KEGG   DGROUP: CYP3A4 substrate
Entry
DG02913                     DGroup                                 
Name
CYP3A4 substrate
Type
Metabolism
Member
Dexamethasone
 D00292  
Dexamethasone (JP18/USP/INN)  <JP/US>
 D00975  
Dexamethasone sodium phosphate (JAN/USP)  <JP/US>
 D01510  
Dexamethasone metasulfobenzoate sodium (JAN)  <JP>
 D01615  
Dexamethasone palmitate (JAN)  <JP>
 D01632  
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN)  <JP>
 D01948  
Dexamethasone valerate (JAN)  <JP>
 D02174  
Dexamethasone acetate (JAN/USP)
 D02591  
Dexamethasone acefurate (USAN/INN)
 D02592  
Dexamethasone beloxil (USAN)
 D07073  
Dexamethasone cipecilate (JAN/INN)  <JP>
 D07796  
Dexamethasone 21-acetate
 D07797  
Dexamethasone isonicotinate
 D07798  
Dexamethasone sodium hemisulfate
 D07799  
Dexamethasone 21-tebutate
 D07800  
Dexamethasone 21-valerate
 D07801  
Dexamethasone phenylpropionate
 D07802  
Dexamethasone phosphate
D01131  
Lafutidine (JP18/INN)  <JP>
Omeprazole
 D00455  
Omeprazole (JP18/USP/INN)  <JP/US>
 D01207  
Omeprazole sodium (USAN)
 D05261  
Omeprazole sodium injection (JAN)  <JP>
 D05259  
Omeprazole magnesium (USP)  <US>
Pantoprazole
 D05353  
Pantoprazole (USAN/INN)
 D02593  
Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN)  <US>
D00355  
Lansoprazole (JP18/USP/INN)  <JP/US>
Rabeprazole
 D08463  
Rabeprazole (INN)
 D00724  
Rabeprazole sodium (JP18/USP)  <JP/US>
Esomeprazole
 D07917  
Esomeprazole (INN)
 D01984  
Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN)  <JP/US>
 D04056  
Esomeprazole sodium (USAN)  <US>
 D09339  
Esomeprazole potassium (USAN)
 D10120  
Esomeprazole strontium (USAN)  <US>
 D11114  
Esomeprazole magnesium dihydrate  <US>
D08903  
Dexlansoprazole (INN/USAN)  <US>
Vonoprazan
 D11784  
Vonoprazan (USAN/INN)
 D10466  
Vonoprazan fumarate (JAN/USAN)  <JP>
D09742  
Lansoprazole, amoxicillin hydrate and metronidazole
D10246  
Omeprazole, clarithromycin and amoxicillin  <US>
D08774  
Amoxicillin hydrate, clarithromycin and lansoprazole  <US>
D10519  
Rabeprazole, amoxicillin and clarithromycin  <JP>
D10520  
Rabeprazole, amoxicillin and metronidazole  <JP>
D10775  
Vonoprazan, amoxicillin and clarithromycin  <JP/US>
D10774  
Vonoprazan, amoxicillin and metronidazole  <JP>
D01121  
Rebamipide (JP18/INN)  <JP>
Alosetron
 D07129  
Alosetron (INN)
 D02829  
Alosetron hydrochloride (USAN)  <US>
Domperidone
 D01745  
Domperidone (JP18/USAN/INN)  <JP>
 D07868  
Domperidone maleate
Mosapride
 D01994  
Mosapride citrate hydrate (JP18)  <JP>
 D08236  
Mosapride (INN)
Ondansetron
 D00456  
Ondansetron (JAN/USP/INN)  <US>
 D00678  
Ondansetron hydrochloride hydrate (JAN/USP)  <JP/US>
Granisetron
 D04370  
Granisetron (JAN/USAN/INN)  <US>
 D00677  
Granisetron hydrochloride (JAN/USP)  <JP/US>
Palonosetron
 D07175  
Palonosetron (INN)
 D05343  
Palonosetron hydrochloride (JAN/USP)  <JP/US>
D10572  
Fosnetupitant and palonosetron hydrochloride  <US>
Aprepitant
 D02968  
Aprepitant (JAN/USP/INN)  <JP/US>
 D10895  
Fosaprepitant (INN)
 D06597  
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN)  <JP/US>
Rolapitant
 D10742  
Rolapitant (USAN/INN)
 D08988  
Rolapitant hydrochloride (USAN)  <US>
Naldemedine
 D10188  
Naldemedine (USAN/INN)
 D10478  
Naldemedine tosylate (JAN/USAN)  <JP/US>
Tenapanor
 D11652  
Tenapanor (USAN/INN)
 D11653  
Tenapanor hydrochloride (JAN/USAN)  <US>
D02554  
Rifaximin (JAN/USAN/INN)  <JP/US>
Loperamide
 D08144  
Loperamide (INN)
 D00729  
Loperamide hydrochloride (JAN/USP)  <JP/US>
 D07113  
Loperamide oxide (INN)
D00246  
Budesonide (JAN/USP/INN)  <JP/US>
D00689  
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18)  <JP/US>
D11572  
Beclomethasone dipropionate monohydrate  <US>
Fenfluramine
 D07945  
Fenfluramine (INN)
 D04148  
Fenfluramine hydrochloride (JAN/USAN)  <US>
D00336  
Glyburide (USP); Glibenclamide (JP18/INN)  <JP/US>
D10263  
Metformin hydrochloride and saxagliptin hydrochloride  <US>
Saxagliptin
 D08996  
