Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
   Ligand-gated ion channels
     Acetylcholine (nicotinic)
     Serotonin
     GABA (ionotropic)
       GABR [HSA:2554 2555 2556 2557 2558 2559 2560 2561 2562 2563 2564 2565 2566 2567 2568 55879] [KO:K05175 K05181 K05184 K05185 K05186 K05189 K05192]
         D01071  Hexobarbital (JAN/INN)
         D00714  Thiopental sodium (JP18/USP/INN) <JP>
         D00549  Propofol (JAN/USP/INN) <JP/US>
         D04257  Fospropofol disodium (USAN)
         D00700  Mephobarbital (JAN/USP)
         D00506  Phenobarbital (JP18/USP/INN) <JP>
         D00701  Phenobarbital sodium (JAN/USP/INN) <JP/US>
         D08356  Phenobarbital diethylamine
         D07298  Barbexaclone (INN)
         D01382  Metharbital (JAN/INN)
         D00280  Clonazepam (JP18/USP/INN) <JP/US>
         D00058  gamma-Aminobutyric acid (JAN) <JP>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D04300  Ganaxolone (USAN/INN) <US>
         D00293  Diazepam (JP18/USP/INN) <JP/US>
         D00267  Chlordiazepoxide (JP18/USP/INN) <JP>
         D00693  Chlordiazepoxide hydrochloride (JAN/USP) <US>
         D01292  Medazepam (JP18/INN) <JP>
         D04882  Medazepam hydrochloride (USAN)
         D00464  Oxazepam (JAN/USP/INN) <US>
         D00694  Clorazepate dipotassium (JP18/USP) <JP/US>
         D03562  Clorazepate monopotassium (USAN)
         D00365  Lorazepam (JP18/USP/INN) <JP/US>
         D02770  Adinazolam (USAN/INN)
         D02771  Adinazolam mesylate (USAN)
         D01245  Bromazepam (JP18/USAN/INN) <JP>
         D01253  Clobazam (JAN/USAN/INN) <JP/US>
         D04650  Ketazolam (USAN/INN)
         D00470  Prazepam (JP18/USAN/INN)
         D00225  Alprazolam (JP18/USP/INN) <JP/US>
         D00338  Halazepam (USAN/INN)
         D08283  Nordazepam (INN)
         D01354  Fludiazepam (JP18/INN) <JP>
         D01293  Ethyl loflazepate (JP18/INN) <JP>
         D01514  Etizolam (JP18/INN) <JP>
         D01328  Clotiazepam (JP18/INN) <JP>
         D01268  Cloxazolam (JP18/INN) <JP>
         D01254  Tofisopam (JP18/INN) <JP>
         D01316  Mexazolam (JAN/INN) <JP>
         D00376  Meprobamate (JAN/USP/INN) <US>
         D00499  Pentobarbital (USP/INN)
         D00500  Pentobarbital sodium (JAN/USP) <US>
         D02253  Pentobarbital calcium (JP18) <JP>
         D00555  Amobarbital (JP18/INN) <JP>
         D02252  Amobarbital sodium (JAN/USP)
         D02618  Butobarbital (BAN)
         D01740  Barbital (JP18/INN)
         D00698  Aprobarbital (INN)
         D00430  Secobarbital (USP/INN)
         D01310  Secobarbital sodium (JAN/USP) <JP>
         D06887  Talbutal (INN)
         D00329  Flurazepam (JAN/INN)
         D00695  Flurazepam hydrochloride (USP) <US>
         D01408  Flurazepam hydrochloride (JP18) <JP>
         D00531  Nitrazepam (JP18/USAN/INN) <JP>
         D01230  Flunitrazepam (JP18/USAN/INN) <JP>
         D00311  Estazolam (JP18/USP/INN) <JP/US>
         D00387  Triazolam (JP18/USP/INN) <JP/US>
         D01657  Lormetazepam (JAN/USAN/INN) <JP>
         D00370  Temazepam (USP/INN) <US>
         D00550  Midazolam (JAN/USP/INN) <JP/US>
         D00696  Midazolam hydrochloride (USAN) <US>
         D05028  Midazolam maleate (USAN)
         D01744  Brotizolam (JP18/USAN/INN) <JP>
         D00457  Quazepam (JAN/USP/INN) <JP/US>
         D07326  Loprazolam (INN)
         D08145  Loprazolam mesilate
         D07328  Cinolazepam (INN)
         D11788  Remimazolam (USAN/INN)
         D10194  Remimazolam besylate (USAN) <JP/US>
         D01593  Nimetazepam (JAN/INN)
         D00532  Glutethimide (JAN/INN)
         D01372  Zopiclone (JP18/INN) <JP>
         D08690  Zolpidem (INN)
         D00706  Zolpidem tartrate (JP18/USP) <JP/US>
         D02624  Eszopiclone (JAN/USP/INN) <JP/US>
         D11149  Brexanolone (USAN/INN) <US>
         D00697  Flumazenil (JAN/USP/INN) <JP/US>
         D00699  Butabarbital sodium (USP)
         D00713  Thiamylal sodium (JP18) <JP>
         D01278  Oxazolam (JP18/INN) <JP>
         D01279  Flutoprazepam (JP18/INN)
         D01286  Flutazolam (JAN/INN) <JP>
         D01564  Rilmazafone hydrochloride hydrate (JP18) <JP>
         D01758  Haloxazolam (JP18/INN) <JP>
         D02283  Iomazenil (123I) (JAN/INN) <JP>
         D02594  Abecarnil (INN)
         D02616  Pagoclone (USAN/INN)
         D02617  Ocinaplon (USAN/INN)
         D02640  Indiplon (USAN/INN)
         D02833  Alpidem (USAN/INN)
         D03155  Bretazenil (USAN/INN)
         D03180  Butabarbital (USP)
         D03737  Dextofisopam (USAN/INN)
         D04282  Gaboxadol (USAN/INN)
         D04721  Levotofisopam (USAN/INN)
         D05346  Panadiplon (USAN/INN)
         D05378  Pazinaclone (USAN/INN)
         D05980  Suritozole (USAN/INN)
         D06106  Thiamylal
         D07784  Delorazepam (INN)
         D08481  Rilmazafone (INN)
         D08507  Sarmazenil (INN)
         D08840  Adipiplon (USAN)
         D12146  Darigabat (USAN)
         D12449  Cipepofol (USAN/INN)
       GABRA1 [HSA:2554] [KO:K05175]
       GABRA5 [HSA:2558] [KO:K05175]
     Glycine
     Glutamate (ionotropic), non-NMDA
     Glutamate (ionotropic), NMDA
     Epithelial sodium channel (SCNN)
     ATP-gated cation channel (P2X)
   Voltage-gated ion channels
   Other ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 17, 2024

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