G Protein-coupled receptors
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Rhodopsin family
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Acetylcholine (muscarinic)
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Adrenaline
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ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
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ADRA1A [HSA:148] [KO:K04135]
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ADRA1D [HSA:146] [KO:K04137]
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ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
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D00095 Epinephrine (USP/INN) <JP/US>
D00996 Epinephrine hydrochloride (JAN)
D02149 Epinephrine bitartrate (JAN/USP)
D07931 Etilefrine (INN)
D01573 Etilefrine hydrochloride (JP18) <JP>
D00076 Noradrenaline (JP18) <JP>
D05206 Norepinephrine bitartrate (USP) <US>
D08284 Norepinephrine hydrochoride
D09794 Norepinephrine hydrochloride (JAN)
D08192 Metaraminol (INN)
D01019 Metaraminol bitartrate (JAN/USP)
D00124 Ephedrine (USP)
D01386 Ephedrine hydrochloride (JP18/USP) <JP/US>
D04018 Ephedrine sulfate (USP) <US>
D01277 Droxidopa (JP18/USAN/INN) <JP/US>
D08205 Methyldopa (INN)
D00405 Methyldopa (USP) <JP/US>
D00281 Clonidine (JAN/USP/INN) <US>
D00604 Clonidine hydrochloride (JP18/USP) <JP/US>
D05087 Moxonidine (USAN/INN)
D08482 Rilmenidine (INN)
D01603 Bethanidine sulfate (JAN/USAN)
D08362 Phentolamine (INN)
D00509 Phentolamine mesylate (USP) <JP/US>
D08614 Tolazoline (INN)
D00997 Tolazoline hydrochloride (JAN/USP)
D02268 Ergoloid mesylates (USP)
D07834 Dihydroergocristine (BAN)
D07833 Dihydroergocristine mesilate (BAN)
D08358 Phenoxybenzamine (INN)
D00507 Phenoxybenzamine hydrochloride (USP) <US>
D07540 Brimonidine (INN)
D02076 Brimonidine tartrate (JAN/USAN) <JP/US>
D08207 Methylergometrine (INN)
D00680 Methylergonovine maleate (USP) <JP/US>
D07905 Ergometrine (INN)
D01163 Ergonovine maleate (USP)
D08685 Yohimbine (DCF)
D06671 Yohimbine hydrochloride (USP)
D08611 Tizanidine (INN)
D00776 Tizanidine hydrochloride (JP18/USP) <JP/US>
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D00283 Clozapine (JAN/USP/INN) <JP/US>
D00514 Dexmedetomidine (USAN/INN)
D01205 Dexmedetomidine hydrochloride (JAN/USP) <JP/US>
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D00563 Mirtazapine (JAN/USP/INN) <JP/US>
D11056 Mirtazapine hydrate (JAN)
D08141 Lofexidine (INN)
D04765 Lofexidine hydrochloride (USAN) <US>
D08684 Xylometazoline (INN)
D00757 Xylometazoline hydrochloride (USP)
D08624 Tramazoline (INN)
D01347 Tramazoline hydrochloride (JAN/USAN) <JP>
D08368 Phenylpropanolamine (INN)
D01224 Phenylpropanolamine hydrochloride (JAN/USP)
D05466 Phenylpropanolamine polistirex (USAN)
D08449 Pseudoephedrine (INN)
D00485 Pseudoephedrine hydrochloride (USP)
D05648 Pseudoephedrine polistirex (USAN)
D05649 Pseudoephedrine sulfate (USP)
D02349 Dipivefrin (USAN)
D01017 Dipivefrin hydrochloride (USP)
D07461 Apraclonidine (INN)
D01008 Apraclonidine hydrochloride (JAN/USP) <JP/US>
D00605 Guanabenz acetate (JP18/USP) <JP>
D00607 Guanadrel sulfate (USAN)
D01952 L-Methylephedrine hydrochloride (JAN)
D02034 Setiptiline maleate (JAN) <JP>
D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
D02388 Levonordefrin (USP)
D02407 Lidamidine hydrochloride (USAN)
D02569 Sunepitron hydrochloride (USAN)
D02972 Aptazapine maleate (USAN)
D03002 Atipamezole (USAN/INN)
D03672 Delequamine hydrochloride (USAN)
D03702 Detomidine hydrochloride (USAN)
D03887 Domazoline fumarate (USAN)
D04026 Epinephryl borate (USP)
D04124 Fadolmidine hydrochloride (USAN)
D04223 Fluparoxan hydrochloride (USAN)
D04375 Guanabenz (USAN/INN)
D04883 Medetomidine hydrochloride (USAN)
D05119 Napamezole hydrochloride (USAN)
D05228 Octodrine (USAN/INN)
D05637 Propylhexedrine (USP/INN)
D05688 Racepinephrine (USP/INN)
D05689 Racepinephrine hydrochloride (USP)
D06344 Xylazine hydrochloride (USP)
D07795 Detomidine (INN)
D08029 Guanadrel (INN)
D08126 Lidamidine (INN)
D08165 Medetomidine (INN)
D08206 Methylephedrine (BAN)
D08444 Propylhexedrine hydrochloride
D08487 Romifidine (INN)
D08511 Setiptiline (INN)
D08683 Xylazine (USP/INN)
D08982 Racephedrine hydrochloride (USAN)
D09842 dl-Methylephedrine saccharinate (JAN)
D11320 Vatinoxan (USAN)
D11321 Vatinoxan hydrochloride (USAN)
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ADRA2A [HSA:150] [KO:K04138]
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ADRA2B [HSA:151] [KO:K04139]
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ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
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ADRB1 [HSA:153] [KO:K04141]
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ADRB2 [HSA:154] [KO:K04142]
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ADRB3 [HSA:155] [KO:K04143]
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Dopamine
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DRD [HSA:1812 1813 1814 1815 1816] [KO:K04144 K04145 K04146 K04147 K05840]
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DRD1 [HSA:1812] [KO:K04144]
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DRD2 [HSA:1813] [KO:K04145]
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DRD3 [HSA:1814] [KO:K04146]
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DRD4 [HSA:1815] [KO:K04147]