Saxagliptin (USAN/INN)
 D09753  
Saxagliptin hydrate (JAN)  <JP>
 D10262  
Saxagliptin hydrochloride  <US>
Teneligliptin
 D08616  
Teneligliptin (INN)
 D09756  
Teneligliptin hydrobromide hydrate (JAN)  <JP>
 D11968  
Teneligliptin hydrobromide (JAN)
D00594  
Repaglinide (JAN/USP/INN)  <JP/US>
Eliglustat
 D09893  
Eliglustat (USAN/INN)
 D09894  
Eliglustat tartrate (JAN/USAN)  <JP/US>
Clopidogrel
 D07729  
Clopidogrel (USP/INN)
 D00769  
Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18)  <JP/US>
 D10823  
Clopidogrel hydrochloride
 D10824  
Clopidogrel besilate
D01896  
Cilostazol (JP18/USP/INN)  <JP/US>
Vorapaxar
 D09765  
Vorapaxar (USAN/INN)
 D09766  
Vorapaxar sulfate (JAN/USAN)  <US>
D09994  
Selexipag (JAN/USAN/INN)  <JP/US>
D10513  
Clopidogrel sulfate and aspirin  <JP>
D10527  
Acetylsalicylic acid and lansoprazole  <JP>
Argatroban
 C04931  
Argatroban
 D00181  
Argatroban (USP); Argatroban hydrate (JP18)  <JP/US>
D07086  
Rivaroxaban (JAN/USAN/INN)  <JP/US>
D03213  
Apixaban (JAN/USAN/INN)  <JP/US>
Avatrombopag
 D10306  
Avatrombopag (USAN/INN)
 D10307  
Avatrombopag maleate (JAN/USAN)  <US>
D11330  
Voxelotor (USAN)  <US>
Disopyramide
 D00303  
Disopyramide (JP18/USAN/INN)  <JP>
 D00637  
Disopyramide phosphate (JAN/USP)  <JP/US>
Lidocaine
 D00358  
Lidocaine (JP18/USP/INN)  <JP/US>
 D02086  
Lidocaine hydrochloride (JAN/USP)  <JP/US>
 D08127  
Lidocaine hydrochloride monohydrate  <JP/US>
Propafenone
 D08435  
Propafenone (INN)
 D00640  
Propafenone hydrochloride (JP18/USP)  <JP/US>
Amiodarone
 D02910  
Amiodarone (USAN/INN)
 D00636  
Amiodarone hydrochloride (JP18/USP)  <JP/US>
Cibenzoline
 D03492  
Cifenline (USAN); Cibenzoline (INN)
 D01455  
Cifenline succinate (USAN); Cibenzoline succinate (JP18)  <JP>
Ivabradine
 D07165  
Ivabradine (USAN/INN)
 D08095  
Ivabradine hydrochloride (JAN/USAN)  <JP/US>
Guanfacine
 D08031  
Guanfacine (INN)
 D00606  
Guanfacine hydrochloride (JAN/USP)  <JP/US>
Bosentan
 D07538  
Bosentan (INN)
 D01227  
Bosentan (USAN); Bosentan hydrate (JAN)  <JP/US>
D10135  
Macitentan (JAN/USAN)  <JP/US>
D01115  
Eplerenone (JP18/USAN/INN)  <JP/US>
D10633  
Finerenone (JAN/USAN/INN)  <JP/US>
D01213  
Tolvaptan (JAN/USAN/INN)  <JP/US>
Diltiazem
 D07845  
Diltiazem (INN)
 D00616  
Diltiazem hydrochloride (JP18/USP)  <JP/US>
 D03830  
Diltiazem malate (USAN)
Carvedilol
 D00255  
Carvedilol (JP18/USP/INN)  <JP/US>
 D03415  
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN)  <US>
Amlodipine
 D07450  
Amlodipine (USP/INN)
 D00615  
Amlodipine besylate (USP); Amlodipine besilate (JP18)  <JP/US>
 D02914  
Amlodipine maleate (USAN)
 D11881  
Amlodipine benzoate  <US>
D00319  
Felodipine (JP18/USP/INN)  <JP/US>
Nicardipine
 D08270  
Nicardipine (INN)
 D00617  
Nicardipine hydrochloride (JP18/USAN)  <JP/US>
D00437  
Nifedipine (JP18/USP/INN)  <JP/US>
D00438  
Nimodipine (USP/INN)  <US>
D00618  
Nisoldipine (JAN/USAN/INN)  <US>
D00629  
Nitrendipine (JP18/USAN/INN)  <JP>
D01908  
Nilvadipine (JP18/USAN/INN)  <JP>
Manidipine
 D08155  
Manidipine (INN)
 D01553  
Manidipine hydrochloride (JP18)  <JP>
Barnidipine
 D07494  
Barnidipine (INN)
 D01104  
Barnidipine hydrochloride (JAN)  <JP>
D01173  
Cilnidipine (JP18/INN)  <JP>
Benidipine
 D07509  
Benidipine (INN)
 D02045  
Benidipine hydrochloride (JP18)  <JP>
Verapamil
 D02356  
Verapamil (USAN/INN)
 D00619  
Verapamil hydrochloride (JP18/USP)  <JP/US>
Bepridil
 D07520  
Bepridil (INN)
 D00631  
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN)  <JP>
D09745  
Valsartan and amlodipine besilate  <JP/US>
D09743  
Telmisartan and amlodipine besilate (JP18)  <JP/US>
D10243  
Irbesartan and amlodipine besilate (JP18)  <JP>
D07569  
Candesartan cilexetil and anmlodipine besylate (JP18)  <JP>
Aliskiren
 D03208  
Aliskiren (USAN/INN)
 D06412  
Aliskiren fumarate (JAN/USAN)  <JP/US>
D00434  
Simvastatin (JP18/USP/INN)  <JP/US>
D00359  
Lovastatin (USP/INN)  <US>
Fluvastatin
 D07983  
Fluvastatin (INN)
 D00892  
Fluvastatin sodium (JAN/USP)  <JP/US>
