Target-based Classification of Drugs

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 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
     Adrenaline
       ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
       ADRA1A [HSA:148] [KO:K04135]
       ADRA1D [HSA:146] [KO:K04137]
       ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
         D00095  Epinephrine (USP/INN) <JP/US>
         D00996  Epinephrine hydrochloride (JAN)
         D02149  Epinephrine bitartrate (JAN/USP)
         D07931  Etilefrine (INN)
         D01573  Etilefrine hydrochloride (JP18) <JP>
         D00076  Noradrenaline (JP18) <JP>
         D05206  Norepinephrine bitartrate (USP) <US>
         D08284  Norepinephrine hydrochoride
         D09794  Norepinephrine hydrochloride (JAN)
         D08192  Metaraminol (INN)
         D01019  Metaraminol bitartrate (JAN/USP)
         D00124  Ephedrine (USP)
         D01386  Ephedrine hydrochloride (JP18/USP) <JP/US>
         D04018  Ephedrine sulfate (USP) <US>
         D01277  Droxidopa (JP18/USAN/INN) <JP/US>
         D08205  Methyldopa (INN)
         D00405  Methyldopa (USP) <JP/US>
         D00281  Clonidine (JAN/USP/INN) <US>
         D00604  Clonidine hydrochloride (JP18/USP) <JP/US>
         D05087  Moxonidine (USAN/INN)
         D08482  Rilmenidine (INN)
         D01603  Bethanidine sulfate (JAN/USAN)
         D08362  Phentolamine (INN)
         D00509  Phentolamine mesylate (USP) <JP/US>
         D08614  Tolazoline (INN)
         D00997  Tolazoline hydrochloride (JAN/USP)
         D02268  Ergoloid mesylates (USP)
         D07834  Dihydroergocristine (BAN)
         D07833  Dihydroergocristine mesilate (BAN)
         D08358  Phenoxybenzamine (INN)
         D00507  Phenoxybenzamine hydrochloride (USP) <US>
         D07540  Brimonidine (INN)
         D02076  Brimonidine tartrate (JAN/USAN) <JP/US>
         D08207  Methylergometrine (INN)
         D00680  Methylergonovine maleate (USP) <JP/US>
         D07905  Ergometrine (INN)
         D01163  Ergonovine maleate (USP)
         D08685  Yohimbine (DCF)
         D06671  Yohimbine hydrochloride (USP)
         D08611  Tizanidine (INN)
         D00776  Tizanidine hydrochloride (JP18/USP) <JP/US>
         D00270  Chlorpromazine (USP/INN)
         D00789  Chlorpromazine hydrochloride (JP18/USP) <JP/US>
         D03274  Chlorpromazine hibenzate (JAN)
         D04034  Chlorpromazine phenolphthalinate (JAN) <JP>
         D09819  Chlorpromazine tannate (JAN)
         D00283  Clozapine (JAN/USP/INN) <JP/US>
         D00514  Dexmedetomidine (USAN/INN)
         D01205  Dexmedetomidine hydrochloride (JAN/USP) <JP/US>
         D08216  Mianserin (INN)
         D01358  Mianserin hydrochloride (JAN/USAN) <JP>
         D00563  Mirtazapine (JAN/USP/INN) <JP/US>
         D11056  Mirtazapine hydrate (JAN)
         D08141  Lofexidine (INN)
         D04765  Lofexidine hydrochloride (USAN) <US>
         D08684  Xylometazoline (INN)
         D00757  Xylometazoline hydrochloride (USP)
         D08624  Tramazoline (INN)
         D01347  Tramazoline hydrochloride (JAN/USAN) <JP>
         D08368  Phenylpropanolamine (INN)
         D01224  Phenylpropanolamine hydrochloride (JAN/USP)
         D05466  Phenylpropanolamine polistirex (USAN)
         D08449  Pseudoephedrine (INN)
         D00485  Pseudoephedrine hydrochloride (USP)
         D05648  Pseudoephedrine polistirex (USAN)
         D05649  Pseudoephedrine sulfate (USP)
         D02349  Dipivefrin (USAN)
