G Protein-coupled receptors
|
Rhodopsin family
|
Acetylcholine (muscarinic)
|
Adrenaline
|
Dopamine
|
DRD [HSA:1812 1813 1814 1815 1816] [KO:K04144 K04145 K04146 K04147 K05840]
|
DRD1 [HSA:1812] [KO:K04144]
|
DRD2 [HSA:1813] [KO:K04145]
|
D00726 Metoclopramide (JP18/INN) <JP>
D02213 Metoclopramide hydrochloride (JAN) <JP>
D05008 Metoclopramide hydrochloride (USP) <US>
D01745 Domperidone (JP18/USAN/INN) <JP>
D07868 Domperidone maleate
D07101 Bromopride (INN)
D07102 Alizapride (INN)
D07563 Alizapride hydrochloride
D03534 Clebopride (USAN)
D01742 Clebopride malate (JP18)
D08094 Itopride (INN)
D02729 Itopride hydrochloride (JAN) <JP>
D05010 Metopimazine (USAN/INN)
D04488 Ibopamine (USAN/INN)
D08057 Ibopamine hydrochloride
D03165 Bromocriptine (USAN/INN)
D00780 Bromocriptine mesylate (USP) <JP/US>
D08132 Lisuride (INN)
D01462 Lisuride maleate (JAN)
D00987 Cabergoline (JP18/USP/INN) <JP/US>
D07217 Quinagolide (INN/BAN)
D08457 Quinagolide hydrochloride (BAN)
D01348 Terguride (JAN/INN)
D07460 Apomorphine (BAN)
D02004 Apomorphine hydrochloride (USP) <JP/US>
D08339 Pergolide (INN)
D00502 Pergolide mesylate (USP) <JP>
D07836 Dihydroergocryptine mesilate
D08489 Ropinirole (USAN/INN)
D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
D05575 Pramipexole (USAN/INN)
D00559 Pramipexole dihydrochloride (USP) <JP/US>
D07305 Piribedil (INN)
D05768 Rotigotine (JAN/USAN/INN) <JP/US>
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D00403 Methotrimeprazine (USP)
D01520 Levomepromazine hydrochloride (JAN/USAN) <JP>
D02248 Levomepromazine maleate (JP18/USAN) <JP>
D08430 Promazine (INN)
D00797 Promazine hydrochloride (USP)
D07065 Acepromazine (INN)
D02604 Acepromazine maleate (USP)
D00390 Triflupromazine (USP/INN)
D00800 Triflupromazine hydrochloride (JAN/USP)
D07977 Fluphenazine (INN)
D00791 Fluphenazine hydrochloride (JAN/USP) <US>
D00792 Fluphenazine enanthate (JP18/USP)
D00793 Fluphenazine decanoate (JAN/USP) <JP/US>
D02163 Fluphenazine maleate (JAN) <JP>
D00503 Perphenazine (JP18/USP/INN) <JP/US>
D02037 Perphenazine maleate (JP18) <JP>
D04038 Perphenazine fendizoate (JAN) <JP>
D04965 Perphenazine hydrochloride <JP>
D08341 Perphenazine decanoate
D08342 Perphenazine enantate
D00493 Prochlorperazine (JAN/USP/INN) <US>
D00479 Prochlorperazine maleate (JP18/USP) <JP/US>
D02022 Prochlorperazine mesilate (JAN) <JP>
D02609 Prochlorperazine edisylate (USP) <US>
D08636 Trifluoperazine (INN)
D00799 Trifluoperazine hydrochloride (JAN/USP) <US>
D01448 Trifluoperazine maleate (JAN)
D00788 Acetophenazine maleate (USAN)
D08585 Thioproperazine (INN)
D01447 Thioproperazine mesilate (JAN)
D01412 Perazine maleate (JAN)
D01860 Perazine dimalonate (JAN)
D02608 Perazine fendizoate (JAN)
D01485 Propericiazine (JAN) <JP>
D00373 Thioridazine (USP/INN)
D00798 Thioridazine hydrochloride (JP18/USP) <US>
D02671 Mesoridazine (USAN/INN)
D00795 Mesoridazine besylate (USP)
D08385 Pipotiazine (INN)
D02680 Pipotiazine palmitate (USAN)
D00136 Haloperidol (JP18/USP/INN) <JP/US>
D01898 Haloperidol decanoate (JAN/USP) <JP/US>
D08035 Haloperidol lactate <US>
D02625 Trifluperidol (USAN/INN)
D08637 Trifluperidol hydrochloride
D07309 Melperone (INN)
D08172 Melperone hydrochloride
D02623 Moperone (INN)
D01105 Moperone hydrochloride (JAN)