Atorvastatin
 D07474  
Atorvastatin (INN)
 D00887  
Atorvastatin calcium anhydorous
 D02258  
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18)  <JP/US>
 D11095  
Atorvastatin calcium propylene glycol solvate  <US>
Cerivastatin
 D07661  
Cerivastatin (INN)
 D00889  
Cerivastatin sodium (JAN/USAN)
Lomitapide
 D09637  
Lomitapide (USAN/INN)
 D09638  
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN)  <JP/US>
D10385  
Ezetimibe and atorvastatin  <JP/US>
D08488  
Amlodipine besilate and atorvastatin calcium  <JP/US>
D00351  
Ketoconazole (JP18/USP)  <JP/US>
Terbinafine
 D02375  
Terbinafine (USAN/INN)
 D02219  
Terbinafine hydrochloride (JP18/USP)  <JP/US>
D09544  
Ozenoxacin (JAN/USAN/INN)  <JP/US>
Methylprednisolone
 D00407  
Methylprednisolone (JP18/USP/INN)  <JP/US>
 D00751  
Methylprednisolone sodium succinate (JAN/USP)  <JP/US>
 D00979  
Methylprednisolone acetate (JAN/USP)  <JP/US>
 D05000  
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18)
 D05001  
Methylprednisolone sodium phosphate (USAN)
 D05002  
Methylprednisolone suleptanate (USAN/INN)
 D07203  
Methylprednisolone aceponate (INN)
Mometasone
 D08227  
Mometasone (INN)
 D00690  
Mometasone furoate (JAN/USP)  <JP/US>
 D03325  
Mometasone furoate hydrate (JAN)  <JP>
Fluticasone
 D07981  
Fluticasone (INN)
 D01708  
Fluticasone propionate (JAN/USP)  <JP/US>
 D06315  
Fluticasone furoate (JAN/USAN/INN)  <JP/US>
D00592  
Dapsone (USP); Diaphenylsulfone (JAN)  <JP/US>
Tacrolimus
 D08556  
Tacrolimus (INN)
 D00107  
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18)  <JP/US>
D00321  
Finasteride (JAN/USP/INN)  <JP/US>
D00804  
Ivermectin (JAN/USP/INN)  <JP/US>
Caffeine
 D00528  
Caffeine (USP); Anhydrous caffeine (JP18)  <JP>
 D01453  
Caffeine hydrate (JP18)  <JP>
 D07603  
Caffeine citrate (USP)  <US>
Methylergometrine
 D08207  
Methylergometrine (INN)
 D00680  
Methylergonovine maleate (USP); Methylergometrine maleate (JP18)  <JP/US>
Ergometrine
 D07905  
Ergometrine (INN)
 D01163  
Ergonovine maleate (USP); Ergometrine maleate (JP18)
Bromocriptine
 D03165  
Bromocriptine (USAN/INN)
 D00780  
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18)  <JP/US>
D00987  
Cabergoline (JP18/USP/INN)  <JP/US>
D02577  
Flibanserin (USAN/INN)  <US>
D04463  
Norgestrel and ethinylestradiol tablets (JP18)  <JP/US>
D03917  
Drospirenone (JAN/USP/INN)
Ethinylestradiol
 D00554  
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN)  <JP>
 D07928  
Ethinylestradiol propanesulfonate
Estradiol
 D00105  
Estradiol (JAN/USP/INN)  <JP/US>
 D01413  
Estradiol valerate (JAN/USP/INN)  <JP/US>
 D01617  
Estradiol dipropionate (JAN)
 D01953  
Estradiol benzoate (JP18/USP)
 D04061  
Estradiol acetate (USAN)  <US>
 D04063  
Estradiol cypionate (USP)  <US>
 D04064  
Estradiol enanthate (USAN)
 D04065  
Estradiol undecylate (USAN/INN)
 D07918  
Estradiol hemihydrate  <US>
 D07919  
Estradiol 17 beta-hemisuccinate
Estrone
 D00067  
Estrone (JAN/USP/INN)
 D00312  
Estrone sodium sulfate
 D00948  
Estropipate (USP)
Conjugated estrogen
 D04070  
Estrogens, conjugated (JAN/USP)  <JP/US>
 D05987  
Synthetic conjugated estrogens, B (USAN)
D00066  
Progesterone (JP18/USP/INN)  <JP/US>
D01217  
Dydrogesterone (JP18/USP/INN)  <JP>
D03799  
Dienogest (JAN/USAN/INN)  <JP>
D09188  
Estradiol and norethindrone  <JP/US>
D09187  
Estradiol and levonorgestrel  <JP/US>
D09741  
Drospirenone and ethinylestradiol  <JP/US>
D00585  
Mifepristone (JAN/USAN/INN)  <US>
Oxybutynin
 D00465  
Oxybutynin (USAN/INN)  <US>
 D00722  
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JAN)  <JP/US>
Propiverine
 D08441  
Propiverine (INN)
 D01007  
Propiverine hydrochloride (JP18)  <JP>
Tolterodine
 D00646  
Tolterodine (USAN/INN)
 D01148  
Tolterodine tartrate (JAN/USP)  <JP/US>
Solifenacin
 D08522  
Solifenacin (INN)
 D01269  
Solifenacin succinate (JAN/USAN/INN)  <JP/US>
Darifenacin
 D03654  
Darifenacin (USAN/INN)
 D01699  
Darifenacin hydrobromide (JAN/USAN)  <US>