         D01017  Dipivefrin hydrochloride (USP)
         D07461  Apraclonidine (INN)
         D01008  Apraclonidine hydrochloride (JAN/USP) <JP/US>
         D00605  Guanabenz acetate (JP18/USP) <JP>
         D00607  Guanadrel sulfate (USAN)
         D01952  L-Methylephedrine hydrochloride (JAN)
         D02034  Setiptiline maleate (JAN) <JP>
         D02109  dl-Methylephedrine hydrochloride (JP18) <JP>
         D02388  Levonordefrin (USP)
         D02407  Lidamidine hydrochloride (USAN)
         D02569  Sunepitron hydrochloride (USAN)
         D02972  Aptazapine maleate (USAN)
         D03002  Atipamezole (USAN/INN)
         D03672  Delequamine hydrochloride (USAN)
         D03702  Detomidine hydrochloride (USAN)
         D03887  Domazoline fumarate (USAN)
         D04026  Epinephryl borate (USP)
         D04124  Fadolmidine hydrochloride (USAN)
         D04223  Fluparoxan hydrochloride (USAN)
         D04375  Guanabenz (USAN/INN)
         D04883  Medetomidine hydrochloride (USAN)
         D05119  Napamezole hydrochloride (USAN)
         D05228  Octodrine (USAN/INN)
         D05637  Propylhexedrine (USP/INN)
         D05688  Racepinephrine (USP/INN)
         D05689  Racepinephrine hydrochloride (USP)
         D06344  Xylazine hydrochloride (USP)
         D07795  Detomidine (INN)
         D08029  Guanadrel (INN)
         D08126  Lidamidine (INN)
         D08165  Medetomidine (INN)
         D08206  Methylephedrine (BAN)
         D08444  Propylhexedrine hydrochloride
         D08487  Romifidine (INN)
         D08511  Setiptiline (INN)
         D08683  Xylazine (USP/INN)
         D08982  Racephedrine hydrochloride (USAN)
         D09842  dl-Methylephedrine saccharinate (JAN)
         D11320  Vatinoxan (USAN)
         D11321  Vatinoxan hydrochloride (USAN)
       ADRA2A [HSA:150] [KO:K04138]
       ADRA2B [HSA:151] [KO:K04139]
       ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
       ADRB1 [HSA:153] [KO:K04141]
       ADRB2 [HSA:154] [KO:K04142]
       ADRB3 [HSA:155] [KO:K04143]
     Dopamine
       DRD [HSA:1812 1813 1814 1815 1816] [KO:K04144 K04145 K04146 K04147 K05840]
       DRD1 [HSA:1812] [KO:K04144]
       DRD2 [HSA:1813] [KO:K04145]
       DRD3 [HSA:1814] [KO:K04146]
       DRD4 [HSA:1815] [KO:K04147]
         D08132  Lisuride (INN)
         D01462  Lisuride maleate (JAN)
         D08489  Ropinirole (USAN/INN)
         D00784  Ropinirole hydrochloride (JAN/USP) <JP/US>
         D05575  Pramipexole (USAN/INN)
         D00559  Pramipexole dihydrochloride (USP) <JP/US>
         D00283  Clozapine (JAN/USP/INN) <JP/US>
         D00454  Olanzapine (JAN/USP/INN) <JP/US>
         D06623  Olanzapine pamoate (USAN) <US>
         D02656  Fananserin (USAN/INN)
         D05891  Sonepiprazole mesylate (USAN)
       DRD5 [HSA:1816] [KO:K05840]
     Histamine
     Serotonin
       HTR1 [HSA:3350 3351 3352 3354 3355] [KO:K04153]
       HTR1A [HSA:3350] [KO:K04153]
       HTR1B [HSA:3351] [KO:K04153]
       HTR1D [HSA:3352] [KO:K04153]
       HTR1F [HSA:3355] [KO:K04153]
       HTR2 [HSA:3356 3357 3358] [KO:K04157]
       HTR2A [HSA:3356] [KO:K04157]
         D00274  Cisapride (USP/INN)
         D02092  Cisapride (JAN)
         D07945  Fenfluramine (INN)
         D04148  Fenfluramine hydrochloride (JAN/USAN) <JP/US>
         D02363  Ketanserin (USAN/INN)
         D08099  Ketanserin tartrate
         D08244  Naftidrofuryl (INN)
         D05107  Nafronyl oxalate (USAN)
         D07307  Cyamemazine (INN)
