Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
   Oxidoreductases (EC1)
   Transferases (EC2)
     Methyltransferases [EC:2.1.1.-]
     Acyltransferases [EC:2.3.1.-]
     gamma-Glutamyltransferase [EC:2.3.2.2]
     E3 ubiquitin-protein ligase [EC:2.3.2.27]
     ATP citrate synthase [EC:2.3.3.8]
     Hexosyltransferases [EC:2.4.1.-]
     Pentosyltransferases [EC:2.4.2.-]
     Alkyl/Aryl transferases [EC:2.5.1.-]
       FDPS [HSA:2224] [KO:K00787]
         D07281  Pamidronic acid (INN)
         D00941  Pamidronate disodium (USP) <JP/US>
         D07119  Alendronic acid (INN)
         D00939  Alendronate sodium (USP) <JP/US>
         D08056  Ibandronic acid (INN)
         D04486  Ibandronate sodium (USAN) <JP/US>
         D08484  Risedronic acid (INN)
         D00942  Risedronate sodium (USP) <US>
         D03234  Sodium risedronate hydrate (JP18) <JP/US>
         D11570  Risedronate sodium monohydrate <US>
         D08689  Zoledronic acid (INN)
         D01968  Zoledronic acid (USAN) <JP/US>
         D06378  Zoledronate disodium (USAN)
         D06379  Zoledronate trisodium (USAN)
         D10515  Zoledronic acid hemipentahydrate (JAN)
         D07123  Incadronate disodium hydrate (JAN)
         D08073  Incadronic acid (INN)
         D09198  Minodronic acid hydrate (JAN) <JP>
       GSTP1 [HSA:2950] [KO:K23790]
       FDFT1 [HSA:2222] [KO:K00801]
       FNT [HSA:2339 2342] [KO:K05955 K05954]
     Aminotransferase [EC:2.6.1.-]
     Phosphotransferase [EC:2.7.1.-]
     DNA polymerase [EC:2.7.7.7]
     Reverse transcriptase [EC:2.7.7.49]
   Hydrolases (EC3)
   Lyases (EC4)
   Isomerases (EC5)
   Ligases (EC6)
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 20, 2024

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