G Protein-coupled receptors
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Rhodopsin family
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Acetylcholine (muscarinic)
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Adrenaline
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ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
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D00095 Epinephrine (USP/INN) <JP/US>
D00996 Epinephrine hydrochloride (JAN)
D02149 Epinephrine bitartrate (JAN/USP)
D02774 Adrenalone (USAN/INN)
D07560 Adrenalone hydrochloride
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D07931 Etilefrine (INN)
D01573 Etilefrine hydrochloride (JP18) <JP>
D00076 Noradrenaline (JP18) <JP>
D05206 Norepinephrine bitartrate (USP) <US>
D08284 Norepinephrine hydrochoride
D09794 Norepinephrine hydrochloride (JAN)
D08286 Norfenefrine (INN)
D01405 Norfenefrine hydrochloride (JAN)
D08365 Phenylephrine (INN)
D00511 Phenylephrine hydrochloride (JP18/USP) <JP/US>
D08366 Phenylephrine tartrate
D08966 Phenylephrine bitartrate (USP)
D08192 Metaraminol (INN)
D01019 Metaraminol bitartrate (JAN/USP)
D08201 Methoxamine (BAN)
D01020 Methoxamine hydrochloride (JAN)
D08220 Midodrine (INN)
D01307 Midodrine hydrochloride (JAN/USP) <JP/US>
D00124 Ephedrine (USP)
D01386 Ephedrine hydrochloride (JP18/USP) <JP/US>
D04018 Ephedrine sulfate (USP) <US>
D01277 Droxidopa (JP18/USAN/INN) <JP/US>
D08411 Prazosin (INN)
D00609 Prazosin hydrochloride (JP18/USP) <JP/US>
D04531 Indoramin (USAN/INN)
D04532 Indoramin hydrochloride (USAN)
D08212 Trimazosin (INN)
D06234 Trimazosin hydrochloride (USAN)
D07874 Doxazosin (INN)
D00608 Doxazosin mesylate (USP) <JP/US>
D01333 Urapidil (JP18/INN) <JP>
D08662 Urapidil hydrochloride
D08362 Phentolamine (INN)
D00509 Phentolamine mesylate (USP) <JP/US>
D08614 Tolazoline (INN)
D00997 Tolazoline hydrochloride (JAN/USP)
D02268 Ergoloid mesylates (USP)
D01290 Nicergoline (JP18/USAN/INN) <JP>
D08271 Nicergoline tartrate
D07834 Dihydroergocristine (BAN)
D07833 Dihydroergocristine mesilate (BAN)
D08358 Phenoxybenzamine (INN)
D00507 Phenoxybenzamine hydrochloride (USP) <US>
D08239 Moxisylyte (INN)
D01571 Moxisylyte hydrochloride (JAN)
D08064 Ifenprodil (INN)
D01445 Ifenprodil tartrate (JP18) <JP>
D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
D08106 Labetalol (INN)
D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
D00255 Carvedilol (JP18/USP/INN) <JP/US>
D03415 Carvedilol phosphate (USAN) <US>
D08207 Methylergometrine (INN)
D00680 Methylergonovine maleate (USP) <JP/US>
D07906 Ergotamine (INN)
D07905 Ergometrine (INN)
D01163 Ergonovine maleate (USP)
D08560 Tamsulosin (INN)
D01024 Tamsulosin hydrochloride (JP18/USP) <JP/US>
D08569 Terazosin (INN)
D00610 Terazosin hydrochloride (USP) <JP/US>
D11585 Terazosin hydrochloride anhydrous <US>
D00679 Ergotamine tartrate (JP18/USP) <US>
D01485 Propericiazine (JAN) <JP>
D00308 Droperidol (JP18/USP/INN) <JP/US>
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D08257 Nefazodone (INN)
D00819 Nefazodone hydrochloride (USP) <US>
D08578 Tetryzoline (INN)
D00756 Tetrahydrozoline nitrate (JAN)
D01023 Tetrahydrozoline hydrochloride (JAN/USP)
D08684 Xylometazoline (INN)
D00757 Xylometazoline hydrochloride (USP)
D08253 Naphazoline (INN)
D00743 Naphazoline hydrochloride (JP18/USP)
D01021 Naphazoline nitrate (JP18) <JP>
D08624 Tramazoline (INN)
D01347 Tramazoline hydrochloride (JAN/USAN) <JP>
D08368 Phenylpropanolamine (INN)
D01224 Phenylpropanolamine hydrochloride (JAN/USP)
D05466 Phenylpropanolamine polistirex (USAN)
D08449 Pseudoephedrine (INN)
D00485 Pseudoephedrine hydrochloride (USP)
D05648 Pseudoephedrine polistirex (USAN)
D05649 Pseudoephedrine sulfate (USP)
D02349 Dipivefrin (USAN)