         D07756  Cyamemazine tartrate
         D02671  Mesoridazine (USAN/INN)
         D00795  Mesoridazine besylate (USP)
         D08385  Pipotiazine (INN)
         D02680  Pipotiazine palmitate (USAN)
         D11169  Lumateperone (USAN/INN)
         D11170  Lumateperone tosylate (USAN) <US>
         D00561  Sertindole (USAN/INN)
         D08687  Ziprasidone (INN)
         D01939  Ziprasidone hydrochloride (USP) <US>
         D02100  Ziprasidone mesylate (USAN) <US>
         D04820  Lurasidone hydrochloride (JAN/USAN) <JP/US>
         D02340  Loxapine (USAN/INN) <US>
         D00794  Loxapine succinate (USP) <US>
         D08148  Loxapine hydrochloride
         D00283  Clozapine (JAN/USP/INN) <JP/US>
         D08456  Quetiapine (INN)
         D00458  Quetiapine fumarate (JP18/USP) <JP/US>
         D11769  Asenapine (INN) <US>
         D02995  Asenapine maleate (JAN/USAN) <JP/US>
         D00426  Risperidone (JP18/USP/INN) <JP/US>
         D08235  Mosapramine (INN)
         D01548  Mosapramine hydrochloride (JAN) <JP>
         D01164  Aripiprazole (JAN/USP/INN) <JP/US>
         D10355  Aripiprazole cavoxil (USAN)
         D10364  Aripiprazole lauroxil (USAN) <US>
         D10516  Aripiprazole hydrate (JAN) <JP/US>
         D05339  Paliperidone (JAN/USP/INN) <JP/US>
         D05340  Paliperidone palmitate (JAN/USAN) <JP/US>
         D09997  Cariprazine (USAN/INN)
         D09876  Cariprazine hydrochloride (JAN/USAN) <US>
         D10309  Brexpiprazole (JAN/USAN/INN) <JP/US>
         D08969  Pimavanserin tartrate (USAN) <US>
         D08216  Mianserin (INN)
         D01358  Mianserin hydrochloride (JAN/USAN) <JP>
         D08257  Nefazodone (INN)
         D00819  Nefazodone hydrochloride (USP) <US>
         D01176  Blonanserin (JAN/INN) <JP>
         D01624  Sarpogrelate hydrochloride (JP18) <JP>
         D02372  Perospirone hydrochloride hydrate (JAN) <JP>
         D02656  Fananserin (USAN/INN)
         D02836  Altanserin tartrate (USAN)
         D02893  Amesergide (USAN/INN)
         D03005  Atiprosin maleate (USAN)
         D04055  Esmirtazapine maleate (USAN)
         D04788  Lubazodone hydrochloride (USAN)
         D05738  Ritanserin (USAN/INN)
         D06632  Pruvanserin (USAN/INN)
         D06633  Pruvanserin hydrochloride (USAN)
         D08508  Sarpogrelate (INN)
         D09645  Nelotanserin (USAN/INN)
         D09976  Temanogrel (USAN/INN)
         D09977  Temanogrel hydrochloride (USAN)
         D10006  Eplivanserin (USAN/INN)
         D10329  Zicronapine (USAN/INN)
         D10495  Zicronapine succinate (USAN)
       HTR2C [HSA:3358] [KO:K04157]
         D07945  Fenfluramine (INN)
         D04148  Fenfluramine hydrochloride (JAN/USAN) <JP/US>
         D06613  Lorcaserin hydrochloride (USAN)
         D11566  Lorcaserin hydrochloride hemihydrate
         D07307  Cyamemazine (INN)
         D07756  Cyamemazine tartrate
         D00283  Clozapine (JAN/USP/INN) <JP/US>
         D02995  Asenapine maleate (JAN/USAN) <JP/US>
         D08969  Pimavanserin tartrate (USAN) <US>
         D07316  Captodiame (BAN)
         D08216  Mianserin (INN)
         D01358  Mianserin hydrochloride (JAN/USAN) <JP>
         D08257  Nefazodone (INN)
         D00819  Nefazodone hydrochloride (USP) <US>
         D02578  Agomelatine (INN)
         D02893  Amesergide (USAN/INN)
         D05738  Ritanserin (USAN/INN)
         D06660  Vabicaserin hydrochloride (USAN)
         D10170  Tedatioxetine (USAN)
