Target-based Classification of Drugs

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 G Protein-coupled receptors
   Rhodopsin family
     Acetylcholine (muscarinic)
     Adrenaline
       ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
         D00095  Epinephrine (USP/INN) <JP/US>
         D00996  Epinephrine hydrochloride (JAN)
         D02149  Epinephrine bitartrate (JAN/USP)
         D02774  Adrenalone (USAN/INN)
         D07560  Adrenalone hydrochloride
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D02537  Dronedarone (INN)
         D03914  Dronedarone hydrochloride (USP) <US>
         D07931  Etilefrine (INN)
         D01573  Etilefrine hydrochloride (JP18) <JP>
         D00076  Noradrenaline (JP18) <JP>
         D05206  Norepinephrine bitartrate (USP) <US>
         D08284  Norepinephrine hydrochoride
         D09794  Norepinephrine hydrochloride (JAN)
         D08286  Norfenefrine (INN)
         D01405  Norfenefrine hydrochloride (JAN)
         D08365  Phenylephrine (INN)
         D00511  Phenylephrine hydrochloride (JP18/USP) <JP/US>
         D08366  Phenylephrine tartrate
         D08966  Phenylephrine bitartrate (USP)
         D08192  Metaraminol (INN)
         D01019  Metaraminol bitartrate (JAN/USP)
         D08201  Methoxamine (BAN)
         D01020  Methoxamine hydrochloride (JAN)
         D08220  Midodrine (INN)
         D01307  Midodrine hydrochloride (JAN/USP) <JP/US>
         D00124  Ephedrine (USP)
         D01386  Ephedrine hydrochloride (JP18/USP) <JP/US>
         D04018  Ephedrine sulfate (USP) <US>
         D01277  Droxidopa (JP18/USAN/INN) <JP/US>
         D08411  Prazosin (INN)
         D00609  Prazosin hydrochloride (JP18/USP) <JP/US>
         D04531  Indoramin (USAN/INN)
         D04532  Indoramin hydrochloride (USAN)
         D08212  Trimazosin (INN)
         D06234  Trimazosin hydrochloride (USAN)
         D07874  Doxazosin (INN)
         D00608  Doxazosin mesylate (USP) <JP/US>
         D01333  Urapidil (JP18/INN) <JP>
         D08662  Urapidil hydrochloride
         D08362  Phentolamine (INN)
         D00509  Phentolamine mesylate (USP) <JP/US>
         D08614  Tolazoline (INN)
         D00997  Tolazoline hydrochloride (JAN/USP)
         D02268  Ergoloid mesylates (USP)
         D01290  Nicergoline (JP18/USAN/INN) <JP>
         D08271  Nicergoline tartrate
         D07834  Dihydroergocristine (BAN)
         D07833  Dihydroergocristine mesilate (BAN)
         D08358  Phenoxybenzamine (INN)
         D00507  Phenoxybenzamine hydrochloride (USP) <US>
         D08239  Moxisylyte (INN)
         D01571  Moxisylyte hydrochloride (JAN)
         D08064  Ifenprodil (INN)
         D01445  Ifenprodil tartrate (JP18) <JP>
         D01369  Bevantolol hydrochloride (JAN/USAN) <JP>
         D08106  Labetalol (INN)
         D00600  Labetalol hydrochloride (JP18/USP) <JP/US>
         D00255  Carvedilol (JP18/USP/INN) <JP/US>
         D03415  Carvedilol phosphate (USAN) <US>
         D08207  Methylergometrine (INN)
         D00680  Methylergonovine maleate (USP) <JP/US>
         D07906  Ergotamine (INN)
         D07905  Ergometrine (INN)
         D01163  Ergonovine maleate (USP)
         D08560  Tamsulosin (INN)
         D01024  Tamsulosin hydrochloride (JP18/USP) <JP/US>
         D08569  Terazosin (INN)
         D00610  Terazosin hydrochloride (USP) <JP/US>
         D11585  Terazosin hydrochloride anhydrous <US>
         D00679  Ergotamine tartrate (JP18/USP) <US>
         D01485  Propericiazine (JAN) <JP>
         D00308  Droperidol (JP18/USP/INN) <JP/US>
         D00454  Olanzapine (JAN/USP/INN) <JP/US>
         D06623  Olanzapine pamoate (USAN) <US>