Fesoterodine
 D07226  
Fesoterodine (INN)
 D08923  
Fesoterodine fumarate (JAN/USAN)  <JP/US>
D09535  
Mirabegron (USAN/JAN)  <JP/US>
Sildenafil
 D08514  
Sildenafil (INN)
 D02229  
Sildenafil citrate (JAN/USP)  <JP/US>
D02008  
Tadalafil (JAN/USP/INN)  <JP/US>
Vardenafil
 D08668  
Vardenafil (USAN/INN)
 D02731  
Vardenafil dihydrochoride (USAN)
 D03260  
Vardenafil hydrochloride hydrate (JAN)  <JP/US>
 D09989  
Vardenafil hydrochloride (USP)
D03217  
Avanafil (USAN/INN)  <US>
Alfuzosin
 D07124  
Alfuzosin (INN)
 D01692  
Alfuzosin hydrochloride (JAN/USAN)  <US>
D01965  
Silodosin (JP18/INN)  <JP/US>
D11389  
Dutasteride and tamsulosin  <US>
D03820  
Dutasteride (JAN/USP/INN)  <JP/US>
D03671  
Deflazacort (USAN/INN)  <US>
Osilodrostat
 D11061  
Osilodrostat (USAN/INN)
 D11062  
Osilodrostat phosphate (JAN/USAN)  <JP/US>
Cinacalcet
 D03504  
Cinacalcet (USAN)
 D03505  
Cinacalcet hydrochloride (JAN/USAN)  <JP/US>
D01322  
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN)
Clarithromycin
 D00276  
Clarithromycin (JP18/USP/INN)  <JP/US>
 D07710  
Clarithromycin lactobionate
Ofloxacin
 D00453  
Ofloxacin (JP18/USP/INN)  <JP/US>
 D08291  
Ofloxacin hydrochloride
Lefamulin
 D11631  
Lefamulin (USAN/INN)
 D11632  
Lefamulin acetate (USAN)  <US>
D00350  
Itraconazole (JP18/USP)  <JP/US>
D00424  
Rifabutin (JAN/USP/INN)  <JP/US>
Bedaquiline
 D09872  
Bedaquiline (USAN/INN)
 D09873  
Bedaquiline fumarate (JAN/USAN)  <JP/US>
D09785  
Delamanid (JAN/USAN)  <JP>
Saquinavir
 D00429  
Saquinavir (JAN/USP/INN)
 D01160  
Saquinavir mesylate (USP); Saquinavir mesilate (JAN)  <US>
Indinavir
 C07051  
Indinavir
 D03833  
Indinavir (USAN)
 D00897  
Indinavir sulfate (USP)  <US>
 D02861  
Indinavir sulfate ethanolate (JAN)
Nelfinavir
 D08259  
Nelfinavir (INN)
 D00899  
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN)  <US>
D00894  
Amprenavir (JAN/USAN/INN)
Fosamprenavir
 D02497  
Fosamprenavir (INN)
 D02867  
Fosamprenavir calcium hydrate (JAN)  <JP>
 D03835  
Fosamprenavir calcium (USAN)  <US>
 D03837  
Fosamprenavir sodium (USAN)
Darunavir
 D03656  
Darunavir (USAN/INN)
 D06478  
Darunavir ethanolate (JAN)  <JP/US>
D00435  
Nevirapine (JAN/USP/INN)  <JP/US>
D00896  
Efavirenz (JAN/USP/INN)  <JP/US>
D04112  
Etravirine (JAN/USAN/INN)  <JP/US>
Dolutegravir
 D10066  
Dolutegravir (USAN)
 D10113  
Dolutegravir sodium (JAN/USAN)  <JP/US>
D09012  
Telaprevir (JAN/USAN/INN)
Daclatasvir
 D10065  
Daclatasvir (USAN)
 D10105  
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN)
D10745  
Ombitasvir, paritaprevir and ritonavir
D10827  
Sofosbuvir and velpatasvir  <JP/US>
D10600  
Dolutegravir, abacavir and lamivudine  <JP/US>
D10753  
Atazanavir and cobicistat  <US>
D06670  
Maraviroc (JAN/INN)  <JP/US>
D04859  
Maribavir (JAN/USAN/INN)  <US>
Cyclophosphamide
 D07760  
Cyclophosphamide (INN)
 D00287  
Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18)  <JP/US>
D00343  
Ifosfamide (JAN/USP/INN)  <JP/US>
Vinblastine
 D08675  
Vinblastine (INN)
 D01068  
Vinblastine sulfate (JP18/USP)  <JP/US>
Vinorelbine
 D08680  
Vinorelbine (INN)
 D01935  
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN)  <JP/US>
Paclitaxel
 D00491  
Paclitaxel (JAN/USP/INN)  <JP/US>
 D05333  
Paclitaxel poliglumex (USAN/INN)
Docetaxel
 D07866  
Docetaxel (JAN/INN)  <JP/US>
 D02165  
Docetaxel (USP); Docetaxel hydrate (JP18)  <JP/US>
Irinotecan
 D08086  
Irinotecan (INN)
 D01061  
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18)  <JP/US>
 D10642  
Irinotecan sucrosofate (USAN)
D06199  
Trabectedin (JAN/USAN/INN)  <JP/US>
D04645  
Ixabepilone (JAN/USAN/INN)  <US>
Imatinib
 D08066  
Imatinib (INN)
 D01441  
Imatinib mesylate (USAN); Imatinib mesilate (JAN)  <JP/US>
Dasatinib
 D03658  
Dasatinib (JAN/INN)  <JP>
 D06414  
Dasatinib (USAN); Dasatinib hydrate (JAN)  <JP/US>
Nilotinib
 D08953  
Nilotinib (USAN/INN)
 D06413  
Nilotinib hydrochloride hydrate (JAN)  <JP/US>
Bosutinib
 D03252  
Bosutinib (USAN)
 D09728  