D02622 Pipamperone (USAN/INN)
D01482 Pipamperone hydrochloride (JAN) <JP>
D01101 Bromperidol (JAN/USAN/INN) <JP>
D02626 Bromperidol decanoate (USAN)
D02627 Benperidol (USAN/INN)
D00308 Droperidol (JP18/USP/INN) <JP/US>
D11169 Lumateperone (USAN/INN)
D11170 Lumateperone tosylate (USAN) <US>
D08226 Molindone (INN)
D00796 Molindone hydrochloride (USP) <US>
D00561 Sertindole (USAN/INN)
D08687 Ziprasidone (INN)
D01939 Ziprasidone hydrochloride (USP) <US>
D02100 Ziprasidone mesylate (USAN) <US>
D04820 Lurasidone hydrochloride (JAN/USAN) <JP/US>
D01044 Flupentixol (INN)
D02236 Flupentixol dihydrochloride (JAN)
D07976 Flupentixol decanoate
D02613 Clopenthixol (USAN)
D00790 Chlorprothixene (JAN/USAN/INN)
D02162 Chlorprothixene hydrochloride (JAN)
D07686 Chlorprothixene acetate
D07687 Chlorprothixene citrate
D00374 Thiothixene (USP) <US>
D02612 Thiothixene hydrochloride (USP)
D03556 Zuclopenthixol (INN)
D08691 Zuclopenthixol acetate
D08692 Zuclopenthixol decanoate
D08693 Zuclopenthixol dihydrochloride
D00560 Pimozide (JP18/USP/INN) <US>
D02340 Loxapine (USAN/INN) <US>
D00794 Loxapine succinate (USP) <US>
D08148 Loxapine hydrochloride
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D08456 Quetiapine (INN)
D00458 Quetiapine fumarate (JP18/USP) <JP/US>
D11769 Asenapine (INN) <US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D01226 Sulpiride (JP18/USAN/INN) <JP>
D08549 Sultopride (INN)
D02208 Sultopride hydrochloride (JAN) <JP>
D08590 Tiapride (INN)
D01522 Tiapride hydrochloride (JP18) <JP>
D02682 Remoxipride (USAN)
D02683 Remoxipride hydrochloride (USAN)
D07310 Amisulpride (INN) <US>
D07312 Levosulpiride (INN)
D00426 Risperidone (JP18/USP/INN) <JP/US>
D08235 Mosapramine (INN)
D01548 Mosapramine hydrochloride (JAN) <JP>
D01321 Zotepine (JAN/INN) <JP>
D01164 Aripiprazole (JAN/USP/INN) <JP/US>
D10355 Aripiprazole cavoxil (USAN)
D10364 Aripiprazole lauroxil (USAN) <US>
D10516 Aripiprazole hydrate (JAN) <JP/US>
D05339 Paliperidone (JAN/USP/INN) <JP/US>
D05340 Paliperidone palmitate (JAN/USAN) <JP/US>
D02666 Iloperidone (USAN/INN) <US>
D09997 Cariprazine (USAN/INN)
D09876 Cariprazine hydrochloride (JAN/USAN) <US>
D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
D07593 Buspirone (INN)
D00702 Buspirone hydrochloride (USP) <US>
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D02354 Thiethylperazine (USAN/INN)
D01130 Thiethylperazine maleate (JAN/USP)
D02610 Thiethylperazine malate (JAN)
D01051 Spiperone (JAN/USAN) <JP>
D01176 Blonanserin (JAN/INN) <JP>
D01468 Nemonapride (JAN/INN) <JP>
D01505 Talipexole hydrochloride (JAN)
D02035 Timiperone (JAN) <JP>
D02371 Clocapramine hydrochloride hydrate (JP18) <JP>
D02372 Perospirone hydrochloride hydrate (JAN) <JP>
D02605 Methoxypromazine maleate
D02634 Alentemol hydrobromide (USAN)
D02641 Butaclamol hydrochloride (USAN)
D02644 Carphenazine maleate (USAN)
D02645 Carvotroline hydrochloride (USAN)
D02670 Mazapertine succinate (USAN)
D02675 Ocaperidone (USAN)
D02681 Piquindone hydrochloride (USAN)
D02688 Tiospirone hydrochloride (USAN)
D03214 Aplindore fumarate (USAN)
D03494 Ciladopa hydrochloride (USAN)
D04693 Lergotrile (USAN/INN)
D04694 Lergotrile mesylate (USAN)
D05124 Naxagolide hydrochloride (USAN)