         D08257  Nefazodone (INN)
         D00819  Nefazodone hydrochloride (USP) <US>
         D08578  Tetryzoline (INN)
         D00756  Tetrahydrozoline nitrate (JAN)
         D01023  Tetrahydrozoline hydrochloride (JAN/USP)
         D08684  Xylometazoline (INN)
         D00757  Xylometazoline hydrochloride (USP)
         D08253  Naphazoline (INN)
         D00743  Naphazoline hydrochloride (JP18/USP)
         D01021  Naphazoline nitrate (JP18) <JP>
         D08624  Tramazoline (INN)
         D01347  Tramazoline hydrochloride (JAN/USAN) <JP>
         D08368  Phenylpropanolamine (INN)
         D01224  Phenylpropanolamine hydrochloride (JAN/USP)
         D05466  Phenylpropanolamine polistirex (USAN)
         D08449  Pseudoephedrine (INN)
         D00485  Pseudoephedrine hydrochloride (USP)
         D05648  Pseudoephedrine polistirex (USAN)
         D05649  Pseudoephedrine sulfate (USP)
         D02349  Dipivefrin (USAN)
         D01017  Dipivefrin hydrochloride (USP)
         D08115  Levobunolol (INN)
         D01025  Levobunolol hydrochloride (JAN/USP) <JP/US>
         D07775  Dapiprazole (INN)
         D03648  Dapiprazole hydrochloride (USAN) <US>
         D00607  Guanadrel sulfate (USAN)
         D01171  Monatepil maleate (JAN/USAN)
         D01444  Bunitrolol hydrochloride (JAN)
         D01469  Amosulalol hydrochloride (JP18) <JP>
         D01674  Naftopidil (JP18/INN) <JP>
         D01691  Nipradilol (JAN/INN) <JP>
         D01830  Arotinolol hydrochloride (JP18) <JP>
         D01887  Bunazosin hydrochloride (JP18) <JP>
         D01952  L-Methylephedrine hydrochloride (JAN)
         D02109  dl-Methylephedrine hydrochloride (JP18) <JP>
         D02568  Flesinoxan (INN)
         D02901  Amidephrine mesylate (USAN)
         D03887  Domazoline fumarate (USAN)
         D04026  Epinephryl borate (USP)
         D05228  Octodrine (USAN/INN)
         D05395  Pelanserin hydrochloride (USAN)
         D05637  Propylhexedrine (USP/INN)
         D05688  Racepinephrine (USP/INN)
         D05689  Racepinephrine hydrochloride (USP)
         D07451  Amosulalol (INN)
         D07465  Arotinolol (INN)
         D07550  Bunazosin (INN)
         D08029  Guanadrel (INN)
         D08206  Methylephedrine (BAN)
         D08444  Propylhexedrine hydrochloride
         D08982  Racephedrine hydrochloride (USAN)
         D09842  dl-Methylephedrine saccharinate (JAN)
       ADRA1A [HSA:148] [KO:K04135]
       ADRA1D [HSA:146] [KO:K04137]
       ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
       ADRA2A [HSA:150] [KO:K04138]
       ADRA2B [HSA:151] [KO:K04139]
       ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
       ADRB1 [HSA:153] [KO:K04141]
         D02910  Amiodarone (USAN/INN)
         D00636  Amiodarone hydrochloride (JP18/USP) <JP/US>
         D02537  Dronedarone (INN)
         D03914  Dronedarone hydrochloride (USP) <US>
         D03879  Dobutamine (USAN/INN)
         D00632  Dobutamine hydrochloride (JP18/USP) <JP/US>
         D03880  Dobutamine lactobionate (USAN)
         D03881  Dobutamine tartrate (USAN)
         D06328  Xamoterol (USAN)
         D06329  Xamoterol fumarate (USAN)
         D08600  Timolol (INN)
         D00378  Timolol (USAN) <US>
         D00603  Timolol maleate (JP18/USP) <JP/US>
         D08525  Sotalol (INN)
         D01026  Sotalol hydrochloride (JAN/USP) <JP/US>
         D00432  Nadolol (JP18/USP/INN) <JP/US>
         D05587  Practolol (USAN)
         D02358  Metoprolol (USAN/INN)
         D00601  Metoprolol tartrate (JP18/USP) <JP/US>
         D00635  Metoprolol succinate (USP) <US>
         D05011  Metoprolol fumarate (USP)