         D10171  Tedatioxetine hydrobromide (USAN)
         D10710  Idalopirdine (USAN/INN)
       HTR4 [HSA:3360] [KO:K04160]
       HTR6 [HSA:3362] [KO:K04162]
       HTR7 [HSA:3363] [KO:K04163]
     Trace amine
     Angiotensin
     Bradykinin
     Cholecystokinin
     Endothelin
     Follicle stimulating hormone
     Ghrelin
     Gonadotropin-releasing hormone
     Lutropin-choriogonadotropic hormone
     Melanocortin
     Motilin
     Neuropeptide Y
     Opioid
     Orexin
     Oxytocin
     Relaxin
     Somatostatin
     Tachykinin
     Thrombin
     Thyrotropin-releasing hormone
     Vasopressin
     Purine / pyrimidine
     Adenosine
     Cysteinyl leukotriene
     Free fatty acid
     Leukotriene
     Lysophosphatidic acid
     Prostaglandin
     Prostacyclin
     Sphingolipid
     Thromboxane
     Cannabinoid
     Melatonin
     Platelet activating factor
     R-spondin
   Secretin receptor family
   Metabotropic glutamate receptor family
   Frizzled / Smoothened family
   Others
 
 Ion channels
   Ligand-gated ion channels
     Acetylcholine (nicotinic)
     Serotonin
       HTR3 [HSA:3359 9177 170572 200909 285242] [KO:K04819]
         D07129  Alosetron (INN)
         D02829  Alosetron hydrochloride (USAN) <US>
         D03495  Cilansetron (USAN/INN)
         D03496  Cilansetron hydrochloride (USAN)
         D00456  Ondansetron (JAN/USP/INN) <US>
         D00678  Ondansetron hydrochloride hydrate (JAN/USP) <JP/US>
         D02130  Tropisetron (INN)
         D02041  Tropisetron hydrochloride (JAN)
         D07867  Dolasetron (INN)
         D00725  Dolasetron mesylate (USP) <US>
         D07175  Palonosetron (INN)
         D05343  Palonosetron hydrochloride (JAN/USP) <JP/US>
         D00283  Clozapine (JAN/USP/INN) <JP/US>
         D08216  Mianserin (INN)
         D01358  Mianserin hydrochloride (JAN/USAN) <JP>
         D00563  Mirtazapine (JAN/USP/INN) <JP/US>
         D11056  Mirtazapine hydrate (JAN)
         D10184  Vortioxetine (USAN)
         D10185  Vortioxetine hydrobromide (JAN/USAN) <JP/US>
         D12544  Vortioxetine hemihydrobromide (USAN)
         D01613  Azasetron hydrochloride (JAN)
         D01838  Fabesetron hydrochloride (JAN)
         D02016  Ramosetron hydrochloride (JAN) <JP>
         D02632  Indisetron hydrochloride (JAN)
         D03060  Batanopride hydrochloride (USAN)
         D03073  Bemesetron (USAN/INN)
         D03662  Dazopride fumarate (USAN)
         D04294  Galdansetron hydrochloride (USAN)
         D04642  Itasetron (USAN/INN)
         D04821  Lurosetron mesylate (USAN)
         D05050  Mirisetron maleate (USAN)
         D05348  Pancopride (USAN/INN)
         D05685  Quipazine maleate (USAN)
         D06253  Tropanserin hydrochloride (USAN)
         D06353  Zacopride hydrochloride (USAN)
         D06358  Zatosetron maleate (USAN)
         D06396  Renzapride (INN)
         D07481  Azasetron (INN)
         D08466  Ramosetron (INN)
         D09749  Itasetron hydrochloride hydrate (JAN)
         D10170  Tedatioxetine (USAN)
         D10171  Tedatioxetine hydrobromide (USAN)
       HTR3A [HSA:3359] [KO:K04819]
       HTR3B [HSA:9177] [KO:K04819]
     GABA (ionotropic)
     Glycine
     Glutamate (ionotropic), non-NMDA
     Glutamate (ionotropic), NMDA
     Epithelial sodium channel (SCNN)
     ATP-gated cation channel (P2X)
   Voltage-gated ion channels
   Other ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: March 26, 2024

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