Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
 
 Nuclear receptors
 
 Protein kinases
   Serine/threonine kinases
   Receptor serine/threonine kinases (RSTK)
   Receptor tyrosine kinases (RTK)
     EGFR family
     INSR family
     PDGFR family
       PDGFR [HSA:5156 5159] [KO:K04363 K05089]
       PDGFRA [HSA:5156] [KO:K04363]
       PDGFRA* [HSA_VAR:5156v2] [HSA:5156] [KO:K04363]
       FIP1L1-PDGFRA [HSA:5156] [KO:K04363]
       PDGFRB [HSA:5159] [KO:K05089]
       KIT (CD117) [HSA:3815] [KO:K05091]
       KIT* (CD117) [HSA_VAR:3815v1] [HSA:3815] [KO:K05091]
       FLT3 (CD135) [HSA:2322] [KO:K05092]
         D11768  Pacritinib (USAN/INN) <US>
         D08552  Sunitinib (INN)
         D06402  Sunitinib malate (JAN/USAN) <JP/US>
         D08524  Sorafenib (USAN/INN)
         D06272  Sorafenib tosylate (USAN) <JP/US>
         D09955  Quizartinib (USAN/INN)
         D10709  Gilteritinib (USAN/INN)
         D04696  Lestaurtinib (USAN/INN)
         D05819  Semaxanib (USAN/INN)
         D06005  Tandutinib (USAN/INN)
         D08279  Tozasertib (USAN)
         D08344  Tozasertib lactate (USAN)
         D08907  Dovitinib lactate (USAN)
         D10102  Crenolanib (USAN)
         D10103  Crenolanib besylate (USAN)
         D11599  Zotiraciclib (USAN)
         D11600  Zotiraciclib citrate (USAN)
         D12476  Tuspetinib (USAN/INN)
         D12641  Emirodatamab (USAN/INN)
       FLT3* (CD135) [HSA_VAR:2322v1 2322v2] [HSA:2322] [KO:K05092]
       FLT3* (CD135) [HSA_VAR:2322v2] [HSA:2322] [KO:K05092]
     FGFR family
     VEGFR family
     MET family
     TRK family
     EPH family
     AXL family
     ALK family
     TIE family
     ROR family
     RET family
     CCK family
   Non-receptor tyrosine kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 25, 2024

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