction: CYP3A |
D11977 |
Fruquintinib (JAN/USAN); Fruzaqla (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP3A |
D12001 |
Mobocertinib (USAN/INN) |
(P) CYP induction: CYP3A |
D12015 |
St. John's wort; SJW |
(P) unclassified |
D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) CYP induction: CYP3A |
D12130 |
Drospirenone, ethinyl estradiol and levomefolate calcium; Beyaz (TN); Safyral (TN); Tydemy (TN) |
(P) unclassified |
D12137 |
Elagolix, estradiol and norethisterone; Oriahnn (TN) |
(P) CYP induction: CYP3A |
D12161 |
Lenacapavir (USAN/INN) |
(P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D12162 |
Lenacapavir sodium (JAN/USAN); Sunlenca (TN) |
(CI,P) CYP induction: CYP3A / Transporter induction: ABCB1 |
D12265 |
Mavacamten (JAN/USAN/INN); Camzyos (TN) |
(P) Enzyme: CYP2C9 |
D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(CI,P) unclassified |
D12294 |
Sitagliptin phosphate (JAN) |
(P) unclassified |
D12301 |
Adagrasib (USAN/INN); Krazati (TN) |
(P) unclassified |
D12312 |
Codeine phosphate and chlorpheniramine maleate; Tuxarin (TN) |
(P) unclassified |
D12313 |
Chlorpheniramine polistirex and codeine polistirex; Tuzistra (TN) |
(P) unclassified |
D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(CI,P) CYP induction: CYP3A |
D12388 |
Fosifloxuridine nafalbenamide |
(P) unclassified |
D12403 |
Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) |
(P) unclassified |
D12442 |
Tucatinib ethanolate (JAN); Tucatinib hemiethanolate |
(P) unclassified |
D12444 |
Nilotinib hydrochloride dihydrate (JAN) |
(P) Transporter induction: ABCB1 |
D12483 |
Olutasidenib (USAN/INN); Rezlidhia (TN) |
(P) unclassified |
D12484 |
Carfloglitazar (INN) |
(P) unclassified |
D12486 |
Finasteride and tadalafil; Entadfi (TN) |
(P) unclassified |
D12497 |
Drospirenone and estradiol; Angeliq (TN) |
(P) unclassified |
D12544 |
Vortioxetine hemihydrobromide (USAN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(CI,P) CYP induction: CYP3A |
D12609 |
Dasatinib laurylsulfate (USAN) |
(P) unclassified |
D12619 |
Ensitrelvir (USAN/INN) |
(P) CYP induction: CYP3A |
D12637 |
Darunavir hydrate |
(P) unclassified |
D12703 |
Linagliptin hydrate (JAN); Linagliptin hemihydrate |
(P) unclassified |
D12704 |
Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate |
(P) CYP induction: CYP3A |
D12752 |
Darunavir propylene glycolate |
(P) unclassified |
D12756 |
Vonoprazan and amoxicillin; Voquezna (TN) |
(P) Enzyme: CYP2C9 / CYP induction: CYP2B6 |
D12816 |
Dexlansoprazole sesquihydrate |
(P) unclassified |
D12854 |
Nilotinib laurylsulfate (USAN) |
(P) Transporter induction: ABCB1 |