Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
   Serine/threonine kinases
   Receptor serine/threonine kinases (RSTK)
   Receptor tyrosine kinases (RTK)
     EGFR family
       EGFR [HSA:1956] [KO:K04361]
       EGFR* [HSA_VAR:1956v2] [HSA:1956] [KO:K04361]
         D01977  Gefitinib (JP18/USAN/INN) <JP/US>
         D04023  Erlotinib hydrochloride (JAN/USAN) <JP/US>
         D09733  Afatinib dimaleate (USAN) <JP/US>
         D10766  Osimertinib mesylate (USAN) <JP/US>
         D10514  Dacomitinib (USAN) <JP/US>
         D11980  Lazertinib (USAN)
         D12245  Lazertinib mesilate hydrate (JAN)
         D11969  Mobocertinib succinate (JAN) <US>
         D12258  Aumolertinib (USAN/INN)
         D12259  Aumolertinib mesylate (USAN)
         D11894  Amivantamab (USAN/INN) <US>
         D12506  Sunvozertinib (USAN/INN)
         D12730  Tigozertinib (USAN)
         D12859  Pebezertinib (USAN)
       ERBB2 (HER2, CD340) [HSA:2064] [KO:K05083]
         D09724  Afatinib (USAN/INN)
         D09733  Afatinib dimaleate (USAN) <JP/US>
         D09883  Dacomitinib (INN)
         D10514  Dacomitinib (USAN) <JP/US>
         D08108  Lapatinib (INN)
         D08950  Neratinib (USAN/INN)
         D11375  Trastuzumab duocarmazine (USAN/INN)
         D03350  Canertinib dihydrochloride (USAN)
         D04025  Mubritinib (USAN/INN)
         D06610  Lapuleucel-T (USAN)
         D09689  Varlitinib (USAN/INN)
         D09690  Varlitinib tosylate (USAN)
         D10344  Nelipepimut-S (USAN)
         D11772  Tesevatinib (USAN/INN)
         D11773  Tesevatinib tosylate (USAN)
         D11991  Zenocutuzumab (USAN/INN)
         D12011  Zanidatamab (USAN/INN)
         D12229  Poziotinib (USAN/INN)
         D12230  Poziotinib hydrochloride (USAN)
         D12236  Runimotamab (USAN/INN)
         D12457  Tuxobertinib (USAN/INN)
         D12583  Anvatabart opadotin (USAN/INN)
         D12584  Anvatabart pactil (USAN/INN)
       ERBB2* (HER2, CD340) [HSA_VAR:2064v1] [HSA:2064] [KO:K05083]
       ERBB2* (HER2, CD340) [HSA_VAR:2064v1 2064v3] [HSA:2064] [KO:K05083]
       ERBB3 (HER3) [HSA:2065] [KO:K05084]
       ERBB4 (HER4) [HSA:2066] [KO:K05085]
         D09724  Afatinib (USAN/INN)
         D09733  Afatinib dimaleate (USAN) <JP/US>
         D09883  Dacomitinib (INN)
         D10514  Dacomitinib (USAN) <JP/US>
         D08950  Neratinib (USAN/INN)
         D10898  Neratinib maleate <US>
         D03350  Canertinib dihydrochloride (USAN)
         D09689  Varlitinib (USAN/INN)
         D09690  Varlitinib tosylate (USAN)
     INSR family
     PDGFR family
     FGFR family
     VEGFR family
     MET family
     TRK family
     EPH family
     AXL family
     ALK family
     TIE family
     ROR family
     RET family
     CCK family
   Non-receptor tyrosine kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 18, 2024

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