D05677 Quinelorane hydrochloride (USAN)
D05682 Quinpirole hydrochloride (USAN)
D05690 Raclopride C11 (USAN)
D05804 Sarizotan hydrochloride (USAN)
D05832 Sibenadet hydrochloride (USAN)
D06566 Bifeprunox (USAN/INN)
D06567 Bifeprunox mesylate (USAN)
D07718 Clocapramine (INN)
D07835 Dihydroergocryptine
D08558 Talipexole (INN)
D09366 Pardoprunox hydrochloride (USAN)
D09397 Pardoprunox (USAN/INN)
D09953 Pridopidine (USAN/INN)
D09954 Pridopidine hydrochloride (USAN)
D10329 Zicronapine (USAN/INN)
D10495 Zicronapine succinate (USAN)
D11982 Trazpiroben (USAN/INN)
D12733 Dordaviprone (USAN/INN)
D12734 Dordaviprone hydrochloride (JAN/USAN)
D12813 Brilaroxazine (USAN/INN)
D12814 Brilaroxazine hydrochloride (USAN)
|
DRD3 [HSA:1814] [KO:K04146]
|
DRD4 [HSA:1815] [KO:K04147]
|
DRD5 [HSA:1816] [KO:K05840]
|
Histamine
|
HRH1 [HSA:3269] [KO:K04149]
|
D08587 Thonzylamine (INN)
D01801 Thonzylamine hydrochloride (JAN/USAN)
D08183 Mepyramine (INN)
D05660 Pyrilamine maleate (USP)
D07194 Thenalidine (INN)
D08645 Tripelennamine (INN)
D02091 Tripelennamine hydrochloride (USP)
D06246 Tripelennamine citrate
D07195 Chloropyramine (INN)
D07679 Chloropyramine hydrochloride
D00494 Promethazine (JAN/INN)
D00480 Promethazine hydrochloride (JP18/USP) <JP/US>
D01242 Promethazine teoclate (JAN/INN)
D03290 Promethazine methylenedisalicylate (JAN) <JP>
D08432 Promethazine maleate
D08768 Promethazine hibenzate <JP>
D07196 Tolpropamine (INN)
D07853 Dimetindene (INN)
D01343 Dimethindene maleate (USAN)
D03535 Clemastine (USAN)
D00666 Clemastine fumarate (JP18/USP) <JP/US>
D07197 Bamipine (INN)
D07492 Bamipine dihydrochloride
D07493 Bamipine lactate
D08355 Pheniramine (INN)
D01174 Pheniramine maleate (JAN/USP)
D08091 Isothipendyl (INN)
D01143 Isothipendyl hydrochloride (JAN)
D00300 Diphenhydramine (JP18/INN) <JP>
D00669 Diphenhydramine hydrochloride (JP18/USP) <JP/US>
D02419 Diphenhydramine salicylate (JAN)
D03285 Diphenhydramine tannate (JP18)
D03360 Diphenhydramine laurylsulfate (JAN) <JP>
D03854 Diphenhydramine citrate (USP)
D07198 Chlorphenoxamine (INN)
D07684 Chlorphenoxamine hydrochloride
D07875 Doxepin (INN)
D00814 Doxepin hydrochloride (USP) <US>
D00774 Orphenadrine citrate (USP) <US>
D07854 Dimetotiazine (INN)
D01902 Fonazine mesylate (USAN) <JP>
D02599 Orphenadrine hydrochloride
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D08054 Hydroxyzine (INN)
D00672 Hydroxyzine hydrochloride (JP18/USP) <JP/US>
D01096 Hydroxyzine pamoate (JP18/USP) <JP/US>
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D07522 Betahistine (INN)
D01592 Betahistine mesilate (JP18) <JP>
D03102 Betahistine hydrochloride (USP)
D01295 Cinnarizine (JAN/USAN/INN)
D07734 Cinnarizine dihydrochloride
D08117 Levocabastine (INN)
D01717 Levocabastine hydrochloride (JAN/USP) <JP>
D07483 Azelastine (INN)
D00659 Azelastine hydrochloride (JP18/USP) <JP/US>
D07458 Antazoline (INN)
D02950 Antazoline phosphate (USP)
D07459 Antazoline hydrochloride
D08293 Olopatadine (INN)
D01192 Olopatadine hydrochloride (JP18/USP) <JP/US>
D03166 Bromodiphenhydramine hydrochloride (USP)
D07862 Diphenylpyraline (INN)
D01172 Diphenylpyraline hydrochloride (JAN)
D01627 Diphenylpyraline teoclate (JAN)
D07617 Carbinoxamine (INN)
D01336 Carbinoxamine maleate (JAN/USP) <US>