D01017 Dipivefrin hydrochloride (USP)
D08115 Levobunolol (INN)
D01025 Levobunolol hydrochloride (JAN/USP) <JP/US>
D07775 Dapiprazole (INN)
D03648 Dapiprazole hydrochloride (USAN) <US>
D00607 Guanadrel sulfate (USAN)
D01171 Monatepil maleate (JAN/USAN)
D01444 Bunitrolol hydrochloride (JAN)
D01469 Amosulalol hydrochloride (JP18) <JP>
D01674 Naftopidil (JP18/INN) <JP>
D01691 Nipradilol (JAN/INN) <JP>
D01830 Arotinolol hydrochloride (JP18) <JP>
D01887 Bunazosin hydrochloride (JP18) <JP>
D01952 L-Methylephedrine hydrochloride (JAN)
D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
D02568 Flesinoxan (INN)
D02901 Amidephrine mesylate (USAN)
D03887 Domazoline fumarate (USAN)
D04026 Epinephryl borate (USP)
D05228 Octodrine (USAN/INN)
D05395 Pelanserin hydrochloride (USAN)
D05637 Propylhexedrine (USP/INN)
D05688 Racepinephrine (USP/INN)
D05689 Racepinephrine hydrochloride (USP)
D07451 Amosulalol (INN)
D07465 Arotinolol (INN)
D07550 Bunazosin (INN)
D08029 Guanadrel (INN)
D08206 Methylephedrine (BAN)
D08444 Propylhexedrine hydrochloride
D08982 Racephedrine hydrochloride (USAN)
D09842 dl-Methylephedrine saccharinate (JAN)
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ADRA1A [HSA:148] [KO:K04135]
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ADRA1D [HSA:146] [KO:K04137]
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ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
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ADRA2A [HSA:150] [KO:K04138]
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ADRA2B [HSA:151] [KO:K04139]
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ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
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ADRB1 [HSA:153] [KO:K04141]
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D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D03879 Dobutamine (USAN/INN)
D00632 Dobutamine hydrochloride (JP18/USP) <JP/US>
D03880 Dobutamine lactobionate (USAN)
D03881 Dobutamine tartrate (USAN)
D06328 Xamoterol (USAN)
D06329 Xamoterol fumarate (USAN)
D08600 Timolol (INN)
D00378 Timolol (USAN) <US>
D00603 Timolol maleate (JP18/USP) <JP/US>
D08525 Sotalol (INN)
D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
D00432 Nadolol (JP18/USP/INN) <JP/US>
D05587 Practolol (USAN)
D02358 Metoprolol (USAN/INN)
D00601 Metoprolol tartrate (JP18/USP) <JP/US>
D00635 Metoprolol succinate (USP) <US>
D05011 Metoprolol fumarate (USP)
D00235 Atenolol (JP18/USP/INN) <JP/US>
D02338 Acebutolol (USAN/INN)
D00597 Acebutolol hydrochloride (JP18/USP) <US>
D07526 Betaxolol (INN)
D00598 Betaxolol hydrochloride (JP18/USP) <JP/US>
D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
D02342 Bisoprolol (JAN/USAN/INN) <JP>
D00634 Bisoprolol fumarate (JP18/USP) <JP/US>
D07660 Celiprolol (INN)
D01741 Celiprolol hydrochloride (JAN/USAN) <JP>
D07916 Esmolol (INN)
D00644 Esmolol hydrochloride (JAN/USP) <JP/US>
D06646 Epanolol (USAN/INN)
D01471 Esatenolol (JAN/INN)
D05127 Nebivolol (USAN/INN)
D06622 Nebivolol hydrochloride (USAN) <US>
D01847 Landiolol hydrochloride (JAN/USAN) <JP>
D12410 Landiolol (USAN/INN)
D08106 Labetalol (INN)
D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
D00255 Carvedilol (JP18/USP/INN) <JP/US>
D03415 Carvedilol phosphate (USAN) <US>
D01469 Amosulalol hydrochloride (JP18) <JP>
D01492 Bucumolol hydrochloride (JP18)
D01830 Arotinolol hydrochloride (JP18) <JP>
D01903 Docarpamine (JAN/INN) <JP>
D01958 Indenolol hydrochloride (JP18)
D02389 Primidolol (USAN/INN)
D02614 Denopamine (JAN/INN) <JP>
D03177 Bunolol hydrochloride (USAN)
D03195 Butopamine (USAN/INN)
D03449 Cetamolol hydrochloride (USAN)
D03490 Cicloprolol hydrochloride (USAN)
D04708 Levdobutamine lactobionate (USAN)