         D00235  Atenolol (JP18/USP/INN) <JP/US>
         D02338  Acebutolol (USAN/INN)
         D00597  Acebutolol hydrochloride (JP18/USP) <US>
         D07526  Betaxolol (INN)
         D00598  Betaxolol hydrochloride (JP18/USP) <JP/US>
         D01369  Bevantolol hydrochloride (JAN/USAN) <JP>
         D02342  Bisoprolol (JAN/USAN/INN) <JP>
         D00634  Bisoprolol fumarate (JP18/USP) <JP/US>
         D07660  Celiprolol (INN)
         D01741  Celiprolol hydrochloride (JAN/USAN) <JP>
         D07916  Esmolol (INN)
         D00644  Esmolol hydrochloride (JAN/USP) <JP/US>
         D06646  Epanolol (USAN/INN)
         D01471  Esatenolol (JAN/INN)
         D05127  Nebivolol (USAN/INN)
         D06622  Nebivolol hydrochloride (USAN) <US>
         D01847  Landiolol hydrochloride (JAN/USAN) <JP>
         D12410  Landiolol (USAN/INN)
         D08106  Labetalol (INN)
         D00600  Labetalol hydrochloride (JP18/USP) <JP/US>
         D00255  Carvedilol (JP18/USP/INN) <JP/US>
         D03415  Carvedilol phosphate (USAN) <US>
         D01469  Amosulalol hydrochloride (JP18) <JP>
         D01492  Bucumolol hydrochloride (JP18)
         D01830  Arotinolol hydrochloride (JP18) <JP>
         D01903  Docarpamine (JAN/INN) <JP>
         D01958  Indenolol hydrochloride (JP18)
         D02389  Primidolol (USAN/INN)
         D02614  Denopamine (JAN/INN) <JP>
         D03177  Bunolol hydrochloride (USAN)
         D03195  Butopamine (USAN/INN)
         D03449  Cetamolol hydrochloride (USAN)
         D03490  Cicloprolol hydrochloride (USAN)
         D04708  Levdobutamine lactobionate (USAN)
         D04710  Levobetaxolol hydrochloride (USAN)
         D07451  Amosulalol (INN)
         D07465  Arotinolol (INN)
         D08078  Indenolol (INN)
       ADRB2 [HSA:154] [KO:K04142]
         D03891  Dopexamine (USAN/INN)
         D03892  Dopexamine hydrochloride (USAN)
         D08092  Isoxsuprine (INN)
         D01748  Isoxsuprine hydrochloride (JP18/USP) <JP>
         D08093  Isoxsuprine lactate
         D08600  Timolol (INN)
         D00378  Timolol (USAN) <US>
         D00603  Timolol maleate (JP18/USP) <JP/US>
         D08525  Sotalol (INN)
         D01026  Sotalol hydrochloride (JAN/USP) <JP/US>
         D00432  Nadolol (JP18/USP/INN) <JP/US>
         D08106  Labetalol (INN)
         D00600  Labetalol hydrochloride (JP18/USP) <JP/US>
         D00255  Carvedilol (JP18/USP/INN) <JP/US>
         D03415  Carvedilol phosphate (USAN) <US>
         D02359  Ritodrine (USAN/INN)
         D01263  Ritodrine hydrochloride (JP18/USP) <JP>
         D04157  Fenoterol (USAN/INN)
         D01428  Fenoterol hydrobromide (JAN) <JP>
         D08300  Orciprenaline (INN)
         D00685  Metaproterenol sulfate (USP)
         D04954  Metaproterenol polistirex (USAN)
         D02147  Albuterol (USP)
         D00683  Albuterol sulfate (USP) <JP/US>
         D08570  Terbutaline (INN)
         D00688  Terbutaline sulfate (JP18/USP) <JP/US>
         D05730  Rimiterol hydrobromide (USAN)
         D08039  Hexoprenaline (INN)
         D02396  Hexoprenaline sulfate (USAN)
         D04625  Isoetharine (USP)
         D02093  Isoetharine hydrochloride (USP)
         D04626  Isoetharine mesylate (USP)
         D08387  Pirbuterol (INN)
         D00686  Pirbuterol acetate (USAN)
         D01349  Pirbuterol hydrochloride (JAN/USAN)
         D08629  Tretoquinol (INN)
         D01978  Trimetoquinol hydrochloride
         D05037  Trimetoquinol hydrochloride hydrate (JP18) <JP>
         D03402  Carbuterol hydrochloride (USAN)
         D02151  Tulobuterol (JP18/INN) <JP>
         D01362  Tulobuterol hydrochloride (JP18) <JP>
         D05792  Salmeterol (USAN/INN)
