Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
   Ligand-gated ion channels
     Acetylcholine (nicotinic)
     Serotonin
     GABA (ionotropic)
     Glycine
     Glutamate (ionotropic), non-NMDA
     Glutamate (ionotropic), NMDA
       GRIN (NMDAR) [HSA:2902 2903 2904 2905 2906 116443 116444] [KO:K05208 K05209 K05210 K05211 K05212 K05213 K05214]
       GRIN (NMDAR) [HSA:2902 2903 2904 2905 2906] [KO:K05208 K05209 K05210 K05211 K05212]
         D08098  Ketamine (INN)
         D00711  Ketamine hydrochloride (JP18/USP) <JP/US>
         D07283  Esketamine (USAN/INN)
         D10627  Esketamine hydrochloride (JAN/USAN) <US>
         D07441  Amantadine (INN)
         D00777  Amantadine hydrochloride (JP18/USP) <JP/US>
         D07306  Budipine (INN)
         D07589  Budipine hydrochloride
         D08174  Memantine (INN)
         D04905  Memantine hydrochloride (JAN/USP) <JP/US>
         D07058  Acamprosate (INN)
         D02780  Acamprosate calcium (JAN/USAN) <JP/US>
         D08195  Methadone (BAN)
         D02102  Methadone hydrochloride (JAN/USP) <JP/US>
         D08121  Levomethadone (INN)
         D08122  Levomethadone hydrochloride
         D00775  Riluzole (JAN/USP/INN) <JP/US>
         D11414  Troriluzole (USAN)
         D11415  Troriluzole hydrochloride (USAN)
         D03742  Dextromethorphan (USP)
         D00848  Dextromethorphan hydrobromide (USP) <JP>
         D03744  Dextromethorphan polistirex (USAN)
         D02410  Selfotel (USAN/INN)
         D02973  Aptiganel hydrochloride (USAN)
         D03679  Delucemine hydrochloride (USAN)
         D03746  Dextrorphan hydrochloride (USAN)
         D03878  Dizocilpine maleate (USAN)
         D04308  Gavestinel (USAN/INN)
         D04728  Licostinel (USAN/INN)
         D05447  Perzinfotel (USAN/INN)
         D05453  Phencyclidine hydrochloride (USAN)
         D05714  Remacemide hydrochloride (USAN)
         D06146  Tiletamine hydrochloride (USP)
         D08596  Tiletamine (INN)
         D09917  Latrepirdine (USAN/INN)
         D09918  Latrepirdine dihydrochloride (USAN)
         D11299  Apimostinel (USAN)
         D12214  Esmethadone (USAN)
         D12215  Esmethadone hydrochloride (USAN)
         D12553  Nevadistinel (USAN)
         D12554  Risevistinel (USAN)
         D12702  Tenocyclidine (INN)
       GRIN2B (NMDAR2B) [HSA:2904] [KO:K05210]
     Epithelial sodium channel (SCNN)
     ATP-gated cation channel (P2X)
   Voltage-gated ion channels
   Other ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 20, 2024

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