D04710 Levobetaxolol hydrochloride (USAN)
D07451 Amosulalol (INN)
D07465 Arotinolol (INN)
D08078 Indenolol (INN)
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ADRB2 [HSA:154] [KO:K04142]
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D03891 Dopexamine (USAN/INN)
D03892 Dopexamine hydrochloride (USAN)
D08092 Isoxsuprine (INN)
D01748 Isoxsuprine hydrochloride (JP18/USP) <JP>
D08093 Isoxsuprine lactate
D08600 Timolol (INN)
D00378 Timolol (USAN) <US>
D00603 Timolol maleate (JP18/USP) <JP/US>
D08525 Sotalol (INN)
D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
D00432 Nadolol (JP18/USP/INN) <JP/US>
D08106 Labetalol (INN)
D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
D00255 Carvedilol (JP18/USP/INN) <JP/US>
D03415 Carvedilol phosphate (USAN) <US>
D02359 Ritodrine (USAN/INN)
D01263 Ritodrine hydrochloride (JP18/USP) <JP>
D04157 Fenoterol (USAN/INN)
D01428 Fenoterol hydrobromide (JAN) <JP>
D08300 Orciprenaline (INN)
D00685 Metaproterenol sulfate (USP)
D04954 Metaproterenol polistirex (USAN)
D02147 Albuterol (USP)
D00683 Albuterol sulfate (USP) <JP/US>
D08570 Terbutaline (INN)
D00688 Terbutaline sulfate (JP18/USP) <JP/US>
D05730 Rimiterol hydrobromide (USAN)
D08039 Hexoprenaline (INN)
D02396 Hexoprenaline sulfate (USAN)
D04625 Isoetharine (USP)
D02093 Isoetharine hydrochloride (USP)
D04626 Isoetharine mesylate (USP)
D08387 Pirbuterol (INN)
D00686 Pirbuterol acetate (USAN)
D01349 Pirbuterol hydrochloride (JAN/USAN)
D08629 Tretoquinol (INN)
D01978 Trimetoquinol hydrochloride
D05037 Trimetoquinol hydrochloride hydrate (JP18) <JP>
D03402 Carbuterol hydrochloride (USAN)
D02151 Tulobuterol (JP18/INN) <JP>
D01362 Tulobuterol hydrochloride (JP18) <JP>
D05792 Salmeterol (USAN/INN)
D00687 Salmeterol xinafoate (JAN/USP) <JP/US>
D07990 Formoterol (INN)
D01373 Formoterol fumarate (USP) <US>
D05277 Formoterol fumarate hydrate (JP18) <JP/US>
D07713 Clenbuterol (INN)
D01360 Clenbuterol hydrochloride (JAN/USP) <JP>
D08474 Reproterol (INN)
D05718 Reproterol hydrochloride (USAN)
D08424 Procaterol (INN)
D02404 Procaterol hydrochloride (USAN)
D05366 Procaterol hydrochloride hydrate (JP18) <JP>
D07534 Bitolterol (INN)
D00684 Bitolterol mesylate (USAN)
D09318 Indacaterol (USAN/INN)
D09319 Indacaterol maleate (JAN/USAN) <JP>
D11009 Indacaterol acetate (JAN)
D10145 Olodaterol (USAN/INN)
D10020 Olodaterol hydrochloride (JAN/USAN) <US>
D01635 Methoxyphenamine hydrochloride (JAN)
D07377 Bambuterol (INN)
D07489 Bambuterol hydrochloride
D01469 Amosulalol hydrochloride (JP18) <JP>
D01492 Bucumolol hydrochloride (JP18)
D01589 Mabuterol hydrochloride (JAN)
D01830 Arotinolol hydrochloride (JP18) <JP>
D01835 Clorprenaline hydrochloride (JAN/USAN)
D01958 Indenolol hydrochloride (JP18)
D02281 Levalbuterol hydrochloride (USP) <US>
D02981 Arformoterol tartrate (USAN) <US>
D03170 Bucindolol hydrochloride (USAN)
D03177 Bunolol hydrochloride (USAN)
D03198 Butoxamine hydrochloride (USAN)
D03587 Colterol mesylate (USAN)
D04072 Etafedrine hydrochloride (USAN)
D04701 Levalbuterol sulfate (USAN)
D04703 Levalbuterol tartrate (USAN) <US>
D04953 Metalol hydrochloride (USAN)
D05476 Picumeterol fumarate (USAN)
D05691 Ractopamine hydrochloride (USP)
D05832 Sibenadet hydrochloride (USAN)
D05902 Soterenol hydrochloride (USAN)
D06374 Zinterol hydrochloride (USAN)
D06562 Bedoradrine sulfate (USAN)
D07451 Amosulalol (INN)
D07463 Arformoterol (INN)
D07465 Arotinolol (INN)
D07608 Carazolol (INN)
D08078 Indenolol (INN)
D08124 Levosalbutamol (INN)
D08945 Milveterol hydrochloride (USAN)
D09696 Vilanterol (USAN/INN)
D09697 Vilanterol trifenatate (JAN/USAN)
D10219 Abediterol (USAN/INN)
D10220 Abediterol napadisylate (USAN)
D10545 Batefenterol (USAN)
D10546 Batefenterol succinate (USAN)