Bosutinib hydrate (JAN)  <JP/US>
Asciminib
 D11403  
Asciminib (USAN/INN)
 D11404  
Asciminib hydrochloride (JAN/USAN)  <JP/US>
Erlotinib
 D07907  
Erlotinib (INN)
 D04023  
Erlotinib hydrochloride (JAN/USAN)  <JP/US>
Dabrafenib
 D10064  
Dabrafenib (USAN)
 D10104  
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN)  <JP/US>
D11053  
Encorafenib (JAN/USAN/INN)  <JP/US>
D09731  
Crizotinib (JAN/USAN/INN)  <JP/US>
Alectinib
 D10542  
Alectinib (USAN/INN)
 D10450  
Alectinib hydrochloride (JAN)  <JP/US>
D10866  
Brigatinib (JAN/USAN)  <JP/US>
Selumetinib
 D09666  
Selumetinib (USAN/INN)
 D10024  
Selumetinib sulfate (JAN/USAN)  <US>
Ribociclib
 D10883  
Ribociclib (USAN/INN)
 D10979  
Ribociclib succinate (USAN)  <US>
D06068  
Temsirolimus (JAN/USAN/INN)  <JP/US>
D02714  
Everolimus (JAN/USAN/INN)  <JP/US>
Lapatinib
 D08108  
Lapatinib (INN)
 D04024  
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN)  <JP/US>
Ruxolitinib
 D09959  
Ruxolitinib (USAN/INN)
 D09960  
Ruxolitinib phosphate (JAN/USAN)  <JP/US>
Fedratinib
 D10630  
Fedratinib (USAN/INN)
 D11296  
Fedratinib hydrochloride (USAN)  <US>
D11768  
Pacritinib (USAN/INN)  <US>
D03218  
Axitinib (JAN/USAN)  <JP/US>
Tivozanib
 D09683  
Tivozanib (USAN/INN)
 D10190  
Tivozanib hydrochloride (USAN)  <US>
D10927  
Erdafitinib (JAN/USAN/INN)  <US>
D11417  
Pemigatinib (JAN/USAN/INN)  <JP/US>
Sunitinib
 D08552  
Sunitinib (INN)
 D06402  
Sunitinib malate (JAN/USAN)  <JP/US>
D06407  
Vandetanib (JAN/USAN/INN)  <JP/US>
Regorafenib
 D10138  
Regorafenib (USAN/INN)
 D10137  
Regorafenib hydrate (JAN)  <JP/US>
D05029  
Midostaurin (JAN/USAN/INN)  <US>
Gilteritinib
 D10709  
Gilteritinib (USAN/INN)
 D10800  
Gilteritinib fumarate (JAN/USAN)  <JP/US>
D10926  
Entrectinib (JAN/USAN/INN)  <JP/US>
Pexidartinib
 D11270  
Pexidartinib (USAN/INN)
 D11271  
Pexidartinib hydrochloride (JAN/USAN)  <US>
Capmatinib
 D10696  
Capmatinib (USAN/INN)
 D10891  
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN)  <JP/US>
Tepotinib
 D11717  
Tepotinib (USAN/INN)
 D11073  
Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN)  <JP/US>
D11713  
Selpercatinib (JAN/USAN/INN)  <JP/US>
D03259  
Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN)  <JP/US>
Panobinostat
 D10319  
Panobinostat (USAN/INN)
 D10019  
Panobinostat lactate (JAN)  <JP/US>
D08870  
Belinostat (USAN/INN)  <US>
D08914  
Eribulin mesylate (USAN); Eribulin mesilate (JAN)  <JP/US>
D11222  
Selinexor (USAN/INN)  <US>
D11954  
Belzutifan (JAN/USAN/INN)  <US>
Tamoxifen
 D08559  
Tamoxifen (INN)
 D00966  
Tamoxifen citrate (JP18/USP)  <JP/US>
Toremifene
 D08620  
Toremifene (INN)
 D00967  
Toremifene citrate (JAN/USAN)  <JP/US>
D01161  
Fulvestrant (JAN/USP/INN)  <JP/US>
D10218  
Enzalutamide (JAN/USAN)  <JP/US>
D11040  
Apalutamide (JAN/INN)  <JP/US>
D00964  
Letrozole (JAN/USP/INN)  <JP/US>
D00963  
Exemestane (JAN/USP/INN)  <JP/US>
D09701  
Abiraterone acetate (JAN/USP)  <JP/US>
D00753  
Sirolimus (JAN/USAN/INN)  <JP/US>
D00749  
Leflunomide (JAN/USP/INN)  <JP/US>
Tofacitinib
 D09970  
Tofacitinib (USAN)
 D09783  
Tofacitinib citrate (JAN/USAN)  <JP/US>
Siponimod
 D11460  
Siponimod (USAN/INN)
 D11072  
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN)  <JP/US>
Upadacitinib
 D10994  
Upadacitinib (USAN/INN)  <US>
 D10995  
Upadacitinib tartrate (USAN)
 D11048  
Upadacitinib hydrate (JAN)  <JP>
D00184  
Cyclosporine (USP); Ciclosporin (JP18)  <JP/US>
D09033  
Voclosporin (JAN/USAN/INN)  <US>
D08976  
Pomalidomide (JAN/USAN/INN)  <JP/US>
D00969  
Meloxicam (JAN/USP/INN)  <JP/US>
D11576  
Naproxen and esomeprazole magnesium  <US>
D00570  
Colchicine (JP18/USP)  <JP/US>
D11406  
Risdiplam (JAN/USAN/INN)  <JP/US>
D00542  
Halothane (JP18/USP/INN)
Fentanyl
 D00320  
Fentanyl (JAN/USP/INN)  <JP/US>
 D01399  
Fentanyl citrate (JP18/USP)  <JP/US>
 D10811  
Fentanyl hydrochloride (JAN)
D03852  
Droperidol and fentanyl citrate
Esketamine
 D07283  
Esketamine (USAN/INN)
 D10627  
Esketamine hydrochloride (JAN/USAN)  <US>