D09808 Carbinoxamine diphenyldisulfonate (JAN)
D07878 Doxylamine (INN)
D02327 Doxylamine succinate (USP)
D00520 Dimenhydrinate (JP18/USP/INN) <JP/US>
D07543 Brompheniramine (INN)
D00663 Brompheniramine maleate (USP)
D07803 Dexchlorpheniramine (INN)
D00668 Dexchlorpheniramine maleate (USP) <JP/US>
D07398 Chlorphenamine (INN)
D00665 Chlorpheniramine maleate (JP18/USP) <JP>
D03475 Chlorpheniramine polistirex (USAN)
D03704 Dexbrompheniramine maleate (USP)
D07400 Histapyrrodine (INN)
D07125 Alimemazine (INN)
D02245 Trimeprazine tartrate (USP) <JP>
D04979 Methdilazine (INN)
D04980 Methdilazine hydrochloride (USP)
D01324 Mequitazine (JP18/INN) <JP>
D07401 Oxomemazine (INN)
D07547 Buclizine (INN)
D02089 Buclizine hydrochloride (USAN)
D03621 Cyclizine (INN)
D02090 Cyclizine lactate (BAN)
D03622 Cyclizine hydrochloride (USP)
D08163 Meclozine (BAN)
D01317 Meclizine hydrochloride (JAN/USP) <US>
D07662 Cetirizine (INN)
D00664 Cetirizine hydrochloride (JP18/USP) <JP/US>
D07402 Levocetirizine (USAN/INN)
D08118 Levocetirizine dihydrochloride (USP) <JP/US>
D07765 Cyproheptadine (INN)
D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
D08353 Phenindamine (INN)
D02148 Phenindamine tartrate (USAN)
D08648 Triprolidine (INN)
D01782 Triprolidine hydrochloride (USP)
D07403 Pyrrobutamine (BAN)
D07482 Azatadine (INN)
D00662 Azatadine maleate (USP)
D00234 Astemizole (JAN/USP/INN)
D00521 Terfenadine (JAN/USAN/INN)
D00364 Loratadine (JAN/USP/INN) <JP>
D08161 Mebhydrolin (INN)
D01786 Mebhydrolin napadisilate (JAN)
D07404 Deptropine (INN)
D07790 Deptropine citrate
D08105 Ketotifen (INN)
D01332 Ketotifen fumarate (JP18/USAN) <JP>
D02760 Acrivastine (USAN/INN)
D01478 Ebastine (JP18/USAN/INN) <JP>
D07406 Pimethixene (INN)
D07900 Epinastine (INN)
D01713 Epinastine hydrochloride (JAN) <JP/US>
D01117 Mizolastine (JAN/INN)
D07958 Fexofenadine (INN)
D00671 Fexofenadine hydrochloride (JP18/USP) <JP/US>
D03693 Desloratadine (JAN/USP/INN) <JP/US>
D07407 Rupatadine (INN)
D08497 Rupatadine fumarate (JAN) <JP>
D09570 Bilastine (JAN/INN) <JP>
D10230 Quifenadine (INN)
D10510 Sequifenadine
D07890 Emedastine (INN)
D02249 Emedastine difumarate (JP18/USP) <JP>
D06552 Alcaftadine (JAN/USAN/INN) <US>
D04445 Histamine phosphate (USP) <US>
D01460 Homochlorcyclizine hydrochloride (JP18) <JP>
D01654 Bepotastine besylate (USAN) <JP/US>
D01701 Difeterol hydrochloride (JAN)
D02067 Diphenylimidazole (JAN)
D03056 Barmastine (USAN/INN)
D03491 Cidoxepin hydrochloride (USAN)
D03568 Closiramine aceturate (USAN)
D03620 Cycliramine maleate (USAN)
D03893 Dorastine hydrochloride (USAN)
D03963 Efletirizine dihydrochloride (USAN)
D04055 Esmirtazapine maleate (USAN)
D04494 Icotidine (USAN)
D05196 Noberastine (USAN/INN)
D05664 Pyroxamine maleate (USAN)
D05742 Rocastine hydrochloride (USAN)
D05769 Rotoxamine (USAN/INN)
D06012 Tazifylline hydrochloride (USAN)
D06021 Tecastemizole (USAN/INN)
D06063 Temelastine (USAN/INN)
D06084 Tesmilifene hydrochloride (USAN)
D06376 Zolamine hydrochloride (USAN)
D07532 Bisulepin
D07533 Bisulepin hydrochloride
D07860 Dioxopromethazine hydrochloride
D07889 Embramine (INN)
D08040 Histamine (DCF) <US>
D08041 Homochlorcyclizine (INN)
D08305 Orphenadrine (INN)
D08967 Phenyltoloxamine citrate (USP)
D09705 Bepotastine (USAN/INN)