D11900 Navafenterol (USAN)
D11901 Navafenterol saccharinate (USAN)
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ADRB3 [HSA:155] [KO:K04143]
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Dopamine
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Histamine
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Serotonin
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Trace amine
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Angiotensin
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Bradykinin
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Cholecystokinin
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Endothelin
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Follicle stimulating hormone
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Ghrelin
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Gonadotropin-releasing hormone
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Lutropin-choriogonadotropic hormone
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Melanocortin
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Motilin
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Neuropeptide Y
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Opioid
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Orexin
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Oxytocin
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Relaxin
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Somatostatin
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Tachykinin
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Thrombin
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Thyrotropin-releasing hormone
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Vasopressin
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Purine / pyrimidine
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Adenosine
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Cysteinyl leukotriene
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Free fatty acid
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Leukotriene
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Lysophosphatidic acid
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Prostaglandin
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Prostacyclin
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Sphingolipid
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Thromboxane
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Cannabinoid
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Melatonin
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Platelet activating factor
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R-spondin
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Secretin receptor family
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Metabotropic glutamate receptor family
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Frizzled / Smoothened family
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Others
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Ion channels
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Nuclear receptors
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Protein kinases
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Cytokines and receptors
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Cell surface molecules and ligands
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Transporters
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Enzymes
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Nucleic acids
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Not elsewhere classified
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