Bupivacaine
 D07552  
Bupivacaine (USAN/INN)  <US>
 D01450  
Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18)  <JP/US>
Ropivacaine
 D08490  
Ropivacaine (INN)
 D04048  
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN)  <JP/US>
Levobupivacaine
 D08116  
Levobupivacaine (INN)
 D01287  
Levobupivacaine hydrochloride (JAN/USAN)  <JP>
D02740  
Lidocaine and prilocaine  <JP/US>
Oxycodone
 D05312  
Oxycodone (USAN/INN)
 D00847  
Oxycodone hydrochloride (USP)  <US>
 D02175  
Compound oxycodone (JP18)
 D03783  
Oxycodone terephthalate (USP)
 D05462  
Oxycodone hydrochloride hydrate (JP18)  <JP>
Dihydrocodeine
 D07831  
Dihydrocodeine (INN)
 D01481  
Dihydrocodeine phosphate (JP18)  <JP>
 D03825  
Dihydrocodeine bitartrate (USP)
 D07832  
Dihydrocodeine thiocyanate
D08695  
dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea  <JP>
Buprenorphine
 D07132  
Buprenorphine (JAN/INN)  <JP/US>
 D00836  
Buprenorphine hydrochloride (JP18/USP)  <JP/US>
D09999  
Tramadol hydrochloride and acetaminophen  <JP/US>
D11573  
Oxycodone and ibuprofen
Tramadol
 D08623  
Tramadol (INN)
 D01355  
Tramadol hydrochloride (JP18/USP)  <JP/US>
D00544  
Methoxyflurane (USP/INN)
Dihydroergotamine
 D07837  
Dihydroergotamine (INN)
 D02211  
Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18)  <US>
 D07838  
Dihydroergotamine tartrate
Ergotamine
 D07906  
Ergotamine (INN)
 D00679  
Ergotamine tartrate (JP18/USP)  <US>
D07585  
Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine  <JP>
Naratriptan
 D08255  
Naratriptan (INN)
 D00674  
Naratriptan hydrochloride (JAN/USP)  <JP/US>
Almotriptan
 D02824  
Almotriptan (USAN)
 D02825  
Almotriptan malate (USP)  <US>
Eletriptan
 D07887  
Eletriptan (INN)
 D01973  
Eletriptan hydrobromide (JAN/USAN)  <JP/US>
 D11617  
Eletriptan hydrobromide monohydrate  <US>
D10673  
Ubrogepant (USAN/INN)  <US>
Rimegepant
 D10662  
Rimegepant (USAN/INN)
 D10663  
Rimegepant sulfate (USAN)  <US>
D11313  
Atogepant (USAN)  <US>
D00539  
Ethosuximide (JP18/USP/INN)  <JP/US>
D00252  
Carbamazepine (JP18/USP/INN)  <JP/US>
D00537  
Topiramate (JAN/USP/INN)  <JP/US>
D05928  
Stiripentol (JAN/USAN/INN)  <JP/US>
D07299  
Lacosamide (JAN/USAN/INN)  <JP/US>
D10915  
Cannabidiol (USAN/INN)  <US>
D11150  
Cenobamate (USAN/INN)  <US>
D04300  
Ganaxolone (USAN/INN)  <US>
Selegiline
 D03731  
Selegiline (USAN/INN)  <US>
 D00785  
Selegiline hydrochloride (JAN/USP)  <JP/US>
Safinamide
 D10158  
Safinamide (USAN/INN)
 D10191  
Safinamide mesylate (USAN); Safinamide mesilate (JAN)  <JP/US>
D04641  
Istradefylline (JAN/USAN/INN)  <JP/US>
Haloperidol
 D00136  
Haloperidol (JP18/USP/INN)  <JP/US>
 D01898  
Haloperidol decanoate (JAN/USP)  <JP/US>
 D08035  
Haloperidol lactate  <US>
Bromperidol
 D01101  
Bromperidol (JAN/USAN/INN)  <JP>
 D02626  
Bromperidol decanoate (USAN)
D04820  
Lurasidone hydrochloride (JAN/USAN)  <JP/US>
D00560  
Pimozide (JP18/USP/INN)  <US>
Loxapine
 D02340  
Loxapine (USAN/INN)  <US>
 D00794  
Loxapine succinate (USP)  <US>
 D08148  
Loxapine hydrochloride
D00283  
Clozapine (JAN/USP/INN)  <JP/US>
Quetiapine
 D08456  
Quetiapine (INN)
 D00458  
Quetiapine fumarate (JP18/USP)  <JP/US>
D00426  
Risperidone (JP18/USP/INN)  <JP/US>
Aripiprazole
 D01164  
Aripiprazole (JAN/USP/INN)  <JP/US>
 D10355  
Aripiprazole cavoxil (USAN)
 D10364  
Aripiprazole lauroxil (USAN)  <US>
 D10516  
Aripiprazole hydrate (JAN)  <JP/US>
D02666  
Iloperidone (USAN/INN)  <US>
Cariprazine
 D09997  
Cariprazine (USAN/INN)
 D09876  
Cariprazine hydrochloride (JAN/USAN)  <US>
D10309  
Brexpiprazole (JAN/USAN/INN)  <JP/US>
D08969  
Pimavanserin tartrate (USAN)  <US>
D00293  
Diazepam (JP18/USP/INN)  <JP/US>
D01253  
Clobazam (JAN/USAN/INN)  <JP/US>
D08283  
Nordazepam (INN)
D01293  
Ethyl loflazepate (JP18/INN)  <JP>
D01514  
Etizolam (JP18/INN)  <JP>
D01316  
Mexazolam (JAN/INN)  <JP>
D00387  
Triazolam (JP18/USP/INN)  <JP/US>
Midazolam
 D00550  
Midazolam (JAN/USP/INN)  <JP/US>
 D00696  
Midazolam hydrochloride (USAN)  <US>
