Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
   Serine/threonine kinases
   Receptor serine/threonine kinases (RSTK)
   Receptor tyrosine kinases (RTK)
     EGFR family
       EGFR [HSA:1956] [KO:K04361]
         D07907  Erlotinib (INN)
         D09724  Afatinib (USAN/INN)
         D10858  Rociletinib (USAN/INN)
         D10859  Olmutinib (USAN/INN)
         D11115  Olmutinib hydrochloride (USAN)
         D09883  Dacomitinib (INN)
         D11251  Icotinib
         D12001  Mobocertinib (USAN/INN)
         D08108  Lapatinib (INN)
         D04024  Lapatinib ditosylate (USAN) <JP/US>
         D08950  Neratinib (USAN/INN)
         D10898  Neratinib maleate <US>
         D06407  Vandetanib (JAN/USAN/INN) <JP/US>
         D03455  Cetuximab (USAN/INN) <JP/US>
         D05350  Panitumumab (USAN/INN) <JP/US>
         D10018  Necitumumab (USAN/INN) <JP/US>
         D11894  Amivantamab (USAN/INN) <US>
         D04862  Masoprocol (USAN/INN)
         D03350  Canertinib dihydrochloride (USAN)
         D05399  Pelitinib (USAN/INN)
         D09660  Rindopepimut (USAN)
         D09689  Varlitinib (USAN/INN)
         D09690  Varlitinib tosylate (USAN)
         D10031  Zalutumumab (USAN/INN)
         D10439  Imgatuzumab (USAN/INN)
         D10886  Naquotinib mesylate (USAN)
         D10958  Naquotinib (USAN/INN)
         D11125  Modotuximab (USAN/INN)
         D11368  Mavelertinib (USAN/INN)
         D11410  Lifirafenib (USAN/INN)
         D11411  Lifirafenib maleate (USAN)
         D11430  Nazartinib (USAN/INN)
         D11434  Nazartinib mesylate (USAN)
         D11750  Duligotuzumab (USAN)
         D11772  Tesevatinib (USAN/INN)
         D11773  Tesevatinib tosylate (USAN)
         D11803  Cetuximab sarotalocan (USAN/INN)
         D11805  Cetuximab sarotalocan sodium (genetical recombination) (JAN) <JP>
         D11872  Serclutamab (USAN/INN)
         D11874  Serclutamab talirine (USAN/INN)
         D12229  Poziotinib (USAN/INN)
         D12230  Poziotinib hydrochloride (USAN)
         D12416  Petosemtamab (USAN/INN)
         D12457  Tuxobertinib (USAN/INN)
         D12709  Dalmitamig (USAN)
         D12768  Ficerafusp alfa (USAN)
         D12809  Bafisontamab (USAN/INN)
       EGFR* [HSA_VAR:1956v2] [HSA:1956] [KO:K04361]
       ERBB2 (HER2, CD340) [HSA:2064] [KO:K05083]
         D09724  Afatinib (USAN/INN)
         D09733  Afatinib dimaleate (USAN) <JP/US>
         D09883  Dacomitinib (INN)
         D10514  Dacomitinib (USAN) <JP/US>
         D08108  Lapatinib (INN)
         D08950  Neratinib (USAN/INN)
         D11375  Trastuzumab duocarmazine (USAN/INN)
         D03350  Canertinib dihydrochloride (USAN)
         D04025  Mubritinib (USAN/INN)
         D06610  Lapuleucel-T (USAN)
         D09689  Varlitinib (USAN/INN)
         D09690  Varlitinib tosylate (USAN)
         D10344  Nelipepimut-S (USAN)
         D11772  Tesevatinib (USAN/INN)
         D11773  Tesevatinib tosylate (USAN)
         D11991  Zenocutuzumab (USAN/INN)
         D12011  Zanidatamab (USAN/INN)
         D12229  Poziotinib (USAN/INN)
         D12230  Poziotinib hydrochloride (USAN)
         D12236  Runimotamab (USAN/INN)
         D12457  Tuxobertinib (USAN/INN)
         D12583  Anvatabart opadotin (USAN/INN)
         D12584  Anvatabart pactil (USAN/INN)
         D12879  Zongertinib (USAN/INN)
       ERBB2* (HER2, CD340) [HSA_VAR:2064v1] [HSA:2064] [KO:K05083]
       ERBB2* (HER2, CD340) [HSA_VAR:2064v1 2064v3] [HSA:2064] [KO:K05083]
       ERBB3 (HER3) [HSA:2065] [KO:K05084]
       ERBB4 (HER4) [HSA:2066] [KO:K05085]
         D09724  Afatinib (USAN/INN)
         D09733  Afatinib dimaleate (USAN) <JP/US>
         D09883  Dacomitinib (INN)
         D10514  Dacomitinib (USAN) <JP/US>
         D08950  Neratinib (USAN/INN)
         D10898  Neratinib maleate <US>
         D03350  Canertinib dihydrochloride (USAN)
         D09689  Varlitinib (USAN/INN)
         D09690  Varlitinib tosylate (USAN)
     INSR family
     PDGFR family
     FGFR family
     VEGFR family
     MET family
     TRK family
     EPH family
     AXL family
     ALK family
     TIE family
     ROR family
     RET family
     CCK family
   Non-receptor tyrosine kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 25, 2024

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