         D00687  Salmeterol xinafoate (JAN/USP) <JP/US>
         D07990  Formoterol (INN)
         D01373  Formoterol fumarate (USP) <US>
         D05277  Formoterol fumarate hydrate (JP18) <JP/US>
         D07713  Clenbuterol (INN)
         D01360  Clenbuterol hydrochloride (JAN/USP) <JP>
         D08474  Reproterol (INN)
         D05718  Reproterol hydrochloride (USAN)
         D08424  Procaterol (INN)
         D02404  Procaterol hydrochloride (USAN)
         D05366  Procaterol hydrochloride hydrate (JP18) <JP>
         D07534  Bitolterol (INN)
         D00684  Bitolterol mesylate (USAN)
         D09318  Indacaterol (USAN/INN)
         D09319  Indacaterol maleate (JAN/USAN) <JP>
         D11009  Indacaterol acetate (JAN)
         D10145  Olodaterol (USAN/INN)
         D10020  Olodaterol hydrochloride (JAN/USAN) <US>
         D01635  Methoxyphenamine hydrochloride (JAN)
         D07377  Bambuterol (INN)
         D07489  Bambuterol hydrochloride
         D01469  Amosulalol hydrochloride (JP18) <JP>
         D01492  Bucumolol hydrochloride (JP18)
         D01589  Mabuterol hydrochloride (JAN)
         D01830  Arotinolol hydrochloride (JP18) <JP>
         D01835  Clorprenaline hydrochloride (JAN/USAN)
         D01958  Indenolol hydrochloride (JP18)
         D02281  Levalbuterol hydrochloride (USP) <US>
         D02981  Arformoterol tartrate (USAN) <US>
         D03170  Bucindolol hydrochloride (USAN)
         D03177  Bunolol hydrochloride (USAN)
         D03198  Butoxamine hydrochloride (USAN)
         D03587  Colterol mesylate (USAN)
         D04072  Etafedrine hydrochloride (USAN)
         D04701  Levalbuterol sulfate (USAN)
         D04703  Levalbuterol tartrate (USAN) <US>
         D04953  Metalol hydrochloride (USAN)
         D05476  Picumeterol fumarate (USAN)
         D05691  Ractopamine hydrochloride (USP)
         D05832  Sibenadet hydrochloride (USAN)
         D05902  Soterenol hydrochloride (USAN)
         D06374  Zinterol hydrochloride (USAN)
         D06562  Bedoradrine sulfate (USAN)
         D07451  Amosulalol (INN)
         D07463  Arformoterol (INN)
         D07465  Arotinolol (INN)
         D07608  Carazolol (INN)
         D08078  Indenolol (INN)
         D08124  Levosalbutamol (INN)
         D08945  Milveterol hydrochloride (USAN)
         D09696  Vilanterol (USAN/INN)
         D09697  Vilanterol trifenatate (JAN/USAN)
         D10219  Abediterol (USAN/INN)
         D10220  Abediterol napadisylate (USAN)
         D10545  Batefenterol (USAN)
         D10546  Batefenterol succinate (USAN)
         D11900  Navafenterol (USAN)
         D11901  Navafenterol saccharinate (USAN)
       ADRB3 [HSA:155] [KO:K04143]
     Dopamine
     Histamine
     Serotonin
     Trace amine
     Angiotensin
     Bradykinin
     Cholecystokinin
     Endothelin
     Follicle stimulating hormone
     Ghrelin
     Gonadotropin-releasing hormone
     Lutropin-choriogonadotropic hormone
     Melanocortin
     Motilin
     Neuropeptide Y
     Opioid
     Orexin
     Oxytocin
     Relaxin
     Somatostatin
     Tachykinin
     Thrombin
     Thyrotropin-releasing hormone
     Vasopressin
     Purine / pyrimidine
     Adenosine
     Cysteinyl leukotriene
     Free fatty acid
     Leukotriene
     Lysophosphatidic acid
     Prostaglandin
     Prostacyclin
     Sphingolipid
     Thromboxane
     Cannabinoid
     Melatonin
     Platelet activating factor
     R-spondin
   Secretin receptor family
   Metabotropic glutamate receptor family
   Frizzled / Smoothened family
   Others
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 18, 2024

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