 D05028  
Midazolam maleate (USAN)
D01744  
Brotizolam (JP18/USAN/INN)  <JP>
D00457  
Quazepam (JAN/USP/INN)  <JP/US>
D01372  
Zopiclone (JP18/INN)  <JP>
Zolpidem
 D08690  
Zolpidem (INN)
 D00706  
Zolpidem tartrate (JP18/USP)  <JP/US>
D00530  
Zaleplon (JAN/USP/INN)  <US>
D02624  
Eszopiclone (JAN/USP/INN)  <JP/US>
D09388  
Tasimelteon (USAN/INN)  <US>
D11022  
Lemborexant (JAN/USAN/INN)  <JP/US>
Imipramine
 D08070  
Imipramine (INN)
 D00815  
Imipramine hydrochloride (JP18/USP)  <JP/US>
 D08071  
Imipramine pamoate (USP)  <US>
Clomipramine
 D07727  
Clomipramine (INN)
 D00811  
Clomipramine hydrochloride (JP18/USP)  <JP/US>
Amitriptyline
 D07448  
Amitriptyline (INN)
 D00809  
Amitriptyline hydrochloride (JP18/USP)  <JP/US>
Citalopram
 D07704  
Citalopram (USP/INN)
 D00822  
Citalopram hydrobromide (USP)  <US>
 D07705  
Citalopram hydrochloride
Sertraline
 D02360  
Sertraline (INN)
 D00825  
Sertraline hydrochloride (JAN/USP)  <JP/US>
Escitalopram
 D07913  
Escitalopram (INN)
 D02567  
Escitalopram oxalate (JAN/USP)  <JP/US>
Mianserin
 D08216  
Mianserin (INN)
 D01358  
Mianserin hydrochloride (JAN/USAN)  <JP>
Trazodone
 D08626  
Trazodone (INN)
 D00820  
Trazodone hydrochloride (JAN/USP)  <JP/US>
Mirtazapine
 D00563  
Mirtazapine (JAN/USP/INN)  <JP/US>
 D11056  
Mirtazapine hydrate (JAN)
Venlafaxine
 D08670  
Venlafaxine (INN)
 D00821  
Venlafaxine hydrochloride (JAN/USP)  <JP/US>
 D12403  
Venlafaxine besylate monohydrate  <US>
Desvenlafaxine
 D07793  
Desvenlafaxine (INN)  <US>
 D02570  
Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN)  <US>
 D11619  
Desvenlafaxine succinate anhydrous  <US>
Vilazodone
 D09698  
Vilazodone (USAN/INN)
 D09699  
Vilazodone hydrochloride (USAN)  <US>
Vortioxetine
 D10184  
Vortioxetine (USAN)
 D10185  
Vortioxetine hydrobromide (JAN/USAN)  <JP/US>
D01832  
Modafinil (JAN/USP/INN)  <JP/US>
D03215  
Armodafinil (USAN/INN)  <US>
Donepezil
 D07869  
Donepezil (JAN/INN)
 D00670  
Donepezil hydrochloride (JP18/USP)  <JP/US>
Galantamine
 D04292  
Galantamine (USAN/INN)
 D02173  
Galantamine hydrobromide (JAN/USP)  <JP/US>
Cevimeline
 D07667  
Cevimeline (INN)
 D00661  
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN)  <JP/US>
Methadone
 D08195  
Methadone (BAN)
 D02102  
Methadone hydrochloride (JAN/USP)  <JP/US>
Levacetylmethadol
 D04716  
Levomethadyl acetate (USAN); Levacetylmethadol (INN)
 D00840  
Levomethadyl acetate hydrochloride (USAN)
D08575  
Tetrabenazine (JAN/INN)  <JP/US>
Pitolisant
 D10749  
Pitolisant (USAN/INN)
 D11490  
Pitolisant hydrochloride (USAN)  <US>
Valbenazine
 D10675  
Valbenazine (USAN/INN)
 D10999  
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN)  <JP/US>
Hydroxychloroquine
 D08050  
Hydroxychloroquine (INN)
 D02114  
Hydroxychloroquine sulfate (JAN/USP)  <JP/US>
Quinine
 D08460  
Quinine (BAN)
 D01663  
Quinine ethylcarbonate (JP18)
 D02261  
Quinine hydrochloride hydrate (JP18)
 D02262  
Quinine sulfate (USP); Quinine sulfate hydrate (JP18)  <US>
 D05681  
Quinine ascorbate (USAN)
 D08461  
Quinine dihydrochloride
D11252  
Fexinidazole (USAN/INN)  <US>
D00471  
Praziquantel (JAN/USP/INN)  <JP/US>
Flunisolide
 C07005  
Flunisolide
 D00324  
Flunisolide (JAN/USP)  <US>
 D04214  
Flunisolide acetate (USAN)
D01703  
Ciclesonide (JAN/USAN/INN)  <JP/US>
D08699  
Salmeterol xinafoate and fluticasone propionate  <JP/US>
Salmeterol
 D05792  
Salmeterol (USAN/INN)
 D00687  
Salmeterol xinafoate (JAN/USP)  <JP/US>
Procaterol
 D08424  
Procaterol (INN)
 D02404  
Procaterol hydrochloride (USAN)
 D05366  
Procaterol hydrochloride hydrate (JP18)  <JP>
Indacaterol
 D09318  
Indacaterol (USAN/INN)
 D09319  
Indacaterol maleate (JAN/USAN)  <JP>
 D11009  
Indacaterol acetate (JAN)
D09595  
Budesonide and formoterol fumarate dihydrate  <JP/US>
D10501  
Fluticasone furoate and vilanterol trifenatate  <JP/US>
D10506  
Fluticasone propionate and formoterol fumarate hydrate  <JP>
D10533  
Umeclidinium bromide and vilanterol  <JP/US>