D09747 Difeterol phosphate (JAN)
D09748 Difeterol (JAN/INN)
D09838 Broizine (JAN)
|
HRH2 [HSA:3274] [KO:K04150]
|
HRH3 [HSA:11255] [KO:K04151]
|
HRH4 [HSA:59340] [KO:K04152]
|
Serotonin
|
HTR1 [HSA:3350 3351 3352 3354 3355] [KO:K04153]
|
HTR1A [HSA:3350] [KO:K04153]
|
HTR1B [HSA:3351] [KO:K04153]
|
HTR1D [HSA:3352] [KO:K04153]
|
HTR1F [HSA:3355] [KO:K04153]
|
HTR2 [HSA:3356 3357 3358] [KO:K04157]
|
D07700 Cinitapride (INN)
D07701 Cinitapride tartrate
D02577 Flibanserin (USAN/INN) <US>
D02357 Methysergide (USAN/INN)
D00681 Methysergide maleate (USP)
D05523 Pizotyline (USAN)
D08397 Pizotifen malate
D07854 Dimetotiazine (INN)
D01902 Fonazine mesylate (USAN) <JP>
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D01485 Propericiazine (JAN) <JP>
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D02666 Iloperidone (USAN/INN) <US>
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D08626 Trazodone (INN)
D00820 Trazodone hydrochloride (JAN/USP) <JP/US>
D00563 Mirtazapine (JAN/USP/INN) <JP/US>
D11056 Mirtazapine hydrate (JAN)
D07765 Cyproheptadine (INN)
D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
D02675 Ocaperidone (USAN)
D02686 Setoperone (USAN/INN)
D02688 Tiospirone hydrochloride (USAN)
D02767 Adatanserin hydrochloride (USAN)
D04320 Glemanserin (USAN/INN)
D05015 Metrenperone (USAN/INN)
D05395 Pelanserin hydrochloride (USAN)
D05829 Sergolexole maleate (USAN)
D06253 Tropanserin hydrochloride (USAN)
D06343 Xylamidine tosylate (USAN)
D12707 Brolamfetamine (INN)
|
HTR2A [HSA:3356] [KO:K04157]
|
HTR2C [HSA:3358] [KO:K04157]
|
HTR4 [HSA:3360] [KO:K04160]
|
HTR6 [HSA:3362] [KO:K04162]
|
HTR7 [HSA:3363] [KO:K04163]
|
Trace amine
|
Angiotensin
|
Bradykinin
|
Cholecystokinin
|
Endothelin
|
Follicle stimulating hormone
|
Ghrelin
|
Gonadotropin-releasing hormone
|
Lutropin-choriogonadotropic hormone
|
Melanocortin
|
Motilin
|
Neuropeptide Y
|
Opioid
|
Orexin
|
Oxytocin
|
Relaxin
|
Somatostatin
|
Tachykinin
|
Thrombin
|
Thyrotropin-releasing hormone
|
Vasopressin
|
Purine / pyrimidine
|
Adenosine
|
Cysteinyl leukotriene
|
Free fatty acid
|
Leukotriene
|
Lysophosphatidic acid
|
Prostaglandin
|
Prostacyclin
|
Sphingolipid
|
Thromboxane
|
Cannabinoid
|
Melatonin
|
Platelet activating factor
|
R-spondin
|
Secretin receptor family
|
Metabotropic glutamate receptor family
|
Frizzled / Smoothened family
|
Others
|
|
Ion channels
|
|
Nuclear receptors
|
|
Protein kinases
|
|
Cytokines and receptors
|
|
Cell surface molecules and ligands
|
|
Transporters
|
ABC transporters
|
Solute carrier family
|
Major facilitator superfamily
|
Other transporters
|
Channels and pores (TC:1)
|
Auxiliary transport proteins (TC:8.A)
|
SIGMAR1 [HSA:10280] [KO:K20719]
|
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D07316 Captodiame (BAN)
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D03742 Dextromethorphan (USP)
D00848 Dextromethorphan hydrobromide (USP) <JP>
D03744 Dextromethorphan polistirex (USAN)
D02684 Rimcazole hydrochloride (USAN)
D02688 Tiospirone hydrochloride (USAN)
D04502 Igmesine hydrochloride (USAN)
D11383 Blarcamesine (USAN)
D11549 Blarcamesine hydrochloride (USAN)
|
KLB [HSA:152831] [KO:K22404]
|
Others
|
|
Enzymes
|
|
Nucleic acids
|
|
Not elsewhere classified
|