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D08132 Lisuride (INN)
D01462 Lisuride maleate (JAN)
D08489 Ropinirole (USAN/INN)
D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
D05575 Pramipexole (USAN/INN)
D00559 Pramipexole dihydrochloride (USP) <JP/US>
D00283 Clozapine (JAN/USP/INN) <JP/US>
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D02656 Fananserin (USAN/INN)
D05891 Sonepiprazole mesylate (USAN)
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DRD5 [HSA:1816] [KO:K05840]
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Histamine
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Serotonin
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HTR1 [HSA:3350 3351 3352 3354 3355] [KO:K04153]
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HTR1A [HSA:3350] [KO:K04153]
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HTR1B [HSA:3351] [KO:K04153]
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HTR1D [HSA:3352] [KO:K04153]
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HTR1F [HSA:3355] [KO:K04153]
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HTR2 [HSA:3356 3357 3358] [KO:K04157]
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HTR2A [HSA:3356] [KO:K04157]
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D00274 Cisapride (USP/INN)
D02092 Cisapride (JAN)
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D02363 Ketanserin (USAN/INN)
D08099 Ketanserin tartrate
D08244 Naftidrofuryl (INN)
D05107 Nafronyl oxalate (USAN)
D07307 Cyamemazine (INN)
D07756 Cyamemazine tartrate
D02671 Mesoridazine (USAN/INN)
D00795 Mesoridazine besylate (USP)
D08385 Pipotiazine (INN)
D02680 Pipotiazine palmitate (USAN)
D11169 Lumateperone (USAN/INN)
D11170 Lumateperone tosylate (USAN) <US>
D00561 Sertindole (USAN/INN)
D08687 Ziprasidone (INN)
D01939 Ziprasidone hydrochloride (USP) <US>
D02100 Ziprasidone mesylate (USAN) <US>
D04820 Lurasidone hydrochloride (JAN/USAN) <JP/US>
D02340 Loxapine (USAN/INN) <US>
D00794 Loxapine succinate (USP) <US>
D08148 Loxapine hydrochloride
D00283 Clozapine (JAN/USP/INN) <JP/US>
D08456 Quetiapine (INN)
D00458 Quetiapine fumarate (JP18/USP) <JP/US>
D11769 Asenapine (INN) <US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D00426 Risperidone (JP18/USP/INN) <JP/US>
D08235 Mosapramine (INN)
D01548 Mosapramine hydrochloride (JAN) <JP>
D01164 Aripiprazole (JAN/USP/INN) <JP/US>
D10355 Aripiprazole cavoxil (USAN)
D10364 Aripiprazole lauroxil (USAN) <US>
D10516 Aripiprazole hydrate (JAN) <JP/US>
D05339 Paliperidone (JAN/USP/INN) <JP/US>
D05340 Paliperidone palmitate (JAN/USAN) <JP/US>
D09997 Cariprazine (USAN/INN)
D09876 Cariprazine hydrochloride (JAN/USAN) <US>
D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
D08969 Pimavanserin tartrate (USAN) <US>
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D08257 Nefazodone (INN)
D00819 Nefazodone hydrochloride (USP) <US>
D01176 Blonanserin (JAN/INN) <JP>
D01624 Sarpogrelate hydrochloride (JP18) <JP>
D02372 Perospirone hydrochloride hydrate (JAN) <JP>
D02656 Fananserin (USAN/INN)
D02836 Altanserin tartrate (USAN)
D02893 Amesergide (USAN/INN)
D03005 Atiprosin maleate (USAN)
D04055 Esmirtazapine maleate (USAN)
D04788 Lubazodone hydrochloride (USAN)
D05738 Ritanserin (USAN/INN)
D06632 Pruvanserin (USAN/INN)
D06633 Pruvanserin hydrochloride (USAN)
D08508 Sarpogrelate (INN)
D09645 Nelotanserin (USAN/INN)
D09976 Temanogrel (USAN/INN)
D09977 Temanogrel hydrochloride (USAN)
D10006 Eplivanserin (USAN/INN)
D10329 Zicronapine (USAN/INN)
D10495 Zicronapine succinate (USAN)
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HTR2C [HSA:3358] [KO:K04157]
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D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D06613 Lorcaserin hydrochloride (USAN)
D11566 Lorcaserin hydrochloride hemihydrate
D07307 Cyamemazine (INN)
D07756 Cyamemazine tartrate
D00283 Clozapine (JAN/USP/INN) <JP/US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D08969 Pimavanserin tartrate (USAN) <US>
D07316 Captodiame (BAN)
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D08257 Nefazodone (INN)
D00819 Nefazodone hydrochloride (USP) <US>
D02578 Agomelatine (INN)
D02893 Amesergide (USAN/INN)
D05738 Ritanserin (USAN/INN)
D06660 Vabicaserin hydrochloride (USAN)
D10170 Tedatioxetine (USAN)
D10171 Tedatioxetine hydrobromide (USAN)
D10710 Idalopirdine (USAN/INN)
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HTR4 [HSA:3360] [KO:K04160]
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HTR6 [HSA:3362] [KO:K04162]
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HTR7 [HSA:3363] [KO:K04163]
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Trace amine
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Angiotensin
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Bradykinin
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Cholecystokinin
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Endothelin
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Follicle stimulating hormone
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Ghrelin
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Gonadotropin-releasing hormone
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Lutropin-choriogonadotropic hormone
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Melanocortin
