Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
   Ligand-gated ion channels
   Voltage-gated ion channels
     Sodium channels
       SCN1A [HSA:6323] [KO:K04833]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN2A [HSA:6326] [KO:K04834]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN3A [HSA:6328] [KO:K04836]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D07299  Lacosamide (JAN/USAN/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN4A [HSA:6329] [KO:K04837]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN5A [HSA:6331] [KO:K04838]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D05077  Moricizine (USAN)
         D02087  Moricizine hydrochloride (USP)
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D06665  Vernakalant hydrochloride (USAN)
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN8A [HSA:6334] [KO:K04840]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN9A [HSA:6335] [KO:K04841]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D07299  Lacosamide (JAN/USAN/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D11156  Funapide (USAN/INN)
         D11179  Vixotrigine (USAN/INN)
         D11180  Vixotrigine hydrochloride (USAN)
         D12616  Bliretrigine (JAN/INN)
       SCN10A [HSA:6336] [KO:K04842]
         D08458  Quinidine (BAN)
         D00642  Quinidine gluconate (USP) <US>
         D00643  Quinidine polygalacturonate
         D02272  Quinidine sulfate (USP) <JP/US>
         D08459  Quinidine phenylethylbarbiturate
         D08421  Procainamide (INN)
         D00477  Procainamide hydrochloride (JP18/USP) <JP/US>
         D00303  Disopyramide (JP18/USAN/INN) <JP>
         D00637  Disopyramide phosphate (JAN/USP) <JP/US>
         D01041  Sparteine (INN)
         D02239  Sparteine sulfate (JAN/USAN)
         D00199  Ajmaline (JP18)
         D04774  Lorajmine hydrochloride (USAN)
         D00358  Lidocaine (JP18/USP/INN) <JP/US>
         D02086  Lidocaine hydrochloride (JAN/USP) <JP/US>
         D08127  Lidocaine hydrochloride monohydrate <JP/US>
         D08215  Mexiletine (INN)
         D00639  Mexiletine hydrochloride (JP18/USP) <JP/US>
         D06172  Tocainide (USAN/INN)
         D02088  Tocainide hydrochloride (USP)
         D02969  Aprindine (USAN/INN)
         D01326  Aprindine hydrochloride (JP18/USAN) <JP>
         D08435  Propafenone (INN)
         D00640  Propafenone hydrochloride (JP18/USP) <JP/US>
         D07962  Flecainide (INN)
         D00638  Flecainide acetate (JP18/USP) <JP/US>
         D07894  Encainide (INN)
         D03991  Encainide hydrochloride (USAN)
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D03492  Cifenline (USAN)
         D01455  Cifenline succinate (USAN) <JP>
         D00551  Tetracaine (USP/INN)
         D00741  Tetracaine hydrochloride (JP18/USP) <JP/US>
         D00552  Benzocaine (USP/INN) <JP>
         D00733  Dibucaine (USP)
         D02220  Dibucaine hydrochloride (JP18/USP)
         D08422  Procaine (INN)
         D00740  Procaine hydrochloride (JP18/USP) <JP>
         D01152  Oxethazaine (JP18/USAN) <JP>
         D08311  Oxetacaine hydrochloride
         D08407  Pramocaine (INN)
         D00739  Pramoxine hydrochloride (USP)
         D02456  Aminobenzoic acid (USP)
         D02906  Aminobenzoate potassium (USP)
         D02907  Aminobenzoate sodium (USP)
         D08319  Oxybuprocaine (INN)
         D01768  Benoxinate hydrochloride (USP) <JP>
         D07678  Chloroprocaine (INN)
         D00732  Chloroprocaine hydrochloride (USP) <US>
         D07552  Bupivacaine (USAN/INN) <US>
         D01450  Bupivacaine hydrochloride (USP) <JP/US>
         D08181  Mepivacaine (INN)
         D00738  Mepivacaine hydrochloride (JP18/USP) <JP/US>
         D00553  Prilocaine (USP/INN)
         D01243  Prilocaine hydrochloride (USP) <US>
         D04095  Etidocaine (USAN/INN)
         D00737  Etidocaine hydrochloride
         D07468  Articaine (INN)
         D02991  Articaine hydrochloride (JAN/USP)
         D08490  Ropivacaine (INN)
         D04048  Ropivacaine hydrochloride (USP) <JP/US>
         D08116  Levobupivacaine (INN)
         D01287  Levobupivacaine hydrochloride (JAN/USAN) <JP>
         D00110  Cocaine (USP)
         D02182  Cocaine hydrochloride (JP18/USP) <US>
         D00512  Phenytoin (JP18/USP/INN) <JP/US>
         D02103  Phenytoin sodium (USP) <JP/US>
         D00375  Mephenytoin (USP/INN)
         D07993  Fosphenytoin (INN)
         D02096  Fosphenytoin sodium (USP) <US>
         D07595  Fosphenytoin sodium hydrate (JAN) <JP>
         D00252  Carbamazepine (JP18/USP/INN) <JP/US>
         D00533  Oxcarbazepine (JAN/USP/INN) <US>
         D05775  Rufinamide (JAN/USP/INN) <JP/US>
         D09215  Eslicarbazepine (USAN/INN)
         D09612  Eslicarbazepine acetate (USAN) <US>
         D00354  Lamotrigine (JAN/USP/INN) <JP/US>
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D00538  Zonisamide (JP18/USP/INN) <JP/US>
         D07299  Lacosamide (JAN/USAN/INN) <JP/US>
         D11150  Cenobamate (USAN/INN) <US>
         D08448  Proxymetacaine (INN)
         D02098  Proparacaine hydrochloride (USP) <US>
         D01519  Ethyl piperidinoacetylaminobenzoate (JAN) <JP>
         D01554  Pilsicainide hydrochloride hydrate (JP18) <JP>
         D01785  Pirmenol hydrochloride hydrate (JAN) <JP>
         D01967  p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN) <JP>
         D02762  Actisomide (USAN/INN)
         D04521  Indecainide hydrochloride (USAN)
         D05708  Recainam hydrochloride (USAN)
         D05709  Recainam tosylate (USAN)
         D06203  Transcainide (USAN/INN)
         D06517  Pirmenol hydrochloride (USAN)
         D08377  Pilsicainide (INN)
         D08394  Pirmenol (INN)
         D09833  Levosemotiadil fumarate (JAN)
         D11155  Eleclazine (USAN/INN)
         D12616  Bliretrigine (JAN/INN)
       SCN11A [HSA:11280] [KO:K04843]
     Calcium channels
     Potassium channels
     Inward rectifier channels (Kir)
     Ryanodine receptors (RYR)
     Transient receptor potential channels
   Other ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

[ DRUG | BRITE | KEGG2 | KEGG ]
Last updated: March 28, 2024

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