D10505  
Glycopyrronium bromide and indacaterol maleate  <JP>
Pranlukast
 D08408  
Pranlukast (INN)
 D02732  
Pranlukast hydrate (JP18)  <JP>
Montelukast
 D08229  
Montelukast (INN)
 D00529  
Montelukast sodium (JP18/USP)  <JP/US>
D05744  
Roflumilast (JAN/USAN/INN)  <US>
Ethylmorphine
 D07929  
Ethylmorphine (BAN)
 D02205  
Ethylmorphine hydrochloride hydrate (JP18)
Hydrocodone
 D08045  
Hydrocodone (INN)
 D03725  
Hydrocodone bitartrate (USP)  <US>
 D04461  
Hydrocodone polistirex (USAN)
 D08046  
Hydrocodone hydrochloride
Codeine
 C06174  
Codeine
 D00195  
Codeine (USP)
 D02101  
Codeine phosphate (USP); Codeine phosphate hydrate (JP18)  <JP>
 D03579  
Codeine polistirex (USAN)
 D03580  
Codeine sulfate (USP)  <US>
 D07740  
Codeine hydrochloride
D04340  
Dextromethorphan hydrobromide and potassium cresolsulfonate  <JP>
D04447  
Betamethasone and d-chlorpheniramine maleate  <JP>
D04313  
Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate  <JP>
Levocetirizine
 D07402  
Levocetirizine (USAN/INN)
 D08118  
Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN)  <JP/US>
D00364  
Loratadine (JAN/USP/INN)  <JP/US>
D01478  
Ebastine (JP18/USAN/INN)  <JP>
Rupatadine
 D07407  
Rupatadine (INN)
 D08497  
Rupatadine fumarate (JAN)  <JP>
Doxapram
 D07873  
Doxapram (INN)
 D01872  
Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18)  <JP/US>
Dorzolamide
 D07871  
Dorzolamide (INN)
 D00653  
Dorzolamide hydrochloride (JP18/USP)  <JP/US>
D10512  
Brinzolamide and timolol maleate  <JP>
D08493  
Dorzolamide hydrochloride and timolol maleate (JP18)  <JP/US>
D06405  
Nalfurafine hydrochloride (JAN/USAN)  <JP>
Rilmazafone
 D08481  
Rilmazafone (INN)
 D01564  
Rilmazafone hydrochloride hydrate (JP18)  <JP>
Sarpogrelate
 D08508  
Sarpogrelate (INN)
 D01624  
Sarpogrelate hydrochloride (JP18)  <JP>
D01098  
Maxacalcitol (JAN/USAN/INN)  <JP>
D01145  
Azelnidipine (JP18/INN)  <JP>
D01176  
Blonanserin (JAN/INN)  <JP>
D01418  
Tamibarotene (JAN/USAN/INN)  <JP>
D01468  
Nemonapride (JAN/INN)  <JP>
D01562  
Aranidipine (JAN/INN)  <JP>
D01855  
Mozavaptane hydrochloride (JAN)
D04052  
Epinephrine and lidocaine hydrochloride  <JP/US>
D04338  
Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride  <JP>
D04446  
Betamethasone acetate and betamethasone sodium phosphate  <JP/US>
D04813  
Lidocaine hydrochloride and epinephrine bitartrate  <JP/US>
D06273  
Imidafenacin (JAN/INN)  <JP>
D08697  
Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate  <JP>
D09594  
Olmesartan medoxomil and azelnidipine  <JP>
D10433  
Vibegron (JAN/USAN)  <JP/US>
D10524  
Azilsartan and amlodipine besilate  <JP>
D10525  
Valsartan and cilnidipine  <JP>
D10805  
Telmisartan, amlodipine and hydrochlorothiazide  <JP>
D10897  
Teneligliptin and canagliflozin  <JP>
D08856  
Anamorelin hydrochloride (JAN/USAN)  <JP>
D11093  
Avacopan (JAN/USAN/INN)  <JP/US>
D11553  
Lidocaine and tetracaine  <US>
D11616  
Aspirin and omeprazole  <US>
D11628  
Benzhydrocodone and acetaminophen  <US>
D11656  
Azelastine hydrochloride and fluticasone propionate  <US>
D11706  
Omeprazole and sodium bicarbonate  <US>
D11710  
Phentermine and topiramate  <US>
D11851  
Butalbital, acetaminophen, caffeine and codeine phosphate  <US>
D11860  
Butalbital, aspirin, caffeine and codeine  <US>
D12130  
Drospirenone, ethinyl estradiol and levomefolate calcium  <US>
D12265  
Mavacamten (USAN/INN)  <US>
D12269  
Nirmatrelvir and ritonavir  <JP/US>
D12312  
Codeine phosphate and chlorpheniramine maleate  <US>
D12313  
Chlorpheniramine polistirex and codeine polistirex  <US>
Dihydroergotoxine
 D07839  
Dihydroergotoxine
 D02268  
Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18)
Benzhydrocodone
 D10612  
Benzhydrocodone (USAN/INN)
 D10692  
Benzhydrocodone hydrochloride (USAN)
D11886  
Daridorexant (USAN/INN)
 » expand
Class
Metabolizing enzyme substrate
 DG01633  CYP3A/CYP3A4 substrate

» Japanese version

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