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Motilin
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Neuropeptide Y
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Opioid
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Orexin
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Oxytocin
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Relaxin
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Somatostatin
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Tachykinin
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Thrombin
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Thyrotropin-releasing hormone
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Vasopressin
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Purine / pyrimidine
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Adenosine
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Cysteinyl leukotriene
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Free fatty acid
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Leukotriene
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Lysophosphatidic acid
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Prostaglandin
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Prostacyclin
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Sphingolipid
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Thromboxane
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Cannabinoid
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Melatonin
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Platelet activating factor
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R-spondin
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Secretin receptor family
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Metabotropic glutamate receptor family
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Frizzled / Smoothened family
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Others
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Ion channels
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Ligand-gated ion channels
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Acetylcholine (nicotinic)
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Serotonin
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HTR3 [HSA:3359 9177 170572 200909 285242] [KO:K04819]
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D07129 Alosetron (INN)
D02829 Alosetron hydrochloride (USAN) <US>
D03495 Cilansetron (USAN/INN)
D03496 Cilansetron hydrochloride (USAN)
D00456 Ondansetron (JAN/USP/INN) <US>
D00678 Ondansetron hydrochloride hydrate (JAN/USP) <JP/US>
D02130 Tropisetron (INN)
D02041 Tropisetron hydrochloride (JAN)
D07867 Dolasetron (INN)
D00725 Dolasetron mesylate (USP) <US>
D07175 Palonosetron (INN)
D05343 Palonosetron hydrochloride (JAN/USP) <JP/US>
D00283 Clozapine (JAN/USP/INN) <JP/US>
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D00563 Mirtazapine (JAN/USP/INN) <JP/US>
D11056 Mirtazapine hydrate (JAN)
D10184 Vortioxetine (USAN)
D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
D12544 Vortioxetine hemihydrobromide (USAN)
D01613 Azasetron hydrochloride (JAN)
D01838 Fabesetron hydrochloride (JAN)
D02016 Ramosetron hydrochloride (JAN) <JP>
D02632 Indisetron hydrochloride (JAN)
D03060 Batanopride hydrochloride (USAN)
D03073 Bemesetron (USAN/INN)
D03662 Dazopride fumarate (USAN)
D04294 Galdansetron hydrochloride (USAN)
D04642 Itasetron (USAN/INN)
D04821 Lurosetron mesylate (USAN)
D05050 Mirisetron maleate (USAN)
D05348 Pancopride (USAN/INN)
D05685 Quipazine maleate (USAN)
D06253 Tropanserin hydrochloride (USAN)
D06353 Zacopride hydrochloride (USAN)
D06358 Zatosetron maleate (USAN)
D06396 Renzapride (INN)
D07481 Azasetron (INN)
D08466 Ramosetron (INN)
D09749 Itasetron hydrochloride hydrate (JAN)
D10170 Tedatioxetine (USAN)
D10171 Tedatioxetine hydrobromide (USAN)
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HTR3A [HSA:3359] [KO:K04819]
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HTR3B [HSA:9177] [KO:K04819]
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GABA (ionotropic)
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Glycine
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Glutamate (ionotropic), non-NMDA
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Glutamate (ionotropic), NMDA
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Epithelial sodium channel (SCNN)
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ATP-gated cation channel (P2X)
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Voltage-gated ion channels
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Other ion channels
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Nuclear receptors
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Protein kinases
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Cytokines and receptors
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Cell surface molecules and ligands
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Transporters
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Enzymes
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Nucleic acids
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Not elsewhere classified
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